Calcitriol//Vitamin D-binding protein//Vitamin transporter activity
Ergocalciferol//Vitamin D-binding protein//Vitamin transporter activity
Cholecalciferol//Vitamin D-binding protein//Vitamin transporter activity
Flunisolide//Corticosteroid-binding globulin//Steroid binding
Lovastatin//Serum albumin//Toxic substance binding
Enflurane//Serum albumin//Toxic substance binding
Alclometasone//Corticosteroid-binding globulin//Steroid binding
Benzatropine//Serum albumin//Toxic substance binding
Diethylstilbestrol//Transthyretin//Identical protein binding
Metoprolol//Serum albumin//Toxic substance binding
Dicoumarol//Serum albumin//Toxic substance binding
Argatroban//Serum albumin//Toxic substance binding
Atomoxetine//Serum albumin//Toxic substance binding
Atomoxetine//High affinity immunoglobulin gamma Fc receptor I//Receptor signaling protein activity
Etonogestrel//Serum albumin//Toxic substance binding
Etonogestrel//Sex hormone-binding globulin//Androgen binding
Morphine//Serum albumin//Toxic substance binding
Acetaminophen//Serum albumin//Toxic substance binding
Gefitinib//Serum albumin//Toxic substance binding
Amitriptyline//Serum albumin//Toxic substance binding
Floxuridine//Thyroxine-binding globulin//Serine-type endopeptidase inhibitor activity
Fluorometholone//Corticosteroid-binding globulin//Steroid binding
Hydromorphone//Serum albumin//Toxic substance binding
Indomethacin//Serum albumin//Toxic substance binding
Ipratropiumbromide//Serum albumin//Toxic substance binding
Methadone//Serum albumin//Toxic substance binding
Diltiazem//Serum albumin//Toxic substance binding
Beclomethasonedipropionate//Corticosteroid-binding globulin//Steroid binding
Acetohexamide//Serum albumin//Toxic substance binding
Betamethasone//Serum albumin//Toxic substance binding
Betamethasone//Corticosteroid-binding globulin//Steroid binding
Levothyroxine//Transthyretin//Identical protein binding
Levothyroxine//Thyroxine-binding globulin//Serine-type endopeptidase inhibitor activity
Levothyroxine//Serum albumin//Toxic substance binding
Imipramine//Serum albumin//Toxic substance binding
Acitretin//Serum albumin//Toxic substance binding
Nabumetone//Serum albumin//Toxic substance binding
Fluoxetine//Serum albumin//Toxic substance binding
Duloxetine//Serum albumin//Toxic substance binding
Chlorpromazine//Serum albumin//Toxic substance binding
Buspirone//Serum albumin//Toxic substance binding
Cisplatin//Serum albumin//Toxic substance binding
Alitretinoin//Cellular retinoic acid-binding protein 2//Transporter activity
Alitretinoin//Cellular retinoic acid-binding protein 1//Transporter activity
Erlotinib//Serum albumin//Toxic substance binding
Ciprofloxacin//Serum albumin//Toxic substance binding
Fluorouracil//Serum albumin//Toxic substance binding
Fluorouracil//Thyroxine-binding globulin//Serine-type endopeptidase inhibitor activity
Lamotrigine//Serum albumin//Toxic substance binding
Hydroxyzine//Serum albumin//Toxic substance binding
Methotrexate//Serum albumin//Toxic substance binding
Clonidine//Serum albumin//Toxic substance binding
Enalapril//Serum albumin//Toxic substance binding
Diclofenac//Transthyretin//Identical protein binding
Diclofenac//Serum albumin//Toxic substance binding
Fluticasonepropionate//Corticosteroid-binding globulin//Steroid binding
Fluticasonepropionate//Solute carrier organic anion transporter family member 1B1//Sodium-independent organic anion transmembrane transporter activity
Fluocinoloneacetonide//Corticosteroid-binding globulin//Steroid binding
Labetalol//Serum albumin//Toxic substance binding
Medroxyprogesteroneacetate//Serum albumin//Toxic substance binding
Chloroquine//Serum albumin//Toxic substance binding
Imatinib//Serum albumin//Toxic substance binding
Niacin//Thyroxine-binding globulin//Serine-type endopeptidase inhibitor activity
Clofibrate//Thyroxine-binding globulin//Serine-type endopeptidase inhibitor activity
Mitotane//Sex hormone-binding globulin//Androgen binding
Mitotane//Corticosteroid-binding globulin//Steroid binding
Mitotane//Thyroxine-binding globulin//Serine-type endopeptidase inhibitor activity
Estrone//Serum albumin//Toxic substance binding
Isoflurophate//Serum albumin//Toxic substance binding
Losartan//Serum albumin//Toxic substance binding
Furosemide//Serum albumin//Toxic substance binding
Furosemide//Thyroxine-binding globulin//Serine-type endopeptidase inhibitor activity
Flurbiprofen//Serum albumin//Toxic substance binding
Apomorphine//Serum albumin//Toxic substance binding
Nateglinide//Serum albumin//Toxic substance binding
Meclizine//Serum albumin//Toxic substance binding
Hydrocortisone//Sex hormone-binding globulin//Androgen binding
Hydrocortisone//Corticosteroid-binding globulin//Steroid binding
Etodolac//Serum albumin//Toxic substance binding
Isoflurane//Serum albumin//Toxic substance binding
Ethotoin//Thyroxine-binding globulin//Serine-type endopeptidase inhibitor activity
Irinotecan//Serum albumin//Toxic substance binding
Estradiol//Sex hormone-binding globulin//Androgen binding
Estradiol//Serum albumin//Toxic substance binding
Estradiol//Fatty acid-binding protein, intestinal//Transporter activity
Mefenamicacid//Serum albumin//Toxic substance binding
Naproxen//Serum albumin//Toxic substance binding
Alfentanil//Serum albumin//Toxic substance binding
Indapamide//Serum albumin//Toxic substance binding
Fentanyl//Serum albumin//Toxic substance binding
Meloxicam//Serum albumin//Toxic substance binding
Diazepam//Serum albumin//Toxic substance binding
Clofazimine//Serum albumin//Toxic substance binding
Diflunisal//Transthyretin//Identical protein binding
Diflunisal//Serum albumin//Toxic substance binding
Etacrynicacid//Serum albumin//Toxic substance binding
Cyclobenzaprine//Serum albumin//Toxic substance binding
Fexofenadine//Serum albumin//Toxic substance binding
Isoniazid//Serum albumin//Toxic substance binding
Methylprednisolone//Serum albumin//Toxic substance binding
Ethinylestradiol//Serum albumin//Toxic substance binding
Ethinylestradiol//Sex hormone-binding globulin//Androgen binding
Formoterol//Serum albumin//Toxic substance binding
Azathioprine//Serum albumin//Toxic substance binding
Doxorubicin//Serum albumin//Toxic substance binding
Letrozole//Serum albumin//Toxic substance binding
Ketoprofen//Serum albumin//Toxic substance binding
Clobetasolpropionate//Corticosteroid-binding globulin//Steroid binding
Clobetasolpropionate//Serum albumin//Toxic substance binding
Glyburide//Serum albumin//Toxic substance binding
Ketoconazole//Serum albumin//Toxic substance binding
Ketoconazole//Sex hormone-binding globulin//Androgen binding
Irbesartan//Serum albumin//Toxic substance binding
Fenofibrate//Serum albumin//Toxic substance binding
Ibuprofen//Serum albumin//Toxic substance binding
Glipizide//Serum albumin//Toxic substance binding
Clonazepam//Serum albumin//Toxic substance binding
Atorvastatin//Serum albumin//Toxic substance binding
Miconazole//Serum albumin//Toxic substance binding
Amiodarone//Serum albumin//Toxic substance binding
Gliclazide//Serum albumin//Toxic substance binding
Dutasteride//Serum albumin//Toxic substance binding
Carvedilol//Serum albumin//Toxic substance binding
Levofloxacin//Serum albumin//Toxic substance binding
Doxepin//Serum albumin//Toxic substance binding
Halothane//Serum albumin//Toxic substance binding
Arsenictrioxide//Serum albumin//Toxic substance binding
Naloxone//Serum albumin//Toxic substance binding
Flecainide//Serum albumin//Toxic substance binding
Captopril//Serum albumin//Toxic substance binding
Ceftriaxone//Serum albumin//Toxic substance binding
Dantrolene//Thyroxine-binding globulin//Serine-type endopeptidase inhibitor activity
Budesonide//Corticosteroid-binding globulin//Steroid binding
Budesonide//Serum albumin//Toxic substance binding
Dexamethasone//Serum albumin//Toxic substance binding
Levodopa//Serum albumin//Toxic substance binding
Aripiprazole//Serum albumin//Toxic substance binding
Gemfibrozil//Serum albumin//Toxic substance binding
Clomipramine//Serum albumin//Toxic substance binding
Hydralazine//Serum albumin//Toxic substance binding
Fosphenytoin//Serum albumin//Toxic substance binding
Fosphenytoin//Thyroxine-binding globulin//Serine-type endopeptidase inhibitor activity
Cefazolin//Serum albumin//Toxic substance binding
Ephedrine//Serum albumin//Toxic substance binding
Colchicine//Serum albumin//Toxic substance binding
Digitoxin//Serum albumin//Toxic substance binding
Danazol//Sex hormone-binding globulin//Androgen binding
Ciclesonide//Corticosteroid-binding globulin//Steroid binding
Acenocoumarol//Serum albumin//Toxic substance binding
Liotrix//Transthyretin//Identical protein binding
Liotrix//Thyroxine-binding globulin//Serine-type endopeptidase inhibitor activity
Liotrix//Serum albumin//Toxic substance binding
Ketazolam//Serum albumin//Toxic substance binding
Hydroxychloroquine//Serum albumin//Toxic substance binding
Estronesulfate//Sex hormone-binding globulin//Androgen binding
Estronesulfate//Serum albumin//Toxic substance binding
Dronedarone//Serum albumin//Toxic substance binding
Nebivolol//Serum albumin//Toxic substance binding
Abiraterone//Serum albumin//Toxic substance binding
Asenapine//Serum albumin//Toxic substance binding
Levocetirizine//Serum albumin//Toxic substance binding
Methyltestosterone//Serum albumin//Toxic substance binding
Methyltestosterone//Sex hormone-binding globulin//Androgen binding
Fospropofol//Serum albumin//Toxic substance binding
Ivacaftor//Serum albumin//Toxic substance binding
Mirabegron//Serum albumin//Toxic substance binding
Enzalutamide//Serum albumin//Toxic substance binding
Enzalutamide//Thyroxine-binding globulin//Serine-type endopeptidase inhibitor activity
Fluticasonefuroate//Corticosteroid-binding globulin//Steroid binding
Fluticasonefuroate//Multidrug resistance protein 1//Xenobiotic-transporting atpase activity
Fluticasonefuroate//Solute carrier organic anion transporter family member 1B1//Sodium-independent organic anion transmembrane transporter activity
Macitentan//Serum albumin//Toxic substance binding
Ibrutinib//Serum albumin//Toxic substance binding
Lorpiprazole//Serum albumin//Toxic substance binding
Blonanserin//Serum albumin//Toxic substance binding
Aranidipine//Serum albumin//Toxic substance binding
Imidafenacin//Serum albumin//Toxic substance binding
Lumacaftor//Serum albumin//Toxic substance binding
Dexchlorpheniraminemaleate//Solute carrier family 22 member 1//Secondary active organic cation transmembrane transporter activity
Dexchlorpheniraminemaleate//Solute carrier family 22 member 2//Quaternary ammonium group transmembrane transporter activity
Butamben//Serum albumin//Toxic substance binding
Ertugliflozin//Serum albumin//Toxic substance binding
Neratinib//Serum albumin//Toxic substance binding
Abemaciclib//Serum albumin//Toxic substance binding
Copanlisib//Serum albumin//Toxic substance binding
Estradiolacetate//Sex hormone-binding globulin//Androgen binding
Estradiolacetate//Serum albumin//Toxic substance binding
Estradiolacetate//Fatty acid-binding protein, intestinal//Transporter activity
Estradiolbenzoate//Sex hormone-binding globulin//Androgen binding
Estradiolbenzoate//Serum albumin//Toxic substance binding
Estradiolbenzoate//Fatty acid-binding protein, intestinal//Transporter activity
Estradiolcypionate//Sex hormone-binding globulin//Androgen binding
Estradiolcypionate//Serum albumin//Toxic substance binding
Estradiolcypionate//Fatty acid-binding protein, intestinal//Transporter activity
Estradioldienanthate//Sex hormone-binding globulin//Androgen binding
Estradioldienanthate//Serum albumin//Toxic substance binding
Estradioldienanthate//Fatty acid-binding protein, intestinal//Transporter activity
Estradiolvalerate//Sex hormone-binding globulin//Androgen binding
Estradiolvalerate//Serum albumin//Toxic substance binding
Estradiolvalerate//Fatty acid-binding protein, intestinal//Transporter activity
Cyclosporine//Multidrug resistance protein 1//Xenobiotic-transporting atpase activity
Cyclosporine//Bile salt export pump//Transporter activity
Cyclosporine//Sodium/bile acid cotransporter//Virus receptor activity
Cyclosporine//Solute carrier family 22 member 6//Sodium-independent organic anion transmembrane transporter activity
Cyclosporine//Multidrug resistance-associated protein 7//Atpase activity, coupled to transmembrane movement of substances
Cyclosporine//Canalicular multispecific organic anion transporter 1//Organic anion transmembrane transporter activity
Cyclosporine//ATP-binding cassette sub-family G member 2//Xenobiotic-transporting atpase activity
Cyclosporine//Solute carrier organic anion transporter family member 1B1//Sodium-independent organic anion transmembrane transporter activity
Cyclosporine//Solute carrier organic anion transporter family member 1B3//Sodium-independent organic anion transmembrane transporter activity
Cyanocobalamin//Protein amnionless//Receptor binding
Cyanocobalamin//Transcobalamin-1//Cobalamin binding
Cyanocobalamin//Transcobalamin-2//Metal ion binding
Cyanocobalamin//Gastric intrinsic factor//Cobalamin binding
Cyanocobalamin//Cubilin//Transporter activity
Cyanocobalamin//Low-density lipoprotein receptor-related protein 2//Calcium ion binding
Cyanocobalamin//Multidrug resistance-associated protein 1//Transporter activity
Choline//Solute carrier family 22 member 2//Quaternary ammonium group transmembrane transporter activity
Choline//Solute carrier family 22 member 1//Secondary active organic cation transmembrane transporter activity
Choline//Solute carrier family 22 member 3//Toxin transporter activity
Choline//Solute carrier family 22 member 5//Symporter activity
Choline//Solute carrier family 22 member 4//Symporter activity
Choline//Choline transporter-like protein 2//Signal transducer activity
    Lglutamine//Sodium-coupled neutral amino acid transporter 3//Symporter activity
    Lglutamine//Neutral amino acid transporter B(0)//Virus receptor activity
    Lglutamine//Large neutral amino acids transporter small subunit 1//Peptide antigen binding
    Lglutamine//Large neutral amino acids transporter small subunit 2//Toxin transporter activity
    Lglutamine//b(0,+)-type amino acid transporter 1//Peptide antigen binding
    Lglutamine//Monocarboxylate transporter 10//Transporter activity
Methionine//Monocarboxylate transporter 10//Transporter activity
Ltryptophan//Monocarboxylate transporter 8//Transporter activity
Ltryptophan//Monocarboxylate transporter 10//Transporter activity
Folicacid//ATP-binding cassette sub-family C member 11//Purine nucleotide transmembrane transporter activity
Folicacid//Canalicular multispecific organic anion transporter 2//Organic anion transmembrane transporter activity
Folicacid//Solute carrier family 22 member 6//Sodium-independent organic anion transmembrane transporter activity
Folicacid//Multidrug resistance-associated protein 4//Atpase activity, coupled to transmembrane movement of substances
Folicacid//ATP-binding cassette sub-family G member 2//Xenobiotic-transporting atpase activity
Fluvoxamine//Multidrug resistance protein 1//Xenobiotic-transporting atpase activity
Fluvoxamine//Bile salt export pump//Transporter activity
Amphetamine//Solute carrier family 22 member 3//Toxin transporter activity
Amphetamine//Solute carrier family 22 member 5//Symporter activity
Bortezomib//Multidrug resistance protein 1//Xenobiotic-transporting atpase activity
Bortezomib//Solute carrier organic anion transporter family member 1B3//Sodium-independent organic anion transmembrane transporter activity
Erythromycin//Solute carrier organic anion transporter family member 1B3//Sodium-independent organic anion transmembrane transporter activity
Erythromycin//Bile salt export pump//Transporter activity
Erythromycin//Multidrug resistance protein 1//Xenobiotic-transporting atpase activity
Erythromycin//Solute carrier organic anion transporter family member 1B1//Sodium-independent organic anion transmembrane transporter activity
Erythromycin//Canalicular multispecific organic anion transporter 1//Organic anion transmembrane transporter activity
Erythromycin//Solute carrier organic anion transporter family member 1A2//Sodium-independent organic anion transmembrane transporter activity
Caffeine//ATP-binding cassette sub-family G member 2//Xenobiotic-transporting atpase activity
Dofetilide//Solute carrier family 22 member 2//Quaternary ammonium group transmembrane transporter activity
Azithromycin//Multidrug resistance protein 1//Xenobiotic-transporting atpase activity
Azithromycin//Canalicular multispecific organic anion transporter 1//Organic anion transmembrane transporter activity
Midodrine//Solute carrier family 15 member 1//Proton-dependent oligopeptide secondary active transmembrane transporter activity
Citalopram//Multidrug resistance protein 1//Xenobiotic-transporting atpase activity
Eletriptan//Multidrug resistance protein 1//Xenobiotic-transporting atpase activity
Glimepiride//Bile salt export pump//Transporter activity
Lovastatin//Multidrug resistance protein 1//Xenobiotic-transporting atpase activity
Lovastatin//Solute carrier organic anion transporter family member 1A2//Sodium-independent organic anion transmembrane transporter activity
Lovastatin//Solute carrier organic anion transporter family member 1B1//Sodium-independent organic anion transmembrane transporter activity
Lovastatin//Canalicular multispecific organic anion transporter 1//Organic anion transmembrane transporter activity
Lovastatin//Bile salt export pump//Transporter activity
Lovastatin//Solute carrier organic anion transporter family member 2B1//Sodium-independent organic anion transmembrane transporter activity
Lovastatin//Solute carrier organic anion transporter family member 1B3//Sodium-independent organic anion transmembrane transporter activity
Cladribine//ATP-binding cassette sub-family G member 2//Xenobiotic-transporting atpase activity
Cladribine//Solute carrier family 28 member 3//Pyrimidine- and adenine-specific:sodium symporter activity
Cabergoline//Multidrug resistance protein 1//Xenobiotic-transporting atpase activity
Doxycycline//Solute carrier family 22 member 6//Sodium-independent organic anion transmembrane transporter activity
Doxycycline//ATP-binding cassette sub-family B member 5//Efflux transmembrane transporter activity
Diethylstilbestrol//ATP-binding cassette sub-family G member 2//Xenobiotic-transporting atpase activity
Diethylstilbestrol//Multidrug resistance protein 1//Xenobiotic-transporting atpase activity
Diethylstilbestrol//Solute carrier organic anion transporter family member 1B1//Sodium-independent organic anion transmembrane transporter activity
Diethylstilbestrol//Solute carrier organic anion transporter family member 2B1//Sodium-independent organic anion transmembrane transporter activity
Diethylstilbestrol//Bile salt export pump//Transporter activity
Clotrimazole//Multidrug resistance protein 1//Xenobiotic-transporting atpase activity
Clotrimazole//Bile salt export pump//Transporter activity
Clotrimazole//Solute carrier organic anion transporter family member 1B1//Sodium-independent organic anion transmembrane transporter activity
Clotrimazole//Solute carrier organic anion transporter family member 1B3//Sodium-independent organic anion transmembrane transporter activity
Metoprolol//Solute carrier family 22 member 2//Quaternary ammonium group transmembrane transporter activity
Isradipine//Bile salt export pump//Transporter activity
Amsacrine//Multidrug resistance protein 1//Xenobiotic-transporting atpase activity
Disopyramide//Solute carrier family 22 member 1//Secondary active organic cation transmembrane transporter activity
Disopyramide//Solute carrier family 22 member 2//Quaternary ammonium group transmembrane transporter activity
Lidocaine//Solute carrier family 22 member 5//Symporter activity
Lidocaine//Multidrug resistance protein 1//Xenobiotic-transporting atpase activity
Morphine//Multidrug resistance protein 1//Xenobiotic-transporting atpase activity
Acetaminophen//Multidrug resistance protein 1//Xenobiotic-transporting atpase activity
Gefitinib//Multidrug resistance protein 1//Xenobiotic-transporting atpase activity
Gefitinib//ATP-binding cassette sub-family G member 2//Xenobiotic-transporting atpase activity
Codeine//Solute carrier family 22 member 1//Secondary active organic cation transmembrane transporter activity
Dihydroergotamine//Multidrug resistance protein 1//Xenobiotic-transporting atpase activity
Amitriptyline//Multidrug resistance protein 1//Xenobiotic-transporting atpase activity
Indomethacin//Canalicular multispecific organic anion transporter 2//Organic anion transmembrane transporter activity
Indomethacin//Multidrug resistance-associated protein 4//Atpase activity, coupled to transmembrane movement of substances
Indomethacin//Multidrug resistance-associated protein 6//Transporter activity
Indomethacin//Multidrug resistance protein 1//Xenobiotic-transporting atpase activity
Indomethacin//Multidrug resistance-associated protein 1//Transporter activity
Indomethacin//Solute carrier organic anion transporter family member 1A2//Sodium-independent organic anion transmembrane transporter activity
Indomethacin//Solute carrier family 22 member 6//Sodium-independent organic anion transmembrane transporter activity
Indomethacin//Solute carrier family 22 member 8//Sodium-independent organic anion transmembrane transporter activity
Indomethacin//Canalicular multispecific organic anion transporter 1//Organic anion transmembrane transporter activity
Indomethacin//ATP-binding cassette sub-family C member 11//Purine nucleotide transmembrane transporter activity
Indomethacin//Solute carrier family 22 member 11//Sodium-independent organic anion transmembrane transporter activity
Indomethacin//Sodium/bile acid cotransporter//Virus receptor activity
Indomethacin//Solute carrier family 22 member 7//Sodium-independent organic anion transmembrane transporter activity
Indomethacin//Solute carrier organic anion transporter family member 1B1//Sodium-independent organic anion transmembrane transporter activity
Indomethacin//Bile salt export pump//Transporter activity
Ipratropiumbromide//Solute carrier family 22 member 5//Symporter activity
Ipratropiumbromide//Solute carrier family 22 member 4//Symporter activity
Methadone//Multidrug resistance protein 1//Xenobiotic-transporting atpase activity
Diltiazem//Multidrug resistance protein 1//Xenobiotic-transporting atpase activity
Mefloquine//Multidrug resistance protein 1//Xenobiotic-transporting atpase activity
Clozapine//Multidrug resistance protein 1//Xenobiotic-transporting atpase activity
Mirtazapine//Sodium-dependent serotonin transporter//Serotonin:sodium symporter activity
Amlodipine//Multidrug resistance protein 1//Xenobiotic-transporting atpase activity
Digoxin//Multidrug resistance protein 1//Xenobiotic-transporting atpase activity
Digoxin//Solute carrier organic anion transporter family member 4C1//Sodium-independent organic anion transmembrane transporter activity
Digoxin//Bile salt export pump//Transporter activity
Digoxin//Solute carrier organic anion transporter family member 1A2//Sodium-independent organic anion transmembrane transporter activity
Digoxin//Organic solute transporter subunit alpha//Transporter activity
Digoxin//Organic solute transporter subunit beta//Transporter activity
Digoxin//Solute carrier organic anion transporter family member 1B1//Sodium-independent organic anion transmembrane transporter activity
Beclomethasonedipropionate//Multidrug resistance protein 1//Xenobiotic-transporting atpase activity
Beclomethasonedipropionate//ATP-binding cassette sub-family G member 2//Xenobiotic-transporting atpase activity
Beclomethasonedipropionate//Solute carrier organic anion transporter family member 1B1//Sodium-independent organic anion transmembrane transporter activity
Beclomethasonedipropionate//Solute carrier organic anion transporter family member 1B3//Sodium-independent organic anion transmembrane transporter activity
Allopurinol//Solute carrier family 22 member 8//Sodium-independent organic anion transmembrane transporter activity
Allopurinol//Solute carrier family 22 member 7//Sodium-independent organic anion transmembrane transporter activity
Allopurinol//ATP-binding cassette sub-family G member 2//Xenobiotic-transporting atpase activity
Allopurinol//Solute carrier family 22 member 2//Quaternary ammonium group transmembrane transporter activity
Cerivastatin//Multidrug resistance protein 1//Xenobiotic-transporting atpase activity
Cerivastatin//Canalicular multispecific organic anion transporter 1//Organic anion transmembrane transporter activity
Cerivastatin//ATP-binding cassette sub-family G member 2//Xenobiotic-transporting atpase activity
Cerivastatin//Solute carrier organic anion transporter family member 1B1//Sodium-independent organic anion transmembrane transporter activity
Cerivastatin//Bile salt export pump//Transporter activity
Gemcitabine//Multidrug resistance protein 1//Xenobiotic-transporting atpase activity
Gemcitabine//Multidrug resistance-associated protein 7//Atpase activity, coupled to transmembrane movement of substances
Gemcitabine//Equilibrative nucleoside transporter 1//Nucleoside transmembrane transporter activity
Gemcitabine//Sodium/nucleoside cotransporter 1//Pyrimidine- and adenine-specific:sodium symporter activity
Gemcitabine//Equilibrative nucleoside transporter 2//Nucleoside transmembrane transporter activity
Gemcitabine//Solute carrier family 28 member 3//Pyrimidine- and adenine-specific:sodium symporter activity
Betamethasone//Multidrug resistance protein 1//Xenobiotic-transporting atpase activity
Epirubicin//Multidrug resistance-associated protein 1//Transporter activity
Chloramphenicol//Solute carrier family 22 member 6//Sodium-independent organic anion transmembrane transporter activity
Lansoprazole//ATP-binding cassette sub-family G member 2//Xenobiotic-transporting atpase activity
Lansoprazole//Multidrug resistance protein 1//Xenobiotic-transporting atpase activity
Lansoprazole//Solute carrier family 22 member 8//Sodium-independent organic anion transmembrane transporter activity
Lansoprazole//Solute carrier family 22 member 1//Secondary active organic cation transmembrane transporter activity
Lansoprazole//Solute carrier family 22 member 2//Quaternary ammonium group transmembrane transporter activity
Lansoprazole//Solute carrier family 22 member 3//Toxin transporter activity
Levothyroxine//Solute carrier organic anion transporter family member 1C1//Thyroid hormone transmembrane transporter activity
Levothyroxine//Monocarboxylate transporter 8//Transporter activity
Levothyroxine//Multidrug resistance protein 1//Xenobiotic-transporting atpase activity
Levothyroxine//Solute carrier organic anion transporter family member 1A2//Sodium-independent organic anion transmembrane transporter activity
Levothyroxine//Solute carrier organic anion transporter family member 1B1//Sodium-independent organic anion transmembrane transporter activity
Levothyroxine//Solute carrier organic anion transporter family member 1B3//Sodium-independent organic anion transmembrane transporter activity
Levothyroxine//Solute carrier organic anion transporter family member 4A1//Thyroid hormone transmembrane transporter activity
Levothyroxine//Solute carrier organic anion transporter family member 4C1//Sodium-independent organic anion transmembrane transporter activity
Levothyroxine//Large neutral amino acids transporter small subunit 1//Peptide antigen binding
Levothyroxine//Solute carrier organic anion transporter family member 2B1//Sodium-independent organic anion transmembrane transporter activity
Loratadine//Multidrug resistance protein 1//Xenobiotic-transporting atpase activity
Loratadine//Bile salt export pump//Transporter activity
Imipramine//Multidrug resistance protein 1//Xenobiotic-transporting atpase activity
Imipramine//Solute carrier family 22 member 2//Quaternary ammonium group transmembrane transporter activity
Imipramine//Solute carrier family 22 member 3//Toxin transporter activity
Imipramine//Solute carrier family 22 member 4//Symporter activity
Dronabinol//Multidrug resistance protein 1//Xenobiotic-transporting atpase activity
Dronabinol//ATP-binding cassette sub-family G member 2//Xenobiotic-transporting atpase activity
Montelukast//Solute carrier organic anion transporter family member 2B1//Sodium-independent organic anion transmembrane transporter activity
Fluoxetine//Multidrug resistance protein 1//Xenobiotic-transporting atpase activity
Duloxetine//Multidrug resistance protein 1//Xenobiotic-transporting atpase activity
Chlorpromazine//Multidrug resistance protein 1//Xenobiotic-transporting atpase activity
Chlorpromazine//Bile salt export pump//Transporter activity
Celecoxib//Multidrug resistance-associated protein 4//Atpase activity, coupled to transmembrane movement of substances
Celecoxib//Bile salt export pump//Transporter activity
Celecoxib//Multidrug resistance protein 1//Xenobiotic-transporting atpase activity
Celecoxib//ATP-binding cassette sub-family G member 2//Xenobiotic-transporting atpase activity
Buspirone//Multidrug resistance protein 1//Xenobiotic-transporting atpase activity
Cimetidine//Multidrug resistance protein 1//Xenobiotic-transporting atpase activity
Cimetidine//Solute carrier family 22 member 2//Quaternary ammonium group transmembrane transporter activity
Cimetidine//Solute carrier family 22 member 1//Secondary active organic cation transmembrane transporter activity
Cimetidine//Solute carrier family 22 member 3//Toxin transporter activity
Cimetidine//Solute carrier family 22 member 5//Symporter activity
Cimetidine//Solute carrier family 22 member 6//Sodium-independent organic anion transmembrane transporter activity
Cimetidine//Solute carrier family 22 member 8//Sodium-independent organic anion transmembrane transporter activity
Cimetidine//Multidrug and toxin extrusion protein 1//Monovalent cation:proton antiporter activity
Cimetidine//Solute carrier family 22 member 4//Symporter activity
Cimetidine//Solute carrier family 22 member 11//Sodium-independent organic anion transmembrane transporter activity
Cimetidine//Solute carrier family 22 member 7//Sodium-independent organic anion transmembrane transporter activity
Cimetidine//Bile salt export pump//Transporter activity
Cimetidine//Multidrug and toxin extrusion protein 2//Drug transmembrane transporter activity
Haloperidol//Multidrug resistance protein 1//Xenobiotic-transporting atpase activity
Cisplatin//Canalicular multispecific organic anion transporter 2//Organic anion transmembrane transporter activity
Cisplatin//Multidrug resistance-associated protein 5//Organic anion transmembrane transporter activity
Cisplatin//Canalicular multispecific organic anion transporter 1//Organic anion transmembrane transporter activity
Cisplatin//Solute carrier family 22 member 2//Quaternary ammonium group transmembrane transporter activity
Cisplatin//Multidrug resistance-associated protein 6//Transporter activity
Cisplatin//Multidrug resistance protein 1//Xenobiotic-transporting atpase activity
Cisplatin//ATP-binding cassette sub-family G member 2//Xenobiotic-transporting atpase activity
Albendazole//Multidrug resistance protein 1//Xenobiotic-transporting atpase activity
Alitretinoin//Multidrug resistance protein 1//Xenobiotic-transporting atpase activity
Erlotinib//ATP-binding cassette sub-family G member 2//Xenobiotic-transporting atpase activity
Erlotinib//Multidrug resistance protein 1//Xenobiotic-transporting atpase activity
Erlotinib//Solute carrier organic anion transporter family member 2B1//Sodium-independent organic anion transmembrane transporter activity
Ciprofloxacin//Multidrug resistance protein 1//Xenobiotic-transporting atpase activity
Ciprofloxacin//Multidrug and toxin extrusion protein 1//Monovalent cation:proton antiporter activity
Ciprofloxacin//Multidrug and toxin extrusion protein 2//Drug transmembrane transporter activity
Benazepril//Solute carrier family 15 member 1//Proton-dependent oligopeptide secondary active transmembrane transporter activity
Benazepril//Solute carrier family 15 member 2//Peptide:proton symporter activity
Fluorouracil//Solute carrier family 22 member 7//Sodium-independent organic anion transmembrane transporter activity
Fluorouracil//Equilibrative nucleoside transporter 1//Nucleoside transmembrane transporter activity
Fluorouracil//ATP-binding cassette sub-family G member 2//Xenobiotic-transporting atpase activity
Fluorouracil//Canalicular multispecific organic anion transporter 2//Organic anion transmembrane transporter activity
Fluorouracil//Multidrug resistance-associated protein 4//Atpase activity, coupled to transmembrane movement of substances
Fluorouracil//Multidrug resistance-associated protein 5//Organic anion transmembrane transporter activity
Lamotrigine//Multidrug resistance protein 1//Xenobiotic-transporting atpase activity
Lamotrigine//Solute carrier family 22 member 2//Quaternary ammonium group transmembrane transporter activity
Lamotrigine//Solute carrier family 22 member 1//Secondary active organic cation transmembrane transporter activity
Hydroxyzine//Multidrug resistance protein 1//Xenobiotic-transporting atpase activity
Bosentan//Bile salt export pump//Transporter activity
Methotrexate//Canalicular multispecific organic anion transporter 2//Organic anion transmembrane transporter activity
Methotrexate//Multidrug resistance-associated protein 4//Atpase activity, coupled to transmembrane movement of substances
Methotrexate//Multidrug resistance-associated protein 1//Transporter activity
Methotrexate//Solute carrier family 22 member 6//Sodium-independent organic anion transmembrane transporter activity
Methotrexate//Multidrug resistance-associated protein 7//Atpase activity, coupled to transmembrane movement of substances
Methotrexate//Solute carrier family 22 member 8//Sodium-independent organic anion transmembrane transporter activity
Methotrexate//Canalicular multispecific organic anion transporter 1//Organic anion transmembrane transporter activity
Methotrexate//Multidrug resistance protein 1//Xenobiotic-transporting atpase activity
Methotrexate//Solute carrier organic anion transporter family member 1A2//Sodium-independent organic anion transmembrane transporter activity
Methotrexate//Monocarboxylate transporter 1//Symporter activity
Methotrexate//ATP-binding cassette sub-family C member 11//Purine nucleotide transmembrane transporter activity
Methotrexate//Solute carrier organic anion transporter family member 1B3//Sodium-independent organic anion transmembrane transporter activity
Methotrexate//Solute carrier family 22 member 11//Sodium-independent organic anion transmembrane transporter activity
Methotrexate//Solute carrier organic anion transporter family member 1C1//Thyroid hormone transmembrane transporter activity
Methotrexate//Solute carrier organic anion transporter family member 3A1//Sodium-independent organic anion transmembrane transporter activity
Methotrexate//ATP-binding cassette sub-family G member 2//Xenobiotic-transporting atpase activity
Methotrexate//Solute carrier family 22 member 7//Sodium-independent organic anion transmembrane transporter activity
Methotrexate//Solute carrier organic anion transporter family member 1B1//Sodium-independent organic anion transmembrane transporter activity
Methotrexate//Solute carrier organic anion transporter family member 4C1//Sodium-independent organic anion transmembrane transporter activity
Methotrexate//Folate receptor alpha//Receptor activity
Methotrexate//Solute carrier family 15 member 1//Proton-dependent oligopeptide secondary active transmembrane transporter activity
Carbamazepine//Multidrug resistance protein 1//Xenobiotic-transporting atpase activity
Carbamazepine//RalA-binding protein 1//Transmembrane transporter activity
Carbamazepine//Canalicular multispecific organic anion transporter 1//Organic anion transmembrane transporter activity
Atropine//Bile salt export pump//Transporter activity
Clonidine//Solute carrier family 22 member 3//Toxin transporter activity
Clonidine//Solute carrier family 22 member 5//Symporter activity
Clonidine//Solute carrier family 22 member 4//Symporter activity
Clonidine//Multidrug resistance protein 1//Xenobiotic-transporting atpase activity
Enalapril//Multidrug resistance protein 1//Xenobiotic-transporting atpase activity
Enalapril//Solute carrier family 15 member 1//Proton-dependent oligopeptide secondary active transmembrane transporter activity
Enalapril//Solute carrier family 22 member 6//Sodium-independent organic anion transmembrane transporter activity
Enalapril//Solute carrier family 22 member 8//Sodium-independent organic anion transmembrane transporter activity
Enalapril//Solute carrier family 22 member 7//Sodium-independent organic anion transmembrane transporter activity
Enalapril//Solute carrier organic anion transporter family member 1A2//Sodium-independent organic anion transmembrane transporter activity
Diclofenac//Solute carrier family 22 member 6//Sodium-independent organic anion transmembrane transporter activity
Diclofenac//Multidrug resistance-associated protein 4//Atpase activity, coupled to transmembrane movement of substances
Diclofenac//Multidrug resistance-associated protein 1//Transporter activity
Diclofenac//Solute carrier family 22 member 8//Sodium-independent organic anion transmembrane transporter activity
Diclofenac//Solute carrier family 22 member 11//Sodium-independent organic anion transmembrane transporter activity
Diclofenac//Solute carrier organic anion transporter family member 1C1//Thyroid hormone transmembrane transporter activity
Diclofenac//Solute carrier organic anion transporter family member 1B1//Sodium-independent organic anion transmembrane transporter activity
Diclofenac//Bile salt export pump//Transporter activity
Diclofenac//Sodium channel protein type 4 subunit alpha//Voltage-gated sodium channel activity
Diclofenac//Acid-sensing ion channel 1//Ligand-gated sodium channel activity
Diclofenac//Potassium voltage-gated channel subfamily KQT member 2//Voltage-gated potassium channel activity
Diclofenac//Potassium voltage-gated channel subfamily KQT member 3//Voltage-gated potassium channel activity
Diclofenac//Multidrug resistance protein 1//Xenobiotic-transporting atpase activity
Fluticasonepropionate//Multidrug resistance protein 1//Xenobiotic-transporting atpase activity
Fluticasonepropionate//Solute carrier organic anion transporter family member 1B1//Sodium-independent organic anion transmembrane transporter activity
Doxazosin//Multidrug resistance protein 1//Xenobiotic-transporting atpase activity
Doxazosin//Solute carrier family 22 member 1//Secondary active organic cation transmembrane transporter activity
Amiloride//Solute carrier family 22 member 2//Quaternary ammonium group transmembrane transporter activity
Amiloride//Solute carrier family 22 member 4//Symporter activity
Labetalol//ATP-binding cassette sub-family B member 5//Efflux transmembrane transporter activity
Ivermectin//Multidrug resistance protein 1//Xenobiotic-transporting atpase activity
Ivermectin//Multidrug resistance-associated protein 1//Transporter activity
Ivermectin//Canalicular multispecific organic anion transporter 1//Organic anion transmembrane transporter activity
Ivermectin//ATP-binding cassette sub-family G member 2//Xenobiotic-transporting atpase activity
Ivermectin//Solute carrier organic anion transporter family member 1B1//Sodium-independent organic anion transmembrane transporter activity
Ivermectin//Solute carrier organic anion transporter family member 1B3//Sodium-independent organic anion transmembrane transporter activity
Medroxyprogesteroneacetate//Multidrug resistance protein 1//Xenobiotic-transporting atpase activity
Chloroquine//Multidrug resistance protein 1//Xenobiotic-transporting atpase activity
Bisoprolol//Multidrug resistance protein 1//Xenobiotic-transporting atpase activity
Amodiaquine//Multidrug resistance protein 1//Xenobiotic-transporting atpase activity
Imatinib//Solute carrier family 22 member 1//Secondary active organic cation transmembrane transporter activity
Imatinib//Multidrug resistance protein 1//Xenobiotic-transporting atpase activity
Imatinib//Solute carrier family 22 member 2//Quaternary ammonium group transmembrane transporter activity
Imatinib//ATP-binding cassette sub-family G member 2//Xenobiotic-transporting atpase activity
Imatinib//ATP-binding cassette sub-family A member 3//Transporter activity
Imatinib//Bile salt export pump//Transporter activity
Nicardipine//Multidrug resistance protein 1//Xenobiotic-transporting atpase activity
Nicardipine//Solute carrier organic anion transporter family member 1B1//Sodium-independent organic anion transmembrane transporter activity
Nicardipine//Bile salt export pump//Transporter activity
Fluphenazine//Multidrug resistance protein 1//Xenobiotic-transporting atpase activity
Niacin//Solute carrier family 22 member 5//Symporter activity
Niacin//Solute carrier organic anion transporter family member 2B1//Sodium-independent organic anion transmembrane transporter activity
Niacin//Monocarboxylate transporter 1//Symporter activity
Niacin//Sodium-coupled monocarboxylate transporter 1//Symporter activity
Niacin//Monocarboxylate transporter 4//Symporter activity
Clofarabine//ATP-binding cassette sub-family G member 2//Xenobiotic-transporting atpase activity
Astemizole//Multidrug resistance protein 1//Xenobiotic-transporting atpase activity
Astemizole//Bile salt export pump//Transporter activity
Adenosine//Solute carrier family 28 member 3//Pyrimidine- and adenine-specific:sodium symporter activity
Mitotane//Multidrug resistance protein 1//Xenobiotic-transporting atpase activity
Estrone//Solute carrier organic anion transporter family member 2B1//Sodium-independent organic anion transmembrane transporter activity
Estrone//Multidrug resistance protein 1//Xenobiotic-transporting atpase activity
Estrone//Solute carrier organic anion transporter family member 1A2//Sodium-independent organic anion transmembrane transporter activity
Estrone//ATP-binding cassette sub-family G member 2//Xenobiotic-transporting atpase activity
Estrone//Solute carrier organic anion transporter family member 1B1//Sodium-independent organic anion transmembrane transporter activity
Estrone//Solute carrier family 22 member 8//Sodium-independent organic anion transmembrane transporter activity
Epinephrine//Solute carrier family 22 member 2//Quaternary ammonium group transmembrane transporter activity
Epinephrine//Solute carrier family 22 member 1//Secondary active organic cation transmembrane transporter activity
Chlorpropamide//Solute carrier family 15 member 1//Proton-dependent oligopeptide secondary active transmembrane transporter activity
Chlorpropamide//Solute carrier family 15 member 2//Peptide:proton symporter activity
Chlorpropamide//Solute carrier family 22 member 6//Sodium-independent organic anion transmembrane transporter activity
Galantamine//Multidrug resistance protein 1//Xenobiotic-transporting atpase activity
Losartan//Multidrug resistance protein 1//Xenobiotic-transporting atpase activity
Losartan//Solute carrier family 22 member 6//Sodium-independent organic anion transmembrane transporter activity
Losartan//Bile salt export pump//Transporter activity
Mycophenolatemofetil//Solute carrier organic anion transporter family member 1B1//Sodium-independent organic anion transmembrane transporter activity
Mycophenolatemofetil//Solute carrier organic anion transporter family member 1B3//Sodium-independent organic anion transmembrane transporter activity
Mycophenolatemofetil//ATP-binding cassette sub-family G member 2//Xenobiotic-transporting atpase activity
Mycophenolatemofetil//Multidrug resistance protein 1//Xenobiotic-transporting atpase activity
Mycophenolatemofetil//Canalicular multispecific organic anion transporter 1//Organic anion transmembrane transporter activity
Flurazepam//Multidrug resistance protein 1//Xenobiotic-transporting atpase activity
Flurazepam//Solute carrier family 22 member 2//Quaternary ammonium group transmembrane transporter activity
Daunorubicin//Multidrug resistance protein 1//Xenobiotic-transporting atpase activity
Daunorubicin//Multidrug resistance-associated protein 1//Transporter activity
Daunorubicin//Multidrug resistance-associated protein 7//Atpase activity, coupled to transmembrane movement of substances
Daunorubicin//Canalicular multispecific organic anion transporter 1//Organic anion transmembrane transporter activity
Daunorubicin//Multidrug resistance-associated protein 6//Transporter activity
Daunorubicin//Bile salt export pump//Transporter activity
Daunorubicin//ATP-binding cassette sub-family G member 2//Xenobiotic-transporting atpase activity
Furosemide//Solute carrier family 22 member 6//Sodium-independent organic anion transmembrane transporter activity
Furosemide//Solute carrier family 22 member 5//Symporter activity
Furosemide//Solute carrier family 22 member 8//Sodium-independent organic anion transmembrane transporter activity
Furosemide//Canalicular multispecific organic anion transporter 1//Organic anion transmembrane transporter activity
Furosemide//Solute carrier organic anion transporter family member 2A1//Sodium-independent organic anion transmembrane transporter activity
Furosemide//Solute carrier family 22 member 11//Sodium-independent organic anion transmembrane transporter activity
Ergotamine//Multidrug resistance protein 1//Xenobiotic-transporting atpase activity
Methazolamide//Solute carrier family 22 member 6//Sodium-independent organic anion transmembrane transporter activity
Flurbiprofen//Multidrug resistance-associated protein 4//Atpase activity, coupled to transmembrane movement of substances
Flurbiprofen//Solute carrier family 22 member 6//Sodium-independent organic anion transmembrane transporter activity
Apomorphine//Synaptic vesicular amine transporter//Monoamine transmembrane transporter activity
Nateglinide//Multidrug resistance-associated protein 4//Atpase activity, coupled to transmembrane movement of substances
Nateglinide//Monocarboxylate transporter 1//Symporter activity
Nateglinide//Solute carrier family 15 member 1//Proton-dependent oligopeptide secondary active transmembrane transporter activity
Nateglinide//Solute carrier family 15 member 2//Peptide:proton symporter activity
Nateglinide//Solute carrier family 22 member 6//Sodium-independent organic anion transmembrane transporter activity
Esomeprazole//Multidrug resistance protein 1//Xenobiotic-transporting atpase activity
Esomeprazole//Solute carrier family 22 member 8//Sodium-independent organic anion transmembrane transporter activity
Hydrocortisone//Multidrug resistance protein 1//Xenobiotic-transporting atpase activity
Hydrocortisone//Solute carrier organic anion transporter family member 1A2//Sodium-independent organic anion transmembrane transporter activity
Hydrocortisone//Solute carrier family 22 member 8//Sodium-independent organic anion transmembrane transporter activity
Etodolac//Solute carrier family 22 member 6//Sodium-independent organic anion transmembrane transporter activity
Epinastine//Multidrug resistance protein 1//Xenobiotic-transporting atpase activity
Clopidogrel//Multidrug resistance protein 1//Xenobiotic-transporting atpase activity
Clopidogrel//Solute carrier family 22 member 1//Secondary active organic cation transmembrane transporter activity
Clopidogrel//Solute carrier family 22 member 2//Quaternary ammonium group transmembrane transporter activity
Irinotecan//Solute carrier family 22 member 3//Toxin transporter activity
Irinotecan//Solute carrier organic anion transporter family member 1B1//Sodium-independent organic anion transmembrane transporter activity
Irinotecan//Multidrug resistance-associated protein 1//Transporter activity
Irinotecan//ATP-binding cassette sub-family G member 2//Xenobiotic-transporting atpase activity
Irinotecan//Multidrug resistance protein 1//Xenobiotic-transporting atpase activity
Irinotecan//Canalicular multispecific organic anion transporter 1//Organic anion transmembrane transporter activity
Etoposide//Canalicular multispecific organic anion transporter 2//Organic anion transmembrane transporter activity
Etoposide//Multidrug resistance-associated protein 6//Transporter activity
Etoposide//Multidrug resistance protein 1//Xenobiotic-transporting atpase activity
Etoposide//Multidrug resistance-associated protein 1//Transporter activity
Etoposide//Multidrug resistance-associated protein 7//Atpase activity, coupled to transmembrane movement of substances
Etoposide//Canalicular multispecific organic anion transporter 1//Organic anion transmembrane transporter activity
Etoposide//ATP-binding cassette sub-family G member 2//Xenobiotic-transporting atpase activity
Estradiol//Solute carrier family 22 member 2//Quaternary ammonium group transmembrane transporter activity
Estradiol//Solute carrier family 22 member 3//Toxin transporter activity
Estradiol//Multidrug resistance-associated protein 7//Atpase activity, coupled to transmembrane movement of substances
Estradiol//Solute carrier family 22 member 11//Sodium-independent organic anion transmembrane transporter activity
Estradiol//ATP-binding cassette sub-family G member 2//Xenobiotic-transporting atpase activity
Estradiol//Solute carrier organic anion transporter family member 1B1//Sodium-independent organic anion transmembrane transporter activity
Estradiol//Multidrug resistance protein 1//Xenobiotic-transporting atpase activity
Estradiol//Solute carrier family 22 member 8//Sodium-independent organic anion transmembrane transporter activity
Estradiol//Solute carrier organic anion transporter family member 1B3//Sodium-independent organic anion transmembrane transporter activity
Estradiol//Solute carrier organic anion transporter family member 1C1//Thyroid hormone transmembrane transporter activity
Naproxen//Solute carrier organic anion transporter family member 1A2//Sodium-independent organic anion transmembrane transporter activity
Naproxen//Solute carrier family 22 member 6//Sodium-independent organic anion transmembrane transporter activity
Naproxen//Bile salt export pump//Transporter activity
Naproxen//Multidrug resistance protein 1//Xenobiotic-transporting atpase activity
Naproxen//Solute carrier family 22 member 8//Sodium-independent organic anion transmembrane transporter activity
Candesartancilexetil//Multidrug resistance protein 1//Xenobiotic-transporting atpase activity
Alfentanil//Multidrug resistance protein 1//Xenobiotic-transporting atpase activity
Fentanyl//Multidrug resistance protein 1//Xenobiotic-transporting atpase activity
Meloxicam//Multidrug resistance-associated protein 4//Atpase activity, coupled to transmembrane movement of substances
Acetazolamide//Solute carrier family 22 member 6//Sodium-independent organic anion transmembrane transporter activity
Disulfiram//Bile salt export pump//Transporter activity
Diazepam//Multidrug resistance protein 1//Xenobiotic-transporting atpase activity
Mifepristone//Multidrug resistance protein 1//Xenobiotic-transporting atpase activity
Mifepristone//Multidrug resistance-associated protein 1//Transporter activity
Mifepristone//Bile salt export pump//Transporter activity
Mifepristone//Solute carrier organic anion transporter family member 1B1//Sodium-independent organic anion transmembrane transporter activity
Mifepristone//Solute carrier organic anion transporter family member 1B3//Sodium-independent organic anion transmembrane transporter activity
Loperamide//Multidrug resistance protein 1//Xenobiotic-transporting atpase activity
Donepezil//ATP-binding cassette sub-family G member 2//Xenobiotic-transporting atpase activity
Clofazimine//Multidrug resistance protein 1//Xenobiotic-transporting atpase activity
Clofazimine//ATP-binding cassette sub-family G member 2//Xenobiotic-transporting atpase activity
Clofazimine//Multidrug resistance-associated protein 1//Transporter activity
Diflunisal//Solute carrier family 22 member 6//Sodium-independent organic anion transmembrane transporter activity
Conivaptan//Multidrug resistance protein 1//Xenobiotic-transporting atpase activity
Flupentixol//Multidrug resistance protein 1//Xenobiotic-transporting atpase activity
Eprosartan//Canalicular multispecific organic anion transporter 1//Organic anion transmembrane transporter activity
Clomifene//Multidrug resistance protein 1//Xenobiotic-transporting atpase activity
Bumetanide//Sodium/bile acid cotransporter//Virus receptor activity
Bumetanide//Solute carrier family 22 member 6//Sodium-independent organic anion transmembrane transporter activity
Bumetanide//Solute carrier family 22 member 8//Sodium-independent organic anion transmembrane transporter activity
Bumetanide//Solute carrier family 22 member 11//Sodium-independent organic anion transmembrane transporter activity
Bumetanide//Solute carrier family 22 member 7//Sodium-independent organic anion transmembrane transporter activity
Bumetanide//Solute carrier organic anion transporter family member 1A2//Sodium-independent organic anion transmembrane transporter activity
Etacrynicacid//Solute carrier family 22 member 6//Sodium-independent organic anion transmembrane transporter activity
Cocaine//Solute carrier family 22 member 2//Quaternary ammonium group transmembrane transporter activity
Cocaine//Sodium-dependent dopamine transporter//Monoamine transmembrane transporter activity
Amantadine//Solute carrier family 22 member 2//Quaternary ammonium group transmembrane transporter activity
Amantadine//Solute carrier family 22 member 1//Secondary active organic cation transmembrane transporter activity
Metronidazole//Multidrug resistance protein 1//Xenobiotic-transporting atpase activity
Dinoprostone//Solute carrier family 22 member 2//Quaternary ammonium group transmembrane transporter activity
Dinoprostone//Multidrug resistance-associated protein 5//Organic anion transmembrane transporter activity
Dinoprostone//Solute carrier family 22 member 6//Sodium-independent organic anion transmembrane transporter activity
Dinoprostone//Solute carrier family 22 member 8//Sodium-independent organic anion transmembrane transporter activity
Dinoprostone//Solute carrier family 22 member 11//Sodium-independent organic anion transmembrane transporter activity
Dinoprostone//Solute carrier family 22 member 7//Sodium-independent organic anion transmembrane transporter activity
Dinoprostone//Multidrug resistance-associated protein 4//Atpase activity, coupled to transmembrane movement of substances
Dinoprostone//Solute carrier organic anion transporter family member 2B1//Sodium-independent organic anion transmembrane transporter activity
Dinoprostone//Solute carrier organic anion transporter family member 1A2//Sodium-independent organic anion transmembrane transporter activity
Dinoprostone//Organic solute transporter subunit alpha//Transporter activity
Dinoprostone//Organic solute transporter subunit beta//Transporter activity
Dinoprostone//Solute carrier organic anion transporter family member 2A1//Sodium-independent organic anion transmembrane transporter activity
Dinoprostone//Solute carrier organic anion transporter family member 4A1//Thyroid hormone transmembrane transporter activity
Dinoprostone//Solute carrier organic anion transporter family member 1C1//Thyroid hormone transmembrane transporter activity
Dinoprostone//Solute carrier organic anion transporter family member 3A1//Sodium-independent organic anion transmembrane transporter activity
Dinoprostone//Solute carrier organic anion transporter family member 1B1//Sodium-independent organic anion transmembrane transporter activity
Buprenorphine//Multidrug resistance protein 1//Xenobiotic-transporting atpase activity
Buprenorphine//ATP-binding cassette sub-family G member 2//Xenobiotic-transporting atpase activity
Famotidine//Solute carrier family 22 member 6//Sodium-independent organic anion transmembrane transporter activity
Famotidine//Solute carrier family 22 member 8//Sodium-independent organic anion transmembrane transporter activity
Famotidine//Solute carrier family 22 member 2//Quaternary ammonium group transmembrane transporter activity
Famotidine//Multidrug and toxin extrusion protein 1//Monovalent cation:proton antiporter activity
Acetylsalicylicacid//Solute carrier family 22 member 6//Sodium-independent organic anion transmembrane transporter activity
Acetylsalicylicacid//Multidrug resistance protein 1//Xenobiotic-transporting atpase activity
Acetylsalicylicacid//Solute carrier family 22 member 8//Sodium-independent organic anion transmembrane transporter activity
Fexofenadine//Multidrug resistance protein 1//Xenobiotic-transporting atpase activity
Fexofenadine//Solute carrier organic anion transporter family member 1B1//Sodium-independent organic anion transmembrane transporter activity
Fexofenadine//Solute carrier organic anion transporter family member 1B3//Sodium-independent organic anion transmembrane transporter activity
Fexofenadine//Solute carrier organic anion transporter family member 2B1//Sodium-independent organic anion transmembrane transporter activity
Fexofenadine//Solute carrier organic anion transporter family member 1A2//Sodium-independent organic anion transmembrane transporter activity
Fexofenadine//Canalicular multispecific organic anion transporter 1//Organic anion transmembrane transporter activity
Fexofenadine//Canalicular multispecific organic anion transporter 2//Organic anion transmembrane transporter activity
Fexofenadine//Solute carrier family 22 member 8//Sodium-independent organic anion transmembrane transporter activity
Methylprednisolone//Multidrug resistance protein 1//Xenobiotic-transporting atpase activity
Desloratadine//Multidrug resistance protein 1//Xenobiotic-transporting atpase activity
Methyldopa//Solute carrier family 15 member 1//Proton-dependent oligopeptide secondary active transmembrane transporter activity
Azelastine//Multidrug resistance protein 1//Xenobiotic-transporting atpase activity
Ezetimibe//Multidrug resistance protein 1//Xenobiotic-transporting atpase activity
Ezetimibe//Canalicular multispecific organic anion transporter 1//Organic anion transmembrane transporter activity
Ezetimibe//Canalicular multispecific organic anion transporter 2//Organic anion transmembrane transporter activity
Ezetimibe//Solute carrier organic anion transporter family member 1B1//Sodium-independent organic anion transmembrane transporter activity
Ezetimibe//ATP-binding cassette sub-family G member 2//Xenobiotic-transporting atpase activity
Ezetimibe//Bile salt export pump//Transporter activity
Ethinylestradiol//Bile salt export pump//Transporter activity
Ethinylestradiol//Sodium/bile acid cotransporter//Virus receptor activity
Ethinylestradiol//Canalicular multispecific organic anion transporter 1//Organic anion transmembrane transporter activity
Ethinylestradiol//Multidrug resistance protein 1//Xenobiotic-transporting atpase activity
Ethinylestradiol//Solute carrier organic anion transporter family member 1A2//Sodium-independent organic anion transmembrane transporter activity
Lomefloxacin//Solute carrier family 22 member 5//Symporter activity
Lomefloxacin//Canalicular multispecific organic anion transporter 1//Organic anion transmembrane transporter activity
Formoterol//Solute carrier family 22 member 1//Secondary active organic cation transmembrane transporter activity
Formoterol//Solute carrier family 22 member 3//Toxin transporter activity
Formoterol//Solute carrier family 22 member 4//Symporter activity
Formoterol//Solute carrier family 22 member 5//Symporter activity
Cytarabine//Solute carrier family 22 member 4//Symporter activity
Cytarabine//Multidrug resistance-associated protein 7//Atpase activity, coupled to transmembrane movement of substances
Cytarabine//Equilibrative nucleoside transporter 1//Nucleoside transmembrane transporter activity
Dopamine//Solute carrier family 22 member 2//Quaternary ammonium group transmembrane transporter activity
Dopamine//Solute carrier family 22 member 1//Secondary active organic cation transmembrane transporter activity
Dopamine//Solute carrier family 22 member 3//Toxin transporter activity
Dopamine//Solute carrier family 22 member 5//Symporter activity
Dopamine//POU domain, class 5, transcription factor 1//Ubiquitin protein ligase binding
Azathioprine//Equilibrative nucleoside transporter 2//Nucleoside transmembrane transporter activity
Azathioprine//Solute carrier family 28 member 3//Pyrimidine- and adenine-specific:sodium symporter activity
Azathioprine//Multidrug resistance protein 1//Xenobiotic-transporting atpase activity
Gabapentin//Large neutral amino acids transporter small subunit 1//Peptide antigen binding
Doxorubicin//Multidrug resistance protein 1//Xenobiotic-transporting atpase activity
Doxorubicin//Multidrug resistance-associated protein 1//Transporter activity
Doxorubicin//Canalicular multispecific organic anion transporter 2//Organic anion transmembrane transporter activity
Doxorubicin//Multidrug resistance-associated protein 6//Transporter activity
Doxorubicin//ATP-binding cassette sub-family G member 2//Xenobiotic-transporting atpase activity
Doxorubicin//Multidrug resistance-associated protein 7//Atpase activity, coupled to transmembrane movement of substances
Doxorubicin//ATP-binding cassette sub-family B member 8, mitochondrial//Transporter activity
Doxorubicin//Bile salt export pump//Transporter activity
Doxorubicin//RalA-binding protein 1//Transmembrane transporter activity
Doxorubicin//Canalicular multispecific organic anion transporter 1//Organic anion transmembrane transporter activity
Letrozole//Multidrug resistance protein 1//Xenobiotic-transporting atpase activity
Ketoprofen//Multidrug resistance-associated protein 4//Atpase activity, coupled to transmembrane movement of substances
Ketoprofen//Solute carrier organic anion transporter family member 1A2//Sodium-independent organic anion transmembrane transporter activity
Ketoprofen//Solute carrier family 22 member 6//Sodium-independent organic anion transmembrane transporter activity
Ketoprofen//Solute carrier family 22 member 8//Sodium-independent organic anion transmembrane transporter activity
Ketoprofen//Solute carrier family 22 member 11//Sodium-independent organic anion transmembrane transporter activity
Ketoprofen//Solute carrier family 22 member 7//Sodium-independent organic anion transmembrane transporter activity
Metyrapone//Canalicular multispecific organic anion transporter 2//Organic anion transmembrane transporter activity
Glyburide//Canalicular multispecific organic anion transporter 2//Organic anion transmembrane transporter activity
Glyburide//Bile salt export pump//Transporter activity
Glyburide//Multidrug resistance protein 1//Xenobiotic-transporting atpase activity
Glyburide//Multidrug resistance-associated protein 1//Transporter activity
Glyburide//Solute carrier family 15 member 1//Proton-dependent oligopeptide secondary active transmembrane transporter activity
Glyburide//Solute carrier organic anion transporter family member 1A2//Sodium-independent organic anion transmembrane transporter activity
Glyburide//Solute carrier family 15 member 2//Peptide:proton symporter activity
Glyburide//Solute carrier family 22 member 6//Sodium-independent organic anion transmembrane transporter activity
Glyburide//Canalicular multispecific organic anion transporter 1//Organic anion transmembrane transporter activity
Glyburide//ATP-binding cassette sub-family G member 2//Xenobiotic-transporting atpase activity
Glyburide//Solute carrier family 22 member 7//Sodium-independent organic anion transmembrane transporter activity
Glyburide//Solute carrier organic anion transporter family member 2B1//Sodium-independent organic anion transmembrane transporter activity
Guanfacine//Multidrug and toxin extrusion protein 1//Monovalent cation:proton antiporter activity
Guanfacine//Solute carrier family 22 member 1//Secondary active organic cation transmembrane transporter activity
Guanfacine//Solute carrier family 22 member 2//Quaternary ammonium group transmembrane transporter activity
Felodipine//Multidrug resistance protein 1//Xenobiotic-transporting atpase activity
Felodipine//Bile salt export pump//Transporter activity
Ketoconazole//Multidrug resistance protein 1//Xenobiotic-transporting atpase activity
Ketoconazole//Solute carrier organic anion transporter family member 1B1//Sodium-independent organic anion transmembrane transporter activity
Ketoconazole//Bile salt export pump//Transporter activity
Mercaptopurine//Solute carrier family 22 member 8//Sodium-independent organic anion transmembrane transporter activity
Mercaptopurine//Multidrug resistance-associated protein 4//Atpase activity, coupled to transmembrane movement of substances
Mercaptopurine//Multidrug resistance-associated protein 5//Organic anion transmembrane transporter activity
Mercaptopurine//Solute carrier family 28 member 3//Pyrimidine- and adenine-specific:sodium symporter activity
Mercaptopurine//Equilibrative nucleoside transporter 1//Nucleoside transmembrane transporter activity
Mercaptopurine//Equilibrative nucleoside transporter 2//Nucleoside transmembrane transporter activity
Fenofibrate//Bile salt export pump//Transporter activity
Memantine//Solute carrier family 22 member 2//Quaternary ammonium group transmembrane transporter activity
Memantine//Solute carrier family 22 member 4//Symporter activity
Memantine//Multidrug and toxin extrusion protein 1//Monovalent cation:proton antiporter activity
Ibuprofen//Solute carrier organic anion transporter family member 2B1//Sodium-independent organic anion transmembrane transporter activity
Ibuprofen//Multidrug resistance protein 1//Xenobiotic-transporting atpase activity
Ibuprofen//Multidrug resistance-associated protein 4//Atpase activity, coupled to transmembrane movement of substances
Ibuprofen//Multidrug resistance-associated protein 1//Transporter activity
Ibuprofen//Solute carrier organic anion transporter family member 1A2//Sodium-independent organic anion transmembrane transporter activity
Ibuprofen//Solute carrier family 22 member 6//Sodium-independent organic anion transmembrane transporter activity
Ibuprofen//Solute carrier family 22 member 8//Sodium-independent organic anion transmembrane transporter activity
Ibuprofen//Solute carrier family 22 member 11//Sodium-independent organic anion transmembrane transporter activity
Melatonin//Solute carrier family 22 member 8//Sodium-independent organic anion transmembrane transporter activity
Glipizide//Bile salt export pump//Transporter activity
Diphenhydramine//Solute carrier family 22 member 2//Quaternary ammonium group transmembrane transporter activity
Diphenhydramine//Solute carrier family 22 member 5//Symporter activity
Atorvastatin//Multidrug resistance protein 1//Xenobiotic-transporting atpase activity
Atorvastatin//Solute carrier organic anion transporter family member 1A2//Sodium-independent organic anion transmembrane transporter activity
Atorvastatin//Solute carrier organic anion transporter family member 1B1//Sodium-independent organic anion transmembrane transporter activity
Atorvastatin//Multidrug resistance-associated protein 4//Atpase activity, coupled to transmembrane movement of substances
Atorvastatin//Multidrug resistance-associated protein 5//Organic anion transmembrane transporter activity
Atorvastatin//Multidrug resistance-associated protein 1//Transporter activity
Atorvastatin//Solute carrier organic anion transporter family member 2B1//Sodium-independent organic anion transmembrane transporter activity
Atorvastatin//Solute carrier organic anion transporter family member 1B3//Sodium-independent organic anion transmembrane transporter activity
Atorvastatin//Canalicular multispecific organic anion transporter 1//Organic anion transmembrane transporter activity
Atorvastatin//Bile salt export pump//Transporter activity
Benzocaine//Multidrug resistance protein 1//Xenobiotic-transporting atpase activity
Hesperetin//ATP-binding cassette sub-family G member 2//Xenobiotic-transporting atpase activity
Fluvastatin//Solute carrier organic anion transporter family member 1B1//Sodium-independent organic anion transmembrane transporter activity
Fluvastatin//Solute carrier organic anion transporter family member 1B3//Sodium-independent organic anion transmembrane transporter activity
Fluvastatin//Solute carrier organic anion transporter family member 2B1//Sodium-independent organic anion transmembrane transporter activity
Fluvastatin//Solute carrier family 15 member 1//Proton-dependent oligopeptide secondary active transmembrane transporter activity
Fluvastatin//Canalicular multispecific organic anion transporter 1//Organic anion transmembrane transporter activity
Leflunomide//ATP-binding cassette sub-family G member 2//Xenobiotic-transporting atpase activity
Miconazole//Multidrug resistance protein 1//Xenobiotic-transporting atpase activity
Chlorphenamine//Solute carrier family 22 member 2//Quaternary ammonium group transmembrane transporter activity
Chlorphenamine//Solute carrier family 22 member 1//Secondary active organic cation transmembrane transporter activity
Atovaquone//Multidrug resistance protein 1//Xenobiotic-transporting atpase activity
Amiodarone//Multidrug resistance protein 1//Xenobiotic-transporting atpase activity
Amiodarone//Bile salt export pump//Transporter activity
Amiodarone//Solute carrier family 22 member 2//Quaternary ammonium group transmembrane transporter activity
Dutasteride//Sodium-dependent dopamine transporter//Monoamine transmembrane transporter activity
Dutasteride//Synaptic vesicular amine transporter//Monoamine transmembrane transporter activity
Bicalutamide//Multidrug resistance protein 1//Xenobiotic-transporting atpase activity
Carvedilol//Multidrug resistance protein 1//Xenobiotic-transporting atpase activity
Levofloxacin//Multidrug resistance protein 1//Xenobiotic-transporting atpase activity
Levofloxacin//Multidrug and toxin extrusion protein 1//Monovalent cation:proton antiporter activity
Levofloxacin//Multidrug and toxin extrusion protein 2//Drug transmembrane transporter activity
Levofloxacin//Solute carrier family 22 member 1//Secondary active organic cation transmembrane transporter activity
Levofloxacin//Solute carrier family 22 member 2//Quaternary ammonium group transmembrane transporter activity
Levofloxacin//Solute carrier family 22 member 4//Symporter activity
Levofloxacin//Solute carrier organic anion transporter family member 1A2//Sodium-independent organic anion transmembrane transporter activity
Levofloxacin//Solute carrier organic anion transporter family member 4C1//Sodium-independent organic anion transmembrane transporter activity
Doxepin//Multidrug resistance protein 1//Xenobiotic-transporting atpase activity
Nefazodone//Multidrug resistance protein 1//Xenobiotic-transporting atpase activity
Nefazodone//Solute carrier organic anion transporter family member 1B3//Sodium-independent organic anion transmembrane transporter activity
Nefazodone//Solute carrier organic anion transporter family member 2B1//Sodium-independent organic anion transmembrane transporter activity
Nefazodone//Bile salt export pump//Transporter activity
Desipramine//Multidrug resistance protein 1//Xenobiotic-transporting atpase activity
Desipramine//Solute carrier family 22 member 1//Secondary active organic cation transmembrane transporter activity
Desipramine//Solute carrier family 22 member 3//Toxin transporter activity
Desipramine//Solute carrier family 22 member 2//Quaternary ammonium group transmembrane transporter activity
Desipramine//Solute carrier family 22 member 5//Symporter activity
Desipramine//Solute carrier family 22 member 4//Symporter activity
Bupropion//Solute carrier family 22 member 2//Quaternary ammonium group transmembrane transporter activity
Itraconazole//Multidrug resistance protein 1//Xenobiotic-transporting atpase activity
Itraconazole//Solute carrier organic anion transporter family member 2B1//Sodium-independent organic anion transmembrane transporter activity
Arsenictrioxide//Canalicular multispecific organic anion transporter 1//Organic anion transmembrane transporter activity
Arsenictrioxide//Multidrug resistance protein 1//Xenobiotic-transporting atpase activity
Escitalopram//Multidrug resistance protein 1//Xenobiotic-transporting atpase activity
Idarubicin//Multidrug resistance-associated protein 1//Transporter activity
Naloxone//Solute carrier organic anion transporter family member 1A2//Sodium-independent organic anion transmembrane transporter activity
Naloxone//Multidrug resistance protein 1//Xenobiotic-transporting atpase activity
Domperidone//Multidrug resistance protein 1//Xenobiotic-transporting atpase activity
Acebutolol//Multidrug resistance protein 1//Xenobiotic-transporting atpase activity
Flecainide//Multidrug resistance protein 1//Xenobiotic-transporting atpase activity
Flecainide//Multidrug and toxin extrusion protein 1//Monovalent cation:proton antiporter activity
Estramustine//Multidrug resistance protein 1//Xenobiotic-transporting atpase activity
Captopril//Multidrug resistance protein 1//Xenobiotic-transporting atpase activity
Captopril//Solute carrier family 15 member 1//Proton-dependent oligopeptide secondary active transmembrane transporter activity
Captopril//Solute carrier family 22 member 6//Sodium-independent organic anion transmembrane transporter activity
Bromocriptine//Multidrug resistance protein 1//Xenobiotic-transporting atpase activity
Mitoxantrone//Multidrug resistance protein 1//Xenobiotic-transporting atpase activity
Mitoxantrone//Multidrug resistance-associated protein 1//Transporter activity
Mitoxantrone//ATP-binding cassette sub-family G member 2//Xenobiotic-transporting atpase activity
Clarithromycin//Solute carrier family 22 member 7//Sodium-independent organic anion transmembrane transporter activity
Clarithromycin//Multidrug resistance protein 1//Xenobiotic-transporting atpase activity
Clarithromycin//Bile salt export pump//Transporter activity
Clarithromycin//Solute carrier organic anion transporter family member 1B1//Sodium-independent organic anion transmembrane transporter activity
Clarithromycin//Solute carrier organic anion transporter family member 1B3//Sodium-independent organic anion transmembrane transporter activity
Ceftriaxone//Solute carrier family 15 member 1//Proton-dependent oligopeptide secondary active transmembrane transporter activity
Ceftriaxone//Solute carrier family 15 member 2//Peptide:proton symporter activity
Ceftriaxone//Solute carrier family 22 member 6//Sodium-independent organic anion transmembrane transporter activity
Ceftriaxone//Solute carrier family 22 member 8//Sodium-independent organic anion transmembrane transporter activity
Ceftriaxone//Solute carrier family 22 member 11//Sodium-independent organic anion transmembrane transporter activity
Ceftriaxone//Multidrug resistance protein 1//Xenobiotic-transporting atpase activity
Finasteride//Solute carrier family 12 member 5//Protein kinase binding
Anastrozole//Multidrug resistance protein 1//Xenobiotic-transporting atpase activity
Budesonide//Bile salt export pump//Transporter activity
Budesonide//Multidrug resistance protein 1//Xenobiotic-transporting atpase activity
Budesonide//Solute carrier organic anion transporter family member 1A2//Sodium-independent organic anion transmembrane transporter activity
Budesonide//Solute carrier family 22 member 8//Sodium-independent organic anion transmembrane transporter activity
Metoclopramide//Multidrug resistance protein 1//Xenobiotic-transporting atpase activity
Dexamethasone//Multidrug resistance protein 1//Xenobiotic-transporting atpase activity
Dexamethasone//Solute carrier family 22 member 8//Sodium-independent organic anion transmembrane transporter activity
Dexamethasone//Bile salt export pump//Transporter activity
Dexamethasone//Canalicular multispecific organic anion transporter 1//Organic anion transmembrane transporter activity
Dexamethasone//ATP-binding cassette sub-family G member 2//Xenobiotic-transporting atpase activity
Dexamethasone//Solute carrier organic anion transporter family member 1A2//Sodium-independent organic anion transmembrane transporter activity
Levodopa//Solute carrier family 15 member 1//Proton-dependent oligopeptide secondary active transmembrane transporter activity
Levodopa//Monocarboxylate transporter 10//Transporter activity
Levodopa//Large neutral amino acids transporter small subunit 1//Peptide antigen binding
Levodopa//Large neutral amino acids transporter small subunit 2//Toxin transporter activity
Clomipramine//Multidrug resistance protein 1//Xenobiotic-transporting atpase activity
Bepridil//Multidrug resistance protein 1//Xenobiotic-transporting atpase activity
Docetaxel//Multidrug resistance protein 1//Xenobiotic-transporting atpase activity
Docetaxel//Multidrug resistance-associated protein 7//Atpase activity, coupled to transmembrane movement of substances
Docetaxel//Solute carrier organic anion transporter family member 1B3//Sodium-independent organic anion transmembrane transporter activity
Docetaxel//Solute carrier family 22 member 7//Sodium-independent organic anion transmembrane transporter activity
Docetaxel//ATP-binding cassette sub-family G member 2//Xenobiotic-transporting atpase activity
Docetaxel//Canalicular multispecific organic anion transporter 1//Organic anion transmembrane transporter activity
Docetaxel//Multidrug resistance-associated protein 1//Transporter activity
Ergonovine//Multidrug resistance protein 1//Xenobiotic-transporting atpase activity
Dasatinib//Multidrug resistance protein 1//Xenobiotic-transporting atpase activity
Dasatinib//ATP-binding cassette sub-family G member 2//Xenobiotic-transporting atpase activity
Lapatinib//Multidrug resistance protein 1//Xenobiotic-transporting atpase activity
Cefazolin//Multidrug resistance-associated protein 4//Atpase activity, coupled to transmembrane movement of substances
Cefazolin//Solute carrier family 22 member 6//Sodium-independent organic anion transmembrane transporter activity
Cefazolin//Solute carrier family 22 member 8//Sodium-independent organic anion transmembrane transporter activity
Cefazolin//Solute carrier family 22 member 11//Sodium-independent organic anion transmembrane transporter activity
Ephedrine//Synaptic vesicular amine transporter//Monoamine transmembrane transporter activity
Bezafibrate//Solute carrier organic anion transporter family member 1B1//Sodium-independent organic anion transmembrane transporter activity
Colchicine//Multidrug resistance protein 1//Xenobiotic-transporting atpase activity
Digitoxin//Solute carrier organic anion transporter family member 1A2//Sodium-independent organic anion transmembrane transporter activity
Digitoxin//Solute carrier organic anion transporter family member 4C1//Sodium-independent organic anion transmembrane transporter activity
Digitoxin//Multidrug resistance protein 1//Xenobiotic-transporting atpase activity
Acenocoumarol//Multidrug resistance protein 1//Xenobiotic-transporting atpase activity
Antipyrine//Solute carrier family 22 member 6//Sodium-independent organic anion transmembrane transporter activity
Dextroamphetamine//Sodium-dependent dopamine transporter//Monoamine transmembrane transporter activity
Methamphetamine//Solute carrier family 22 member 3//Toxin transporter activity
Methamphetamine//Solute carrier family 22 member 5//Symporter activity
Liotrix//Solute carrier organic anion transporter family member 1A2//Sodium-independent organic anion transmembrane transporter activity
Liotrix//Solute carrier organic anion transporter family member 1B1//Sodium-independent organic anion transmembrane transporter activity
Liotrix//Solute carrier organic anion transporter family member 1B3//Sodium-independent organic anion transmembrane transporter activity
Liotrix//Solute carrier organic anion transporter family member 4C1//Sodium-independent organic anion transmembrane transporter activity
Liotrix//Sodium/bile acid cotransporter//Virus receptor activity
Liotrix//Solute carrier organic anion transporter family member 1C1//Thyroid hormone transmembrane transporter activity
Liotrix//Solute carrier organic anion transporter family member 4A1//Thyroid hormone transmembrane transporter activity
Liotrix//Solute carrier family 22 member 8//Sodium-independent organic anion transmembrane transporter activity
Liotrix//Monocarboxylate transporter 8//Transporter activity
Liotrix//Monocarboxylate transporter 10//Transporter activity
Liotrix//Multidrug resistance protein 1//Xenobiotic-transporting atpase activity
Ketazolam//Multidrug resistance protein 1//Xenobiotic-transporting atpase activity
Everolimus//Solute carrier organic anion transporter family member 1B1//Sodium-independent organic anion transmembrane transporter activity
Everolimus//Solute carrier organic anion transporter family member 1B3//Sodium-independent organic anion transmembrane transporter activity
Everolimus//Solute carrier organic anion transporter family member 1A2//Sodium-independent organic anion transmembrane transporter activity
Everolimus//Multidrug resistance protein 1//Xenobiotic-transporting atpase activity
Hydroxychloroquine//Multidrug resistance protein 1//Xenobiotic-transporting atpase activity
Hydroxychloroquine//Solute carrier organic anion transporter family member 1A2//Sodium-independent organic anion transmembrane transporter activity
Acetylcholine//Solute carrier family 22 member 5//Symporter activity
Acetylcholine//Solute carrier family 22 member 1//Secondary active organic cation transmembrane transporter activity
Estronesulfate//Multidrug and toxin extrusion protein 1//Monovalent cation:proton antiporter activity
Estronesulfate//Multidrug and toxin extrusion protein 2//Drug transmembrane transporter activity
Debrisoquin//Multidrug resistance protein 1//Xenobiotic-transporting atpase activity
Ixabepilone//Multidrug resistance protein 1//Xenobiotic-transporting atpase activity
Dronedarone//Multidrug resistance protein 1//Xenobiotic-transporting atpase activity
Dronedarone//Solute carrier family 22 member 2//Quaternary ammonium group transmembrane transporter activity
Dronedarone//Solute carrier family 22 member 1//Secondary active organic cation transmembrane transporter activity
Dronedarone//Solute carrier organic anion transporter family member 1B1//Sodium-independent organic anion transmembrane transporter activity
Dronedarone//Solute carrier organic anion transporter family member 1B3//Sodium-independent organic anion transmembrane transporter activity
Dronedarone//Solute carrier family 22 member 8//Sodium-independent organic anion transmembrane transporter activity
Flibanserin//Multidrug resistance protein 1//Xenobiotic-transporting atpase activity
Indacaterol//Multidrug resistance protein 1//Xenobiotic-transporting atpase activity
Cobimetinib//Solute carrier organic anion transporter family member 1B1//Sodium-independent organic anion transmembrane transporter activity
Cobimetinib//Solute carrier organic anion transporter family member 1B3//Sodium-independent organic anion transmembrane transporter activity
Cobimetinib//ATP-binding cassette sub-family G member 2//Xenobiotic-transporting atpase activity
Cobimetinib//Multidrug resistance protein 1//Xenobiotic-transporting atpase activity
Histamine//Solute carrier family 22 member 2//Quaternary ammonium group transmembrane transporter activity
Histamine//Solute carrier family 22 member 1//Secondary active organic cation transmembrane transporter activity
Histamine//Solute carrier family 22 member 3//Toxin transporter activity
Histamine//Solute carrier family 22 member 5//Symporter activity
Apremilast//Multidrug resistance protein 1//Xenobiotic-transporting atpase activity
Abiraterone//Multidrug resistance-associated protein 1//Transporter activity
Eltrombopag//Solute carrier organic anion transporter family member 1B1//Sodium-independent organic anion transmembrane transporter activity
Eltrombopag//ATP-binding cassette sub-family G member 2//Xenobiotic-transporting atpase activity
Droxidopa//Sodium-dependent noradrenaline transporter//Norepinephrine:sodium symporter activity
Droxidopa//Monocarboxylate transporter 10//Transporter activity
Amrubicin//ATP-binding cassette sub-family B member 5//Efflux transmembrane transporter activity
Levocetirizine//Solute carrier family 22 member 11//Sodium-independent organic anion transmembrane transporter activity
Dapagliflozin//Multidrug resistance protein 1//Xenobiotic-transporting atpase activity
Ambrisentan//Multidrug resistance protein 1//Xenobiotic-transporting atpase activity
Ambrisentan//Solute carrier organic anion transporter family member 1B1//Sodium-independent organic anion transmembrane transporter activity
Ambrisentan//Solute carrier organic anion transporter family member 1B3//Sodium-independent organic anion transmembrane transporter activity
Apixaban//Multidrug resistance protein 1//Xenobiotic-transporting atpase activity
Apixaban//ATP-binding cassette sub-family G member 2//Xenobiotic-transporting atpase activity
Bosutinib//Multidrug resistance protein 1//Xenobiotic-transporting atpase activity
Axitinib//Multidrug resistance protein 1//Xenobiotic-transporting atpase activity
Axitinib//Solute carrier organic anion transporter family member 1B1//Sodium-independent organic anion transmembrane transporter activity
Dalfampridine//Solute carrier family 22 member 2//Quaternary ammonium group transmembrane transporter activity
Mepyramine//Solute carrier family 22 member 4//Symporter activity
Mepyramine//Solute carrier family 22 member 5//Symporter activity
Dabigatranetexilate//Multidrug resistance protein 1//Xenobiotic-transporting atpase activity
Fesoterodine//Multidrug resistance protein 1//Xenobiotic-transporting atpase activity
Methyltestosterone//Solute carrier organic anion transporter family member 1A2//Sodium-independent organic anion transmembrane transporter activity
Methyltestosterone//Solute carrier family 22 member 8//Sodium-independent organic anion transmembrane transporter activity
Cabazitaxel//Multidrug resistance protein 1//Xenobiotic-transporting atpase activity
Cabazitaxel//ATP-binding cassette sub-family G member 2//Xenobiotic-transporting atpase activity
Cabazitaxel//Solute carrier organic anion transporter family member 1B1//Sodium-independent organic anion transmembrane transporter activity
Cabazitaxel//Solute carrier organic anion transporter family member 1B3//Sodium-independent organic anion transmembrane transporter activity
Ivacaftor//Multidrug resistance protein 1//Xenobiotic-transporting atpase activity
Lomitapide//Multidrug resistance protein 1//Xenobiotic-transporting atpase activity
Crizotinib//Multidrug resistance protein 1//Xenobiotic-transporting atpase activity
Fingolimod//Multidrug resistance protein 1//Xenobiotic-transporting atpase activity
Fingolimod//Multidrug resistance-associated protein 1//Transporter activity
Linagliptin//Multidrug resistance protein 1//Xenobiotic-transporting atpase activity
Linagliptin//Solute carrier family 22 member 1//Secondary active organic cation transmembrane transporter activity
Linagliptin//Solute carrier family 22 member 2//Quaternary ammonium group transmembrane transporter activity
Linagliptin//Solute carrier family 22 member 3//Toxin transporter activity
Mirabegron//Multidrug resistance protein 1//Xenobiotic-transporting atpase activity
Mirabegron//Solute carrier organic anion transporter family member 1A2//Sodium-independent organic anion transmembrane transporter activity
Enzalutamide//Multidrug resistance protein 1//Xenobiotic-transporting atpase activity
Fluticasonefuroate//Multidrug resistance protein 1//Xenobiotic-transporting atpase activity
Fluticasonefuroate//Solute carrier organic anion transporter family member 1B1//Sodium-independent organic anion transmembrane transporter activity
Canagliflozin//Multidrug resistance protein 1//Xenobiotic-transporting atpase activity
Canagliflozin//Canalicular multispecific organic anion transporter 1//Organic anion transmembrane transporter activity
Canagliflozin//ATP-binding cassette sub-family G member 2//Xenobiotic-transporting atpase activity
Dabrafenib//Multidrug resistance protein 1//Xenobiotic-transporting atpase activity
Dabrafenib//ATP-binding cassette sub-family G member 2//Xenobiotic-transporting atpase activity
Dabrafenib//Solute carrier organic anion transporter family member 1B1//Sodium-independent organic anion transmembrane transporter activity
Dabrafenib//Solute carrier organic anion transporter family member 1B3//Sodium-independent organic anion transmembrane transporter activity
Dabrafenib//Solute carrier family 22 member 6//Sodium-independent organic anion transmembrane transporter activity
Dabrafenib//Solute carrier family 22 member 8//Sodium-independent organic anion transmembrane transporter activity
Levomilnacipran//Multidrug resistance protein 1//Xenobiotic-transporting atpase activity
Aliskiren//Multidrug resistance protein 1//Xenobiotic-transporting atpase activity
Eliglustat//Multidrug resistance protein 1//Xenobiotic-transporting atpase activity
Netupitant//Multidrug resistance protein 1//Xenobiotic-transporting atpase activity
Cannabidiol//Multidrug resistance-associated protein 1//Transporter activity
Cannabidiol//ATP-binding cassette sub-family G member 2//Xenobiotic-transporting atpase activity
Cannabidiol//Equilibrative nucleoside transporter 1//Nucleoside transmembrane transporter activity
Ceritinib//Multidrug resistance protein 1//Xenobiotic-transporting atpase activity
Lenvatinib//Multidrug resistance protein 1//Xenobiotic-transporting atpase activity
Lenvatinib//ATP-binding cassette sub-family G member 2//Xenobiotic-transporting atpase activity
Lenvatinib//Solute carrier family 22 member 6//Sodium-independent organic anion transmembrane transporter activity
Lenvatinib//Solute carrier family 22 member 8//Sodium-independent organic anion transmembrane transporter activity
Lenvatinib//Solute carrier family 22 member 2//Quaternary ammonium group transmembrane transporter activity
Lenvatinib//Solute carrier organic anion transporter family member 1B1//Sodium-independent organic anion transmembrane transporter activity
Lenvatinib//Bile salt export pump//Transporter activity
Lobeglitazone//Solute carrier organic anion transporter family member 1B1//Sodium-independent organic anion transmembrane transporter activity
Lobeglitazone//Solute carrier organic anion transporter family member 3A1//Sodium-independent organic anion transmembrane transporter activity
Lobeglitazone//Multidrug resistance protein 1//Xenobiotic-transporting atpase activity
Lumacaftor//Multidrug resistance protein 1//Xenobiotic-transporting atpase activity
Isavuconazole//Multidrug resistance protein 1//Xenobiotic-transporting atpase activity
Isavuconazole//ATP-binding cassette sub-family G member 2//Xenobiotic-transporting atpase activity
Isavuconazole//Solute carrier family 22 member 2//Quaternary ammonium group transmembrane transporter activity
Naldemedine//ATP-binding cassette sub-family B member 5//Efflux transmembrane transporter activity
Baricitinib//Solute carrier family 22 member 8//Sodium-independent organic anion transmembrane transporter activity
Baricitinib//ATP-binding cassette sub-family G member 2//Xenobiotic-transporting atpase activity
Baricitinib//Multidrug and toxin extrusion protein 2//Drug transmembrane transporter activity
Baricitinib//Solute carrier family 22 member 6//Sodium-independent organic anion transmembrane transporter activity
Baricitinib//Solute carrier family 22 member 2//Quaternary ammonium group transmembrane transporter activity
Baricitinib//Solute carrier organic anion transporter family member 1B3//Sodium-independent organic anion transmembrane transporter activity
Baricitinib//Multidrug resistance protein 1//Xenobiotic-transporting atpase activity
Ertugliflozin//Multidrug resistance protein 1//Xenobiotic-transporting atpase activity
Ertugliflozin//ATP-binding cassette sub-family G member 2//Xenobiotic-transporting atpase activity
Neratinib//Multidrug resistance protein 1//Xenobiotic-transporting atpase activity
Apalutamide//Multidrug resistance protein 1//Xenobiotic-transporting atpase activity
Apalutamide//ATP-binding cassette sub-family G member 2//Xenobiotic-transporting atpase activity
Apalutamide//Solute carrier organic anion transporter family member 1B1//Sodium-independent organic anion transmembrane transporter activity
Apalutamide//Solute carrier family 22 member 2//Quaternary ammonium group transmembrane transporter activity
Apalutamide//Solute carrier family 22 member 8//Sodium-independent organic anion transmembrane transporter activity
Apalutamide//Multidrug and toxin extrusion protein 2//Drug transmembrane transporter activity
Apalutamide//Multidrug and toxin extrusion protein 1//Monovalent cation:proton antiporter activity
Abemaciclib//Multidrug and toxin extrusion protein 1//Monovalent cation:proton antiporter activity
Abemaciclib//Multidrug and toxin extrusion protein 2//Drug transmembrane transporter activity
Abemaciclib//Solute carrier family 22 member 2//Quaternary ammonium group transmembrane transporter activity
Abemaciclib//ATP-binding cassette sub-family G member 2//Xenobiotic-transporting atpase activity
Abemaciclib//Multidrug resistance protein 1//Xenobiotic-transporting atpase activity
Fostamatinib//ATP-binding cassette sub-family G member 2//Xenobiotic-transporting atpase activity
Fostamatinib//ATP-binding cassette sub-family B member 5//Efflux transmembrane transporter activity
Brigatinib//ATP-binding cassette sub-family B member 5//Efflux transmembrane transporter activity
Brigatinib//ATP-binding cassette sub-family G member 2//Xenobiotic-transporting atpase activity
Brigatinib//Solute carrier family 22 member 1//Secondary active organic cation transmembrane transporter activity
Brigatinib//Multidrug and toxin extrusion protein 1//Monovalent cation:proton antiporter activity
Brigatinib//Multidrug and toxin extrusion protein 2//Drug transmembrane transporter activity
Betrixaban//Multidrug resistance protein 1//Xenobiotic-transporting atpase activity
Betrixaban//Potassium voltage-gated channel subfamily H member 2//Voltage-gated potassium channel activity involved in ventricular cardiac muscle cell action potential repolarization
Copanlisib//Multidrug resistance protein 1//Xenobiotic-transporting atpase activity
Copanlisib//ATP-binding cassette sub-family G member 2//Xenobiotic-transporting atpase activity
Copanlisib//Multidrug and toxin extrusion protein 2//Drug transmembrane transporter activity
Levosalbutamol//Solute carrier organic anion transporter family member 1B1//Sodium-independent organic anion transmembrane transporter activity
Levosalbutamol//Solute carrier organic anion transporter family member 1B3//Sodium-independent organic anion transmembrane transporter activity
Acemetacin//Multidrug resistance-associated protein 1//Transporter activity
Enasidenib//Multidrug resistance protein 1//Xenobiotic-transporting atpase activity
Enasidenib//ATP-binding cassette sub-family G member 2//Xenobiotic-transporting atpase activity
Enasidenib//Solute carrier family 22 member 6//Sodium-independent organic anion transmembrane transporter activity
Enasidenib//Solute carrier organic anion transporter family member 1B1//Sodium-independent organic anion transmembrane transporter activity
Enasidenib//Solute carrier family 22 member 2//Quaternary ammonium group transmembrane transporter activity
Enasidenib//Solute carrier organic anion transporter family member 1B3//Sodium-independent organic anion transmembrane transporter activity
Enasidenib//Solute carrier family 22 member 8//Sodium-independent organic anion transmembrane transporter activity
Estradiolacetate//Solute carrier family 22 member 2//Quaternary ammonium group transmembrane transporter activity
Estradiolacetate//Solute carrier family 22 member 1//Secondary active organic cation transmembrane transporter activity
Estradiolacetate//Solute carrier family 22 member 3//Toxin transporter activity
Estradiolacetate//Solute carrier organic anion transporter family member 2B1//Sodium-independent organic anion transmembrane transporter activity
Estradiolacetate//Solute carrier organic anion transporter family member 1A2//Sodium-independent organic anion transmembrane transporter activity
Estradiolacetate//Multidrug resistance-associated protein 7//Atpase activity, coupled to transmembrane movement of substances
Estradiolacetate//Solute carrier family 22 member 11//Sodium-independent organic anion transmembrane transporter activity
Estradiolacetate//ATP-binding cassette sub-family G member 2//Xenobiotic-transporting atpase activity
Estradiolacetate//Solute carrier organic anion transporter family member 1B1//Sodium-independent organic anion transmembrane transporter activity
Estradiolacetate//Multidrug resistance protein 1//Xenobiotic-transporting atpase activity
Estradiolacetate//Solute carrier family 22 member 8//Sodium-independent organic anion transmembrane transporter activity
Estradiolacetate//Solute carrier organic anion transporter family member 1B3//Sodium-independent organic anion transmembrane transporter activity
Estradiolacetate//Solute carrier organic anion transporter family member 1C1//Thyroid hormone transmembrane transporter activity
Estradiolacetate//Solute carrier organic anion transporter family member 4A1//Thyroid hormone transmembrane transporter activity
Estradiolbenzoate//Solute carrier family 22 member 2//Quaternary ammonium group transmembrane transporter activity
Estradiolbenzoate//Solute carrier family 22 member 1//Secondary active organic cation transmembrane transporter activity
Estradiolbenzoate//Solute carrier family 22 member 3//Toxin transporter activity
Estradiolbenzoate//Solute carrier organic anion transporter family member 2B1//Sodium-independent organic anion transmembrane transporter activity
Estradiolbenzoate//Solute carrier organic anion transporter family member 1A2//Sodium-independent organic anion transmembrane transporter activity
Estradiolbenzoate//Multidrug resistance-associated protein 7//Atpase activity, coupled to transmembrane movement of substances
Estradiolbenzoate//Solute carrier family 22 member 11//Sodium-independent organic anion transmembrane transporter activity
Estradiolbenzoate//ATP-binding cassette sub-family G member 2//Xenobiotic-transporting atpase activity
Estradiolbenzoate//Solute carrier organic anion transporter family member 1B1//Sodium-independent organic anion transmembrane transporter activity
Estradiolbenzoate//Multidrug resistance protein 1//Xenobiotic-transporting atpase activity
Estradiolbenzoate//Solute carrier family 22 member 8//Sodium-independent organic anion transmembrane transporter activity
Estradiolbenzoate//Solute carrier organic anion transporter family member 1B3//Sodium-independent organic anion transmembrane transporter activity
Estradiolbenzoate//Solute carrier organic anion transporter family member 1C1//Thyroid hormone transmembrane transporter activity
Estradiolbenzoate//Solute carrier organic anion transporter family member 4A1//Thyroid hormone transmembrane transporter activity
Estradiolcypionate//Solute carrier family 22 member 2//Quaternary ammonium group transmembrane transporter activity
Estradiolcypionate//Solute carrier family 22 member 1//Secondary active organic cation transmembrane transporter activity
Estradiolcypionate//Solute carrier family 22 member 3//Toxin transporter activity
Estradiolcypionate//Solute carrier organic anion transporter family member 2B1//Sodium-independent organic anion transmembrane transporter activity
Estradiolcypionate//Solute carrier organic anion transporter family member 1A2//Sodium-independent organic anion transmembrane transporter activity
Estradiolcypionate//Multidrug resistance-associated protein 7//Atpase activity, coupled to transmembrane movement of substances
Estradiolcypionate//Solute carrier family 22 member 11//Sodium-independent organic anion transmembrane transporter activity
Estradiolcypionate//ATP-binding cassette sub-family G member 2//Xenobiotic-transporting atpase activity
Estradiolcypionate//Solute carrier organic anion transporter family member 1B1//Sodium-independent organic anion transmembrane transporter activity
Estradiolcypionate//Multidrug resistance protein 1//Xenobiotic-transporting atpase activity
Estradiolcypionate//Solute carrier family 22 member 8//Sodium-independent organic anion transmembrane transporter activity
Estradiolcypionate//Solute carrier organic anion transporter family member 1B3//Sodium-independent organic anion transmembrane transporter activity
Estradiolcypionate//Solute carrier organic anion transporter family member 1C1//Thyroid hormone transmembrane transporter activity
Estradiolcypionate//Solute carrier organic anion transporter family member 4A1//Thyroid hormone transmembrane transporter activity
Estradioldienanthate//Solute carrier family 22 member 2//Quaternary ammonium group transmembrane transporter activity
Estradioldienanthate//Solute carrier family 22 member 1//Secondary active organic cation transmembrane transporter activity
Estradioldienanthate//Solute carrier family 22 member 3//Toxin transporter activity
Estradioldienanthate//Solute carrier organic anion transporter family member 2B1//Sodium-independent organic anion transmembrane transporter activity
Estradioldienanthate//Solute carrier organic anion transporter family member 1A2//Sodium-independent organic anion transmembrane transporter activity
Estradioldienanthate//Multidrug resistance-associated protein 7//Atpase activity, coupled to transmembrane movement of substances
Estradioldienanthate//Solute carrier family 22 member 11//Sodium-independent organic anion transmembrane transporter activity
Estradioldienanthate//ATP-binding cassette sub-family G member 2//Xenobiotic-transporting atpase activity
Estradioldienanthate//Solute carrier organic anion transporter family member 1B1//Sodium-independent organic anion transmembrane transporter activity
Estradioldienanthate//Multidrug resistance protein 1//Xenobiotic-transporting atpase activity
Estradioldienanthate//Solute carrier family 22 member 8//Sodium-independent organic anion transmembrane transporter activity
Estradioldienanthate//Solute carrier organic anion transporter family member 1B3//Sodium-independent organic anion transmembrane transporter activity
Estradioldienanthate//Solute carrier organic anion transporter family member 1C1//Thyroid hormone transmembrane transporter activity
Estradioldienanthate//Solute carrier organic anion transporter family member 4A1//Thyroid hormone transmembrane transporter activity
Estradiolvalerate//Solute carrier family 22 member 2//Quaternary ammonium group transmembrane transporter activity
Estradiolvalerate//Solute carrier family 22 member 1//Secondary active organic cation transmembrane transporter activity
Estradiolvalerate//Solute carrier family 22 member 3//Toxin transporter activity
Estradiolvalerate//Solute carrier organic anion transporter family member 2B1//Sodium-independent organic anion transmembrane transporter activity
Estradiolvalerate//Solute carrier organic anion transporter family member 1A2//Sodium-independent organic anion transmembrane transporter activity
Estradiolvalerate//Multidrug resistance-associated protein 7//Atpase activity, coupled to transmembrane movement of substances
Estradiolvalerate//Solute carrier family 22 member 11//Sodium-independent organic anion transmembrane transporter activity
Estradiolvalerate//ATP-binding cassette sub-family G member 2//Xenobiotic-transporting atpase activity
Estradiolvalerate//Solute carrier organic anion transporter family member 1B1//Sodium-independent organic anion transmembrane transporter activity
Estradiolvalerate//Multidrug resistance protein 1//Xenobiotic-transporting atpase activity
Estradiolvalerate//Solute carrier family 22 member 8//Sodium-independent organic anion transmembrane transporter activity
Estradiolvalerate//Solute carrier organic anion transporter family member 1B3//Sodium-independent organic anion transmembrane transporter activity
Estradiolvalerate//Solute carrier organic anion transporter family member 1C1//Thyroid hormone transmembrane transporter activity
Estradiolvalerate//Solute carrier organic anion transporter family member 4A1//Thyroid hormone transmembrane transporter activity
Cholinesalicylate//Solute carrier family 22 member 2//Quaternary ammonium group transmembrane transporter activity
Cholinesalicylate//Solute carrier family 22 member 1//Secondary active organic cation transmembrane transporter activity
Cholinesalicylate//Solute carrier family 22 member 3//Toxin transporter activity
Cholinesalicylate//Solute carrier family 22 member 5//Symporter activity
Cholinesalicylate//Solute carrier family 22 member 4//Symporter activity
Nabiximols//Multidrug resistance-associated protein 1//Transporter activity
Nabiximols//ATP-binding cassette sub-family G member 2//Xenobiotic-transporting atpase activity
Nabiximols//Equilibrative nucleoside transporter 1//Nucleoside transmembrane transporter activity
Bivalirudin//Myeloperoxidase//Peroxidase activity
Desmopressin//Prostaglandin G/H synthase 1//Prostaglandin-endoperoxide synthase activity
Desmopressin//Prostaglandin G/H synthase 2//Prostaglandin-endoperoxide synthase activity
Cyclosporine//Cytochrome P450 3A5//Oxygen binding
Cyclosporine//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Cyclosporine//Cytochrome P450 2C19//Steroid hydroxylase activity
Cyclosporine//Cytochrome P450 2D6//Steroid hydroxylase activity
Choline//Choline/ethanolaminephosphotransferase 1//Metal ion binding
Choline//Choline kinase alpha//Signal transducer activity
    Lglutamine//Coagulation factor XIII A chain//Protein-glutamine gamma-glutamyltransferase activity
    Lglutamine//Protein-glutamine gamma-glutamyltransferase 2//Protein-glutamine gamma-glutamyltransferase activity
    Lglutamine//Protein-glutamine gamma-glutamyltransferase 5//Protein-glutamine gamma-glutamyltransferase activity
    Lglutamine//Protein-glutamine gamma-glutamyltransferase 6//Protein-glutamine gamma-glutamyltransferase activity
    Lglutamine//Protein-glutamine gamma-glutamyltransferase K//Protein-glutamine gamma-glutamyltransferase activity
    Lglutamine//Protein-glutamine gamma-glutamyltransferase 4//Protein-glutamine gamma-glutamyltransferase activity
    Lglutamine//Protein-glutamine gamma-glutamyltransferase E//Transferase activity, transferring acyl groups
    Lglutamine//Protein-glutamine gamma-glutamyltransferase Z//Protein-glutamine gamma-glutamyltransferase activity
    Lglutamine//GMP synthase [glutamine-hydrolyzing]//Pyrophosphatase activity
    Lglutamine//Asparagine synthetase [glutamine-hydrolyzing]//Protein homodimerization activity
    Lglutamine//CAD protein//Zinc ion binding
Methionine//Glutamine synthetase//Manganese ion binding
Methionine//Methylenetetrahydrofolate reductase//Protein complex binding
Methionine//S-adenosylmethionine synthase isoform type-2//Methionine adenosyltransferase activity
Methionine//Methionine-R-sulfoxide reductase B2, mitochondrial//Zinc ion binding
Methionine//S-adenosylmethionine synthase isoform type-1//Methionine adenosyltransferase activity
Methionine//Methionine-R-sulfoxide reductase B1//Zinc ion binding
Methionine//Methionine--tRNA ligase, cytoplasmic//Trna binding
Methionine//S-methylmethionine--homocysteine S-methyltransferase BHMT2//Zinc ion binding
Calcitriol//1,25-dihydroxyvitamin D(3) 24-hydroxylase, mitochondrial//Oxidoreductase activity
Calcitriol//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Calcidiol//25-hydroxyvitamin D-1 alpha hydroxylase, mitochondrial//Iron ion binding
Calcidiol//1,25-dihydroxyvitamin D(3) 24-hydroxylase, mitochondrial//Oxidoreductase activity
Ltryptophan//Tryptophan 2,3-dioxygenase//Tryptophan 2,3-dioxygenase activity
Ltryptophan//Aromatic-L-amino-acid decarboxylase//Pyridoxal phosphate binding
Ltryptophan//Tryptophan--tRNA ligase//Tryptophan-trna ligase activity
Ltryptophan//Tryptophan--tRNA ligase, mitochondrial//Tryptophan-trna ligase activity
Ltryptophan//Tryptophan--tRNA ligase, cytoplasmic//Tryptophan-trna ligase activity
Ltryptophan//Indoleamine 2,3-dioxygenase 1//Tryptophan 2,3-dioxygenase activity
Ergocalciferol//1,25-dihydroxyvitamin D(3) 24-hydroxylase, mitochondrial//Oxidoreductase activity
Ergocalciferol//25-hydroxyvitamin D-1 alpha hydroxylase, mitochondrial//Iron ion binding
Ergocalciferol//Sterol 26-hydroxylase, mitochondrial//Vitamin d3 25-hydroxylase activity
Ergocalciferol//Vitamin D 25-hydroxylase//Vitamin d3 25-hydroxylase activity
Ergocalciferol//Cholesterol side-chain cleavage enzyme, mitochondrial//Oxidoreductase activity, acting on paired donors, with incorporation or reduction of molecular oxygen, nad(p)h as one donor, and incorporation of one atom of oxygen
Folicacid//Methylenetetrahydrofolate reductase//Protein complex binding
Folicacid//Dihydrofolate reductase//Nadph binding
Lipoicacid//NADPH--cytochrome P450 reductase//Oxidoreductase activity, acting on paired donors, with incorporation or reduction of molecular oxygen, nad(p)h as one donor, and incorporation of one atom of oxygen
Cholecalciferol//Vitamin D 25-hydroxylase//Vitamin d3 25-hydroxylase activity
Cholecalciferol//Sterol 26-hydroxylase, mitochondrial//Vitamin d3 25-hydroxylase activity
Cholecalciferol//Cytochrome P450 2J2//Steroid hydroxylase activity
Cholecalciferol//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Cholecalciferol//Cholesterol side-chain cleavage enzyme, mitochondrial//Oxidoreductase activity, acting on paired donors, with incorporation or reduction of molecular oxygen, nad(p)h as one donor, and incorporation of one atom of oxygen
Cholecalciferol//Cytochrome P450 1A1//Vitamin d 24-hydroxylase activity
Cholecalciferol//Cytochrome P450 2C8//Steroid hydroxylase activity
Menadione//Xanthine dehydrogenase/oxidase//Xanthine oxidase activity
Menadione//Aldehyde oxidase//Xanthine dehydrogenase activity
Menadione//Methylenetetrahydrofolate reductase//Protein complex binding
Menadione//Cytochrome P450 1A1//Vitamin d 24-hydroxylase activity
Menadione//Cytochrome P450 1A2//Oxidoreductase activity, acting on paired donors, with incorporation or reduction of molecular oxygen, reduced flavin or flavoprotein as one donor, and incorporation of one atom of oxygen
Menadione//Cytochrome P450 2A6//Steroid hydroxylase activity
Fluvoxamine//Cytochrome P450 2D6//Steroid hydroxylase activity
Fluvoxamine//Cytochrome P450 1A2//Oxidoreductase activity, acting on paired donors, with incorporation or reduction of molecular oxygen, reduced flavin or flavoprotein as one donor, and incorporation of one atom of oxygen
Fluvoxamine//Cytochrome P450 1A1//Vitamin d 24-hydroxylase activity
Fluvoxamine//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Fluvoxamine//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Fluvoxamine//Cytochrome P450 3A43//Monooxygenase activity
Fluvoxamine//Cytochrome P450 3A5//Oxygen binding
Fluvoxamine//Cytochrome P450 3A7//Oxygen binding
Fluvoxamine//Cytochrome P450 2C9//Steroid hydroxylase activity
Fluvoxamine//Cytochrome P450 2C19//Steroid hydroxylase activity
Fluvoxamine//Cytochrome P450 2B6//Steroid hydroxylase activity
Masoprocol//Arachidonate 5-lipoxygenase//Iron ion binding
Flunisolide//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Amphetamine//Cytochrome P450 2D6//Steroid hydroxylase activity
Amphetamine//Cytochrome P450 2A6//Steroid hydroxylase activity
Cevimeline//Cytochrome P450 2D6//Steroid hydroxylase activity
Cevimeline//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Cevimeline//Dimethylaniline monooxygenase [N-oxide-forming] 1//Nadp binding
Lorazepam//UDP-glucuronosyltransferase 2B15//Glucuronosyltransferase activity
Lorazepam//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Bortezomib//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Bortezomib//Cytochrome P450 2C19//Steroid hydroxylase activity
Bortezomib//Cytochrome P450 2D6//Steroid hydroxylase activity
Bortezomib//Cytochrome P450 1A2//Oxidoreductase activity, acting on paired donors, with incorporation or reduction of molecular oxygen, reduced flavin or flavoprotein as one donor, and incorporation of one atom of oxygen
Bortezomib//Cytochrome P450 2C9//Steroid hydroxylase activity
Betaxolol//Cytochrome P450 1A2//Oxidoreductase activity, acting on paired donors, with incorporation or reduction of molecular oxygen, reduced flavin or flavoprotein as one donor, and incorporation of one atom of oxygen
Betaxolol//Cytochrome P450 2D6//Steroid hydroxylase activity
Erythromycin//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Erythromycin//Cytochrome P450 3A7//Oxygen binding
Erythromycin//Cytochrome P450 3A5//Oxygen binding
Caffeine//Cytochrome P450 1A2//Oxidoreductase activity, acting on paired donors, with incorporation or reduction of molecular oxygen, reduced flavin or flavoprotein as one donor, and incorporation of one atom of oxygen
Caffeine//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Caffeine//Cytochrome P450 2E1//Steroid hydroxylase activity
Caffeine//Cytochrome P450 2C8//Steroid hydroxylase activity
Caffeine//Cytochrome P450 2C9//Steroid hydroxylase activity
Caffeine//Cytochrome P450 1A1//Vitamin d 24-hydroxylase activity
Caffeine//Cytochrome P450 1B1//Oxygen binding
Caffeine//Cytochrome P450 2D6//Steroid hydroxylase activity
Dofetilide//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Azithromycin//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Midodrine//Cytochrome P450 2D6//Steroid hydroxylase activity
Citalopram//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Citalopram//Cytochrome P450 2C19//Steroid hydroxylase activity
Citalopram//Cytochrome P450 2D6//Steroid hydroxylase activity
Citalopram//Cytochrome P450 1A2//Oxidoreductase activity, acting on paired donors, with incorporation or reduction of molecular oxygen, reduced flavin or flavoprotein as one donor, and incorporation of one atom of oxygen
Eletriptan//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Eletriptan//Cytochrome P450 2D6//Steroid hydroxylase activity
Eletriptan//Cytochrome P450 2C9//Steroid hydroxylase activity
Eletriptan//Cytochrome P450 2C19//Steroid hydroxylase activity
Eletriptan//Cytochrome P450 2A6//Steroid hydroxylase activity
Eletriptan//Prostaglandin G/H synthase 1//Prostaglandin-endoperoxide synthase activity
Glimepiride//Cytochrome P450 2C9//Steroid hydroxylase activity
Lovastatin//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Lovastatin//Serum paraoxonase/lactonase 3//Protein homodimerization activity
Lovastatin//Cytochrome P450 2C8//Steroid hydroxylase activity
Lovastatin//UDP-glucuronosyltransferase 1-1//Steroid binding
Lovastatin//UDP-glucuronosyltransferase 1-3//Retinoic acid binding
Lovastatin//UDP-glucuronosyltransferase 2B7//Glucuronosyltransferase activity
Lovastatin//Cytochrome P450 2C19//Steroid hydroxylase activity
Enflurane//Cytochrome P450 2E1//Steroid hydroxylase activity
Aminosalicylicacid//Myeloperoxidase//Peroxidase activity
Alclometasone//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Cladribine//Deoxycytidine kinase//Protein homodimerization activity
Cabergoline//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Doxycycline//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Diethylstilbestrol//Catechol O-methyltransferase//O-methyltransferase activity
Diethylstilbestrol//Aromatase//Oxygen binding
Diethylstilbestrol//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Diethylstilbestrol//Cytochrome P450 2C8//Steroid hydroxylase activity
Diethylstilbestrol//Cytochrome P450 2C9//Steroid hydroxylase activity
Diethylstilbestrol//Cytochrome P450 2E1//Steroid hydroxylase activity
Clotrimazole//Cytochrome P450 2C8//Steroid hydroxylase activity
Clotrimazole//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Clotrimazole//Cytochrome P450 2B6//Steroid hydroxylase activity
Clotrimazole//Cytochrome P450 2D6//Steroid hydroxylase activity
Clotrimazole//Cytochrome P450 2A6//Steroid hydroxylase activity
Clotrimazole//Cytochrome P450 2C9//Steroid hydroxylase activity
Clotrimazole//Cytochrome P450 2E1//Steroid hydroxylase activity
Clotrimazole//Cytochrome P450 3A7//Oxygen binding
Anagrelide//Cytochrome P450 1A2//Oxidoreductase activity, acting on paired donors, with incorporation or reduction of molecular oxygen, reduced flavin or flavoprotein as one donor, and incorporation of one atom of oxygen
Metoprolol//Cytochrome P450 2D6//Steroid hydroxylase activity
Metoprolol//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Dicoumarol//Cytochrome P450 2C9//Steroid hydroxylase activity
Isradipine//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Argatroban//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Argatroban//Cytochrome P450 3A5//Oxygen binding
Disopyramide//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Disopyramide//Cytochrome P450 1A2//Oxidoreductase activity, acting on paired donors, with incorporation or reduction of molecular oxygen, reduced flavin or flavoprotein as one donor, and incorporation of one atom of oxygen
Lidocaine//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Lidocaine//Cytochrome P450 2D6//Steroid hydroxylase activity
Lidocaine//Cytochrome P450 3A5//Oxygen binding
Lidocaine//Cytochrome P450 3A7//Oxygen binding
Lidocaine//Cytochrome P450 1A2//Oxidoreductase activity, acting on paired donors, with incorporation or reduction of molecular oxygen, reduced flavin or flavoprotein as one donor, and incorporation of one atom of oxygen
Lidocaine//Cytochrome P450 2C9//Steroid hydroxylase activity
Lidocaine//Cytochrome P450 2C8//Steroid hydroxylase activity
Lidocaine//Cytochrome P450 2A6//Steroid hydroxylase activity
Lidocaine//Cytochrome P450 2B6//Steroid hydroxylase activity
Clemastine//Cytochrome P450 2D6//Steroid hydroxylase activity
Atomoxetine//Cytochrome P450 2D6//Steroid hydroxylase activity
Atomoxetine//Cytochrome P450 2C19//Steroid hydroxylase activity
Etomidate//Cytochrome P450 11B1, mitochondrial//Steroid 11-beta-monooxygenase activity
Etomidate//Cytochrome P450 11B2, mitochondrial//Steroid 11-beta-monooxygenase activity
Etonogestrel//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Morphine//Cytochrome P450 2C8//Steroid hydroxylase activity
Morphine//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Morphine//UDP-glucuronosyltransferase 2B7//Glucuronosyltransferase activity
Morphine//UDP-glucuronosyltransferase 1-1//Steroid binding
Morphine//UDP-glucuronosyltransferase 1-8//Steroid binding
Morphine//UDP-glucuronosyltransferase 2B15//Glucuronosyltransferase activity
Morphine//UDP-glucuronosyltransferase 2B4//Glucuronosyltransferase activity
Morphine//UDP-glucuronosyltransferase 1-3//Retinoic acid binding
Bupivacaine//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Bupivacaine//Cytochrome P450 2C19//Steroid hydroxylase activity
Bupivacaine//Cytochrome P450 2D6//Steroid hydroxylase activity
Bexarotene//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Bexarotene//Cytochrome P450 2C8//Steroid hydroxylase activity
Acetaminophen//Cytochrome P450 2E1//Steroid hydroxylase activity
Acetaminophen//Cytochrome P450 1A2//Oxidoreductase activity, acting on paired donors, with incorporation or reduction of molecular oxygen, reduced flavin or flavoprotein as one donor, and incorporation of one atom of oxygen
Acetaminophen//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Acetaminophen//Cytochrome P450 2D6//Steroid hydroxylase activity
Acetaminophen//Cytochrome P450 2A6//Steroid hydroxylase activity
Acetaminophen//UDP-glucuronosyltransferase 1-6//Protein homodimerization activity
Acetaminophen//UDP-glucuronosyltransferase 1-1//Steroid binding
Acetaminophen//UDP-glucuronosyltransferase 1-9//Retinoic acid binding
Acetaminophen//UDP-glucuronosyltransferase 2B15//Glucuronosyltransferase activity
Acetaminophen//Sulfotransferase 1A1//Sulfotransferase activity
Acetaminophen//Sulfotransferase 1A3//Sulfotransferase that utilizes 3'-phospho-5'-adenylyl sulfate (PAPS) as sulfonate donor to catalyze the sulfate conjugation of phenolic monoamines (neurotransmitters such as dopamine, norepinephrine and serotonin) and phenolic and catechol drugs.
Acetaminophen//Arylamine N-acetyltransferase 2//Arylamine n-acetyltransferase activity
Acetaminophen//Fatty-acid amide hydrolase 1//Fatty acid amide hydrolase activity
Acetaminophen//Glutathione S-transferase P//S-nitrosoglutathione binding
Acetaminophen//Glutathione S-transferase Mu 1//Protein homodimerization activity
Gefitinib//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Gefitinib//Cytochrome P450 2D6//Steroid hydroxylase activity
Gefitinib//Cytochrome P450 3A5//Oxygen binding
Gefitinib//Cytochrome P450 1A1//Vitamin d 24-hydroxylase activity
Gefitinib//Cytochrome P450 2C9//Steroid hydroxylase activity
Gefitinib//Cytochrome P450 2C19//Steroid hydroxylase activity
Codeine//Cytochrome P450 2D6//Steroid hydroxylase activity
Codeine//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Codeine//UDP-glucuronosyltransferase 2B7//Glucuronosyltransferase activity
Codeine//UDP-glucuronosyltransferase 2B4//Glucuronosyltransferase activity
Dihydroergotamine//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Amitriptyline//Cytochrome P450 2D6//Steroid hydroxylase activity
Amitriptyline//Cytochrome P450 1A2//Oxidoreductase activity, acting on paired donors, with incorporation or reduction of molecular oxygen, reduced flavin or flavoprotein as one donor, and incorporation of one atom of oxygen
Amitriptyline//Cytochrome P450 2C19//Steroid hydroxylase activity
Amitriptyline//Cytochrome P450 2C9//Steroid hydroxylase activity
Amitriptyline//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Amitriptyline//Cytochrome P450 3A5//Oxygen binding
Amitriptyline//Cytochrome P450 2B6//Steroid hydroxylase activity
Amitriptyline//Cytochrome P450 2C8//Steroid hydroxylase activity
Amitriptyline//UDP-glucuronosyltransferase 2B10//UDPGT is of major importance in the conjugation and subsequent elimination of potentially toxic xenobiotics and endogenous compounds.
Amitriptyline//UDP-glucuronosyltransferase 1-4//Protein homodimerization activity
Floxuridine//Thymidine phosphorylase//Transferase activity, transferring pentosyl groups
Floxuridine//Cytochrome P450 2C9//Steroid hydroxylase activity
Fluorometholone//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Fluorometholone//Cytochrome P450 3A5//Oxygen binding
Hydromorphone//Cytochrome P450 2C9//Steroid hydroxylase activity
Hydromorphone//UDP-glucuronosyltransferase 1-3//Retinoic acid binding
Hydromorphone//UDP-glucuronosyltransferase 2B7//Glucuronosyltransferase activity
Indomethacin//Cytochrome P450 2C19//Steroid hydroxylase activity
Indomethacin//Cytochrome P450 2C9//Steroid hydroxylase activity
Indomethacin//Liver carboxylesterase 1//Triglyceride lipase activity
Indomethacin//UDP-glucuronosyltransferase 1-9//Retinoic acid binding
Indomethacin//UDP-glucuronosyltransferase 1-1//Steroid binding
Indomethacin//UDP-glucuronosyltransferase 2B7//Glucuronosyltransferase activity
Methadone//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Methadone//Cytochrome P450 2C19//Steroid hydroxylase activity
Methadone//Cytochrome P450 3A7//Oxygen binding
Methadone//Cytochrome P450 2D6//Steroid hydroxylase activity
Methadone//Cytochrome P450 2B6//Steroid hydroxylase activity
Methadone//Cytochrome P450 2C8//Steroid hydroxylase activity
Methadone//Aromatase//Oxygen binding
Methadone//Cytochrome P450 1A2//Oxidoreductase activity, acting on paired donors, with incorporation or reduction of molecular oxygen, reduced flavin or flavoprotein as one donor, and incorporation of one atom of oxygen
Methadone//Cytochrome P450 2C18//Steroid hydroxylase activity
Methadone//Cytochrome P450 2C9//Steroid hydroxylase activity
Diltiazem//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Diltiazem//Cytochrome P450 3A5//Oxygen binding
Diltiazem//Cytochrome P450 3A7//Oxygen binding
Diltiazem//Cytochrome P450 2C19//Steroid hydroxylase activity
Diltiazem//Cytochrome P450 2D6//Steroid hydroxylase activity
Diltiazem//Cytochrome P450 2C8//Steroid hydroxylase activity
Alfuzosin//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Methylergometrine//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Chlorzoxazone//Cytochrome P450 2E1//Steroid hydroxylase activity
Chlorzoxazone//Cytochrome P450 1A1//Vitamin d 24-hydroxylase activity
Chlorzoxazone//Cytochrome P450 1A2//Oxidoreductase activity, acting on paired donors, with incorporation or reduction of molecular oxygen, reduced flavin or flavoprotein as one donor, and incorporation of one atom of oxygen
Chlorzoxazone//Cytochrome P450 2A6//Steroid hydroxylase activity
Chlorzoxazone//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Chlorzoxazone//Cytochrome P450 2D6//Steroid hydroxylase activity
Aminoglutethimide//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Aminoglutethimide//Cytochrome P450 2C19//Steroid hydroxylase activity
Mefloquine//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Mefloquine//Cholinesterase//Identical protein binding
Mefloquine//Aromatase//Oxygen binding
Mefloquine//Acetylcholinesterase//Serine hydrolase activity
Clozapine//Cytochrome P450 1A2//Oxidoreductase activity, acting on paired donors, with incorporation or reduction of molecular oxygen, reduced flavin or flavoprotein as one donor, and incorporation of one atom of oxygen
Clozapine//Cytochrome P450 2D6//Steroid hydroxylase activity
Clozapine//Cytochrome P450 2C9//Steroid hydroxylase activity
Clozapine//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Clozapine//Cytochrome P450 2C19//Steroid hydroxylase activity
Clozapine//Cytochrome P450 2A6//Steroid hydroxylase activity
Clozapine//Cytochrome P450 2C8//Steroid hydroxylase activity
Clozapine//Dimethylaniline monooxygenase [N-oxide-forming] 3//Trimethylamine monooxygenase activity
Clozapine//UDP-glucuronosyltransferase 1-4//Protein homodimerization activity
Clozapine//Cytochrome P450 1A1//Vitamin d 24-hydroxylase activity
Doxylamine//CYP2B protein//Oxidoreductase activity, acting on paired donors, with incorporation or reduction of molecular oxygen, reduced flavin or flavoprotein as one donor, and incorporation of one atom of oxygen
Levonorgestrel//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Levonorgestrel//Cytochrome P450 3A5//Oxygen binding
Mirtazapine//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Mirtazapine//Cytochrome P450 2D6//Steroid hydroxylase activity
Mirtazapine//Cytochrome P450 1A2//Oxidoreductase activity, acting on paired donors, with incorporation or reduction of molecular oxygen, reduced flavin or flavoprotein as one donor, and incorporation of one atom of oxygen
Mexiletine//Cytochrome P450 1A2//Oxidoreductase activity, acting on paired donors, with incorporation or reduction of molecular oxygen, reduced flavin or flavoprotein as one donor, and incorporation of one atom of oxygen
Mexiletine//Cytochrome P450 2D6//Steroid hydroxylase activity
Mexiletine//Cytochrome P450 2B6//Steroid hydroxylase activity
Mexiletine//Cytochrome P450 2E1//Steroid hydroxylase activity
Mexiletine//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Amlodipine//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Amlodipine//Cytochrome P450 1A1//Vitamin d 24-hydroxylase activity
Amlodipine//Cytochrome P450 2B6//Steroid hydroxylase activity
Amlodipine//Cytochrome P450 3A5//Oxygen binding
Amlodipine//Cytochrome P450 2C8//Steroid hydroxylase activity
Amlodipine//Cytochrome P450 2D6//Steroid hydroxylase activity
Carbimazole//Aromatase//Oxygen binding
Digoxin//Cholesterol side-chain cleavage enzyme, mitochondrial//Oxidoreductase activity, acting on paired donors, with incorporation or reduction of molecular oxygen, nad(p)h as one donor, and incorporation of one atom of oxygen
Ethopropazine//Cholinesterase//Identical protein binding
Beclomethasonedipropionate//Cytochrome P450 3A5//Oxygen binding
Beclomethasonedipropionate//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Carisoprodol//Cytochrome P450 2C19//Steroid hydroxylase activity
Griseofulvin//Cytochrome P450 1A2//Oxidoreductase activity, acting on paired donors, with incorporation or reduction of molecular oxygen, reduced flavin or flavoprotein as one donor, and incorporation of one atom of oxygen
Griseofulvin//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Eszopiclone//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Eszopiclone//Cytochrome P450 2C8//Steroid hydroxylase activity
Carbachol//Cytosolic phospholipase A2//Phospholipase a2 activity
Acetohexamide//Carbonyl reductase [NADPH] 1//Prostaglandin-e2 9-reductase activity
Acetohexamide//Cytochrome P450 2C9//Steroid hydroxylase activity
Cyproheptadine//UDP-glucuronosyltransferase 1-3//Retinoic acid binding
Bendroflumethiazide//Thiopurine S-methyltransferase//Thiopurine s-methyltransferase activity
Allopurinol//Aldehyde oxidase//Xanthine dehydrogenase activity
Allopurinol//Xanthine dehydrogenase/oxidase//Xanthine oxidase activity
Cerivastatin//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Cerivastatin//Cytochrome P450 3A5//Oxygen binding
Cerivastatin//Cytochrome P450 3A7//Oxygen binding
Cerivastatin//Cytochrome P450 2C8//Steroid hydroxylase activity
Cerivastatin//Cytochrome P450 2D6//Steroid hydroxylase activity
Cerivastatin//Cytochrome P450 2C9//Steroid hydroxylase activity
Cerivastatin//Cytochrome P450 2B6//Steroid hydroxylase activity
Cerivastatin//UDP-glucuronosyltransferase 1-1//Steroid binding
Gemcitabine//Cytidine deaminase//Zinc ion binding
Gemcitabine//Deoxycytidine kinase//Protein homodimerization activity
Betamethasone//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Betamethasone//Aromatase//Oxygen binding
Betamethasone//Cytochrome P450 3A5//Oxygen binding
Betamethasone//Cytochrome P450 3A7//Oxygen binding
Betamethasone//Cytochrome P450 2A6//Steroid hydroxylase activity
Betamethasone//Cytochrome P450 1B1//Oxygen binding
Betamethasone//Cytochrome P450 2B6//Steroid hydroxylase activity
Betamethasone//Cytochrome P450 2C8//Steroid hydroxylase activity
Betamethasone//Cytochrome P450 2C9//Steroid hydroxylase activity
Betamethasone//Cytochrome P450 2C19//Steroid hydroxylase activity
Epirubicin//UDP-glucuronosyltransferase 2B7//Glucuronosyltransferase activity
Epirubicin//Cytosolic phospholipase A2//Phospholipase a2 activity
Chloramphenicol//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Chloramphenicol//Cytochrome P450 3A5//Oxygen binding
Chloramphenicol//Cytochrome P450 3A7//Oxygen binding
Chloramphenicol//Cytochrome P450 2C19//Steroid hydroxylase activity
Lansoprazole//Cytochrome P450 1A1//Vitamin d 24-hydroxylase activity
Lansoprazole//Cytochrome P450 1B1//Oxygen binding
Lansoprazole//Cytochrome P450 2C8//Steroid hydroxylase activity
Lansoprazole//Cytochrome P450 2C9//Steroid hydroxylase activity
Lansoprazole//Cytochrome P450 2C18//Steroid hydroxylase activity
Lansoprazole//Cytochrome P450 2D6//Steroid hydroxylase activity
Lansoprazole//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Lansoprazole//Cytochrome P450 2C19//Steroid hydroxylase activity
Levothyroxine//Cytochrome P450 2C8//Steroid hydroxylase activity
Levothyroxine//UDP-glucuronosyltransferase 1-1//Steroid binding
Levothyroxine//Multidrug resistance protein 1//Xenobiotic-transporting atpase activity
Loratadine//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Loratadine//Cytochrome P450 2D6//Steroid hydroxylase activity
Loratadine//Cytochrome P450 1A1//Vitamin d 24-hydroxylase activity
Loratadine//Cytochrome P450 2C19//Steroid hydroxylase activity
Loratadine//Cytochrome P450 2C8//Steroid hydroxylase activity
Loratadine//Cytochrome P450 1A2//Oxidoreductase activity, acting on paired donors, with incorporation or reduction of molecular oxygen, reduced flavin or flavoprotein as one donor, and incorporation of one atom of oxygen
Loratadine//Cytochrome P450 2B6//Steroid hydroxylase activity
Loratadine//Cytochrome P450 2C9//Steroid hydroxylase activity
Loratadine//Cytochrome P450 3A5//Oxygen binding
Loratadine//UDP-glucuronosyltransferase 2B10//UDPGT is of major importance in the conjugation and subsequent elimination of potentially toxic xenobiotics and endogenous compounds.
Loratadine//UDP-glucuronosyltransferase 1-1//Steroid binding
Loratadine//UDP-glucuronosyltransferase 1-3//Retinoic acid binding
Loratadine//UDP-glucuronosyltransferase 2B15//Glucuronosyltransferase activity
Imipramine//Cytochrome P450 2C19//Steroid hydroxylase activity
Imipramine//Cytochrome P450 2D6//Steroid hydroxylase activity
Imipramine//Cytochrome P450 1A2//Oxidoreductase activity, acting on paired donors, with incorporation or reduction of molecular oxygen, reduced flavin or flavoprotein as one donor, and incorporation of one atom of oxygen
Imipramine//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Imipramine//Cytochrome P450 3A7//Oxygen binding
Imipramine//Cytochrome P450 2B6//Steroid hydroxylase activity
Imipramine//Cytochrome P450 2C18//Steroid hydroxylase activity
Imipramine//Cytochrome P450 2E1//Steroid hydroxylase activity
Nabumetone//Myeloperoxidase//Peroxidase activity
Nabumetone//Cytochrome P450 1A2//Oxidoreductase activity, acting on paired donors, with incorporation or reduction of molecular oxygen, reduced flavin or flavoprotein as one donor, and incorporation of one atom of oxygen
Nabumetone//Cytochrome P450 2C9//Steroid hydroxylase activity
Nabumetone//Corticosteroid 11-beta-dehydrogenase isozyme 1//11-beta-hydroxysteroid dehydrogenase [nad(p)] activity
Nabumetone//Aldo-keto reductase family 1 member C1//Trans-1,2-dihydrobenzene-1,2-diol dehydrogenase activity
Nabumetone//Aldo-keto reductase family 1 member C2//Trans-1,2-dihydrobenzene-1,2-diol dehydrogenase activity
Nabumetone//Aldo-keto reductase family 1 member C4//Retinal dehydrogenase activity
Enoxacin//Cytochrome P450 1A2//Oxidoreductase activity, acting on paired donors, with incorporation or reduction of molecular oxygen, reduced flavin or flavoprotein as one donor, and incorporation of one atom of oxygen
Dronabinol//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Dronabinol//Cytochrome P450 2C9//Steroid hydroxylase activity
Dronabinol//Prostaglandin G/H synthase 1//Prostaglandin-endoperoxide synthase activity
Montelukast//Cytochrome P450 2C8//Steroid hydroxylase activity
Montelukast//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Montelukast//Cytochrome P450 2C9//Steroid hydroxylase activity
Montelukast//Prostaglandin G/H synthase 1//Prostaglandin-endoperoxide synthase activity
Montelukast//Cytochrome P450 2A6//Steroid hydroxylase activity
Fluoxetine//Cytochrome P450 2C19//Steroid hydroxylase activity
Fluoxetine//Cytochrome P450 2D6//Steroid hydroxylase activity
Fluoxetine//Cytochrome P450 2C9//Steroid hydroxylase activity
Fluoxetine//CYP2B protein//Oxidoreductase activity, acting on paired donors, with incorporation or reduction of molecular oxygen, reduced flavin or flavoprotein as one donor, and incorporation of one atom of oxygen
Fluoxetine//Cytochrome P450 1A2//Oxidoreductase activity, acting on paired donors, with incorporation or reduction of molecular oxygen, reduced flavin or flavoprotein as one donor, and incorporation of one atom of oxygen
Fluoxetine//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Fluoxetine//Cytochrome P450 2B6//Steroid hydroxylase activity
Fluoxetine//Cytochrome P450 3A5//Oxygen binding
Duloxetine//Cytochrome P450 1A2//Oxidoreductase activity, acting on paired donors, with incorporation or reduction of molecular oxygen, reduced flavin or flavoprotein as one donor, and incorporation of one atom of oxygen
Duloxetine//Cytochrome P450 2D6//Steroid hydroxylase activity
Duloxetine//Cytochrome P450 2C9//Steroid hydroxylase activity
Chlorpromazine//Cytochrome P450 2D6//Steroid hydroxylase activity
Chlorpromazine//Cytochrome P450 1A2//Oxidoreductase activity, acting on paired donors, with incorporation or reduction of molecular oxygen, reduced flavin or flavoprotein as one donor, and incorporation of one atom of oxygen
Chlorpromazine//Cytochrome P450 2E1//Steroid hydroxylase activity
Chlorpromazine//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Chlorpromazine//Cholinesterase//Identical protein binding
Celecoxib//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Celecoxib//Cytochrome P450 2C9//Steroid hydroxylase activity
Celecoxib//Cytochrome P450 2D6//Steroid hydroxylase activity
Celecoxib//Cytochrome P450 2C8//Steroid hydroxylase activity
Brimonidine//Aldehyde oxidase//Xanthine dehydrogenase activity
Nabilone//Cytochrome P450 2E1//Steroid hydroxylase activity
Nabilone//Cytochrome P450 2C8//Steroid hydroxylase activity
Nabilone//Cytochrome P450 2C9//Steroid hydroxylase activity
Buspirone//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Buspirone//Cytochrome P450 3A5//Oxygen binding
Buspirone//Cytochrome P450 3A7//Oxygen binding
Buspirone//Cytochrome P450 2D6//Steroid hydroxylase activity
Entacapone//Catechol O-methyltransferase//O-methyltransferase activity
Entacapone//UDP-glucuronosyltransferase 1-9//Retinoic acid binding
Entacapone//Cytochrome P450 2D6//Steroid hydroxylase activity
Darifenacin//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Darifenacin//Cytochrome P450 2D6//Steroid hydroxylase activity
Flutamide//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Flutamide//Cytochrome P450 1A2//Oxidoreductase activity, acting on paired donors, with incorporation or reduction of molecular oxygen, reduced flavin or flavoprotein as one donor, and incorporation of one atom of oxygen
Flutamide//Cytochrome P450 1A1//Vitamin d 24-hydroxylase activity
Flutamide//Cytochrome P450 1B1//Oxygen binding
Flutamide//Cytochrome P450 2C19//Steroid hydroxylase activity
Flutamide//Cytochrome P450 3A5//Oxygen binding
Cimetidine//Cytochrome P450 1A2//Oxidoreductase activity, acting on paired donors, with incorporation or reduction of molecular oxygen, reduced flavin or flavoprotein as one donor, and incorporation of one atom of oxygen
Cimetidine//Cytochrome P450 2C19//Steroid hydroxylase activity
Cimetidine//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Cimetidine//Cytochrome P450 3A5//Oxygen binding
Cimetidine//Cytochrome P450 2D6//Steroid hydroxylase activity
Cimetidine//Cytochrome P450 11B1, mitochondrial//Steroid 11-beta-monooxygenase activity
Cimetidine//Cytochrome P450 2C8//Steroid hydroxylase activity
Cimetidine//Cytochrome P450 2C9//Steroid hydroxylase activity
Cimetidine//Cytochrome P450 2E1//Steroid hydroxylase activity
Cimetidine//Dimethylaniline monooxygenase [N-oxide-forming] 3//Trimethylamine monooxygenase activity
Cimetidine//Dimethylaniline monooxygenase [N-oxide-forming] 1//Nadp binding
Haloperidol//Cytochrome P450 3A5//Oxygen binding
Haloperidol//Cytochrome P450 3A7//Oxygen binding
Haloperidol//Cytochrome P450 1A2//Oxidoreductase activity, acting on paired donors, with incorporation or reduction of molecular oxygen, reduced flavin or flavoprotein as one donor, and incorporation of one atom of oxygen
Haloperidol//Cytochrome P450 2D6//Steroid hydroxylase activity
Haloperidol//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Haloperidol//Carbonyl reductase [NADPH] 1//Prostaglandin-e2 9-reductase activity
Haloperidol//UDP-glucuronosyltransferase 1-9//Retinoic acid binding
Haloperidol//Cytochrome P450 2C19//Steroid hydroxylase activity
Haloperidol//Cytochrome P450 2C9//Steroid hydroxylase activity
Haloperidol//Cytochrome P450 1A1//Vitamin d 24-hydroxylase activity
Dextromethorphan//Cytochrome P450 2D6//Steroid hydroxylase activity
Dextromethorphan//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Dextromethorphan//Cytochrome P450 3A7//Oxygen binding
Dextromethorphan//Cytochrome P450 2B6//Steroid hydroxylase activity
Dextromethorphan//Cytochrome P450 2C19//Steroid hydroxylase activity
Dextromethorphan//Cytochrome P450 2C9//Steroid hydroxylase activity
Cisplatin//Myeloperoxidase//Peroxidase activity
Cisplatin//Xanthine dehydrogenase/oxidase//Xanthine oxidase activity
Cisplatin//Cytochrome P450 4A11//Leukotriene-b4 20-monooxygenase activity
Cisplatin//Prostaglandin G/H synthase 2//Prostaglandin-endoperoxide synthase activity
Cisplatin//Cytochrome P450 2C9//Steroid hydroxylase activity
Cisplatin//Cytochrome P450 2B6//Steroid hydroxylase activity
Cisplatin//Cholinesterase//Identical protein binding
Cisplatin//Glutathione S-transferase theta-1//Glutathione transferase activity
Cisplatin//Metallothionein-1A//Zinc ion binding
Cisplatin//Metallothionein-2//Zinc ion binding
Cisplatin//Superoxide dismutase [Cu-Zn]//Zinc ion binding
Cisplatin//Glutathione S-transferase P//S-nitrosoglutathione binding
Cisplatin//NAD(P)H dehydrogenase [quinone] 1//Superoxide dismutase activity
Cisplatin//Glutathione S-transferase Mu 1//Protein homodimerization activity
Albendazole//Cytochrome P450 1A1//Vitamin d 24-hydroxylase activity
Albendazole//Cytochrome P450 1A2//Oxidoreductase activity, acting on paired donors, with incorporation or reduction of molecular oxygen, reduced flavin or flavoprotein as one donor, and incorporation of one atom of oxygen
Albendazole//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Albendazole//Cytochrome P450 2C19//Steroid hydroxylase activity
Carteolol//Cytochrome P450 2D6//Steroid hydroxylase activity
Cinchocaine//Cholinesterase//Identical protein binding
Lercanidipine//Cytochrome P450 3A7//Oxygen binding
Lercanidipine//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Lercanidipine//Cytochrome P450 3A5//Oxygen binding
Lercanidipine//Cytochrome P450 2D6//Steroid hydroxylase activity
Erlotinib//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Erlotinib//Cytochrome P450 3A5//Oxygen binding
Erlotinib//Cytochrome P450 1A2//Oxidoreductase activity, acting on paired donors, with incorporation or reduction of molecular oxygen, reduced flavin or flavoprotein as one donor, and incorporation of one atom of oxygen
Erlotinib//Cytochrome P450 1A1//Vitamin d 24-hydroxylase activity
Erlotinib//Cytochrome P450 2D6//Steroid hydroxylase activity
Erlotinib//Cytochrome P450 2C8//Steroid hydroxylase activity
Erlotinib//Cytochrome P450 1B1//Oxygen binding
Erlotinib//UDP-glucuronosyltransferase 1-1//Steroid binding
Cyclophosphamide//Cytochrome P450 2C9//Steroid hydroxylase activity
Cyclophosphamide//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Cyclophosphamide//Cytochrome P450 2B6//Steroid hydroxylase activity
Cyclophosphamide//Cytochrome P450 2C19//Steroid hydroxylase activity
Cyclophosphamide//Cytochrome P450 2A6//Steroid hydroxylase activity
Cyclophosphamide//Cytochrome P450 2C18//Steroid hydroxylase activity
Cyclophosphamide//Cytochrome P450 2C8//Steroid hydroxylase activity
Cyclophosphamide//Cytochrome P450 3A5//Oxygen binding
Ciprofloxacin//Cytochrome P450 1A2//Oxidoreductase activity, acting on paired donors, with incorporation or reduction of molecular oxygen, reduced flavin or flavoprotein as one donor, and incorporation of one atom of oxygen
Ciprofloxacin//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Ciprofloxacin//Cytochrome P450 3A5//Oxygen binding
Ciprofloxacin//Cytochrome P450 3A7//Oxygen binding
Benazepril//Methylenetetrahydrofolate reductase//Protein complex binding
Amoxapine//Cytochrome P450 2D6//Steroid hydroxylase activity
Fluorouracil//Cytochrome P450 2C9//Steroid hydroxylase activity
Fluorouracil//Cytochrome P450 1A2//Oxidoreductase activity, acting on paired donors, with incorporation or reduction of molecular oxygen, reduced flavin or flavoprotein as one donor, and incorporation of one atom of oxygen
Fluorouracil//Thymidine phosphorylase//Transferase activity, transferring pentosyl groups
Fluorouracil//Dihydropyrimidine dehydrogenase [NADP(+)]//Protein homodimerization activity
Fluorouracil//Uridine phosphorylase 1//Uridine phosphorylase activity
Fluorouracil//Uridine phosphorylase 2//Uridine phosphorylase activity
Fluorouracil//Cytochrome P450 2A6//Steroid hydroxylase activity
Fluorouracil//Cytochrome P450 2C8//Steroid hydroxylase activity
Fluorouracil//Methylenetetrahydrofolate reductase//Protein complex binding
Fluorouracil//Thymidylate synthase//Thymidylate synthase activity
Fluorouracil//Amidophosphoribosyltransferase//Metal ion binding
Adinazolam//Cytochrome P450 2C19//Steroid hydroxylase activity
Adinazolam//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Lamotrigine//UDP-glucuronosyltransferase 1-1//Steroid binding
Lamotrigine//UDP-glucuronosyltransferase 1-10//Protein kinase c binding
Lamotrigine//UDP-glucuronosyltransferase 1-3//Retinoic acid binding
Lamotrigine//UDP-glucuronosyltransferase 1-4//Protein homodimerization activity
Lamotrigine//UDP-glucuronosyltransferase 1-6//Protein homodimerization activity
Lamotrigine//UDP-glucuronosyltransferase 1-7//Retinoic acid binding
Lamotrigine//UDP-glucuronosyltransferase 1-8//Steroid binding
Lamotrigine//UDP-glucuronosyltransferase 1-9//Retinoic acid binding
Lamotrigine//UDP-glucuronosyltransferase 2B15//Glucuronosyltransferase activity
Lamotrigine//UDP-glucuronosyltransferase 2B4//Glucuronosyltransferase activity
Lamotrigine//UDP-glucuronosyltransferase 2B7//Glucuronosyltransferase activity
Lamotrigine//Dihydrofolate reductase//Nadph binding
Hydroxyzine//Cytochrome P450 2D6//Steroid hydroxylase activity
Hydroxyzine//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Hydroxyzine//Cytochrome P450 3A5//Oxygen binding
Bosentan//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Bosentan//Cytochrome P450 2C9//Steroid hydroxylase activity
Methotrexate//Dihydrofolate reductase//Nadph binding
Methotrexate//Aldehyde oxidase//Xanthine dehydrogenase activity
Methotrexate//Methylenetetrahydrofolate reductase//Protein complex binding
Methotrexate//6-phosphogluconate dehydrogenase, decarboxylating//Phosphogluconate dehydrogenase (decarboxylating) activity
Methotrexate//Thymidylate synthase//Thymidylate synthase activity
Methotrexate//Bifunctional purine biosynthesis protein PURH//Protein homodimerization activity
Methotrexate//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Carbamazepine//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Carbamazepine//Cytochrome P450 2C8//Steroid hydroxylase activity
Carbamazepine//Cytochrome P450 1A2//Oxidoreductase activity, acting on paired donors, with incorporation or reduction of molecular oxygen, reduced flavin or flavoprotein as one donor, and incorporation of one atom of oxygen
Carbamazepine//Cytochrome P450 2C9//Steroid hydroxylase activity
Carbamazepine//Cytochrome P450 2C19//Steroid hydroxylase activity
Carbamazepine//Cytochrome P450 2B6//Steroid hydroxylase activity
Carbamazepine//Cytochrome P450 3A5//Oxygen binding
Carbamazepine//UDP-glucuronosyltransferase 2B7//Glucuronosyltransferase activity
Carbamazepine//UDP-glucuronosyltransferase 1-1//Steroid binding
Carbamazepine//UDP-glucuronosyltransferase 1-6//Protein homodimerization activity
Carbamazepine//UDP-glucuronosyltransferase 1-7//Retinoic acid binding
Cinnarizine//Cytochrome P450 2D6//Steroid hydroxylase activity
Cinnarizine//Cytochrome P450 2C9//Steroid hydroxylase activity
Cinnarizine//Cytochrome P450 1A2//Oxidoreductase activity, acting on paired donors, with incorporation or reduction of molecular oxygen, reduced flavin or flavoprotein as one donor, and incorporation of one atom of oxygen
Cinnarizine//Cytochrome P450 2B6//Steroid hydroxylase activity
Cinnarizine//Cytochrome P450 2A6//Steroid hydroxylase activity
Cinnarizine//Cytochrome P450 1A1//Vitamin d 24-hydroxylase activity
Cinnarizine//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Fenfluramine//Cytochrome P450 2D6//Steroid hydroxylase activity
Clonidine//Cytochrome P450 2D6//Steroid hydroxylase activity
Clonidine//Cytochrome P450 1A2//Oxidoreductase activity, acting on paired donors, with incorporation or reduction of molecular oxygen, reduced flavin or flavoprotein as one donor, and incorporation of one atom of oxygen
Clonidine//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Clonidine//Cytochrome P450 1A1//Vitamin d 24-hydroxylase activity
Clonidine//Cytochrome P450 3A5//Oxygen binding
Diclofenac//Cytochrome P450 2C9//Steroid hydroxylase activity
Diclofenac//Cytochrome P450 2C19//Steroid hydroxylase activity
Diclofenac//Cytochrome P450 1A2//Oxidoreductase activity, acting on paired donors, with incorporation or reduction of molecular oxygen, reduced flavin or flavoprotein as one donor, and incorporation of one atom of oxygen
Diclofenac//Cytochrome P450 2C8//Steroid hydroxylase activity
Diclofenac//UDP-glucuronosyltransferase 2B7//Glucuronosyltransferase activity
Diclofenac//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Diclofenac//Cytochrome P450 2B6//Steroid hydroxylase activity
Diclofenac//Cytochrome P450 2C18//Steroid hydroxylase activity
Diclofenac//Cytochrome P450 2E1//Steroid hydroxylase activity
Diclofenac//UDP-glucuronosyltransferase 1-3//Retinoic acid binding
Diclofenac//UDP-glucuronosyltransferase 1-9//Retinoic acid binding
Diclofenac//UDP-glucuronosyltransferase 2B4//Glucuronosyltransferase activity
Diclofenac//Arachidonate 5-lipoxygenase//Iron ion binding
Diclofenac//Phospholipase A2, membrane associated//Phospholipid binding
Fluticasonepropionate//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Fluticasonepropionate//Cytochrome P450 3A5//Oxygen binding
Fluticasonepropionate//Cytochrome P450 3A7//Oxygen binding
Fluticasonepropionate//Cytochrome P450 2C8//Steroid hydroxylase activity
Lisuride//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Doxazosin//Cytochrome P450 2C19//Steroid hydroxylase activity
Doxazosin//Cytochrome P450 2D6//Steroid hydroxylase activity
Doxazosin//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Doxazosin//Cytochrome P450 2C9//Steroid hydroxylase activity
Fluocinoloneacetonide//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Ethosuximide//Cytochrome P450 2E1//Steroid hydroxylase activity
Ethosuximide//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Ethosuximide//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Ethosuximide//Cytochrome P450 3A43//Monooxygenase activity
Ethosuximide//Cytochrome P450 3A5//Oxygen binding
Ethosuximide//Cytochrome P450 3A7//Oxygen binding
Amiloride//Amiloride-sensitive amine oxidase [copper-containing]//Zinc ion binding
Amiloride//Amiloride-sensitive amine oxidase [copper-containing]//Zinc ion binding
Labetalol//Cytochrome P450 2D6//Steroid hydroxylase activity
Labetalol//Cytochrome P450 2C19//Steroid hydroxylase activity
Labetalol//UDP-glucuronosyltransferase 1-1//Steroid binding
Labetalol//UDP-glucuronosyltransferase 2B7//Glucuronosyltransferase activity
Labetalol//UDP-glucuronosyltransferase 1-9//Retinoic acid binding
Ivermectin//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Medroxyprogesteroneacetate//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Medroxyprogesteroneacetate//Cytochrome P450 2C8//Steroid hydroxylase activity
Medroxyprogesteroneacetate//Cytochrome P450 2C9//Steroid hydroxylase activity
Cisapride//Cytochrome P450 3A7//Oxygen binding
Cisapride//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Cisapride//Cytochrome P450 3A5//Oxygen binding
Cisapride//Cytochrome P450 2A6//Steroid hydroxylase activity
Cisapride//Cytochrome P450 2B6//Steroid hydroxylase activity
Cisapride//Cytochrome P450 2C19//Steroid hydroxylase activity
Cisapride//Cytochrome P450 2C8//Steroid hydroxylase activity
Cisapride//Cytochrome P450 2C9//Steroid hydroxylase activity
Cisapride//Cytochrome P450 2D6//Steroid hydroxylase activity
Chloroquine//Cytochrome P450 2C8//Steroid hydroxylase activity
Chloroquine//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Chloroquine//Cytochrome P450 3A5//Oxygen binding
Chloroquine//Cytochrome P450 2D6//Steroid hydroxylase activity
Chloroquine//Cytochrome P450 1A1//Vitamin d 24-hydroxylase activity
Bisoprolol//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Amodiaquine//Cytochrome P450 2C8//Steroid hydroxylase activity
Amodiaquine//Cytochrome P450 1A1//Vitamin d 24-hydroxylase activity
Amodiaquine//Cytochrome P450 1B1//Oxygen binding
Amodiaquine//Cytochrome P450 2D6//Steroid hydroxylase activity
Amodiaquine//Cytochrome P450 2C9//Steroid hydroxylase activity
Imatinib//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Imatinib//Cytochrome P450 3A5//Oxygen binding
Imatinib//Cytochrome P450 3A7//Oxygen binding
Imatinib//Cytochrome P450 1A2//Oxidoreductase activity, acting on paired donors, with incorporation or reduction of molecular oxygen, reduced flavin or flavoprotein as one donor, and incorporation of one atom of oxygen
Imatinib//Cytochrome P450 2C9//Steroid hydroxylase activity
Imatinib//Cytochrome P450 2D6//Steroid hydroxylase activity
Imatinib//Cytochrome P450 2C19//Steroid hydroxylase activity
Imatinib//Prostaglandin G/H synthase 1//Prostaglandin-endoperoxide synthase activity
Imatinib//Cytochrome P450 2C8//Steroid hydroxylase activity
Nicardipine//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Nicardipine//Cytochrome P450 2D6//Steroid hydroxylase activity
Nicardipine//Cytochrome P450 2C19//Steroid hydroxylase activity
Nicardipine//Cytochrome P450 2C8//Steroid hydroxylase activity
Nicardipine//Cytochrome P450 2B6//Steroid hydroxylase activity
Nicardipine//Cytochrome P450 2E1//Steroid hydroxylase activity
Nicardipine//Cytochrome P450 3A5//Oxygen binding
Nicardipine//Cytochrome P450 2C9//Steroid hydroxylase activity
Fluphenazine//Cytochrome P450 2D6//Steroid hydroxylase activity
Fluphenazine//Cytochrome P450 2E1//Steroid hydroxylase activity
Niacin//Cytochrome P450 2D6//Steroid hydroxylase activity
Niacin//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Niacin//Cytochrome P450 2E1//Steroid hydroxylase activity
Clorazepate//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Guanabenz//Cytochrome P450 1A2//Oxidoreductase activity, acting on paired donors, with incorporation or reduction of molecular oxygen, reduced flavin or flavoprotein as one donor, and incorporation of one atom of oxygen
Clofarabine//Deoxycytidine kinase//Protein homodimerization activity
Dexmedetomidine//Cytochrome P450 2E1//Steroid hydroxylase activity
Dexmedetomidine//Cytochrome P450 1A2//Oxidoreductase activity, acting on paired donors, with incorporation or reduction of molecular oxygen, reduced flavin or flavoprotein as one donor, and incorporation of one atom of oxygen
Dexmedetomidine//Cytochrome P450 1A1//Vitamin d 24-hydroxylase activity
Dexmedetomidine//Cytochrome P450 2D6//Steroid hydroxylase activity
Clofibrate//Cytochrome P450 2E1//Steroid hydroxylase activity
Clofibrate//Glutathione S-transferase A2//Glutathione transferase activity
Clofibrate//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Clofibrate//Cytochrome P450 1A1//Vitamin d 24-hydroxylase activity
Clofibrate//Cytochrome P450 4A11//Leukotriene-b4 20-monooxygenase activity
Astemizole//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Astemizole//Cytochrome P450 3A5//Oxygen binding
Astemizole//Cytochrome P450 3A7//Oxygen binding
Astemizole//Cytochrome P450 2D6//Steroid hydroxylase activity
Astemizole//Cytochrome P450 2J2//Steroid hydroxylase activity
Adenosine//Adenosine deaminase//Zinc ion binding
Adenosine//Adenosine kinase//Poly(a) rna binding
Mebendazole//Cytochrome P450 1A1//Vitamin d 24-hydroxylase activity
Mebendazole//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Mebendazole//Cytochrome P450 3A43//Monooxygenase activity
Mebendazole//Cytochrome P450 3A5//Oxygen binding
Mebendazole//Cytochrome P450 3A7//Oxygen binding
Dextropropoxyphene//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Dextropropoxyphene//Cytochrome P450 2D6//Steroid hydroxylase activity
Mitotane//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Estrone//Cytochrome P450 1A1//Vitamin d 24-hydroxylase activity
Estrone//Cytochrome P450 1A2//Oxidoreductase activity, acting on paired donors, with incorporation or reduction of molecular oxygen, reduced flavin or flavoprotein as one donor, and incorporation of one atom of oxygen
Estrone//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Estrone//Cytochrome P450 1B1//Oxygen binding
Estrone//Cytochrome P450 2B6//Steroid hydroxylase activity
Estrone//Cytochrome P450 2C9//Steroid hydroxylase activity
Estrone//Cytochrome P450 2E1//Steroid hydroxylase activity
Estrone//Cytochrome P450 3A5//Oxygen binding
Epinephrine//Cytochrome P450 2C9//Steroid hydroxylase activity
Epinephrine//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Epinephrine//Catechol O-methyltransferase//O-methyltransferase activity
Epinephrine//Amine oxidase [flavin-containing] A//Serotonin binding
Epinephrine//Amine oxidase [flavin-containing] B//Primary amine oxidase activity
Chlorpropamide//Cytochrome P450 2C9//Steroid hydroxylase activity
Chlorpropamide//Cytochrome P450 2C19//Steroid hydroxylase activity
Chlorpropamide//Prostaglandin G/H synthase 1//Prostaglandin-endoperoxide synthase activity
Aprepitant//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Aprepitant//Cytochrome P450 2C19//Steroid hydroxylase activity
Aprepitant//Cytochrome P450 2C9//Steroid hydroxylase activity
Galantamine//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Galantamine//Cytochrome P450 2D6//Steroid hydroxylase activity
Isoflurophate//Cholinesterase//Identical protein binding
Losartan//Cytochrome P450 2C9//Steroid hydroxylase activity
Losartan//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Losartan//Cytochrome P450 2C19//Steroid hydroxylase activity
Losartan//UDP-glucuronosyltransferase 1-1//Steroid binding
Losartan//UDP-glucuronosyltransferase 1-3//Retinoic acid binding
Losartan//UDP-glucuronosyltransferase 1-10//Protein kinase c binding
Losartan//UDP-glucuronosyltransferase 2B7//Glucuronosyltransferase activity
Losartan//UDP-glucuronosyltransferase 2B17//Glucuronosyltransferase activity
Losartan//Cytochrome P450 2C8//Steroid hydroxylase activity
Midazolam//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Midazolam//UDP-glucuronosyltransferase 1-4//Protein homodimerization activity
Midazolam//Cytochrome P450 3A5//Oxygen binding
Midazolam//Cytochrome P450 3A7//Oxygen binding
Mycophenolatemofetil//UDP-glucuronosyltransferase 1-1//Steroid binding
Mycophenolatemofetil//UDP-glucuronosyltransferase 1-7//Retinoic acid binding
Mycophenolatemofetil//UDP-glucuronosyltransferase 1-6//Protein homodimerization activity
Mycophenolatemofetil//UDP-glucuronosyltransferase 1-9//Retinoic acid binding
Mycophenolatemofetil//UDP-glucuronosyltransferase 2B7//Glucuronosyltransferase activity
Mycophenolatemofetil//UDP-glucuronosyltransferase 1-8//Steroid binding
Mycophenolatemofetil//UDP-glucuronosyltransferase 1-10//Protein kinase c binding
Mycophenolatemofetil//Liver carboxylesterase 1//Triglyceride lipase activity
Mycophenolatemofetil//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Mycophenolatemofetil//Cytochrome P450 3A5//Oxygen binding
Mycophenolatemofetil//Cytochrome P450 2C8//Steroid hydroxylase activity
Flurazepam//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Flurazepam//Cytochrome P450 2E1//Steroid hydroxylase activity
Flurazepam//Cytochrome P450 2A6//Steroid hydroxylase activity
Daunorubicin//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Daunorubicin//Cytochrome P450 3A5//Oxygen binding
Daunorubicin//Cytochrome P450 1A1//Vitamin d 24-hydroxylase activity
Daunorubicin//Cytochrome P450 1B1//Oxygen binding
Daunorubicin//Xanthine dehydrogenase/oxidase//Xanthine oxidase activity
Daunorubicin//NADPH--cytochrome P450 reductase//Oxidoreductase activity, acting on paired donors, with incorporation or reduction of molecular oxygen, nad(p)h as one donor, and incorporation of one atom of oxygen
Furosemide//6-phosphogluconate dehydrogenase, decarboxylating//Phosphogluconate dehydrogenase (decarboxylating) activity
Furosemide//UDP-glucuronosyltransferase 1-1//Steroid binding
Ergotamine//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Eplerenone//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Eplerenone//Cytochrome P450 3A5//Oxygen binding
Eplerenone//Cytochrome P450 11B2, mitochondrial//Steroid 11-beta-monooxygenase activity
Naltrexone//UDP-glucuronosyltransferase 1-1//Steroid binding
Diethylcarbamazine//Cholinesterase//Identical protein binding
Flurbiprofen//Cytochrome P450 2C9//Steroid hydroxylase activity
Flurbiprofen//UDP-glucuronosyltransferase 2B7//Glucuronosyltransferase activity
Flurbiprofen//UDP-glucuronosyltransferase 1-1//Steroid binding
Flurbiprofen//UDP-glucuronosyltransferase 1-3//Retinoic acid binding
Flurbiprofen//UDP-glucuronosyltransferase 1-9//Retinoic acid binding
Flurbiprofen//UDP-glucuronosyltransferase 2B4//Glucuronosyltransferase activity
Apomorphine//Catechol O-methyltransferase//O-methyltransferase activity
Apomorphine//Sulfotransferase 1A1//Sulfotransferase activity
Apomorphine//Sulfotransferase 1A3//Sulfotransferase that utilizes 3'-phospho-5'-adenylyl sulfate (PAPS) as sulfonate donor to catalyze the sulfate conjugation of phenolic monoamines (neurotransmitters such as dopamine, norepinephrine and serotonin) and phenolic and catechol drugs.
Apomorphine//Estrogen sulfotransferase//Sulfotransferase activity
Apomorphine//Sulfotransferase family cytosolic 1B member 1//Sulfotransferase activity
Apomorphine//Cytochrome P450 2B6//Steroid hydroxylase activity
Apomorphine//Cytochrome P450 2C8//Steroid hydroxylase activity
Apomorphine//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Apomorphine//Cytochrome P450 3A5//Oxygen binding
Apomorphine//UDP-glucuronosyltransferase 1-1//Steroid binding
Apomorphine//UDP-glucuronosyltransferase 1-10//Protein kinase c binding
Apomorphine//UDP-glucuronosyltransferase 1-3//Retinoic acid binding
Apomorphine//UDP-glucuronosyltransferase 1-4//Protein homodimerization activity
Apomorphine//UDP-glucuronosyltransferase 1-6//Protein homodimerization activity
Apomorphine//UDP-glucuronosyltransferase 1-7//Retinoic acid binding
Apomorphine//UDP-glucuronosyltransferase 1-8//Steroid binding
Apomorphine//UDP-glucuronosyltransferase 1-9//Retinoic acid binding
Apomorphine//UDP-glucuronosyltransferase 2B15//Glucuronosyltransferase activity
Apomorphine//UDP-glucuronosyltransferase 2B4//Glucuronosyltransferase activity
Apomorphine//UDP-glucuronosyltransferase 2B7//Glucuronosyltransferase activity
Azatadine//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Clodronicacid//Prostaglandin G/H synthase 2//Prostaglandin-endoperoxide synthase activity
Imiquimod//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Nateglinide//Cytochrome P450 2C9//Steroid hydroxylase activity
Nateglinide//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Nateglinide//Cytochrome P450 3A5//Oxygen binding
Nateglinide//Cytochrome P450 3A7//Oxygen binding
Nateglinide//Prostaglandin G/H synthase 1//Prostaglandin-endoperoxide synthase activity
Nateglinide//UDP-glucuronosyltransferase 1-9//Retinoic acid binding
Nateglinide//Cytochrome P450 2D6//Steroid hydroxylase activity
Esomeprazole//Cytochrome P450 2C19//Steroid hydroxylase activity
Esomeprazole//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Meclizine//Cytochrome P450 2D6//Steroid hydroxylase activity
Hydrocortisone//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Hydrocortisone//Cytochrome P450 3A5//Oxygen binding
Hydrocortisone//Cytochrome P450 3A7//Oxygen binding
Hydrocortisone//Cytochrome P450 11B1, mitochondrial//Steroid 11-beta-monooxygenase activity
Hydrocortisone//Cytochrome P450 11B2, mitochondrial//Steroid 11-beta-monooxygenase activity
Hydrocortisone//Cytochrome P450 2C8//Steroid hydroxylase activity
Hydrocortisone//3-oxo-5-beta-steroid 4-dehydrogenase//Steroid binding
Hydrocortisone//3-oxo-5-alpha-steroid 4-dehydrogenase 2//Sterol 5-alpha reductase activity
Hydrocortisone//Corticosteroid 11-beta-dehydrogenase isozyme 2//Steroid binding
Hydrocortisone//Corticosteroid 11-beta-dehydrogenase isozyme 1//11-beta-hydroxysteroid dehydrogenase [nad(p)] activity
Hydrocortisone//Cytochrome P450 2A6//Steroid hydroxylase activity
Hydrocortisone//Cytochrome P450 1B1//Oxygen binding
Hydrocortisone//Cytochrome P450 2B6//Steroid hydroxylase activity
Hydrocortisone//Cytochrome P450 2C9//Steroid hydroxylase activity
Hydrocortisone//Cytochrome P450 2C19//Steroid hydroxylase activity
Modafinil//Cytochrome P450 2C19//Steroid hydroxylase activity
Modafinil//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Modafinil//Cytochrome P450 1A2//Oxidoreductase activity, acting on paired donors, with incorporation or reduction of molecular oxygen, reduced flavin or flavoprotein as one donor, and incorporation of one atom of oxygen
Modafinil//Cytochrome P450 2B6//Steroid hydroxylase activity
Modafinil//Cytochrome P450 2C9//Steroid hydroxylase activity
Modafinil//Cytochrome P450 3A5//Oxygen binding
Etodolac//Cytochrome P450 2C9//Steroid hydroxylase activity
Etodolac//UDP-glucuronosyltransferase 1-9//Retinoic acid binding
Etodolac//UDP-glucuronosyltransferase 1-3//Retinoic acid binding
Etodolac//UDP-glucuronosyltransferase 1-10//Protein kinase c binding
Etodolac//UDP-glucuronosyltransferase 2B7//Glucuronosyltransferase activity
Epinastine//Cytochrome P450 2B6//Steroid hydroxylase activity
Epinastine//Cytochrome P450 2D6//Steroid hydroxylase activity
Epinastine//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Isoflurane//Cytochrome P450 2E1//Steroid hydroxylase activity
Isoflurane//Cytochrome P450 2B6//Steroid hydroxylase activity
Isoflurane//NADH-ubiquinone oxidoreductase chain 1//Nadh dehydrogenase (ubiquinone) activity
Dolasetron//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Dolasetron//Cytochrome P450 2D6//Steroid hydroxylase activity
Dolasetron//Cytochrome P450 2C9//Steroid hydroxylase activity
Clopidogrel//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Clopidogrel//Cytochrome P450 2B6//Steroid hydroxylase activity
Clopidogrel//Cytochrome P450 3A5//Oxygen binding
Clopidogrel//Cytochrome P450 2C19//Steroid hydroxylase activity
Clopidogrel//Cytochrome P450 2C9//Steroid hydroxylase activity
Clopidogrel//Cytochrome P450 1A2//Oxidoreductase activity, acting on paired donors, with incorporation or reduction of molecular oxygen, reduced flavin or flavoprotein as one donor, and incorporation of one atom of oxygen
Clopidogrel//Cytochrome P450 2C8//Steroid hydroxylase activity
Clopidogrel//Liver carboxylesterase 1//Triglyceride lipase activity
Irinotecan//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Irinotecan//Cytochrome P450 3A5//Oxygen binding
Irinotecan//Cytochrome P450 2B6//Steroid hydroxylase activity
Irinotecan//Cytochrome P450 3A7//Oxygen binding
Irinotecan//UDP-glucuronosyltransferase 1-1//Steroid binding
Irinotecan//UDP-glucuronosyltransferase 1-9//Retinoic acid binding
Irinotecan//Liver carboxylesterase 1//Triglyceride lipase activity
Irinotecan//Cholinesterase//Identical protein binding
Methimazole//Cytochrome P450 1A2//Oxidoreductase activity, acting on paired donors, with incorporation or reduction of molecular oxygen, reduced flavin or flavoprotein as one donor, and incorporation of one atom of oxygen
Methimazole//Cytochrome P450 2A6//Steroid hydroxylase activity
Methimazole//Cytochrome P450 2B6//Steroid hydroxylase activity
Methimazole//Cytochrome P450 2C19//Steroid hydroxylase activity
Methimazole//Cytochrome P450 2C9//Steroid hydroxylase activity
Methimazole//Cytochrome P450 2D6//Steroid hydroxylase activity
Methimazole//Cytochrome P450 2E1//Steroid hydroxylase activity
Methimazole//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Methimazole//Dimethylaniline monooxygenase [N-oxide-forming] 3//Trimethylamine monooxygenase activity
Mometasone//Cytochrome P450 2C8//Steroid hydroxylase activity
Mometasone//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Mometasone//Cytochrome P450 3A5//Oxygen binding
Hydrocortamate//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Malathion//Cytochrome P450 1A2//Oxidoreductase activity, acting on paired donors, with incorporation or reduction of molecular oxygen, reduced flavin or flavoprotein as one donor, and incorporation of one atom of oxygen
Malathion//Cytochrome P450 2B6//Steroid hydroxylase activity
Etoposide//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Etoposide//Cytochrome P450 1A2//Oxidoreductase activity, acting on paired donors, with incorporation or reduction of molecular oxygen, reduced flavin or flavoprotein as one donor, and incorporation of one atom of oxygen
Etoposide//Cytochrome P450 2E1//Steroid hydroxylase activity
Etoposide//Cytochrome P450 3A5//Oxygen binding
Etoposide//UDP-glucuronosyltransferase 1-1//Steroid binding
Etoposide//Glutathione S-transferase theta-1//Glutathione transferase activity
Etoposide//Glutathione S-transferase P//S-nitrosoglutathione binding
Etoposide//Prostaglandin G/H synthase 2//Prostaglandin-endoperoxide synthase activity
Etoposide//Prostaglandin G/H synthase 1//Prostaglandin-endoperoxide synthase activity
Estradiol//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Estradiol//Cytochrome P450 1A2//Oxidoreductase activity, acting on paired donors, with incorporation or reduction of molecular oxygen, reduced flavin or flavoprotein as one donor, and incorporation of one atom of oxygen
Estradiol//Cytochrome P450 3A5//Oxygen binding
Estradiol//Cytochrome P450 3A7//Oxygen binding
Estradiol//UDP-glucuronosyltransferase 1-1//Steroid binding
Estradiol//Cytochrome P450 1A1//Vitamin d 24-hydroxylase activity
Estradiol//Cytochrome P450 1B1//Oxygen binding
Estradiol//Cytochrome P450 2C19//Steroid hydroxylase activity
Estradiol//Cytochrome P450 2C8//Steroid hydroxylase activity
Estradiol//Cytochrome P450 2C9//Steroid hydroxylase activity
Estradiol//UDP-glucuronosyltransferase 2B15//Glucuronosyltransferase activity
Estradiol//Catechol O-methyltransferase//O-methyltransferase activity
Estradiol//UDP-glucuronosyltransferase 1-1//Steroid binding
Estradiol//UDP-glucuronosyltransferase 1-10//Protein kinase c binding
Estradiol//UDP-glucuronosyltransferase 1-3//Retinoic acid binding
Estradiol//UDP-glucuronosyltransferase 1-4//Protein homodimerization activity
Estradiol//UDP-glucuronosyltransferase 1-6//Protein homodimerization activity
Estradiol//UDP-glucuronosyltransferase 1-7//Retinoic acid binding
Estradiol//UDP-glucuronosyltransferase 1-8//Steroid binding
Estradiol//UDP-glucuronosyltransferase 1-9//Retinoic acid binding
Estradiol//UDP-glucuronosyltransferase 2B15//Glucuronosyltransferase activity
Estradiol//UDP-glucuronosyltransferase 2B4//Glucuronosyltransferase activity
Estradiol//UDP-glucuronosyltransferase 2B7//Glucuronosyltransferase activity
Mefenamicacid//Cytochrome P450 2C9//Steroid hydroxylase activity
Mefenamicacid//Cytochrome P450 2C8//Steroid hydroxylase activity
Mefenamicacid//UDP-glucuronosyltransferase 1-9//Retinoic acid binding
Naproxen//Cytochrome P450 2C9//Steroid hydroxylase activity
Naproxen//Cytochrome P450 1A2//Oxidoreductase activity, acting on paired donors, with incorporation or reduction of molecular oxygen, reduced flavin or flavoprotein as one donor, and incorporation of one atom of oxygen
Naproxen//Cytochrome P450 2C8//Steroid hydroxylase activity
Naproxen//UDP-glucuronosyltransferase 2B7//Glucuronosyltransferase activity
Naproxen//UDP-glucuronosyltransferase 1-3//Retinoic acid binding
Naproxen//UDP-glucuronosyltransferase 1-6//Protein homodimerization activity
Naproxen//UDP-glucuronosyltransferase 1-7//Retinoic acid binding
Naproxen//UDP-glucuronosyltransferase 1-8//Steroid binding
Naproxen//UDP-glucuronosyltransferase 1-9//Retinoic acid binding
Naproxen//UDP-glucuronosyltransferase 1-10//Protein kinase c binding
Candesartancilexetil//Cytochrome P450 2C9//Steroid hydroxylase activity
Candesartancilexetil//Cytochrome P450 2C8//Steroid hydroxylase activity
Candesartancilexetil//UDP-glucuronosyltransferase 1-3//Retinoic acid binding
Candesartancilexetil//Prostaglandin G/H synthase 1//Prostaglandin-endoperoxide synthase activity
Alfentanil//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Alfentanil//Cytochrome P450 3A7//Oxygen binding
Alfentanil//Cytochrome P450 3A5//Oxygen binding
Minaprine//Cytochrome P450 2D6//Steroid hydroxylase activity
Indapamide//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Biperiden//Cytochrome P450 2D6//Steroid hydroxylase activity
Fentanyl//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Fentanyl//Cytochrome P450 3A7//Oxygen binding
Meloxicam//Cytochrome P450 2C9//Steroid hydroxylase activity
Meloxicam//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Meloxicam//6-phosphogluconate dehydrogenase, decarboxylating//Phosphogluconate dehydrogenase (decarboxylating) activity
Meloxicam//Cytochrome P450 2C8//Steroid hydroxylase activity
Acetazolamide//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Disulfiram//Cytochrome P450 2E1//Steroid hydroxylase activity
Disulfiram//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Disulfiram//Cytochrome P450 3A5//Oxygen binding
Diazepam//Cytochrome P450 2C9//Steroid hydroxylase activity
Diazepam//Cytochrome P450 3A7//Oxygen binding
Diazepam//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Diazepam//Cytochrome P450 2C19//Steroid hydroxylase activity
Diazepam//Cytochrome P450 3A5//Oxygen binding
Diazepam//Cytochrome P450 2B6//Steroid hydroxylase activity
Diazepam//Prostaglandin G/H synthase 1//Prostaglandin-endoperoxide synthase activity
Diazepam//Cytochrome P450 2C18//Steroid hydroxylase activity
Diazepam//Cytochrome P450 2C8//Steroid hydroxylase activity
Diazepam//Cytochrome P450 2E1//Steroid hydroxylase activity
Mifepristone//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Mifepristone//Cytochrome P450 3A5//Oxygen binding
Mifepristone//Cytochrome P450 2D6//Steroid hydroxylase activity
Mifepristone//Cytochrome P450 2C8//Steroid hydroxylase activity
Mifepristone//Cytochrome P450 2C9//Steroid hydroxylase activity
Loperamide//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Loperamide//Cytochrome P450 2C8//Steroid hydroxylase activity
Loperamide//Cytochrome P450 2B6//Steroid hydroxylase activity
Loperamide//Cytochrome P450 2D6//Steroid hydroxylase activity
Dobutamine//Catechol O-methyltransferase//O-methyltransferase activity
Donepezil//Cytochrome P450 2D6//Steroid hydroxylase activity
Donepezil//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Donepezil//Cytochrome P450 2C9//Steroid hydroxylase activity
Clofazimine//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Clofazimine//Cytochrome P450 3A5//Oxygen binding
Clofazimine//Cytochrome P450 2C8//Steroid hydroxylase activity
Clofazimine//Cytochrome P450 2D6//Steroid hydroxylase activity
Cysteamine//Myeloperoxidase//Peroxidase activity
Methylphenobarbital//Cytochrome P450 2C19//Steroid hydroxylase activity
Methylphenobarbital//Cytochrome P450 2B6//Steroid hydroxylase activity
Dacarbazine//Cytochrome P450 1A1//Vitamin d 24-hydroxylase activity
Dacarbazine//Cytochrome P450 1A2//Oxidoreductase activity, acting on paired donors, with incorporation or reduction of molecular oxygen, reduced flavin or flavoprotein as one donor, and incorporation of one atom of oxygen
Dacarbazine//Cytochrome P450 2E1//Steroid hydroxylase activity
Diflunisal//UDP-glucuronosyltransferase 1-8//Steroid binding
Diflunisal//UDP-glucuronosyltransferase 1-9//Retinoic acid binding
Benzphetamine//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Benzphetamine//Cytochrome P450 2B6//Steroid hydroxylase activity
Benzphetamine//NADPH--cytochrome P450 reductase//Oxidoreductase activity, acting on paired donors, with incorporation or reduction of molecular oxygen, nad(p)h as one donor, and incorporation of one atom of oxygen
Alprenolol//Cytochrome P450 2D6//Steroid hydroxylase activity
Dorzolamide//Cytochrome P450 2C9//Steroid hydroxylase activity
Dorzolamide//Cytochrome P450 2B1//Steroid hydroxylase activity
Dorzolamide//Cytochrome P450 2E1//Steroid hydroxylase activity
Conivaptan//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Flupentixol//Aromatic-L-amino-acid decarboxylase//Pyridoxal phosphate binding
Clomifene//Steroid 17-alpha-hydroxylase/17,20 lyase//Steroid 17-alpha-monooxygenase activity
Isosorbidedinitrate//Cytochrome P450 2E1//Steroid hydroxylase activity
Bumetanide//Prostaglandin G/H synthase 2//Prostaglandin-endoperoxide synthase activity
Granisetron//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Granisetron//Cytochrome P450 1A1//Vitamin d 24-hydroxylase activity
Ethanol//Cytochrome P450 1A1//Vitamin d 24-hydroxylase activity
Ethanol//Cytochrome P450 1A2//Oxidoreductase activity, acting on paired donors, with incorporation or reduction of molecular oxygen, reduced flavin or flavoprotein as one donor, and incorporation of one atom of oxygen
Ethanol//Cytochrome P450 2B6//Steroid hydroxylase activity
Ethanol//Cytochrome P450 2C9//Steroid hydroxylase activity
Ethanol//Cytochrome P450 2C19//Steroid hydroxylase activity
Ethanol//Cytochrome P450 2E1//Steroid hydroxylase activity
Ethanol//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Ethanol//Cytochrome P450 4A11//Leukotriene-b4 20-monooxygenase activity
Ethanol//Alcohol dehydrogenase 1A//Zinc ion binding
Ethanol//Alcohol dehydrogenase 1B//Zinc ion binding
Ethanol//Alcohol dehydrogenase 1C//Zinc ion binding
Ethanol//Alcohol dehydrogenase class-3//Zinc ion binding
Ethanol//Alcohol dehydrogenase 4//Zinc ion binding
Ethanol//Alcohol dehydrogenase class 4 mu/sigma chain//Zinc ion binding
Ethanol//Alcohol dehydrogenase 6//Zinc ion binding
Etacrynicacid//Glutathione S-transferase A2//Glutathione transferase activity
Cocaine//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Cocaine//Cytochrome P450 2D6//Steroid hydroxylase activity
Cocaine//Cytochrome P450 2C8//Steroid hydroxylase activity
Cocaine//Cholinesterase//Identical protein binding
Cocaine//Liver carboxylesterase 1//Triglyceride lipase activity
Amantadine//Aromatic-L-amino-acid decarboxylase//Pyridoxal phosphate binding
Amantadine//Amine oxidase [flavin-containing] B//Primary amine oxidase activity
Metronidazole//Cytochrome P450 2C9//Steroid hydroxylase activity
Metronidazole//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Metronidazole//Cytochrome P450 2C8//Steroid hydroxylase activity
Metronidazole//UDP-glucuronosyltransferase 1-1//Steroid binding
Metronidazole//Cytochrome P450 2A6//Steroid hydroxylase activity
Metronidazole//Cytochrome P450 3A5//Oxygen binding
Metronidazole//Cytochrome P450 3A7//Oxygen binding
Almotriptan//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Almotriptan//Cytochrome P450 2D6//Steroid hydroxylase activity
Almotriptan//Amine oxidase [flavin-containing] A//Serotonin binding
Almotriptan//Dimethylaniline monooxygenase [N-oxide-forming] 3//Trimethylamine monooxygenase activity
Almotriptan//Cytochrome P450 2C19//Steroid hydroxylase activity
Almotriptan//Cytochrome P450 2E1//Steroid hydroxylase activity
Almotriptan//Cytochrome P450 2C8//Steroid hydroxylase activity
Buprenorphine//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Buprenorphine//Cytochrome P450 3A5//Oxygen binding
Buprenorphine//Cytochrome P450 2C9//Steroid hydroxylase activity
Buprenorphine//Cytochrome P450 2C8//Steroid hydroxylase activity
Buprenorphine//Cytochrome P450 3A7//Oxygen binding
Buprenorphine//Cytochrome P450 2D6//Steroid hydroxylase activity
Buprenorphine//Cytochrome P450 2C18//Steroid hydroxylase activity
Buprenorphine//Cytochrome P450 2C19//Steroid hydroxylase activity
Cyclobenzaprine//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Cyclobenzaprine//Cytochrome P450 1A2//Oxidoreductase activity, acting on paired donors, with incorporation or reduction of molecular oxygen, reduced flavin or flavoprotein as one donor, and incorporation of one atom of oxygen
Cyclobenzaprine//Cytochrome P450 2D6//Steroid hydroxylase activity
Cyclobenzaprine//UDP-glucuronosyltransferase 1-4//Protein homodimerization activity
Cyclobenzaprine//UDP-glucuronosyltransferase 2B10//UDPGT is of major importance in the conjugation and subsequent elimination of potentially toxic xenobiotics and endogenous compounds.
Famotidine//Cytochrome P450 1A2//Oxidoreductase activity, acting on paired donors, with incorporation or reduction of molecular oxygen, reduced flavin or flavoprotein as one donor, and incorporation of one atom of oxygen
Azacitidine//Cytidine deaminase//Zinc ion binding
Mesoridazine//Cytochrome P450 2D6//Steroid hydroxylase activity
Maprotiline//Cytochrome P450 2D6//Steroid hydroxylase activity
Maprotiline//Cytochrome P450 1A2//Oxidoreductase activity, acting on paired donors, with incorporation or reduction of molecular oxygen, reduced flavin or flavoprotein as one donor, and incorporation of one atom of oxygen
Acetylsalicylicacid//Cytochrome P450 2C19//Steroid hydroxylase activity
Acetylsalicylicacid//Cytochrome P450 2C9//Steroid hydroxylase activity
Acetylsalicylicacid//UDP-glucuronosyltransferase 1-6//Protein homodimerization activity
Acetylsalicylicacid//Arylamine N-acetyltransferase 2//Arylamine n-acetyltransferase activity
Fulvestrant//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Fulvestrant//UDP-glucuronosyltransferase 1-1//Steroid binding
Felbamate//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Felbamate//Cytochrome P450 2C19//Steroid hydroxylase activity
Felbamate//Cytochrome P450 2E1//Steroid hydroxylase activity
Felbamate//Cytochrome P450 2C9//Steroid hydroxylase activity
Isoniazid//Cytochrome P450 2E1//Steroid hydroxylase activity
Isoniazid//Cytochrome P450 2C9//Steroid hydroxylase activity
Isoniazid//Cytochrome P450 1A2//Oxidoreductase activity, acting on paired donors, with incorporation or reduction of molecular oxygen, reduced flavin or flavoprotein as one donor, and incorporation of one atom of oxygen
Isoniazid//Cytochrome P450 2D6//Steroid hydroxylase activity
Isoniazid//Cytochrome P450 2C19//Steroid hydroxylase activity
Isoniazid//Arylamine N-acetyltransferase 2//Arylamine n-acetyltransferase activity
Isoniazid//Cytochrome P450 2A6//Steroid hydroxylase activity
Isoniazid//Cytochrome P450 2C8//Steroid hydroxylase activity
Naratriptan//Amine oxidase [flavin-containing] A//Serotonin binding
Hydrocodone//Cytochrome P450 2D6//Steroid hydroxylase activity
Hydrocodone//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Hydrocodone//Cytochrome P450 2B6//Steroid hydroxylase activity
Hydrocodone//Cytochrome P450 2C19//Steroid hydroxylase activity
Methylprednisolone//Aldo-keto reductase family 1 member C1//Trans-1,2-dihydrobenzene-1,2-diol dehydrogenase activity
Methylprednisolone//Aldo-keto reductase family 1 member C2//Trans-1,2-dihydrobenzene-1,2-diol dehydrogenase activity
Methylprednisolone//Aldo-keto reductase family 1 member C3//Trans-1,2-dihydrobenzene-1,2-diol dehydrogenase activity
Methylprednisolone//Aldo-keto reductase family 1 member C4//Retinal dehydrogenase activity
Methylprednisolone//Corticosteroid 11-beta-dehydrogenase isozyme 1//11-beta-hydroxysteroid dehydrogenase [nad(p)] activity
Methylprednisolone//Corticosteroid 11-beta-dehydrogenase isozyme 2//Steroid binding
Methylprednisolone//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Methylprednisolone//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Methylprednisolone//Cytochrome P450 3A43//Monooxygenase activity
Methylprednisolone//Cytochrome P450 3A5//Oxygen binding
Methylprednisolone//Cytochrome P450 3A7//Oxygen binding
Methylprednisolone//Cytochrome P450 2A6//Steroid hydroxylase activity
Methylprednisolone//Cytochrome P450 1B1//Oxygen binding
Methylprednisolone//Cytochrome P450 2B6//Steroid hydroxylase activity
Methylprednisolone//Cytochrome P450 2C8//Steroid hydroxylase activity
Methylprednisolone//Cytochrome P450 2C19//Steroid hydroxylase activity
Methylprednisolone//Cytochrome P450 2C9//Steroid hydroxylase activity
Bromfenac//Prostaglandin G/H synthase 2//Prostaglandin-endoperoxide synthase activity
Methyldopa//Catechol O-methyltransferase//O-methyltransferase activity
Alosetron//Cytochrome P450 1A2//Oxidoreductase activity, acting on paired donors, with incorporation or reduction of molecular oxygen, reduced flavin or flavoprotein as one donor, and incorporation of one atom of oxygen
Alosetron//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Alosetron//Cytochrome P450 2C9//Steroid hydroxylase activity
Alosetron//Cytochrome P450 2E1//Steroid hydroxylase activity
Azelastine//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Azelastine//Cytochrome P450 2D6//Steroid hydroxylase activity
Azelastine//Cytochrome P450 1A2//Oxidoreductase activity, acting on paired donors, with incorporation or reduction of molecular oxygen, reduced flavin or flavoprotein as one donor, and incorporation of one atom of oxygen
Azelastine//Cytochrome P450 2C19//Steroid hydroxylase activity
Azelastine//Cytochrome P450 1A1//Vitamin d 24-hydroxylase activity
Azelastine//Cytochrome P450 3A5//Oxygen binding
Azelastine//Cytochrome P450 2C9//Steroid hydroxylase activity
Azelastine//Cytochrome P450 2C8//Steroid hydroxylase activity
Azelastine//Cytochrome P450 2A6//Steroid hydroxylase activity
Azelastine//Cytochrome P450 2E1//Steroid hydroxylase activity
Azelastine//Cytochrome P450 2B6//Steroid hydroxylase activity
Ezetimibe//UDP-glucuronosyltransferase 1-1//Steroid binding
Ezetimibe//UDP-glucuronosyltransferase 1-3//Retinoic acid binding
Ezetimibe//UDP-glucuronosyltransferase 2B15//Glucuronosyltransferase activity
Ezetimibe//UDP-glucuronosyltransferase 2B7//Glucuronosyltransferase activity
Ezetimibe//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Ezetimibe//Cytochrome P450 2C8//Steroid hydroxylase activity
Ethinylestradiol//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Ethinylestradiol//Cytochrome P450 2C8//Steroid hydroxylase activity
Ethinylestradiol//Cytochrome P450 2C9//Steroid hydroxylase activity
Ethinylestradiol//Cytochrome P450 1A2//Oxidoreductase activity, acting on paired donors, with incorporation or reduction of molecular oxygen, reduced flavin or flavoprotein as one donor, and incorporation of one atom of oxygen
Ethinylestradiol//Cytochrome P450 3A5//Oxygen binding
Ethinylestradiol//UDP-glucuronosyltransferase 1-4//Protein homodimerization activity
Ethinylestradiol//UDP-glucuronosyltransferase 1-3//Retinoic acid binding
Ethinylestradiol//UDP-glucuronosyltransferase 1-1//Steroid binding
Ethinylestradiol//UDP-glucuronosyltransferase 1-9//Retinoic acid binding
Ethinylestradiol//UDP-glucuronosyltransferase 2B7//Glucuronosyltransferase activity
Ethinylestradiol//Sulfotransferase 1A3//Sulfotransferase that utilizes 3'-phospho-5'-adenylyl sulfate (PAPS) as sulfonate donor to catalyze the sulfate conjugation of phenolic monoamines (neurotransmitters such as dopamine, norepinephrine and serotonin) and phenolic and catechol drugs.
Ethinylestradiol//Estrogen sulfotransferase//Sulfotransferase activity
Ethinylestradiol//Catechol O-methyltransferase//O-methyltransferase activity
Ethinylestradiol//Cytochrome P450 2C19//Steroid hydroxylase activity
Lomefloxacin//Cytochrome P450 1A2//Oxidoreductase activity, acting on paired donors, with incorporation or reduction of molecular oxygen, reduced flavin or flavoprotein as one donor, and incorporation of one atom of oxygen
Cyclopentolate//Cholinesterase//Identical protein binding
Formoterol//Cytochrome P450 2D6//Steroid hydroxylase activity
Formoterol//Cytochrome P450 2C19//Steroid hydroxylase activity
Formoterol//Cytochrome P450 2C9//Steroid hydroxylase activity
Formoterol//Cytochrome P450 2A6//Steroid hydroxylase activity
Formoterol//UDP-glucuronosyltransferase 1-8//Steroid binding
Formoterol//UDP-glucuronosyltransferase 1-9//Retinoic acid binding
Formoterol//UDP-glucuronosyltransferase 2B7//Glucuronosyltransferase activity
Formoterol//UDP-glucuronosyltransferase 2B15//Glucuronosyltransferase activity
Cytarabine//Cytidine deaminase//Zinc ion binding
Cytarabine//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Cytarabine//Deoxycytidine kinase//Protein homodimerization activity
Cytarabine//Deoxycytidylate deaminase//Zinc ion binding
Dopamine//Amine oxidase [flavin-containing] A//Serotonin binding
Dopamine//Amine oxidase [flavin-containing] B//Primary amine oxidase activity
Dopamine//Catechol O-methyltransferase//O-methyltransferase activity
Dopamine//Dopamine beta-hydroxylase//L-ascorbic acid binding
Exemestane//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Exemestane//Aromatase//Oxygen binding
Azathioprine//Hypoxanthine-guanine phosphoribosyltransferase//Protein homodimerization activity
Azathioprine//Xanthine dehydrogenase/oxidase//Xanthine oxidase activity
Azathioprine//Thiopurine S-methyltransferase//Thiopurine s-methyltransferase activity
Azathioprine//Glutathione S-transferase A1//Glutathione transferase activity
Azathioprine//Glutathione S-transferase A2//Glutathione transferase activity
Azathioprine//Glutathione S-transferase Mu 1//Protein homodimerization activity
Azathioprine//Inosine-5'-monophosphate dehydrogenase 1//Rna binding
Azathioprine//Inosine-5'-monophosphate dehydrogenase 2//Rna binding
Azathioprine//GMP synthase [glutamine-hydrolyzing]//Pyrophosphatase activity
Azathioprine//Cytochrome P450 1A2//Oxidoreductase activity, acting on paired donors, with incorporation or reduction of molecular oxygen, reduced flavin or flavoprotein as one donor, and incorporation of one atom of oxygen
Doxorubicin//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Doxorubicin//Cytochrome P450 2D6//Steroid hydroxylase activity
Doxorubicin//Cytochrome P450 2B6//Steroid hydroxylase activity
Doxorubicin//Cytochrome P450 1B1//Oxygen binding
Doxorubicin//Carbonyl reductase [NADPH] 1//Prostaglandin-e2 9-reductase activity
Doxorubicin//Carbonyl reductase [NADPH] 3//Nadph binding
Doxorubicin//Aldo-keto reductase family 1 member C3//Trans-1,2-dihydrobenzene-1,2-diol dehydrogenase activity
Doxorubicin//NAD(P)H dehydrogenase [quinone] 1//Superoxide dismutase activity
Doxorubicin//Xanthine dehydrogenase/oxidase//Xanthine oxidase activity
Doxorubicin//Nitric oxide synthase, brain//Tetrahydrobiopterin binding
Doxorubicin//Nitric oxide synthase, inducible//Tetrahydrobiopterin binding
Doxorubicin//Nitric oxide synthase, endothelial//Tetrahydrobiopterin binding
Doxorubicin//NADH dehydrogenase [ubiquinone] iron-sulfur protein 2, mitochondrial//Ubiquitin protein ligase binding
Doxorubicin//NADPH--cytochrome P450 reductase//Oxidoreductase activity, acting on paired donors, with incorporation or reduction of molecular oxygen, nad(p)h as one donor, and incorporation of one atom of oxygen
Frovatriptan//Cytochrome P450 1A2//Oxidoreductase activity, acting on paired donors, with incorporation or reduction of molecular oxygen, reduced flavin or flavoprotein as one donor, and incorporation of one atom of oxygen
Levobupivacaine//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Levobupivacaine//Cytochrome P450 1A2//Oxidoreductase activity, acting on paired donors, with incorporation or reduction of molecular oxygen, reduced flavin or flavoprotein as one donor, and incorporation of one atom of oxygen
Hydroxyurea//Cytochrome P450 2D6//Steroid hydroxylase activity
Letrozole//Aromatase//Oxygen binding
Letrozole//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Letrozole//Cytochrome P450 2A6//Steroid hydroxylase activity
Letrozole//Cytochrome P450 2C19//Steroid hydroxylase activity
Letrozole//UDP-glucuronosyltransferase 2B7//Glucuronosyltransferase activity
Ketoprofen//Cytochrome P450 2C9//Steroid hydroxylase activity
Ketoprofen//Cytochrome P450 2C8//Steroid hydroxylase activity
Ketoprofen//UDP-glucuronosyltransferase 1-1//Steroid binding
Metyrapone//Cytochrome P450 11B2, mitochondrial//Steroid 11-beta-monooxygenase activity
Metyrapone//Cytochrome P450 2A6//Steroid hydroxylase activity
Metyrapone//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Metyrapone//Cytochrome P450 11B1, mitochondrial//Steroid 11-beta-monooxygenase activity
Metyrapone//Cytochrome P450 2E1//Steroid hydroxylase activity
Cinacalcet//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Cinacalcet//Cytochrome P450 2D6//Steroid hydroxylase activity
Cinacalcet//Cytochrome P450 1A2//Oxidoreductase activity, acting on paired donors, with incorporation or reduction of molecular oxygen, reduced flavin or flavoprotein as one donor, and incorporation of one atom of oxygen
Clobetasolpropionate//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Clobetasolpropionate//Cytochrome P450 3A5//Oxygen binding
Glyburide//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Glyburide//Cytochrome P450 2C9//Steroid hydroxylase activity
Glyburide//Cytochrome P450 2C19//Steroid hydroxylase activity
Glyburide//Cytochrome P450 3A7//Oxygen binding
Glyburide//Cytochrome P450 3A5//Oxygen binding
Guanfacine//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Guanfacine//Cytochrome P450 2C19//Steroid hydroxylase activity
Isosorbidemononitrate//Glutathione S-transferase Mu 1//Protein homodimerization activity
Isosorbidemononitrate//Xanthine dehydrogenase/oxidase//Xanthine oxidase activity
Isosorbidemononitrate//Alcohol dehydrogenase class-3//Zinc ion binding
Felodipine//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Felodipine//Cytochrome P450 3A5//Oxygen binding
Felodipine//Cytochrome P450 3A7//Oxygen binding
Felodipine//Cytochrome P450 2C8//Steroid hydroxylase activity
Felodipine//Cytochrome P450 2C9//Steroid hydroxylase activity
Felodipine//Cytochrome P450 2D6//Steroid hydroxylase activity
Mycophenolicacid//UDP-glucuronosyltransferase 1-1//Steroid binding
Mycophenolicacid//UDP-glucuronosyltransferase 1-9//Retinoic acid binding
Mycophenolicacid//UDP-glucuronosyltransferase 2B7//Glucuronosyltransferase activity
Mycophenolicacid//UDP-glucuronosyltransferase 1-7//Retinoic acid binding
Mycophenolicacid//UDP-glucuronosyltransferase 1-6//Protein homodimerization activity
Ketoconazole//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Ketoconazole//Cytochrome P450 3A5//Oxygen binding
Ketoconazole//Cytochrome P450 2C19//Steroid hydroxylase activity
Ketoconazole//Cytochrome P450 1A1//Vitamin d 24-hydroxylase activity
Ketoconazole//Cytochrome P450 1A2//Oxidoreductase activity, acting on paired donors, with incorporation or reduction of molecular oxygen, reduced flavin or flavoprotein as one donor, and incorporation of one atom of oxygen
Ketoconazole//Cytochrome P450 2A6//Steroid hydroxylase activity
Ketoconazole//Cytochrome P450 1B1//Oxygen binding
Ketoconazole//Cytochrome P450 2B6//Steroid hydroxylase activity
Ketoconazole//Cytochrome P450 2C8//Steroid hydroxylase activity
Ketoconazole//Cytochrome P450 2C9//Steroid hydroxylase activity
Ketoconazole//Cytochrome P450 2D6//Steroid hydroxylase activity
Ketoconazole//Cytochrome P450 11B1, mitochondrial//Steroid 11-beta-monooxygenase activity
Ketoconazole//UDP-glucuronosyltransferase 1-1//Steroid binding
Ketoconazole//UDP-glucuronosyltransferase 1-7//Retinoic acid binding
Ketoconazole//UDP-glucuronosyltransferase 2B7//Glucuronosyltransferase activity
Ketoconazole//Cytochrome P450 4F12//Leukotriene-b4 20-monooxygenase activity
Ketoconazole//Aromatase//Oxygen binding
Methoxyflurane//Cytochrome P450 2E1//Steroid hydroxylase activity
Methoxyflurane//Cytochrome P450 1A2//Oxidoreductase activity, acting on paired donors, with incorporation or reduction of molecular oxygen, reduced flavin or flavoprotein as one donor, and incorporation of one atom of oxygen
Methoxyflurane//Cytochrome P450 2A6//Steroid hydroxylase activity
Methoxyflurane//Cytochrome P450 2B6//Steroid hydroxylase activity
Methoxyflurane//Cytochrome P450 2C9//Steroid hydroxylase activity
Methoxyflurane//Cytochrome P450 2D6//Steroid hydroxylase activity
Methoxyflurane//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Irbesartan//Cytochrome P450 2C8//Steroid hydroxylase activity
Irbesartan//Cytochrome P450 2C9//Steroid hydroxylase activity
Irbesartan//UDP-glucuronosyltransferase 1-3//Retinoic acid binding
Irbesartan//Prostaglandin G/H synthase 1//Prostaglandin-endoperoxide synthase activity
Irbesartan//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Mercaptopurine//Thiopurine S-methyltransferase//Thiopurine s-methyltransferase activity
Mercaptopurine//Xanthine dehydrogenase/oxidase//Xanthine oxidase activity
Mercaptopurine//Aldehyde oxidase//Xanthine dehydrogenase activity
Fenofibrate//UDP-glucuronosyltransferase 1-9//Retinoic acid binding
Fenofibrate//Liver carboxylesterase 1//Triglyceride lipase activity
Fenofibrate//Carbonyl reductase [NADPH] 1//Prostaglandin-e2 9-reductase activity
Fenofibrate//Cytochrome P450 2C8//Steroid hydroxylase activity
Fenofibrate//Cytochrome P450 2C19//Steroid hydroxylase activity
Fenofibrate//Cytochrome P450 2A6//Steroid hydroxylase activity
Fenofibrate//Aldo-keto reductase family 1 member C1//Trans-1,2-dihydrobenzene-1,2-diol dehydrogenase activity
Fenofibrate//Aldo-keto reductase family 1 member C2//Trans-1,2-dihydrobenzene-1,2-diol dehydrogenase activity
Fenofibrate//Aldo-keto reductase family 1 member C3//Trans-1,2-dihydrobenzene-1,2-diol dehydrogenase activity
Fenofibrate//Cytochrome P450 2C9//Steroid hydroxylase activity
Memantine//Cytochrome P450 2B6//Steroid hydroxylase activity
Memantine//Cytochrome P450 2A6//Steroid hydroxylase activity
Memantine//Cytochrome P450 2C19//Steroid hydroxylase activity
Lubiprostone//Carbonyl reductase [NADPH] 1//Prostaglandin-e2 9-reductase activity
Ibuprofen//Cytochrome P450 2C9//Steroid hydroxylase activity
Ibuprofen//Cytochrome P450 2C8//Steroid hydroxylase activity
Ibuprofen//Cytochrome P450 2C19//Steroid hydroxylase activity
Ibuprofen//UDP-glucuronosyltransferase 1-3//Retinoic acid binding
Ibuprofen//UDP-glucuronosyltransferase 1-9//Retinoic acid binding
Ibuprofen//UDP-glucuronosyltransferase 2B4//Glucuronosyltransferase activity
Ibuprofen//UDP-glucuronosyltransferase 2B7//Glucuronosyltransferase activity
Ibuprofen//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Isoprenaline//Cytochrome P450 1A1//Vitamin d 24-hydroxylase activity
Melatonin//Cytochrome P450 1A1//Vitamin d 24-hydroxylase activity
Melatonin//Cytochrome P450 1A2//Oxidoreductase activity, acting on paired donors, with incorporation or reduction of molecular oxygen, reduced flavin or flavoprotein as one donor, and incorporation of one atom of oxygen
Melatonin//Cytochrome P450 1B1//Oxygen binding
Melatonin//Cytochrome P450 2C19//Steroid hydroxylase activity
Melatonin//Cytochrome P450 2C9//Steroid hydroxylase activity
Melatonin//Acetylserotonin O-methyltransferase//Protein homodimerization activity
Melatonin//Indoleamine 2,3-dioxygenase 1//Tryptophan 2,3-dioxygenase activity
Melatonin//Myeloperoxidase//Peroxidase activity
Melatonin//Aromatase//Oxygen binding
Glipizide//Cytochrome P450 2C9//Steroid hydroxylase activity
Glipizide//UDP-glucuronosyltransferase 1-1//Steroid binding
Clonazepam//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Clonazepam//Cytochrome P450 2E1//Steroid hydroxylase activity
Clonazepam//Arylamine N-acetyltransferase 2//Arylamine n-acetyltransferase activity
Mequitazine//Cytochrome P450 2D6//Steroid hydroxylase activity
Mequitazine//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Diphenhydramine//Cytochrome P450 2D6//Steroid hydroxylase activity
Diphenhydramine//Cytochrome P450 2C9//Steroid hydroxylase activity
Diphenhydramine//Cytochrome P450 2C19//Steroid hydroxylase activity
Diphenhydramine//Prostaglandin G/H synthase 1//Prostaglandin-endoperoxide synthase activity
Atorvastatin//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Atorvastatin//Cytochrome P450 3A5//Oxygen binding
Atorvastatin//Cytochrome P450 3A7//Oxygen binding
Atorvastatin//Cytochrome P450 2C8//Steroid hydroxylase activity
Atorvastatin//Cytochrome P450 2D6//Steroid hydroxylase activity
Atorvastatin//Cytochrome P450 2C9//Steroid hydroxylase activity
Atorvastatin//Cytochrome P450 2C19//Steroid hydroxylase activity
Atorvastatin//Cytochrome P450 2B6//Steroid hydroxylase activity
Atorvastatin//UDP-glucuronosyltransferase 1-1//Steroid binding
Atorvastatin//UDP-glucuronosyltransferase 1-3//Retinoic acid binding
Benzocaine//Liver carboxylesterase 1//Triglyceride lipase activity
Hesperetin//Cytochrome P450 1A2//Oxidoreductase activity, acting on paired donors, with incorporation or reduction of molecular oxygen, reduced flavin or flavoprotein as one donor, and incorporation of one atom of oxygen
Fluvastatin//Cytochrome P450 1A1//Vitamin d 24-hydroxylase activity
Fluvastatin//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Fluvastatin//Cytochrome P450 3A5//Oxygen binding
Fluvastatin//Cytochrome P450 2C8//Steroid hydroxylase activity
Fluvastatin//Cytochrome P450 2C9//Steroid hydroxylase activity
Fluvastatin//Cytochrome P450 2C19//Steroid hydroxylase activity
Fluvastatin//Cytochrome P450 2D6//Steroid hydroxylase activity
Fluvastatin//UDP-glucuronosyltransferase 1-1//Steroid binding
Fluvastatin//UDP-glucuronosyltransferase 1-3//Retinoic acid binding
Fluvastatin//UDP-glucuronosyltransferase 2B7//Glucuronosyltransferase activity
Fluvastatin//Cytochrome P450 2B6//Steroid hydroxylase activity
Leflunomide//Cytochrome P450 2C9//Steroid hydroxylase activity
Leflunomide//Cytochrome P450 1A2//Oxidoreductase activity, acting on paired donors, with incorporation or reduction of molecular oxygen, reduced flavin or flavoprotein as one donor, and incorporation of one atom of oxygen
Capecitabine//Thymidine phosphorylase//Transferase activity, transferring pentosyl groups
Capecitabine//Liver carboxylesterase 1//Triglyceride lipase activity
Capecitabine//Dihydropyrimidine dehydrogenase [NADP(+)]//Protein homodimerization activity
Capecitabine//Cytidine deaminase//Zinc ion binding
Capecitabine//Cytochrome P450 2C9//Steroid hydroxylase activity
Miconazole//Cytochrome P450 2C9//Steroid hydroxylase activity
Miconazole//Cytochrome P450 2C19//Steroid hydroxylase activity
Miconazole//Cytochrome P450 2A6//Steroid hydroxylase activity
Miconazole//Cytochrome P450 2E1//Steroid hydroxylase activity
Miconazole//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Miconazole//Cytochrome P450 2B6//Steroid hydroxylase activity
Miconazole//Cytochrome P450 2D6//Steroid hydroxylase activity
Miconazole//Cytochrome P450 2C8//Steroid hydroxylase activity
Miconazole//Cytochrome P450 11B1, mitochondrial//Steroid 11-beta-monooxygenase activity
Miconazole//Lanosterol 14-alpha demethylase//Sterol 14-demethylase activity
Miconazole//Aromatase//Oxygen binding
Chlorphenamine//Cytochrome P450 3A7//Oxygen binding
Chlorphenamine//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Chlorphenamine//Cytochrome P450 2D6//Steroid hydroxylase activity
Chlorphenamine//Cytochrome P450 3A5//Oxygen binding
Atovaquone//Cytochrome P450 2C9//Steroid hydroxylase activity
Atovaquone//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Amiodarone//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Amiodarone//Cytochrome P450 2C8//Steroid hydroxylase activity
Amiodarone//Cytochrome P450 2D6//Steroid hydroxylase activity
Amiodarone//Cytochrome P450 2C9//Steroid hydroxylase activity
Amiodarone//Cytochrome P450 1A2//Oxidoreductase activity, acting on paired donors, with incorporation or reduction of molecular oxygen, reduced flavin or flavoprotein as one donor, and incorporation of one atom of oxygen
Amiodarone//Cytochrome P450 2C19//Steroid hydroxylase activity
Amiodarone//Cytochrome P450 1A1//Vitamin d 24-hydroxylase activity
Amiodarone//Cytochrome P450 2A6//Steroid hydroxylase activity
Amiodarone//Cytochrome P450 2J2//Steroid hydroxylase activity
Diazoxide//Glutamine synthetase//Manganese ion binding
Gliclazide//Cytochrome P450 2C9//Steroid hydroxylase activity
Gliclazide//Cytochrome P450 2C19//Steroid hydroxylase activity
Ambenonium//Cholinesterase//Identical protein binding
Dutasteride//Cytochrome P450 3A5//Oxygen binding
Econazole//Aromatase//Oxygen binding
Econazole//Cytochrome P450 2E1//Steroid hydroxylase activity
Econazole//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Bicalutamide//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Bicalutamide//Cytochrome P450 2C19//Steroid hydroxylase activity
Bicalutamide//Cytochrome P450 2C9//Steroid hydroxylase activity
Bicalutamide//Cytochrome P450 2D6//Steroid hydroxylase activity
Doxacuriumchloride//Cholinesterase//Identical protein binding
Carvedilol//Xanthine dehydrogenase/oxidase//Xanthine oxidase activity
Carvedilol//Cytochrome P450 2C9//Steroid hydroxylase activity
Carvedilol//Cytochrome P450 2D6//Steroid hydroxylase activity
Carvedilol//Cytochrome P450 1A2//Oxidoreductase activity, acting on paired donors, with incorporation or reduction of molecular oxygen, reduced flavin or flavoprotein as one donor, and incorporation of one atom of oxygen
Carvedilol//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Carvedilol//Cytochrome P450 1A1//Vitamin d 24-hydroxylase activity
Carvedilol//Cytochrome P450 2E1//Steroid hydroxylase activity
Carvedilol//UDP-glucuronosyltransferase 1-1//Steroid binding
Carvedilol//UDP-glucuronosyltransferase 2B4//Glucuronosyltransferase activity
Carvedilol//UDP-glucuronosyltransferase 2B7//Glucuronosyltransferase activity
Levofloxacin//Cytochrome P450 1A2//Oxidoreductase activity, acting on paired donors, with incorporation or reduction of molecular oxygen, reduced flavin or flavoprotein as one donor, and incorporation of one atom of oxygen
Levofloxacin//Cytochrome P450 2C9//Steroid hydroxylase activity
Doxepin//Cytochrome P450 2D6//Steroid hydroxylase activity
Doxepin//Cytochrome P450 2C19//Steroid hydroxylase activity
Doxepin//Cytochrome P450 2C9//Steroid hydroxylase activity
Doxepin//Cytochrome P450 1A2//Oxidoreductase activity, acting on paired donors, with incorporation or reduction of molecular oxygen, reduced flavin or flavoprotein as one donor, and incorporation of one atom of oxygen
Doxepin//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Amifostine//Alkaline phosphatase, tissue-nonspecific isozyme//Pyrophosphatase activity
Nefazodone//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Nefazodone//CYP2B protein//Oxidoreductase activity, acting on paired donors, with incorporation or reduction of molecular oxygen, reduced flavin or flavoprotein as one donor, and incorporation of one atom of oxygen
Nefazodone//Cytochrome P450 2D6//Steroid hydroxylase activity
Nefazodone//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Nefazodone//Cytochrome P450 3A43//Monooxygenase activity
Nefazodone//Cytochrome P450 3A5//Oxygen binding
Nefazodone//Cytochrome P450 3A7//Oxygen binding
Desipramine//Cytochrome P450 2D6//Steroid hydroxylase activity
Desipramine//Cytochrome P450 1A2//Oxidoreductase activity, acting on paired donors, with incorporation or reduction of molecular oxygen, reduced flavin or flavoprotein as one donor, and incorporation of one atom of oxygen
Desipramine//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Desipramine//Cytochrome P450 2B6//Steroid hydroxylase activity
Desipramine//Cytochrome P450 2E1//Steroid hydroxylase activity
Bupropion//Cytochrome P450 2B6//Steroid hydroxylase activity
Bupropion//Cytochrome P450 2D6//Steroid hydroxylase activity
Bupropion//Cytochrome P450 2C9//Steroid hydroxylase activity
Bupropion//Cytochrome P450 2E1//Steroid hydroxylase activity
Halothane//Cytochrome P450 2E1//Steroid hydroxylase activity
Halothane//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Halothane//Cytochrome P450 2A6//Steroid hydroxylase activity
Halothane//Cytochrome P450 2B6//Steroid hydroxylase activity
Halothane//Cytochrome P450 2C9//Steroid hydroxylase activity
Chloroprocaine//Cholinesterase//Identical protein binding
Cilostazol//Cytochrome P450 3A5//Oxygen binding
Cilostazol//Cytochrome P450 3A7//Oxygen binding
Cilostazol//Cytochrome P450 2C19//Steroid hydroxylase activity
Cilostazol//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Cilostazol//Cytochrome P450 1A2//Oxidoreductase activity, acting on paired donors, with incorporation or reduction of molecular oxygen, reduced flavin or flavoprotein as one donor, and incorporation of one atom of oxygen
Cilostazol//Cytochrome P450 2D6//Steroid hydroxylase activity
Itraconazole//Cytochrome P450 3A5//Oxygen binding
Itraconazole//Cytochrome P450 3A7//Oxygen binding
Itraconazole//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Itraconazole//Cytochrome P450 2B6//Steroid hydroxylase activity
Itraconazole//Cytochrome P450 1A1//Vitamin d 24-hydroxylase activity
Itraconazole//Cytochrome P450 2E1//Steroid hydroxylase activity
Arsenictrioxide//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Moclobemide//Amine oxidase [flavin-containing] A//Serotonin binding
Moclobemide//Amine oxidase [flavin-containing] B//Primary amine oxidase activity
Moclobemide//Cytochrome P450 2C19//Steroid hydroxylase activity
Moclobemide//Cytochrome P450 2D6//Steroid hydroxylase activity
Moclobemide//Cytochrome P450 2C9//Steroid hydroxylase activity
Escitalopram//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Escitalopram//Cytochrome P450 2D6//Steroid hydroxylase activity
Escitalopram//Cytochrome P450 2C19//Steroid hydroxylase activity
Escitalopram//Amine oxidase [flavin-containing] A//Serotonin binding
Escitalopram//Amine oxidase [flavin-containing] B//Primary amine oxidase activity
Cyclizine//Cytochrome P450 2C9//Steroid hydroxylase activity
Idarubicin//Cytochrome P450 2C9//Steroid hydroxylase activity
Idarubicin//Cytochrome P450 2D6//Steroid hydroxylase activity
Ifosfamide//Cytochrome P450 2B6//Steroid hydroxylase activity
Ifosfamide//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Ifosfamide//Cytochrome P450 3A5//Oxygen binding
Ifosfamide//Cytochrome P450 2C19//Steroid hydroxylase activity
Ifosfamide//Cytochrome P450 2C9//Steroid hydroxylase activity
Ifosfamide//Cytochrome P450 2C8//Steroid hydroxylase activity
Ifosfamide//Cytochrome P450 2A6//Steroid hydroxylase activity
Ifosfamide//Cytochrome P450 2C18//Steroid hydroxylase activity
Ifosfamide//Prostaglandin G/H synthase 1//Prostaglandin-endoperoxide synthase activity
Naloxone//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Naloxone//UDP-glucuronosyltransferase 1-1//Steroid binding
Domperidone//Cytochrome P450 3A5//Oxygen binding
Domperidone//Cytochrome P450 3A7//Oxygen binding
Domperidone//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Domperidone//Cytochrome P450 1A2//Oxidoreductase activity, acting on paired donors, with incorporation or reduction of molecular oxygen, reduced flavin or flavoprotein as one donor, and incorporation of one atom of oxygen
Domperidone//Cytochrome P450 2B6//Steroid hydroxylase activity
Domperidone//Cytochrome P450 2C8//Steroid hydroxylase activity
Domperidone//Cytochrome P450 2D6//Steroid hydroxylase activity
Dexfenfluramine//Cytochrome P450 2D6//Steroid hydroxylase activity
Dexfenfluramine//Cytochrome P450 1A2//Oxidoreductase activity, acting on paired donors, with incorporation or reduction of molecular oxygen, reduced flavin or flavoprotein as one donor, and incorporation of one atom of oxygen
Dexfenfluramine//Cytochrome P450 2E1//Steroid hydroxylase activity
Acebutolol//Cytochrome P450 2D6//Steroid hydroxylase activity
Brinzolamide//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Flecainide//Cytochrome P450 2D6//Steroid hydroxylase activity
Flecainide//Cytochrome P450 1A2//Oxidoreductase activity, acting on paired donors, with incorporation or reduction of molecular oxygen, reduced flavin or flavoprotein as one donor, and incorporation of one atom of oxygen
Flecainide//Cytochrome P450 2C9//Steroid hydroxylase activity
Estramustine//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Bromocriptine//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Mitoxantrone//Cytochrome P450 2E1//Steroid hydroxylase activity
Mitoxantrone//Cytochrome P450 1B1//Oxygen binding
Mitoxantrone//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Lomustine//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Lomustine//Cytochrome P450 2D6//Steroid hydroxylase activity
Clarithromycin//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Clarithromycin//Cytochrome P450 3A5//Oxygen binding
Ceftriaxone//Glutamine synthetase//Manganese ion binding
Fomepizole//Cytochrome P450 2E1//Steroid hydroxylase activity
Fomepizole//Cytochrome P450 2A6//Steroid hydroxylase activity
Estazolam//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Finasteride//Cytochrome P450 3A5//Oxygen binding
Finasteride//Cytochrome P450 3A7//Oxygen binding
Finasteride//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Anastrozole//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Anastrozole//Cytochrome P450 3A5//Oxygen binding
Anastrozole//Cytochrome P450 2C8//Steroid hydroxylase activity
Anastrozole//UDP-glucuronosyltransferase 1-4//Protein homodimerization activity
Anastrozole//UDP-glucuronosyltransferase 1-3//Retinoic acid binding
Anastrozole//UDP-glucuronosyltransferase 2B7//Glucuronosyltransferase activity
Anastrozole//Cytochrome P450 1A2//Oxidoreductase activity, acting on paired donors, with incorporation or reduction of molecular oxygen, reduced flavin or flavoprotein as one donor, and incorporation of one atom of oxygen
Anastrozole//Cytochrome P450 2C9//Steroid hydroxylase activity
Halofantrine//Cytochrome P450 2D6//Steroid hydroxylase activity
Halofantrine//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Halofantrine//Cytochrome P450 3A5//Oxygen binding
Halofantrine//Cytochrome P450 2C8//Steroid hydroxylase activity
Ketamine//Cytochrome P450 2C9//Steroid hydroxylase activity
Ketamine//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Ketamine//Cytochrome P450 2B6//Steroid hydroxylase activity
Ketamine//Prostaglandin G/H synthase 1//Prostaglandin-endoperoxide synthase activity
Ketamine//Cytochrome P450 2C8//Steroid hydroxylase activity
Budesonide//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Budesonide//Cytochrome P450 3A5//Oxygen binding
Budesonide//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Budesonide//Cytochrome P450 3A43//Monooxygenase activity
Budesonide//Cytochrome P450 3A5//Oxygen binding
Budesonide//Cytochrome P450 3A7//Oxygen binding
Budesonide//Cytochrome P450 2A6//Steroid hydroxylase activity
Budesonide//Cytochrome P450 1B1//Oxygen binding
Budesonide//Cytochrome P450 2B6//Steroid hydroxylase activity
Budesonide//Cytochrome P450 2C8//Steroid hydroxylase activity
Budesonide//Cytochrome P450 2C9//Steroid hydroxylase activity
Budesonide//Cytochrome P450 2C19//Steroid hydroxylase activity
Aminophylline//Cytochrome P450 1A2//Oxidoreductase activity, acting on paired donors, with incorporation or reduction of molecular oxygen, reduced flavin or flavoprotein as one donor, and incorporation of one atom of oxygen
Aminophylline//Cytochrome P450 2E1//Steroid hydroxylase activity
Aminophylline//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Levomethadylacetate//Cytochrome P450 3A5//Oxygen binding
Levomethadylacetate//Cytochrome P450 3A7//Oxygen binding
Levomethadylacetate//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Encainide//Cytochrome P450 2D6//Steroid hydroxylase activity
Metoclopramide//Cytochrome P450 2D6//Steroid hydroxylase activity
Metoclopramide//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Metoclopramide//Cytochrome P450 1A2//Oxidoreductase activity, acting on paired donors, with incorporation or reduction of molecular oxygen, reduced flavin or flavoprotein as one donor, and incorporation of one atom of oxygen
Dexamethasone//Corticosteroid 11-beta-dehydrogenase isozyme 2//Steroid binding
Dexamethasone//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Dexamethasone//Corticosteroid 11-beta-dehydrogenase isozyme 1//11-beta-hydroxysteroid dehydrogenase [nad(p)] activity
Dexamethasone//Cytochrome P450 3A5//Oxygen binding
Dexamethasone//Cytochrome P450 3A7//Oxygen binding
Dexamethasone//Steroid 17-alpha-hydroxylase/17,20 lyase//Steroid 17-alpha-monooxygenase activity
Dexamethasone//Cytochrome P450 1A1//Vitamin d 24-hydroxylase activity
Dexamethasone//Cytochrome P450 2A6//Steroid hydroxylase activity
Dexamethasone//Cytochrome P450 2B6//Steroid hydroxylase activity
Dexamethasone//Cytochrome P450 2C19//Steroid hydroxylase activity
Dexamethasone//Cytochrome P450 2C8//Steroid hydroxylase activity
Dexamethasone//Cytochrome P450 2E1//Steroid hydroxylase activity
Dexamethasone//Cytochrome P450 3A43//Monooxygenase activity
Dexamethasone//Cytochrome P450 4A11//Leukotriene-b4 20-monooxygenase activity
Dexamethasone//Cytochrome P450 11B1, mitochondrial//Steroid 11-beta-monooxygenase activity
Levodopa//Aromatic-L-amino-acid decarboxylase//Pyridoxal phosphate binding
Aripiprazole//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Aripiprazole//Cytochrome P450 3A7//Oxygen binding
Aripiprazole//Cytochrome P450 3A5//Oxygen binding
Aripiprazole//Cytochrome P450 2D6//Steroid hydroxylase activity
Gemfibrozil//Cytochrome P450 2C8//Steroid hydroxylase activity
Gemfibrozil//Cytochrome P450 2C19//Steroid hydroxylase activity
Gemfibrozil//Cytochrome P450 2C9//Steroid hydroxylase activity
Gemfibrozil//Cytochrome P450 1A2//Oxidoreductase activity, acting on paired donors, with incorporation or reduction of molecular oxygen, reduced flavin or flavoprotein as one donor, and incorporation of one atom of oxygen
Gemfibrozil//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Gemfibrozil//UDP-glucuronosyltransferase 2B7//Glucuronosyltransferase activity
Gemfibrozil//UDP-glucuronosyltransferase 1-1//Steroid binding
Gemfibrozil//UDP-glucuronosyltransferase 1-3//Retinoic acid binding
Gemfibrozil//UDP-glucuronosyltransferase 1-9//Retinoic acid binding
Gemfibrozil//UDP-glucuronosyltransferase 2B4//Glucuronosyltransferase activity
Gemfibrozil//UDP-glucuronosyltransferase 2B17//Glucuronosyltransferase activity
Clomipramine//Cytochrome P450 2D6//Steroid hydroxylase activity
Clomipramine//Cytochrome P450 2C19//Steroid hydroxylase activity
Clomipramine//Cytochrome P450 1A2//Oxidoreductase activity, acting on paired donors, with incorporation or reduction of molecular oxygen, reduced flavin or flavoprotein as one donor, and incorporation of one atom of oxygen
Clomipramine//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Bepridil//Cytochrome P450 2D6//Steroid hydroxylase activity
Bepridil//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Decamethonium//Cholinesterase//Identical protein binding
Docetaxel//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Docetaxel//Cytochrome P450 3A5//Oxygen binding
Docetaxel//Cytochrome P450 3A7//Oxygen binding
Docetaxel//Cytochrome P450 1B1//Oxygen binding
Mitiglinide//UDP-glucuronosyltransferase 1-3//Retinoic acid binding
Mitiglinide//UDP-glucuronosyltransferase 2B7//Glucuronosyltransferase activity
Ergonovine//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Dasatinib//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Dasatinib//Cytochrome P450 1A1//Vitamin d 24-hydroxylase activity
Dasatinib//Cytochrome P450 1A2//Oxidoreductase activity, acting on paired donors, with incorporation or reduction of molecular oxygen, reduced flavin or flavoprotein as one donor, and incorporation of one atom of oxygen
Dasatinib//Cytochrome P450 1B1//Oxygen binding
Dasatinib//Cytochrome P450 3A5//Oxygen binding
Dasatinib//Dimethylaniline monooxygenase [N-oxide-forming] 3//Trimethylamine monooxygenase activity
Lapatinib//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Lapatinib//Cytochrome P450 3A5//Oxygen binding
Lapatinib//Cytochrome P450 2C8//Steroid hydroxylase activity
Lapatinib//Cytochrome P450 2C19//Steroid hydroxylase activity
Decitabine//Deoxycytidine kinase//Protein homodimerization activity
Arformoterol//Cytochrome P450 2D6//Steroid hydroxylase activity
Arformoterol//Cytochrome P450 2C19//Steroid hydroxylase activity
Arformoterol//Cytochrome P450 2A6//Steroid hydroxylase activity
Arformoterol//Cytochrome P450 2C9//Steroid hydroxylase activity
Hydralazine//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Nelarabine//Adenosine deaminase//Zinc ion binding
Nelarabine//Deoxycytidine kinase//Protein homodimerization activity
Lumiracoxib//Cytochrome P450 2C9//Steroid hydroxylase activity
Lumiracoxib//Cytochrome P450 2C19//Steroid hydroxylase activity
Lumiracoxib//UDP-glucuronosyltransferase 1-9//Retinoic acid binding
Lumiracoxib//Cytochrome P450 1A2//Oxidoreductase activity, acting on paired donors, with incorporation or reduction of molecular oxygen, reduced flavin or flavoprotein as one donor, and incorporation of one atom of oxygen
Fosphenytoin//Cytochrome P450 2C9//Steroid hydroxylase activity
Fosphenytoin//Cytochrome P450 2C19//Steroid hydroxylase activity
Fosphenytoin//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Fosphenytoin//Cytochrome P450 2B6//Steroid hydroxylase activity
Fosphenytoin//Cytochrome P450 1A2//Oxidoreductase activity, acting on paired donors, with incorporation or reduction of molecular oxygen, reduced flavin or flavoprotein as one donor, and incorporation of one atom of oxygen
Fosphenytoin//UDP-glucuronosyltransferase 1-6//Protein homodimerization activity
Fosphenytoin//UDP-glucuronosyltransferase 1-9//Retinoic acid binding
Cefazolin//Thiopurine S-methyltransferase//Thiopurine s-methyltransferase activity
Hexobarbital//Cytochrome P450 2C19//Steroid hydroxylase activity
Hexobarbital//Cytochrome P450 2C9//Steroid hydroxylase activity
Hexobarbital//Prostaglandin G/H synthase 1//Prostaglandin-endoperoxide synthase activity
Mestranol//Cytochrome P450 2C9//Steroid hydroxylase activity
Mestranol//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Mestranol//Cytochrome P450 2C8//Steroid hydroxylase activity
Ephedrine//Cholinesterase//Identical protein binding
Ephedrine//Acetylcholinesterase//Serine hydrolase activity
Cortisoneacetate//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Cortisoneacetate//Cytochrome P450 3A5//Oxygen binding
Bezafibrate//Cytochrome P450 1A1//Vitamin d 24-hydroxylase activity
Bezafibrate//Cytochrome P450 2C8//Steroid hydroxylase activity
Bezafibrate//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Colchicine//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Colchicine//Cytochrome P450 2B6//Steroid hydroxylase activity
Colchicine//Cytochrome P450 2C8//Steroid hydroxylase activity
Colchicine//Cytochrome P450 2E1//Steroid hydroxylase activity
Drospirenone//Prostaglandin G/H synthase 2//Prostaglandin-endoperoxide synthase activity
Drospirenone//Serum paraoxonase/arylesterase 1//Protein homodimerization activity
Drospirenone//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Digitoxin//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Digitoxin//Cholesterol side-chain cleavage enzyme, mitochondrial//Oxidoreductase activity, acting on paired donors, with incorporation or reduction of molecular oxygen, nad(p)h as one donor, and incorporation of one atom of oxygen
Neostigmine//Cholinesterase//Identical protein binding
Methotrimeprazine//Cytochrome P450 2D6//Steroid hydroxylase activity
Methotrimeprazine//Cytochrome P450 2E1//Steroid hydroxylase activity
Danazol//Aromatase//Oxygen binding
Danazol//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Clenbuterol//Cytochrome P450 1A1//Vitamin d 24-hydroxylase activity
Bambuterol//Cholinesterase//Identical protein binding
Ciclesonide//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Ciclesonide//Cytochrome P450 2D6//Steroid hydroxylase activity
Ciclesonide//Liver carboxylesterase 1//Triglyceride lipase activity
Acenocoumarol//Cytochrome P450 2C9//Steroid hydroxylase activity
Acenocoumarol//Cytochrome P450 1A2//Oxidoreductase activity, acting on paired donors, with incorporation or reduction of molecular oxygen, reduced flavin or flavoprotein as one donor, and incorporation of one atom of oxygen
Acenocoumarol//Cytochrome P450 2C19//Steroid hydroxylase activity
Acenocoumarol//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Aprindine//Cytochrome P450 2D6//Steroid hydroxylase activity
Antipyrine//Cytochrome P450 2C8//Steroid hydroxylase activity
Antipyrine//Cytochrome P450 2C9//Steroid hydroxylase activity
Antipyrine//Cytochrome P450 1A2//Oxidoreductase activity, acting on paired donors, with incorporation or reduction of molecular oxygen, reduced flavin or flavoprotein as one donor, and incorporation of one atom of oxygen
Antipyrine//Cytochrome P450 2C19//Steroid hydroxylase activity
Antipyrine//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Antipyrine//Cytochrome P450 2A6//Steroid hydroxylase activity
Antipyrine//Cytochrome P450 2B6//Steroid hydroxylase activity
Antipyrine//Cytochrome P450 2C18//Steroid hydroxylase activity
Antipyrine//Cytochrome P450 2D6//Steroid hydroxylase activity
Antipyrine//Cytochrome P450 2E1//Steroid hydroxylase activity
Glutethimide//Cholesterol side-chain cleavage enzyme, mitochondrial//Oxidoreductase activity, acting on paired donors, with incorporation or reduction of molecular oxygen, nad(p)h as one donor, and incorporation of one atom of oxygen
Ethylmorphine//Cytochrome P450 2D6//Steroid hydroxylase activity
Ethylmorphine//NADPH--cytochrome P450 reductase//Oxidoreductase activity, acting on paired donors, with incorporation or reduction of molecular oxygen, nad(p)h as one donor, and incorporation of one atom of oxygen
Ethylmorphine//Cytochrome P450 2B6//Steroid hydroxylase activity
Ethylmorphine//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Flunitrazepam//Cytochrome P450 2C19//Steroid hydroxylase activity
Flunitrazepam//Cytochrome P450 2A6//Steroid hydroxylase activity
Flunitrazepam//UDP-glucuronosyltransferase 2B7//Glucuronosyltransferase activity
Flunitrazepam//Cytochrome P450 2B6//Steroid hydroxylase activity
Flunitrazepam//Cytochrome P450 2C9//Steroid hydroxylase activity
Flunitrazepam//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Flunitrazepam//Cytochrome P450 2E1//Steroid hydroxylase activity
Flunitrazepam//UDP-glucuronosyltransferase 1-1//Steroid binding
Flunitrazepam//UDP-glucuronosyltransferase 1-3//Retinoic acid binding
Bromazepam//Cytochrome P450 1A2//Oxidoreductase activity, acting on paired donors, with incorporation or reduction of molecular oxygen, reduced flavin or flavoprotein as one donor, and incorporation of one atom of oxygen
Bromazepam//Cytochrome P450 2C19//Steroid hydroxylase activity
Bromazepam//Cytochrome P450 2E1//Steroid hydroxylase activity
Clotiazepam//Cytochrome P450 2B6//Steroid hydroxylase activity
Clotiazepam//Cytochrome P450 2C18//Steroid hydroxylase activity
Clotiazepam//Cytochrome P450 2C19//Steroid hydroxylase activity
Clotiazepam//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Dextroamphetamine//Cytochrome P450 2D6//Steroid hydroxylase activity
Methamphetamine//Cytochrome P450 2D6//Steroid hydroxylase activity
Liotrix//Cytochrome P450 2C8//Steroid hydroxylase activity
Liotrix//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Ketazolam//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Everolimus//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Everolimus//Cytochrome P450 2D6//Steroid hydroxylase activity
Hydroxychloroquine//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Hydroxychloroquine//Cytochrome P450 2D6//Steroid hydroxylase activity
Hydroxychloroquine//Cytochrome P450 2C8//Steroid hydroxylase activity
Amylnitrite//Aldehyde dehydrogenase, mitochondrial//Electron carrier activity
Etoricoxib//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Etoricoxib//Cytochrome P450 2C9//Steroid hydroxylase activity
Etoricoxib//Cytochrome P450 2D6//Steroid hydroxylase activity
Etoricoxib//Cytochrome P450 1A2//Oxidoreductase activity, acting on paired donors, with incorporation or reduction of molecular oxygen, reduced flavin or flavoprotein as one donor, and incorporation of one atom of oxygen
Etoricoxib//Cytochrome P450 2C19//Steroid hydroxylase activity
Etoricoxib//Cytochrome P450 2E1//Steroid hydroxylase activity
Calcipotriol//Myeloperoxidase//Peroxidase activity
Calcipotriol//1,25-dihydroxyvitamin D(3) 24-hydroxylase, mitochondrial//Oxidoreductase activity
Doconexent//Cytochrome P450 2C9//Steroid hydroxylase activity
Estronesulfate//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Estronesulfate//Cytochrome P450 1A2//Oxidoreductase activity, acting on paired donors, with incorporation or reduction of molecular oxygen, reduced flavin or flavoprotein as one donor, and incorporation of one atom of oxygen
Estronesulfate//Cytochrome P450 2C9//Steroid hydroxylase activity
Bifonazole//Aromatase//Oxygen binding
Bifonazole//Cytochrome P450 2E1//Steroid hydroxylase activity
Bifonazole//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Metamizole//Cytochrome P450 2B6//Steroid hydroxylase activity
Metamizole//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Maraviroc//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Cyproteroneacetate//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Cyproteroneacetate//Aromatase//Oxygen binding
Debrisoquin//Cytochrome P450 2D6//Steroid hydroxylase activity
Debrisoquin//Cytochrome P450 1A1//Vitamin d 24-hydroxylase activity
Flunarizine//Cytochrome P450 2D6//Steroid hydroxylase activity
Flunarizine//Cytochrome P450 2C9//Steroid hydroxylase activity
Flunarizine//Cytochrome P450 1A1//Vitamin d 24-hydroxylase activity
Flunarizine//Cytochrome P450 1A2//Oxidoreductase activity, acting on paired donors, with incorporation or reduction of molecular oxygen, reduced flavin or flavoprotein as one donor, and incorporation of one atom of oxygen
Flunarizine//Cytochrome P450 2A6//Steroid hydroxylase activity
Flunarizine//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Ixabepilone//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Celiprolol//Cytochrome P450 2D6//Steroid hydroxylase activity
Dronedarone//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Dronedarone//Cytochrome P450 2D6//Steroid hydroxylase activity
Dronedarone//Cytochrome P450 3A5//Oxygen binding
Dronedarone//Cytochrome P450 2J2//Steroid hydroxylase activity
Nebivolol//Cytochrome P450 2D6//Steroid hydroxylase activity
Nebivolol//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Nebivolol//Cytochrome P450 2C19//Steroid hydroxylase activity
Lorcaserin//Cytochrome P450 1A2//Oxidoreductase activity, acting on paired donors, with incorporation or reduction of molecular oxygen, reduced flavin or flavoprotein as one donor, and incorporation of one atom of oxygen
Lorcaserin//Cytochrome P450 2A6//Steroid hydroxylase activity
Lorcaserin//Cytochrome P450 2B6//Steroid hydroxylase activity
Lorcaserin//Cytochrome P450 2C19//Steroid hydroxylase activity
Lorcaserin//Cytochrome P450 2D6//Steroid hydroxylase activity
Lorcaserin//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Lorcaserin//Dimethylaniline monooxygenase [N-oxide-forming] 1//Nadp binding
Lorcaserin//Cytochrome P450 1A1//Vitamin d 24-hydroxylase activity
Flibanserin//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Clevidipine//Cytochrome P450 2C9//Steroid hydroxylase activity
Clevidipine//Cytochrome P450 2D6//Steroid hydroxylase activity
Clevidipine//Cytochrome P450 2E1//Steroid hydroxylase activity
Clevidipine//Cytochrome P450 2C19//Steroid hydroxylase activity
Clevidipine//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Clevidipine//Cholinesterase//Identical protein binding
Iloperidone//Cytochrome P450 2D6//Steroid hydroxylase activity
Iloperidone//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Iloperidone//Cytochrome P450 3A5//Oxygen binding
Iloperidone//Cytochrome P450 3A7//Oxygen binding
Iloperidone//Cytochrome P450 2E1//Steroid hydroxylase activity
Ezogabine//UDP-glucuronosyltransferase 1-1//Steroid binding
Ezogabine//UDP-glucuronosyltransferase 1-3//Retinoic acid binding
Ezogabine//UDP-glucuronosyltransferase 1-4//Protein homodimerization activity
Ezogabine//UDP-glucuronosyltransferase 1-9//Retinoic acid binding
Ezogabine//Arylamine N-acetyltransferase 2//Arylamine n-acetyltransferase activity
Indacaterol//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Indacaterol//UDP-glucuronosyltransferase 1-1//Steroid binding
Crisaborole//Cytochrome P450 2B6//Steroid hydroxylase activity
Crisaborole//Cytochrome P450 2C8//Steroid hydroxylase activity
Crisaborole//Cytochrome P450 2C9//Steroid hydroxylase activity
Cobimetinib//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Cobimetinib//Multidrug resistance protein 1//Xenobiotic-transporting atpase activity
Methsuximide//Cytochrome P450 2C19//Steroid hydroxylase activity
Dexlansoprazole//Cytochrome P450 2C19//Steroid hydroxylase activity
Dexlansoprazole//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Brivaracetam//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Brivaracetam//Cytochrome P450 2C19//Steroid hydroxylase activity
Brivaracetam//Cytochrome P450 2B6//Steroid hydroxylase activity
Brivaracetam//Cytochrome P450 2C9//Steroid hydroxylase activity
Apremilast//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Apremilast//Cytochrome P450 2A6//Steroid hydroxylase activity
Apremilast//Cytochrome P450 1A2//Oxidoreductase activity, acting on paired donors, with incorporation or reduction of molecular oxygen, reduced flavin or flavoprotein as one donor, and incorporation of one atom of oxygen
Abiraterone//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Abiraterone//Bile salt sulfotransferase//Sulfotransferase activity
Abiraterone//Cytochrome P450 2D6//Steroid hydroxylase activity
Abiraterone//Cytochrome P450 2C8//Steroid hydroxylase activity
Abiraterone//Cytochrome P450 1A2//Oxidoreductase activity, acting on paired donors, with incorporation or reduction of molecular oxygen, reduced flavin or flavoprotein as one donor, and incorporation of one atom of oxygen
Abiraterone//Cytochrome P450 2C19//Steroid hydroxylase activity
Abiraterone//Cytochrome P450 2C9//Steroid hydroxylase activity
Cariprazine//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Cariprazine//Cytochrome P450 2D6//Steroid hydroxylase activity
Mianserin//Cytochrome P450 2D6//Steroid hydroxylase activity
Mianserin//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Mianserin//Cytochrome P450 1A2//Oxidoreductase activity, acting on paired donors, with incorporation or reduction of molecular oxygen, reduced flavin or flavoprotein as one donor, and incorporation of one atom of oxygen
Mianserin//Cytochrome P450 2B6//Steroid hydroxylase activity
Alogliptin//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Alogliptin//Cytochrome P450 2D6//Steroid hydroxylase activity
Eltrombopag//Cytochrome P450 2C8//Steroid hydroxylase activity
Eltrombopag//Cytochrome P450 1A2//Oxidoreductase activity, acting on paired donors, with incorporation or reduction of molecular oxygen, reduced flavin or flavoprotein as one donor, and incorporation of one atom of oxygen
Eltrombopag//UDP-glucuronosyltransferase 1-1//Steroid binding
Eltrombopag//UDP-glucuronosyltransferase 1-3//Retinoic acid binding
Eltrombopag//UDP-glucuronosyltransferase 1-9//Retinoic acid binding
Asenapine//UDP-glucuronosyltransferase 1-4//Protein homodimerization activity
Asenapine//Cytochrome P450 1A2//Oxidoreductase activity, acting on paired donors, with incorporation or reduction of molecular oxygen, reduced flavin or flavoprotein as one donor, and incorporation of one atom of oxygen
Asenapine//Cytochrome P450 2D6//Steroid hydroxylase activity
Asenapine//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Nalmefene//UDP-glucuronosyltransferase 2B7//Glucuronosyltransferase activity
Nalmefene//UDP-glucuronosyltransferase 1-3//Retinoic acid binding
Nalmefene//UDP-glucuronosyltransferase 1-8//Steroid binding
Avanafil//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Droxidopa//Aromatic-L-amino-acid decarboxylase//Pyridoxal phosphate binding
Amrubicin//NADPH--cytochrome P450 reductase//Oxidoreductase activity, acting on paired donors, with incorporation or reduction of molecular oxygen, nad(p)h as one donor, and incorporation of one atom of oxygen
Amrubicin//Carbonyl reductase [NADPH] 1//Prostaglandin-e2 9-reductase activity
Levocetirizine//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Dapagliflozin//Cytochrome P450 1A1//Vitamin d 24-hydroxylase activity
Dapagliflozin//Cytochrome P450 1A2//Oxidoreductase activity, acting on paired donors, with incorporation or reduction of molecular oxygen, reduced flavin or flavoprotein as one donor, and incorporation of one atom of oxygen
Dapagliflozin//Cytochrome P450 2A6//Steroid hydroxylase activity
Dapagliflozin//Cytochrome P450 2C9//Steroid hydroxylase activity
Dapagliflozin//Cytochrome P450 2D6//Steroid hydroxylase activity
Dapagliflozin//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Dapagliflozin//UDP-glucuronosyltransferase 1-9//Retinoic acid binding
Dapagliflozin//UDP-glucuronosyltransferase 2B4//Glucuronosyltransferase activity
Dapagliflozin//UDP-glucuronosyltransferase 2B7//Glucuronosyltransferase activity
Ambrisentan//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Ambrisentan//Cytochrome P450 2C19//Steroid hydroxylase activity
Ambrisentan//UDP-glucuronosyltransferase 1-9//Retinoic acid binding
Ambrisentan//UDP-glucuronosyltransferase 2B7//Glucuronosyltransferase activity
Ambrisentan//UDP-glucuronosyltransferase 1-3//Retinoic acid binding
Ambrisentan//Cytochrome P450 3A5//Oxygen binding
Doxercalciferol//Sterol 26-hydroxylase, mitochondrial//Vitamin d3 25-hydroxylase activity
Armodafinil//Cytochrome P450 2C19//Steroid hydroxylase activity
Armodafinil//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Armodafinil//Cytochrome P450 3A5//Oxygen binding
Armodafinil//Cytochrome P450 1A2//Oxidoreductase activity, acting on paired donors, with incorporation or reduction of molecular oxygen, reduced flavin or flavoprotein as one donor, and incorporation of one atom of oxygen
Armodafinil//Cytochrome P450 2B6//Steroid hydroxylase activity
Armodafinil//Cytochrome P450 2C9//Steroid hydroxylase activity
Agomelatine//Cytochrome P450 1A2//Oxidoreductase activity, acting on paired donors, with incorporation or reduction of molecular oxygen, reduced flavin or flavoprotein as one donor, and incorporation of one atom of oxygen
Agomelatine//Cytochrome P450 2C9//Steroid hydroxylase activity
Midostaurin//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Midostaurin//Cytochrome P450 3A43//Monooxygenase activity
Midostaurin//Cytochrome P450 3A5//Oxygen binding
Midostaurin//Cytochrome P450 3A7//Oxygen binding
Midostaurin//Cytochrome P450 1A2//Oxidoreductase activity, acting on paired donors, with incorporation or reduction of molecular oxygen, reduced flavin or flavoprotein as one donor, and incorporation of one atom of oxygen
Midostaurin//Cytochrome P450 2B6//Steroid hydroxylase activity
Midostaurin//Cytochrome P450 2C8//Steroid hydroxylase activity
Midostaurin//Cytochrome P450 2C9//Steroid hydroxylase activity
Midostaurin//Cytochrome P450 2C19//Steroid hydroxylase activity
Midostaurin//Cytochrome P450 2D6//Steroid hydroxylase activity
Midostaurin//Cytochrome P450 2E1//Steroid hydroxylase activity
Midostaurin//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Midostaurin//Cytochrome P450 3A5//Oxygen binding
Midostaurin//Cytochrome P450 3A7//Oxygen binding
Midostaurin//Cytochrome P450 3A43//Monooxygenase activity
Apixaban//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Apixaban//Cytochrome P450 1A2//Oxidoreductase activity, acting on paired donors, with incorporation or reduction of molecular oxygen, reduced flavin or flavoprotein as one donor, and incorporation of one atom of oxygen
Apixaban//Cytochrome P450 2C8//Steroid hydroxylase activity
Apixaban//Cytochrome P450 2C9//Steroid hydroxylase activity
Apixaban//Cytochrome P450 2C19//Steroid hydroxylase activity
Apixaban//Cytochrome P450 2J2//Steroid hydroxylase activity
Apixaban//Cytochrome P450 3A5//Oxygen binding
Bosutinib//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Bosutinib//Cytochrome P450 2C8//Steroid hydroxylase activity
Axitinib//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Axitinib//Cytochrome P450 3A5//Oxygen binding
Axitinib//Cytochrome P450 1A2//Oxidoreductase activity, acting on paired donors, with incorporation or reduction of molecular oxygen, reduced flavin or flavoprotein as one donor, and incorporation of one atom of oxygen
Axitinib//Cytochrome P450 2C19//Steroid hydroxylase activity
Axitinib//UDP-glucuronosyltransferase 1-1//Steroid binding
Dalfampridine//Cytochrome P450 2E1//Steroid hydroxylase activity
Mepyramine//Cytochrome P450 2D6//Steroid hydroxylase activity
Dabigatranetexilate//Liver carboxylesterase 1//Triglyceride lipase activity
Dabigatranetexilate//UDP-glucuronosyltransferase 1-9//Retinoic acid binding
Dabigatranetexilate//UDP-glucuronosyltransferase 2B7//Glucuronosyltransferase activity
Dabigatranetexilate//UDP-glucuronosyltransferase 2B15//Glucuronosyltransferase activity
Dabigatranetexilate//Ribosyldihydronicotinamide dehydrogenase [quinone]//Nadph dehydrogenase (quinone) activity
Desvenlafaxine//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Desvenlafaxine//Cytochrome P450 2D6//Steroid hydroxylase activity
Fesoterodine//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Fesoterodine//Cytochrome P450 2D6//Steroid hydroxylase activity
Methyltestosterone//Cytochrome P450 2B6//Steroid hydroxylase activity
Methyltestosterone//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Methyltestosterone//Aromatase//Oxygen binding
Fospropofol//Alkaline phosphatase, tissue-nonspecific isozyme//Pyrophosphatase activity
Lornoxicam//Cytochrome P450 2C9//Steroid hydroxylase activity
Gestodene//Cytochrome P450 3A5//Oxygen binding
Gestodene//Cytochrome P450 3A7//Oxygen binding
Gestodene//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Gestodene//Cytochrome P450 2C19//Steroid hydroxylase activity
Aceclofenac//Cytochrome P450 2C9//Steroid hydroxylase activity
Ketobemidone//Prostaglandin G/H synthase 1//Prostaglandin-endoperoxide synthase activity
Ketobemidone//Cytochrome P450 2C9//Steroid hydroxylase activity
Ketobemidone//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Ketobemidone//UDP-glucuronosyltransferase 1-9//Retinoic acid binding
Ketobemidone//Cytochrome P450 2B6//Steroid hydroxylase activity
Ketobemidone//Cytochrome P450 2C19//Steroid hydroxylase activity
Ketobemidone//Cytochrome P450 2C8//Steroid hydroxylase activity
Cabazitaxel//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Cabazitaxel//Cytochrome P450 3A5//Oxygen binding
Cabazitaxel//Cytochrome P450 2C8//Steroid hydroxylase activity
Capsaicin//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Capsaicin//Prostaglandin G/H synthase 2//Prostaglandin-endoperoxide synthase activity
Capsaicin//Myeloperoxidase//Peroxidase activity
Capsaicin//Cytochrome P450 1A2//Oxidoreductase activity, acting on paired donors, with incorporation or reduction of molecular oxygen, reduced flavin or flavoprotein as one donor, and incorporation of one atom of oxygen
Capsaicin//Cytochrome P450 2E1//Steroid hydroxylase activity
Capsaicin//Amine oxidase [flavin-containing] A//Serotonin binding
Capsaicin//Dopamine beta-hydroxylase//L-ascorbic acid binding
Capsaicin//Glutamine synthetase//Manganese ion binding
Capsaicin//Cholinesterase//Identical protein binding
Chenodeoxycholicacid//Sterol 26-hydroxylase, mitochondrial//Vitamin d3 25-hydroxylase activity
Chenodeoxycholicacid//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Chenodeoxycholicacid//UDP-glucuronosyltransferase 2B7//Glucuronosyltransferase activity
Hydroxyprogesteronecaproate//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Hydroxyprogesteronecaproate//Cytochrome P450 3A5//Oxygen binding
Hydroxyprogesteronecaproate//Cytochrome P450 2C19//Steroid hydroxylase activity
Nandrolonedecanoate//Aromatase//Oxygen binding
Nandrolonedecanoate//Amine oxidase [flavin-containing] B//Primary amine oxidase activity
Nandrolonedecanoate//Amine oxidase [flavin-containing] A//Serotonin binding
Lurasidone//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Ivacaftor//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Ivacaftor//Cytochrome P450 3A5//Oxygen binding
Lomitapide//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Crizotinib//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Crizotinib//Cytochrome P450 3A5//Oxygen binding
Crizotinib//Cytochrome P450 2B6//Steroid hydroxylase activity
Crizotinib//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Crizotinib//Cytochrome P450 3A43//Monooxygenase activity
Crizotinib//Cytochrome P450 3A5//Oxygen binding
Crizotinib//Cytochrome P450 3A7//Oxygen binding
Fingolimod//Sphingosine kinase 1//Sphingosine-1-phosphate receptor activity
Fingolimod//Cytochrome P450 2E1//Steroid hydroxylase activity
Cabozantinib//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Cabozantinib//Cytochrome P450 2C9//Steroid hydroxylase activity
Cabozantinib//Cytochrome P450 2C8//Steroid hydroxylase activity
Linagliptin//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Mirabegron//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Mirabegron//Cytochrome P450 2D6//Steroid hydroxylase activity
Mirabegron//Cholinesterase//Identical protein binding
Aclidinium//Cholinesterase//Identical protein binding
Enzalutamide//Cytochrome P450 2C8//Steroid hydroxylase activity
Enzalutamide//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Enzalutamide//Cytochrome P450 2C9//Steroid hydroxylase activity
Enzalutamide//Cytochrome P450 2C19//Steroid hydroxylase activity
Enzalutamide//Cytochrome P450 2B6//Steroid hydroxylase activity
Enzalutamide//Cytochrome P450 3A5//Oxygen binding
Fluticasonefuroate//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Fluticasonefuroate//Cytochrome P450 3A5//Oxygen binding
Fluticasonefuroate//Cytochrome P450 3A7//Oxygen binding
Fluticasonefuroate//Cytochrome P450 2C8//Steroid hydroxylase activity
Canagliflozin//UDP-glucuronosyltransferase 1-9//Retinoic acid binding
Canagliflozin//UDP-glucuronosyltransferase 2B4//Glucuronosyltransferase activity
Canagliflozin//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Dabrafenib//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Dabrafenib//Cytochrome P450 2C8//Steroid hydroxylase activity
Dabrafenib//Cytochrome P450 2B6//Steroid hydroxylase activity
Dabrafenib//Cytochrome P450 2C9//Steroid hydroxylase activity
Levomilnacipran//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Levomilnacipran//Cytochrome P450 2C8//Steroid hydroxylase activity
Levomilnacipran//Cytochrome P450 2C19//Steroid hydroxylase activity
Levomilnacipran//Cytochrome P450 2D6//Steroid hydroxylase activity
Levomilnacipran//Cytochrome P450 2J2//Steroid hydroxylase activity
Macitentan//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Macitentan//Cytochrome P450 2C19//Steroid hydroxylase activity
Aliskiren//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Miltefosine//Phospholipase D1//Phospholipase d activity
Eliglustat//Cytochrome P450 2D6//Steroid hydroxylase activity
Eliglustat//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Netupitant//Cytochrome P450 3A43//Monooxygenase activity
Netupitant//Cytochrome P450 2C9//Steroid hydroxylase activity
Netupitant//Cytochrome P450 2D6//Steroid hydroxylase activity
Netupitant//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Naloxegol//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Naloxegol//Cytochrome P450 2D6//Steroid hydroxylase activity
Naloxegol//Cytochrome P450 2C19//Steroid hydroxylase activity
Ibrutinib//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Ibrutinib//Cytochrome P450 3A5//Oxygen binding
Ibrutinib//Cytochrome P450 2D6//Steroid hydroxylase activity
Cannabidiol//Cytochrome P450 2C9//Steroid hydroxylase activity
Cannabidiol//Cytochrome P450 2C19//Steroid hydroxylase activity
Cannabidiol//Cytochrome P450 2D6//Steroid hydroxylase activity
Cannabidiol//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Cannabidiol//Cytochrome P450 3A5//Oxygen binding
Cannabidiol//Cytochrome P450 1A1//Vitamin d 24-hydroxylase activity
Cannabidiol//Fatty-acid amide hydrolase 1//Fatty acid amide hydrolase activity
Cannabidiol//Arachidonate 5-lipoxygenase//Iron ion binding
Cannabidiol//Arachidonate 15-lipoxygenase//Phosphatidylinositol-4,5-bisphosphate binding
Cannabidiol//Quinone oxidoreductase//Zinc ion binding
Ceritinib//Cytochrome P450 2C9//Steroid hydroxylase activity
Ceritinib//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Lenvatinib//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Lenvatinib//Aldehyde oxidase//Xanthine dehydrogenase activity
Lenvatinib//Cytochrome P450 2C8//Steroid hydroxylase activity
Lenvatinib//Cytochrome P450 2C9//Steroid hydroxylase activity
Lenvatinib//Cytochrome P450 1A2//Oxidoreductase activity, acting on paired donors, with incorporation or reduction of molecular oxygen, reduced flavin or flavoprotein as one donor, and incorporation of one atom of oxygen
Lenvatinib//Cytochrome P450 2B6//Steroid hydroxylase activity
Lenvatinib//Cytochrome P450 2C19//Steroid hydroxylase activity
Lenvatinib//Cytochrome P450 2D6//Steroid hydroxylase activity
Calciumcarbimide//Catalase//Receptor binding
Eslicarbazepineacetate//Cytochrome P450 2C19//Steroid hydroxylase activity
Eslicarbazepineacetate//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Eslicarbazepineacetate//UDP-glucuronosyltransferase 1-1//Steroid binding
Dienogest//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Brexpiprazole//Cytochrome P450 2D6//Steroid hydroxylase activity
Brexpiprazole//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Etizolam//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Etizolam//Cytochrome P450 2C18//Steroid hydroxylase activity
Etizolam//Cytochrome P450 2C19//Steroid hydroxylase activity
Dosulepin//Cytochrome P450 2D6//Steroid hydroxylase activity
Dosulepin//Cytochrome P450 1A2//Oxidoreductase activity, acting on paired donors, with incorporation or reduction of molecular oxygen, reduced flavin or flavoprotein as one donor, and incorporation of one atom of oxygen
Dosulepin//Cytochrome P450 2C19//Steroid hydroxylase activity
Dosulepin//Cytochrome P450 2C9//Steroid hydroxylase activity
Lorpiprazole//Cytochrome P450 2D6//Steroid hydroxylase activity
Lorpiprazole//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Lobeglitazone//Cytochrome P450 1A2//Oxidoreductase activity, acting on paired donors, with incorporation or reduction of molecular oxygen, reduced flavin or flavoprotein as one donor, and incorporation of one atom of oxygen
Lobeglitazone//Cytochrome P450 2C9//Steroid hydroxylase activity
Lobeglitazone//Cytochrome P450 2C19//Steroid hydroxylase activity
Lobeglitazone//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Lobeglitazone//Cytochrome P450 2C8//Steroid hydroxylase activity
Loxoprofen//Carbonyl reductase [NADPH] 1//Prostaglandin-e2 9-reductase activity
Loxoprofen//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Loxoprofen//Cytochrome P450 3A43//Monooxygenase activity
Loxoprofen//Cytochrome P450 3A5//Oxygen binding
Loxoprofen//Cytochrome P450 3A7//Oxygen binding
Loxoprofen//UDP-glucuronosyltransferase 2B7//Glucuronosyltransferase activity
Dexketoprofen//Prostaglandin G/H synthase 1//Prostaglandin-endoperoxide synthase activity
Dexketoprofen//Prostaglandin G/H synthase 2//Prostaglandin-endoperoxide synthase activity
Blonanserin//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Melperone//Cytochrome P450 2D6//Steroid hydroxylase activity
Aranidipine//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Azelnidipine//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Benidipine//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Benidipine//Cytochrome P450 3A5//Oxygen binding
Cilnidipine//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Efonidipine//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Imidafenacin//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Imidafenacin//UDP-glucuronosyltransferase 1-4//Protein homodimerization activity
Lumacaftor//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Lumacaftor//Cytochrome P450 2B6//Steroid hydroxylase activity
Lumacaftor//Cytochrome P450 2C8//Steroid hydroxylase activity
Lumacaftor//Cytochrome P450 2C9//Steroid hydroxylase activity
Lumacaftor//Cytochrome P450 2C19//Steroid hydroxylase activity
Molsidomine//Guanylate cyclase soluble subunit alpha-2//Heme binding
Molsidomine//cGMP-specific 3',5'-cyclic phosphodiesterase//Metal ion binding
Morniflumate//Arachidonate 5-lipoxygenase//Iron ion binding
Morniflumate//Prostaglandin G/H synthase 2//Prostaglandin-endoperoxide synthase activity
Morniflumate//UDP-glucuronosyltransferase 1-9//Retinoic acid binding
Glycerin//Retinal dehydrogenase 1//Retinal dehydrogenase activity
Glycerin//Cytochrome P450 2E1//Steroid hydroxylase activity
Dexchlorpheniraminemaleate//Cytochrome P450 2D6//Steroid hydroxylase activity
Dexchlorpheniraminemaleate//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Butamben//Cholinesterase//Identical protein binding
Homatropine//Liver carboxylesterase 1//Triglyceride lipase activity
Lesinurad//Cytochrome P450 2C9//Steroid hydroxylase activity
Lesinurad//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Isavuconazole//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Isavuconazole//Cytochrome P450 3A5//Oxygen binding
Isavuconazole//Cytochrome P450 2C8//Steroid hydroxylase activity
Isavuconazole//Cytochrome P450 2C9//Steroid hydroxylase activity
Isavuconazole//Cytochrome P450 2C19//Steroid hydroxylase activity
Isavuconazole//Cytochrome P450 2D6//Steroid hydroxylase activity
Isavuconazole//Cytochrome P450 2B6//Steroid hydroxylase activity
Isavuconazole//UDP-glucuronosyltransferase 1-9//Retinoic acid binding
Isavuconazole//UDP-glucuronosyltransferase 1-8//Steroid binding
Artenimol//UDP-glucuronosyltransferase 1-9//Retinoic acid binding
Artenimol//UDP-glucuronosyltransferase 2B7//Glucuronosyltransferase activity
Artenimol//Cytochrome P450 2D6//Steroid hydroxylase activity
Artenimol//Cytochrome P450 2C19//Steroid hydroxylase activity
Naldemedine//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Naldemedine//Cytochrome P450 3A43//Monooxygenase activity
Naldemedine//Cytochrome P450 3A5//Oxygen binding
Naldemedine//Cytochrome P450 3A7//Oxygen binding
Naldemedine//UDP-glucuronosyltransferase 1-3//Retinoic acid binding
Icotinib//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Icotinib//Cytochrome P450 1A2//Oxidoreductase activity, acting on paired donors, with incorporation or reduction of molecular oxygen, reduced flavin or flavoprotein as one donor, and incorporation of one atom of oxygen
Icotinib//Cytochrome P450 3A5//Oxygen binding
Baricitinib//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Ertugliflozin//UDP-glucuronosyltransferase 1-9//Retinoic acid binding
Ertugliflozin//UDP-glucuronosyltransferase 2B7//Glucuronosyltransferase activity
Ertugliflozin//UDP-glucuronosyltransferase 1-1//Steroid binding
Ertugliflozin//UDP-glucuronosyltransferase 1-4//Protein homodimerization activity
Neratinib//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Neratinib//Dimethylaniline monooxygenase [N-oxide-forming] 3//Trimethylamine monooxygenase activity
Apalutamide//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Apalutamide//Cytochrome P450 2C8//Steroid hydroxylase activity
Apalutamide//Cytochrome P450 2C19//Steroid hydroxylase activity
Apalutamide//Cytochrome P450 2C9//Steroid hydroxylase activity
Abemaciclib//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Abemaciclib//Cytochrome P450 1A2//Oxidoreductase activity, acting on paired donors, with incorporation or reduction of molecular oxygen, reduced flavin or flavoprotein as one donor, and incorporation of one atom of oxygen
Abemaciclib//Cytochrome P450 2B6//Steroid hydroxylase activity
Abemaciclib//Cytochrome P450 2C8//Steroid hydroxylase activity
Abemaciclib//Cytochrome P450 2C9//Steroid hydroxylase activity
Abemaciclib//Cytochrome P450 2D6//Steroid hydroxylase activity
Fostamatinib//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Fostamatinib//UDP-glucuronosyltransferase 1-9//Retinoic acid binding
Deutetrabenazine//Carbonyl reductase [NADPH] 1//Prostaglandin-e2 9-reductase activity
Deutetrabenazine//Carbonyl reductase [NADPH] 3//Nadph binding
Deutetrabenazine//Cytochrome P450 2D6//Steroid hydroxylase activity
Deutetrabenazine//Cytochrome P450 1A2//Oxidoreductase activity, acting on paired donors, with incorporation or reduction of molecular oxygen, reduced flavin or flavoprotein as one donor, and incorporation of one atom of oxygen
Deutetrabenazine//Cytochrome P450 3A5//Oxygen binding
Deutetrabenazine//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Brigatinib//Cytochrome P450 2C8//Steroid hydroxylase activity
Brigatinib//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Brigatinib//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Brigatinib//Cytochrome P450 3A43//Monooxygenase activity
Brigatinib//Cytochrome P450 3A5//Oxygen binding
Brigatinib//Cytochrome P450 3A7//Oxygen binding
Betrixaban//Prothrombin//Thrombospondin receptor activity
Copanlisib//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Copanlisib//Cytochrome P450 3A5//Oxygen binding
Copanlisib//Cytochrome P450 3A7//Oxygen binding
Copanlisib//Cytochrome P450 3A43//Monooxygenase activity
Macimorelin//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Levosalbutamol//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Levosalbutamol//Cytochrome P450 2D6//Steroid hydroxylase activity
Acemetacin//UDP-glucuronosyltransferase 2B7//Glucuronosyltransferase activity
Enasidenib//Cytochrome P450 1A2//Oxidoreductase activity, acting on paired donors, with incorporation or reduction of molecular oxygen, reduced flavin or flavoprotein as one donor, and incorporation of one atom of oxygen
Enasidenib//Cytochrome P450 2B6//Steroid hydroxylase activity
Enasidenib//Cytochrome P450 2C8//Steroid hydroxylase activity
Enasidenib//Cytochrome P450 2C9//Steroid hydroxylase activity
Enasidenib//Cytochrome P450 2C19//Steroid hydroxylase activity
Enasidenib//Cytochrome P450 2D6//Steroid hydroxylase activity
Enasidenib//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Enasidenib//UDP-glucuronosyltransferase 1-1//Steroid binding
Enasidenib//UDP-glucuronosyltransferase 1-3//Retinoic acid binding
Enasidenib//UDP-glucuronosyltransferase 1-4//Protein homodimerization activity
Enasidenib//UDP-glucuronosyltransferase 1-9//Retinoic acid binding
Enasidenib//UDP-glucuronosyltransferase 2B7//Glucuronosyltransferase activity
Enasidenib//UDP-glucuronosyltransferase 2B15//Glucuronosyltransferase activity
Estradiolacetate//Cytochrome P450 1A2//Oxidoreductase activity, acting on paired donors, with incorporation or reduction of molecular oxygen, reduced flavin or flavoprotein as one donor, and incorporation of one atom of oxygen
Estradiolacetate//UDP-glucuronosyltransferase 1-1//Steroid binding
Estradiolacetate//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Estradiolacetate//Cytochrome P450 3A5//Oxygen binding
Estradiolacetate//Cytochrome P450 3A7//Oxygen binding
Estradiolacetate//Cytochrome P450 1A1//Vitamin d 24-hydroxylase activity
Estradiolacetate//Cytochrome P450 1B1//Oxygen binding
Estradiolacetate//Cytochrome P450 2C19//Steroid hydroxylase activity
Estradiolacetate//Cytochrome P450 2C8//Steroid hydroxylase activity
Estradiolacetate//Cytochrome P450 2C9//Steroid hydroxylase activity
Estradiolbenzoate//Cytochrome P450 1A2//Oxidoreductase activity, acting on paired donors, with incorporation or reduction of molecular oxygen, reduced flavin or flavoprotein as one donor, and incorporation of one atom of oxygen
Estradiolbenzoate//UDP-glucuronosyltransferase 1-1//Steroid binding
Estradiolbenzoate//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Estradiolbenzoate//Cytochrome P450 3A5//Oxygen binding
Estradiolbenzoate//Cytochrome P450 3A7//Oxygen binding
Estradiolbenzoate//Cytochrome P450 1A1//Vitamin d 24-hydroxylase activity
Estradiolbenzoate//Cytochrome P450 1B1//Oxygen binding
Estradiolbenzoate//Cytochrome P450 2C19//Steroid hydroxylase activity
Estradiolbenzoate//Cytochrome P450 2C8//Steroid hydroxylase activity
Estradiolbenzoate//Cytochrome P450 2C9//Steroid hydroxylase activity
Estradiolcypionate//Cytochrome P450 1A2//Oxidoreductase activity, acting on paired donors, with incorporation or reduction of molecular oxygen, reduced flavin or flavoprotein as one donor, and incorporation of one atom of oxygen
Estradiolcypionate//UDP-glucuronosyltransferase 1-1//Steroid binding
Estradiolcypionate//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Estradiolcypionate//Cytochrome P450 3A5//Oxygen binding
Estradiolcypionate//Cytochrome P450 3A7//Oxygen binding
Estradiolcypionate//Cytochrome P450 1A1//Vitamin d 24-hydroxylase activity
Estradiolcypionate//Cytochrome P450 1B1//Oxygen binding
Estradiolcypionate//Cytochrome P450 2C19//Steroid hydroxylase activity
Estradiolcypionate//Cytochrome P450 2C8//Steroid hydroxylase activity
Estradiolcypionate//Cytochrome P450 2C9//Steroid hydroxylase activity
Estradioldienanthate//Cytochrome P450 1A2//Oxidoreductase activity, acting on paired donors, with incorporation or reduction of molecular oxygen, reduced flavin or flavoprotein as one donor, and incorporation of one atom of oxygen
Estradioldienanthate//UDP-glucuronosyltransferase 1-1//Steroid binding
Estradioldienanthate//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Estradioldienanthate//Cytochrome P450 3A5//Oxygen binding
Estradioldienanthate//Cytochrome P450 3A7//Oxygen binding
Estradioldienanthate//Cytochrome P450 1A1//Vitamin d 24-hydroxylase activity
Estradioldienanthate//Cytochrome P450 1B1//Oxygen binding
Estradioldienanthate//Cytochrome P450 2C19//Steroid hydroxylase activity
Estradioldienanthate//Cytochrome P450 2C8//Steroid hydroxylase activity
Estradioldienanthate//Cytochrome P450 2C9//Steroid hydroxylase activity
Estradiolvalerate//Cytochrome P450 1A2//Oxidoreductase activity, acting on paired donors, with incorporation or reduction of molecular oxygen, reduced flavin or flavoprotein as one donor, and incorporation of one atom of oxygen
Estradiolvalerate//UDP-glucuronosyltransferase 1-1//Steroid binding
Estradiolvalerate//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Estradiolvalerate//Cytochrome P450 3A5//Oxygen binding
Estradiolvalerate//Cytochrome P450 3A7//Oxygen binding
Estradiolvalerate//Cytochrome P450 1A1//Vitamin d 24-hydroxylase activity
Estradiolvalerate//Cytochrome P450 1B1//Oxygen binding
Estradiolvalerate//Cytochrome P450 2C19//Steroid hydroxylase activity
Estradiolvalerate//Cytochrome P450 2C8//Steroid hydroxylase activity
Estradiolvalerate//Cytochrome P450 2C9//Steroid hydroxylase activity
Cholinesalicylate//Choline/ethanolaminephosphotransferase 1//Metal ion binding
Cholinesalicylate//Choline kinase alpha//Signal transducer activity
Nabiximols//Cytochrome P450 2C9//Steroid hydroxylase activity
Nabiximols//Cytochrome P450 2C19//Steroid hydroxylase activity
Nabiximols//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Nabiximols//Cytochrome P450 3A5//Oxygen binding
Nabiximols//Arachidonate 5-lipoxygenase//Iron ion binding
Nabiximols//Arachidonate 15-lipoxygenase//Phosphatidylinositol-4,5-bisphosphate binding
Nabiximols//Cytochrome P450 2D6//Steroid hydroxylase activity
Bivalirudin//Prothrombin//Thrombospondin receptor activity
Desmopressin//Vasopressin V2 receptor//Vasopressin receptor activity
Desmopressin//Vasopressin V1a receptor//Vasopressin receptor activity
Desmopressin//Vasopressin V1b receptor//Vasopressin receptor activity
Cyclosporine//Calcineurin subunit B type 2//Calcium ion binding
Cyanocobalamin//Methionine synthase//Zinc ion binding
Cyanocobalamin//Methylmalonic aciduria and homocystinuria type C protein//Cobalamin binding
Cyanocobalamin//Methylenetetrahydrofolate reductase//Protein complex binding
Choline//Acetylcholinesterase//Serine hydrolase activity
Choline//Choline-phosphate cytidylyltransferase A//Lipid binding
Choline//Phospholipase D2//Phospholipase d activity
Choline//Cholinesterase//Identical protein binding
Choline//Phospholipase D1//Phospholipase d activity
Choline//Phosphoethanolamine/phosphocholine phosphatase//Pyrophosphatase activity
Choline//Neuronal acetylcholine receptor subunit alpha-7//Toxic substance binding
    Lglutamine//Amidophosphoribosyltransferase//Metal ion binding
    Lglutamine//Glutamine synthetase//Manganese ion binding
Methionine//Methionine synthase//Zinc ion binding
Methionine//Betaine--homocysteine S-methyltransferase 1//Zinc ion binding
Methionine//Methionine aminopeptidase 2//Poly(a) rna binding
Methionine//S-methylmethionine--homocysteine S-methyltransferase BHMT2//Zinc ion binding
Calcitriol//Vitamin D3 receptor//Zinc ion binding
Calcidiol//Vitamin D3 receptor//Zinc ion binding
Ltryptophan//Tryptophan--tRNA ligase, cytoplasmic//Tryptophan-trna ligase activity
Ltryptophan//Tryptophan--tRNA ligase//Tryptophan-trna ligase activity
Ltryptophan//Tryptophan--tRNA ligase, mitochondrial//Tryptophan-trna ligase activity
Ergocalciferol//Vitamin D3 receptor//Zinc ion binding
Ergocalciferol//Voltage-dependent calcium channel gamma-1 subunit//Voltage-gated calcium channel activity
Ergocalciferol//Voltage-dependent calcium channel gamma-2 subunit//Voltage-gated calcium channel activity
Ergocalciferol//Voltage-dependent calcium channel gamma-3 subunit//Regulates the trafficking to the somatodendritic compartment and gating properties of AMPA-selective glutamate receptors (AMPARs). Promotes their targeting to the cell membrane and synapses and modulates their gating properties by slowing their rates of activation, deactivation and desensitization. Does not show subunit-specific AMPA receptor regulation and regulates all AMPAR subunits. Thought to stabilize the calcium channel in an inactivated (closed) state.
Ergocalciferol//Voltage-dependent calcium channel gamma-4 subunit//Regulates the trafficking and gating properties of AMPA-selective glutamate receptors (AMPARs). Promotes their targeting to the cell membrane and synapses and modulates their gating properties by slowing their rates of activation, deactivation and desensitization and by mediating their resensitization. Does not show subunit-specific AMPA receptor regulation and regulates all AMPAR subunits. Thought to stabilize the calcium channel in an inactivated (closed) state.
Ergocalciferol//Voltage-dependent calcium channel gamma-5 subunit//Regulates the gating properties of AMPA-selective glutamate receptors (AMPARs). Modulates their gating properties by accelerating their rates of activation, deactivation and desensitization. Displays subunit-specific AMPA receptor regulation. Shows specificity for GRIA1, GRIA4 and the long isoform of GRIA2. Thought to stabilize the calcium channel in an inactivated (closed) state (By similarity).
Ergocalciferol//Voltage-dependent calcium channel gamma-6 subunit//Thought to stabilize the calcium channel in an inactivated (closed) state.
Ergocalciferol//Voltage-dependent calcium channel gamma-7 subunit//Regulates the trafficking and gating properties of AMPA-selective glutamate receptors (AMPARs). Promotes their targeting to the cell membrane and synapses and modulates their gating properties by slowing their rates of activation, deactivation and desensitization and by mediating their resensitization. Displays subunit-specific AMPA receptor regulation. Shows specificity only for GRIA1 and GRIA2. Thought to stabilize the calcium channel in an inactivated (closed) state.
Ergocalciferol//Voltage-dependent calcium channel gamma-8 subunit//Regulates the trafficking and gating properties of AMPA-selective glutamate receptors (AMPARs). Promotes their targeting to the cell membrane and synapses and modulates their gating properties by slowing their rates of activation, deactivation and desensitization and by mediating their resensitization. Does not show subunit-specific AMPA receptor regulation and regulates all AMPAR subunits. Thought to stabilize the calcium channel in an inactivated (closed) state.
Ergocalciferol//Voltage-dependent calcium channel subunit alpha-2/delta-1//Voltage-gated calcium channel activity
Ergocalciferol//Voltage-dependent calcium channel subunit alpha-2/delta-2//Voltage-gated calcium channel activity
Ergocalciferol//Voltage-dependent calcium channel subunit alpha-2/delta-3//Voltage-gated ion channel activity
Ergocalciferol//Voltage-dependent calcium channel subunit alpha-2/delta-4//The alpha-2/delta subunit of voltage-dependent calcium channels regulates calcium current density and activation/inactivation kinetics of the calcium channel.
Ergocalciferol//Voltage-dependent L-type calcium channel subunit alpha-1C//Voltage-gated calcium channel activity
Ergocalciferol//Voltage-dependent L-type calcium channel subunit alpha-1D//Voltage-gated calcium channel activity involved sa node cell action potential
Ergocalciferol//Voltage-dependent L-type calcium channel subunit alpha-1F//Voltage-gated calcium channel activity
Ergocalciferol//Voltage-dependent L-type calcium channel subunit alpha-1S//Voltage-gated calcium channel activity
Ergocalciferol//Voltage-dependent L-type calcium channel subunit beta-1//Voltage-gated calcium channel activity
Ergocalciferol//Voltage-dependent L-type calcium channel subunit beta-2//Voltage-gated calcium channel activity
Ergocalciferol//Voltage-dependent L-type calcium channel subunit beta-3//Voltage-gated calcium channel activity
Ergocalciferol//Voltage-dependent L-type calcium channel subunit beta-4//Voltage-gated calcium channel activity
Ergocalciferol//Voltage-dependent N-type calcium channel subunit alpha-1B//Voltage-gated calcium channel activity
Ergocalciferol//Voltage-dependent P/Q-type calcium channel subunit alpha-1A//Voltage-gated calcium channel activity
Ergocalciferol//Voltage-dependent R-type calcium channel subunit alpha-1E//Voltage-sensitive calcium channels (VSCC) mediate the entry of calcium ions into excitable cells and are also involved in a variety of calcium-dependent processes, including muscle contraction, hormone or neurotransmitter release, gene expression, cell motility, cell division and cell death. The isoform alpha-1E gives rise to R-type calcium currents. R-type calcium channels belong to the 'high-voltage activated' (HVA) group and are blocked by nickel, and partially by omega-agatoxin-IIIA (omega-Aga-IIIA). They are however insensitive to dihydropyridines (DHP), omega-conotoxin-GVIA (omega-CTx-GVIA), and omega-agatoxin-IVA (omega-Aga-IVA). Calcium channels containing alpha-1E subunit could be involved in the modulation of firing patterns of neurons which is important for information processing.
Ergocalciferol//Voltage-dependent T-type calcium channel subunit alpha-1G//Scaffold protein binding
Ergocalciferol//Voltage-dependent T-type calcium channel subunit alpha-1H//Scaffold protein binding
Ergocalciferol//Voltage-dependent T-type calcium channel subunit alpha-1I//Voltage-gated calcium channel activity
Folicacid//Folate receptor alpha//Receptor activity
Lipoicacid//Lipoyltransferase 1, mitochondrial//Transferase activity, transferring acyl groups
Lipoicacid//Lipoyl synthase, mitochondrial//Metal ion binding
Cholecalciferol//Vitamin D3 receptor//Zinc ion binding
Menadione//Vitamin K epoxide reductase complex subunit 1//Vitamin-k-epoxide reductase (warfarin-sensitive) activity
Menadione//Vitamin K epoxide reductase complex subunit 1-like protein 1//Vitamin-k-epoxide reductase (warfarin-sensitive) activity
Menadione//Prothrombin//Thrombospondin receptor activity
Menadione//Coagulation factor IX//Serine-type endopeptidase activity
Menadione//Vitamin K-dependent protein C//Serine-type endopeptidase activity
Menadione//Ribosyldihydronicotinamide dehydrogenase [quinone]//Nadph dehydrogenase (quinone) activity
Menadione//NAD(P)H dehydrogenase [quinone] 1//Superoxide dismutase activity
Menadione//Osteocalcin//Structural molecule activity
Fluvoxamine//Sodium-dependent serotonin transporter//Serotonin:sodium symporter activity
Fluvoxamine//Potassium voltage-gated channel subfamily H member 2//Voltage-gated potassium channel activity involved in ventricular cardiac muscle cell action potential repolarization
Masoprocol//Arachidonate 5-lipoxygenase//Iron ion binding
Masoprocol//Sex hormone-binding globulin//Androgen binding
Flunisolide//Glucocorticoid receptor//Zinc ion binding
Amphetamine//Synaptic vesicular amine transporter//Monoamine transmembrane transporter activity
Amphetamine//Sodium-dependent dopamine transporter//Monoamine transmembrane transporter activity
Amphetamine//Trace amine-associated receptor 1//Trace-amine receptor activity
Amphetamine//Sodium-dependent noradrenaline transporter//Norepinephrine:sodium symporter activity
Amphetamine//Alpha-1A adrenergic receptor//Protein heterodimerization activity
Amphetamine//Alpha-1B adrenergic receptor//Protein heterodimerization activity
Amphetamine//Alpha-1D adrenergic receptor//Alpha1-adrenergic receptor activity
Amphetamine//Alpha-2A adrenergic receptor//Thioesterase binding
Amphetamine//Alpha-2B adrenergic receptor//Epinephrine binding
Amphetamine//Alpha-2C adrenergic receptor//Protein homodimerization activity
Amphetamine//Beta-1 adrenergic receptor//Receptor signaling protein activity
Amphetamine//Beta-2 adrenergic receptor//Protein homodimerization activity
Amphetamine//Beta-3 adrenergic receptor//Protein homodimerization activity
Amphetamine//D(2) dopamine receptor//Potassium channel regulator activity
Amphetamine//Amine oxidase [flavin-containing] B//Primary amine oxidase activity
Amphetamine//Sodium-dependent serotonin transporter//Serotonin:sodium symporter activity
Amphetamine//Amine oxidase [flavin-containing] A//Serotonin binding
Amphetamine//Amine oxidase [flavin-containing] B//Primary amine oxidase activity
Cevimeline//Muscarinic acetylcholine receptor M3//Receptor activity
Cevimeline//Muscarinic acetylcholine receptor M1//Phosphatidylinositol phospholipase c activity
Lorazepam//Gamma-aminobutyric acid receptor subunit alpha-1//Inhibitory extracellular ligand-gated ion channel activity
Lorazepam//Gamma-aminobutyric acid receptor subunit alpha-2//Inhibitory extracellular ligand-gated ion channel activity
Lorazepam//Gamma-aminobutyric acid receptor subunit alpha-3//Inhibitory extracellular ligand-gated ion channel activity
Lorazepam//Gamma-aminobutyric acid receptor subunit alpha-4//Inhibitory extracellular ligand-gated ion channel activity
Lorazepam//Gamma-aminobutyric acid receptor subunit alpha-5//Transporter activity
Lorazepam//Gamma-aminobutyric acid receptor subunit alpha-6//Inhibitory extracellular ligand-gated ion channel activity
Lorazepam//Gamma-aminobutyric acid receptor subunit beta-1//Ligand-gated ion channel activity
Lorazepam//Gamma-aminobutyric acid receptor subunit beta-2//Inhibitory extracellular ligand-gated ion channel activity
Lorazepam//Gamma-aminobutyric acid receptor subunit beta-3//Gaba-gated chloride ion channel activity
Lorazepam//Gamma-aminobutyric acid receptor subunit delta//Gaba-a receptor activity
Lorazepam//Gamma-aminobutyric acid receptor subunit epsilon//Inhibitory extracellular ligand-gated ion channel activity
Lorazepam//Gamma-aminobutyric acid receptor subunit gamma-1//Inhibitory extracellular ligand-gated ion channel activity
Lorazepam//Gamma-aminobutyric acid receptor subunit gamma-2//Inhibitory extracellular ligand-gated ion channel activity
Lorazepam//Gamma-aminobutyric acid receptor subunit gamma-3//Inhibitory extracellular ligand-gated ion channel activity
Lorazepam//Gamma-aminobutyric acid receptor subunit pi//Gaba-a receptor activity
Lorazepam//Gamma-aminobutyric acid receptor subunit theta//Transmembrane signaling receptor activity
Lorazepam//Gamma-aminobutyric acid receptor subunit alpha-1//Inhibitory extracellular ligand-gated ion channel activity
Lorazepam//Gamma-aminobutyric acid receptor subunit alpha-2//Inhibitory extracellular ligand-gated ion channel activity
Lorazepam//Gamma-aminobutyric acid receptor subunit alpha-3//Inhibitory extracellular ligand-gated ion channel activity
Lorazepam//Gamma-aminobutyric acid receptor subunit alpha-5//Transporter activity
Lorazepam//Gamma-aminobutyric acid receptor subunit gamma-1//Inhibitory extracellular ligand-gated ion channel activity
Lorazepam//Gamma-aminobutyric acid receptor subunit gamma-2//Inhibitory extracellular ligand-gated ion channel activity
Lorazepam//Gamma-aminobutyric acid receptor subunit gamma-3//Inhibitory extracellular ligand-gated ion channel activity
Betaxolol//Beta-1 adrenergic receptor//Receptor signaling protein activity
Betaxolol//Beta-2 adrenergic receptor//Protein homodimerization activity
Erythromycin//Potassium voltage-gated channel subfamily H member 2//Voltage-gated potassium channel activity involved in ventricular cardiac muscle cell action potential repolarization
Caffeine//Adenosine receptor A1//Purine nucleoside binding
Caffeine//cAMP-specific 3',5'-cyclic phosphodiesterase 4B//Metal ion binding
Caffeine//Ryanodine receptor 1//Voltage-gated calcium channel activity
Caffeine//Adenosine receptor A2a//Identical protein binding
Caffeine//Calcium/calmodulin-dependent 3',5'-cyclic nucleotide phosphodiesterase 1A//Metal ion binding
Caffeine//Calcium/calmodulin-dependent 3',5'-cyclic nucleotide phosphodiesterase 1B//Metal ion binding
Caffeine//cAMP and cAMP-inhibited cGMP 3',5'-cyclic phosphodiesterase 10A//Metal ion binding
Caffeine//cAMP-specific 3',5'-cyclic phosphodiesterase 4A//Metal ion binding
Caffeine//cAMP-specific 3',5'-cyclic phosphodiesterase 4B//Metal ion binding
Caffeine//cAMP-specific 3',5'-cyclic phosphodiesterase 4C//Metal ion binding
Caffeine//cAMP-specific 3',5'-cyclic phosphodiesterase 4D//Ubiquitin protein ligase binding
Caffeine//cAMP-specific 3',5'-cyclic phosphodiesterase 7B//Metal ion binding
Caffeine//cGMP-inhibited 3',5'-cyclic phosphodiesterase A//Metal ion binding
Caffeine//cGMP-specific 3',5'-cyclic phosphodiesterase//Metal ion binding
Caffeine//Dual 3',5'-cyclic-AMP and -GMP phosphodiesterase 11A//Metal ion binding
Caffeine//High affinity cAMP-specific 3',5'-cyclic phosphodiesterase 7A//Metal ion binding
Caffeine//High affinity cAMP-specific and IBMX-insensitive 3',5'-cyclic phosphodiesterase 8A//Metal ion binding
Caffeine//High affinity cGMP-specific 3',5'-cyclic phosphodiesterase 9A//Metal ion binding
Caffeine//DNA-dependent protein kinase catalytic subunit//Transcription factor binding
Caffeine//Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform//Phosphatidylinositol-4,5-bisphosphate 3-kinase activity
Caffeine//Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform//Protein serine/threonine kinase activity
Caffeine//Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoform//Phosphatidylinositol-4,5-bisphosphate 3-kinase activity
Caffeine//Serine-protein kinase ATM//Protein serine/threonine kinase activity
Caffeine//Adenosine receptor A2b//G-protein coupled adenosine receptor activity
Caffeine//Adenosine receptor A3//G-protein coupled adenosine receptor activity
Caffeine//Calcium/calmodulin-dependent 3',5'-cyclic nucleotide phosphodiesterase 1B//Metal ion binding
Caffeine//cAMP-specific 3',5'-cyclic phosphodiesterase 4D//Ubiquitin protein ligase binding
Caffeine//cGMP-specific 3',5'-cyclic phosphodiesterase//Metal ion binding
Dofetilide//Potassium voltage-gated channel subfamily H member 2//Voltage-gated potassium channel activity involved in ventricular cardiac muscle cell action potential repolarization
Dofetilide//ATP-sensitive inward rectifier potassium channel 12//Inward rectifier potassium channel activity
Midodrine//Alpha-1A adrenergic receptor//Protein heterodimerization activity
Midodrine//Alpha-1B adrenergic receptor//Protein heterodimerization activity
Midodrine//Alpha-1D adrenergic receptor//Alpha1-adrenergic receptor activity
Citalopram//Sodium-dependent serotonin transporter//Serotonin:sodium symporter activity
Citalopram//Histamine H1 receptor//Histamine receptor activity
Eletriptan//5-hydroxytryptamine receptor 1D//Serotonin receptor activity
Eletriptan//5-hydroxytryptamine receptor 1B//Serotonin receptor activity
Eletriptan//5-hydroxytryptamine receptor 1F//Serotonin receptor activity
Eletriptan//5-hydroxytryptamine receptor 1A//Serotonin receptor activity
Glimepiride//ATP-sensitive inward rectifier potassium channel 11//Voltage-gated potassium channel activity
Glimepiride//ATP-sensitive inward rectifier potassium channel 1//Phosphatidylinositol-4,5-bisphosphate binding
Glimepiride//ATP-binding cassette sub-family C member 8//Sulfonylurea receptor activity
Lovastatin//3-hydroxy-3-methylglutaryl-coenzyme A reductase//Nadph binding
Lovastatin//Integrin alpha-L//Metal ion binding
Lovastatin//Histone deacetylase 2//Transcription factor binding
Enflurane//Gamma-aminobutyric acid receptor subunit alpha-1//Inhibitory extracellular ligand-gated ion channel activity
Enflurane//Gamma-aminobutyric acid receptor subunit alpha-2//Inhibitory extracellular ligand-gated ion channel activity
Enflurane//Gamma-aminobutyric acid receptor subunit alpha-3//Inhibitory extracellular ligand-gated ion channel activity
Enflurane//Gamma-aminobutyric acid receptor subunit alpha-4//Inhibitory extracellular ligand-gated ion channel activity
Enflurane//Gamma-aminobutyric acid receptor subunit alpha-5//Transporter activity
Enflurane//Gamma-aminobutyric acid receptor subunit alpha-6//Inhibitory extracellular ligand-gated ion channel activity
Enflurane//Gamma-aminobutyric acid receptor subunit beta-1//Ligand-gated ion channel activity
Enflurane//Gamma-aminobutyric acid receptor subunit beta-2//Inhibitory extracellular ligand-gated ion channel activity
Enflurane//Gamma-aminobutyric acid receptor subunit beta-3//Gaba-gated chloride ion channel activity
Enflurane//Gamma-aminobutyric acid receptor subunit delta//Gaba-a receptor activity
Enflurane//Gamma-aminobutyric acid receptor subunit epsilon//Inhibitory extracellular ligand-gated ion channel activity
Enflurane//Gamma-aminobutyric acid receptor subunit gamma-1//Inhibitory extracellular ligand-gated ion channel activity
Enflurane//Gamma-aminobutyric acid receptor subunit gamma-2//Inhibitory extracellular ligand-gated ion channel activity
Enflurane//Gamma-aminobutyric acid receptor subunit gamma-3//Inhibitory extracellular ligand-gated ion channel activity
Enflurane//Gamma-aminobutyric acid receptor subunit pi//Gaba-a receptor activity
Enflurane//Gamma-aminobutyric acid receptor subunit theta//Transmembrane signaling receptor activity
Enflurane//Potassium voltage-gated channel subfamily A member 1//Voltage-gated potassium channel activity
Enflurane//Potassium voltage-gated channel subfamily A member 10//Intracellular cyclic nucleotide activated cation channel activity
Enflurane//Potassium voltage-gated channel subfamily A member 2//Voltage-gated potassium channel activity
Enflurane//Potassium voltage-gated channel subfamily A member 3//Voltage-gated ion channel activity
Enflurane//Potassium voltage-gated channel subfamily A member 4//Voltage-gated potassium channel activity
Enflurane//Potassium voltage-gated channel subfamily A member 5//Voltage-gated potassium channel activity involved in sa node cell action potential repolarization
Enflurane//Potassium voltage-gated channel subfamily A member 6//Voltage-gated potassium channel activity
Enflurane//Potassium voltage-gated channel subfamily B member 1//Ubiquitin-like protein binding
Enflurane//Potassium voltage-gated channel subfamily B member 2//Protein heterodimerization activity
Enflurane//Potassium voltage-gated channel subfamily C member 1//Voltage-gated potassium channel activity
Enflurane//Potassium voltage-gated channel subfamily C member 2//Voltage-gated potassium channel activity
Enflurane//Potassium voltage-gated channel subfamily C member 3//Voltage-gated potassium channel activity
Enflurane//Potassium voltage-gated channel subfamily C member 4//Voltage-gated potassium channel activity
Enflurane//Potassium voltage-gated channel subfamily D member 1//Metal ion binding
Enflurane//Potassium voltage-gated channel subfamily D member 2//Voltage-gated potassium channel activity
Enflurane//Potassium voltage-gated channel subfamily D member 3//Metal ion binding
Enflurane//Potassium voltage-gated channel subfamily G member 1//Potassium channel subunit that does not form functional channels by itself. Can form functional heterotetrameric channels with KCNB1; modulates the delayed rectifier voltage-gated potassium channel activation and deactivation rates of KCNB1 (PubMed:19074135).
Enflurane//Potassium voltage-gated channel subfamily G member 2//Potassium channel subunit. Modulates channel activity by shifting the threshold and the half-maximal activation to more negative values.
Enflurane//Potassium voltage-gated channel subfamily G member 4//Potassium channel subunit that does not form functional channels by itself. Can form functional heterotetrameric channels with KCNB1; modulates the delayed rectifier voltage-gated potassium channel activation and deactivation rates of KCNB1 (PubMed:19074135).
Enflurane//Potassium voltage-gated channel subfamily H member 1//Phosphorelay sensor kinase activity
Enflurane//Potassium voltage-gated channel subfamily H member 2//Voltage-gated potassium channel activity involved in ventricular cardiac muscle cell action potential repolarization
Enflurane//Potassium voltage-gated channel subfamily H member 6//Voltage-gated potassium channel activity
Enflurane//Potassium voltage-gated channel subfamily H member 7//Voltage-gated potassium channel activity
Enflurane//Potassium voltage-gated channel subfamily KQT member 1//Voltage-gated potassium channel activity involved in ventricular cardiac muscle cell action potential repolarization
Enflurane//Potassium voltage-gated channel subfamily KQT member 2//Voltage-gated potassium channel activity
Enflurane//Potassium voltage-gated channel subfamily KQT member 3//Voltage-gated potassium channel activity
Enflurane//Potassium voltage-gated channel subfamily KQT member 4//Potassium channel activity
Enflurane//Potassium voltage-gated channel subfamily KQT member 5//Voltage-gated potassium channel activity
Enflurane//Potassium voltage-gated channel subfamily V member 2//Potassium channel subunit. Modulates channel activity by shifting the threshold and the half-maximal activation to more negative values.
Enflurane//Calcium-transporting ATPase type 2C member 1//Signal transducer activity
Enflurane//Sarcoplasmic/endoplasmic reticulum calcium ATPase 1//Protein homodimerization activity
Enflurane//Glutamate receptor ionotropic, NMDA 1//Voltage-gated cation channel activity
Enflurane//Glutamate receptor ionotropic, NMDA 2A//Zinc ion binding
Enflurane//Glutamate receptor ionotropic, NMDA 2B//Zinc ion binding
Enflurane//Glutamate receptor ionotropic, NMDA 2C//Nmda glutamate receptor activity
Enflurane//Glutamate receptor ionotropic, NMDA 2D//Nmda glutamate receptor activity
Enflurane//Glutamate receptor ionotropic, NMDA 3A//Protein phosphatase 2a binding
Enflurane//Glutamate receptor ionotropic, NMDA 3B//Nmda glutamate receptor activity
Enflurane//Voltage-dependent calcium channel gamma-1 subunit//Voltage-gated calcium channel activity
Enflurane//Voltage-dependent calcium channel gamma-2 subunit//Voltage-gated calcium channel activity
Enflurane//Voltage-dependent calcium channel gamma-3 subunit//Regulates the trafficking to the somatodendritic compartment and gating properties of AMPA-selective glutamate receptors (AMPARs). Promotes their targeting to the cell membrane and synapses and modulates their gating properties by slowing their rates of activation, deactivation and desensitization. Does not show subunit-specific AMPA receptor regulation and regulates all AMPAR subunits. Thought to stabilize the calcium channel in an inactivated (closed) state.
Enflurane//Voltage-dependent calcium channel gamma-4 subunit//Regulates the trafficking and gating properties of AMPA-selective glutamate receptors (AMPARs). Promotes their targeting to the cell membrane and synapses and modulates their gating properties by slowing their rates of activation, deactivation and desensitization and by mediating their resensitization. Does not show subunit-specific AMPA receptor regulation and regulates all AMPAR subunits. Thought to stabilize the calcium channel in an inactivated (closed) state.
Enflurane//Voltage-dependent calcium channel gamma-5 subunit//Regulates the gating properties of AMPA-selective glutamate receptors (AMPARs). Modulates their gating properties by accelerating their rates of activation, deactivation and desensitization. Displays subunit-specific AMPA receptor regulation. Shows specificity for GRIA1, GRIA4 and the long isoform of GRIA2. Thought to stabilize the calcium channel in an inactivated (closed) state (By similarity).
Enflurane//Voltage-dependent calcium channel gamma-6 subunit//Thought to stabilize the calcium channel in an inactivated (closed) state.
Enflurane//Voltage-dependent calcium channel gamma-7 subunit//Regulates the trafficking and gating properties of AMPA-selective glutamate receptors (AMPARs). Promotes their targeting to the cell membrane and synapses and modulates their gating properties by slowing their rates of activation, deactivation and desensitization and by mediating their resensitization. Displays subunit-specific AMPA receptor regulation. Shows specificity only for GRIA1 and GRIA2. Thought to stabilize the calcium channel in an inactivated (closed) state.
Enflurane//Voltage-dependent calcium channel gamma-8 subunit//Regulates the trafficking and gating properties of AMPA-selective glutamate receptors (AMPARs). Promotes their targeting to the cell membrane and synapses and modulates their gating properties by slowing their rates of activation, deactivation and desensitization and by mediating their resensitization. Does not show subunit-specific AMPA receptor regulation and regulates all AMPAR subunits. Thought to stabilize the calcium channel in an inactivated (closed) state.
Enflurane//Voltage-dependent calcium channel subunit alpha-2/delta-1//Voltage-gated calcium channel activity
Enflurane//Voltage-dependent calcium channel subunit alpha-2/delta-2//Voltage-gated calcium channel activity
Enflurane//Voltage-dependent calcium channel subunit alpha-2/delta-3//Voltage-gated ion channel activity
Enflurane//Voltage-dependent calcium channel subunit alpha-2/delta-4//The alpha-2/delta subunit of voltage-dependent calcium channels regulates calcium current density and activation/inactivation kinetics of the calcium channel.
Enflurane//Voltage-dependent L-type calcium channel subunit alpha-1C//Voltage-gated calcium channel activity
Enflurane//Voltage-dependent L-type calcium channel subunit alpha-1D//Voltage-gated calcium channel activity involved sa node cell action potential
Enflurane//Voltage-dependent L-type calcium channel subunit alpha-1F//Voltage-gated calcium channel activity
Enflurane//Voltage-dependent L-type calcium channel subunit alpha-1S//Voltage-gated calcium channel activity
Enflurane//Voltage-dependent L-type calcium channel subunit beta-1//Voltage-gated calcium channel activity
Enflurane//Voltage-dependent L-type calcium channel subunit beta-2//Voltage-gated calcium channel activity
Enflurane//Voltage-dependent L-type calcium channel subunit beta-3//Voltage-gated calcium channel activity
Enflurane//Voltage-dependent L-type calcium channel subunit beta-4//Voltage-gated calcium channel activity
Enflurane//Voltage-dependent N-type calcium channel subunit alpha-1B//Voltage-gated calcium channel activity
Enflurane//Voltage-dependent P/Q-type calcium channel subunit alpha-1A//Voltage-gated calcium channel activity
Enflurane//Voltage-dependent R-type calcium channel subunit alpha-1E//Voltage-sensitive calcium channels (VSCC) mediate the entry of calcium ions into excitable cells and are also involved in a variety of calcium-dependent processes, including muscle contraction, hormone or neurotransmitter release, gene expression, cell motility, cell division and cell death. The isoform alpha-1E gives rise to R-type calcium currents. R-type calcium channels belong to the 'high-voltage activated' (HVA) group and are blocked by nickel, and partially by omega-agatoxin-IIIA (omega-Aga-IIIA). They are however insensitive to dihydropyridines (DHP), omega-conotoxin-GVIA (omega-CTx-GVIA), and omega-agatoxin-IVA (omega-Aga-IVA). Calcium channels containing alpha-1E subunit could be involved in the modulation of firing patterns of neurons which is important for information processing.
Enflurane//Voltage-dependent T-type calcium channel subunit alpha-1G//Scaffold protein binding
Enflurane//Voltage-dependent T-type calcium channel subunit alpha-1H//Scaffold protein binding
Enflurane//Voltage-dependent T-type calcium channel subunit alpha-1I//Voltage-gated calcium channel activity
Enflurane//Glycine receptor subunit alpha-1//Transmitter-gated ion channel activity
Aminosalicylicacid//Prostaglandin G/H synthase 2//Prostaglandin-endoperoxide synthase activity
Aminosalicylicacid//Inhibitor of nuclear factor kappa-B kinase subunit alpha//Scaffold protein binding
Aminosalicylicacid//Arachidonate 5-lipoxygenase//Iron ion binding
Aminosalicylicacid//Group IIE secretory phospholipase A2//Phospholipase a2 activity
Alclometasone//Glucocorticoid receptor//Zinc ion binding
Cladribine//Ribonucleoside-diphosphate reductase large subunit//Ribonucleoside-diphosphate reductase activity, thioredoxin disulfide as acceptor
Cladribine//Ribonucleoside-diphosphate reductase subunit M2//Ribonucleoside-diphosphate reductase activity, thioredoxin disulfide as acceptor
Cladribine//Ribonucleoside-diphosphate reductase subunit M2 B//Ribonucleoside-diphosphate reductase activity, thioredoxin disulfide as acceptor
Cladribine//DNA polymerase alpha catalytic subunit//Protein kinase binding
Cladribine//DNA polymerase epsilon catalytic subunit A//Zinc ion binding
Cladribine//DNA polymerase epsilon subunit 2//Dna-directed dna polymerase activity
Cladribine//DNA polymerase epsilon subunit 3//Dna-directed dna polymerase activity
Cladribine//DNA polymerase epsilon subunit 4//Dna-directed dna polymerase activity
Benzatropine//Muscarinic acetylcholine receptor M1//Phosphatidylinositol phospholipase c activity
Benzatropine//Sodium-dependent dopamine transporter//Monoamine transmembrane transporter activity
Benzatropine//Histamine H1 receptor//Histamine receptor activity
Benzatropine//Sodium-dependent serotonin transporter//Serotonin:sodium symporter activity
Benzatropine//Sodium-dependent noradrenaline transporter//Norepinephrine:sodium symporter activity
Cabergoline//D(2) dopamine receptor//Potassium channel regulator activity
Cabergoline//5-hydroxytryptamine receptor 2B//Serotonin receptor activity
Cabergoline//D(3) dopamine receptor//G-protein coupled amine receptor activity
Cabergoline//5-hydroxytryptamine receptor 2A//Virus receptor activity
Cabergoline//Alpha-2B adrenergic receptor//Epinephrine binding
Cabergoline//5-hydroxytryptamine receptor 1D//Serotonin receptor activity
Cabergoline//D(4) dopamine receptor//Sh3 domain binding
Cabergoline//Alpha-2A adrenergic receptor//Thioesterase binding
Cabergoline//5-hydroxytryptamine receptor 1A//Serotonin receptor activity
Cabergoline//Alpha-2C adrenergic receptor//Protein homodimerization activity
Cabergoline//D(1B) dopamine receptor//G-protein coupled amine receptor activity
Cabergoline//D(1A) dopamine receptor//G-protein coupled amine receptor activity
Cabergoline//5-hydroxytryptamine receptor 1B//Serotonin receptor activity
Cabergoline//5-hydroxytryptamine receptor 2C//Serotonin receptor activity
Cabergoline//5-hydroxytryptamine receptor 7//Serotonin receptor activity
Cabergoline//Alpha-1A adrenergic receptor//Protein heterodimerization activity
Cabergoline//Alpha-1B adrenergic receptor//Protein heterodimerization activity
Cabergoline//Alpha-1D adrenergic receptor//Alpha1-adrenergic receptor activity
Cabergoline//Beta-1 adrenergic receptor//Receptor signaling protein activity
Cabergoline//Beta-2 adrenergic receptor//Protein homodimerization activity
Cabergoline//D(1A) dopamine receptor//G-protein coupled amine receptor activity
Cabergoline//D(1B) dopamine receptor//G-protein coupled amine receptor activity
Diethylstilbestrol//Estrogen receptor//Zinc ion binding
Diethylstilbestrol//Estrogen-related receptor gamma//Zinc ion binding
Diethylstilbestrol//Estrogen receptor beta//Zinc ion binding
Diethylstilbestrol//Steroid hormone receptor ERR1//Zinc ion binding
Diethylstilbestrol//Steroid hormone receptor ERR2//Zinc ion binding
Diethylstilbestrol//Nuclear receptor coactivator 2//Transcription coactivator activity
Diethylstilbestrol//Nuclear receptor subfamily 1 group I member 2//Zinc ion binding
Diethylstilbestrol//Androgen receptor//Zinc ion binding
Diethylstilbestrol//Sex hormone-binding globulin//Androgen binding
Clotrimazole//Lanosterol 14-alpha demethylase//Sterol 14-demethylase activity
Clotrimazole//Intermediate conductance calcium-activated potassium channel protein 4//Protein phosphatase binding
Clotrimazole//Nuclear receptor subfamily 1 group I member 2//Zinc ion binding
Anagrelide//cGMP-inhibited 3',5'-cyclic phosphodiesterase A//Metal ion binding
Carmustine//Glutathione reductase, mitochondrial//Nadp binding
Metoprolol//Beta-1 adrenergic receptor//Receptor signaling protein activity
Metoprolol//Beta-2 adrenergic receptor//Protein homodimerization activity
Dicoumarol//Vitamin K epoxide reductase complex subunit 1//Vitamin-k-epoxide reductase (warfarin-sensitive) activity
Dicoumarol//NAD(P)H dehydrogenase [quinone] 1//Superoxide dismutase activity
Dicoumarol//Quinone oxidoreductase//Zinc ion binding
Isradipine//Voltage-dependent L-type calcium channel subunit alpha-1C//Voltage-gated calcium channel activity
Isradipine//Voltage-dependent calcium channel subunit alpha-2/delta-1//Voltage-gated calcium channel activity
Isradipine//Voltage-dependent L-type calcium channel subunit beta-2//Voltage-gated calcium channel activity
Isradipine//Voltage-dependent T-type calcium channel subunit alpha-1H//Scaffold protein binding
Isradipine//Voltage-dependent calcium channel subunit alpha-2/delta-2//Voltage-gated calcium channel activity
Isradipine//Voltage-dependent L-type calcium channel subunit alpha-1D//Voltage-gated calcium channel activity involved sa node cell action potential
Isradipine//Voltage-dependent L-type calcium channel subunit alpha-1S//Voltage-gated calcium channel activity
Amsacrine//DNA topoisomerase 2-alpha//Ubiquitin binding
Amsacrine//Potassium voltage-gated channel subfamily H member 2//Voltage-gated potassium channel activity involved in ventricular cardiac muscle cell action potential repolarization
Amsacrine//Serum albumin//Toxic substance binding
Argatroban//Prothrombin//Thrombospondin receptor activity
Disopyramide//Sodium channel protein type 5 subunit alpha//Voltage-gated sodium channel activity involved in sa node cell action potential
Disopyramide//Muscarinic acetylcholine receptor M1//Phosphatidylinositol phospholipase c activity
Disopyramide//Muscarinic acetylcholine receptor M2//G-protein coupled acetylcholine receptor activity
Disopyramide//Muscarinic acetylcholine receptor M3//Receptor activity
Disopyramide//Potassium voltage-gated channel subfamily D member 2//Voltage-gated potassium channel activity
Disopyramide//Potassium voltage-gated channel subfamily D member 3//Metal ion binding
Disopyramide//Potassium voltage-gated channel subfamily H member 2//Voltage-gated potassium channel activity involved in ventricular cardiac muscle cell action potential repolarization
Lidocaine//Sodium channel protein type 10 subunit alpha//Voltage-gated sodium channel activity
Lidocaine//Sodium channel protein type 9 subunit alpha//Voltage-gated sodium channel activity
Lidocaine//Sodium channel protein type 5 subunit alpha//Voltage-gated sodium channel activity involved in sa node cell action potential
Lidocaine//Epidermal growth factor receptor//Ubiquitin protein ligase binding
Lidocaine//Sodium channel protein type 4 subunit alpha//Voltage-gated sodium channel activity
Clemastine//Histamine H1 receptor//Histamine receptor activity
Atomoxetine//Sodium-dependent noradrenaline transporter//Norepinephrine:sodium symporter activity
Atomoxetine//Sodium-dependent serotonin transporter//Serotonin:sodium symporter activity
Atomoxetine//Glutamate receptor ionotropic, NMDA 1//Voltage-gated cation channel activity
Atomoxetine//Glutamate receptor ionotropic, NMDA 2A//Zinc ion binding
Atomoxetine//Glutamate receptor ionotropic, NMDA 2B//Zinc ion binding
Atomoxetine//Glutamate receptor ionotropic, NMDA 2C//Nmda glutamate receptor activity
Atomoxetine//Glutamate receptor ionotropic, NMDA 2D//Nmda glutamate receptor activity
Atomoxetine//Glutamate receptor ionotropic, NMDA 3A//Protein phosphatase 2a binding
Atomoxetine//Glutamate receptor ionotropic, NMDA 3B//Nmda glutamate receptor activity
Atomoxetine//G protein-activated inward rectifier potassium channel 1//G-protein activated inward rectifier potassium channel activity
Atomoxetine//Kappa-type opioid receptor//Opioid receptor activity
Bleomycin//DNA ligase 1//Metal ion binding
Bleomycin//DNA ligase 3//Zinc ion binding
Etomidate//Gamma-aminobutyric acid receptor subunit alpha-1//Inhibitory extracellular ligand-gated ion channel activity
Etomidate//Alpha-2B adrenergic receptor//Epinephrine binding
Etomidate//Gamma-aminobutyric acid receptor subunit alpha-1//Inhibitory extracellular ligand-gated ion channel activity
Etomidate//Gamma-aminobutyric acid receptor subunit alpha-2//Inhibitory extracellular ligand-gated ion channel activity
Etomidate//Gamma-aminobutyric acid receptor subunit alpha-3//Inhibitory extracellular ligand-gated ion channel activity
Etomidate//Gamma-aminobutyric acid receptor subunit alpha-4//Inhibitory extracellular ligand-gated ion channel activity
Etomidate//Gamma-aminobutyric acid receptor subunit alpha-5//Transporter activity
Etomidate//Gamma-aminobutyric acid receptor subunit alpha-6//Inhibitory extracellular ligand-gated ion channel activity
Etomidate//Gamma-aminobutyric acid receptor subunit beta-1//Ligand-gated ion channel activity
Etomidate//Gamma-aminobutyric acid receptor subunit beta-2//Inhibitory extracellular ligand-gated ion channel activity
Etomidate//Gamma-aminobutyric acid receptor subunit beta-3//Gaba-gated chloride ion channel activity
Etomidate//Gamma-aminobutyric acid receptor subunit delta//Gaba-a receptor activity
Etomidate//Gamma-aminobutyric acid receptor subunit epsilon//Inhibitory extracellular ligand-gated ion channel activity
Etomidate//Gamma-aminobutyric acid receptor subunit gamma-1//Inhibitory extracellular ligand-gated ion channel activity
Etomidate//Gamma-aminobutyric acid receptor subunit gamma-2//Inhibitory extracellular ligand-gated ion channel activity
Etomidate//Gamma-aminobutyric acid receptor subunit gamma-3//Inhibitory extracellular ligand-gated ion channel activity
Etomidate//Gamma-aminobutyric acid receptor subunit pi//Gaba-a receptor activity
Etomidate//Gamma-aminobutyric acid receptor subunit theta//Transmembrane signaling receptor activity
Etonogestrel//Progesterone receptor//Zinc ion binding
Morphine//Mu-type opioid receptor//Voltage-gated calcium channel activity
Morphine//Kappa-type opioid receptor//Opioid receptor activity
Morphine//Delta-type opioid receptor//Opioid receptor activity
Bupivacaine//Sodium channel protein type 10 subunit alpha//Voltage-gated sodium channel activity
Bupivacaine//Prostaglandin E2 receptor EP1 subtype//Prostaglandin e receptor activity
Bexarotene//Retinoic acid receptor RXR-alpha//Zinc ion binding
Bexarotene//Retinoic acid receptor RXR-beta//Zinc ion binding
Bexarotene//Retinoic acid receptor RXR-gamma//Zinc ion binding
Acetaminophen//Prostaglandin G/H synthase 1//Prostaglandin-endoperoxide synthase activity
Acetaminophen//Prostaglandin G/H synthase 2//Prostaglandin-endoperoxide synthase activity
Acetaminophen//Prostaglandin E synthase 3//Unfolded protein binding
Acetaminophen//Transient receptor potential cation channel subfamily V member 1//Transmembrane signaling receptor activity
Gefitinib//Epidermal growth factor receptor//Ubiquitin protein ligase binding
Codeine//Mu-type opioid receptor//Voltage-gated calcium channel activity
Codeine//Kappa-type opioid receptor//Opioid receptor activity
Codeine//Delta-type opioid receptor//Opioid receptor activity
Dihydroergotamine//5-hydroxytryptamine receptor 1D//Serotonin receptor activity
Dihydroergotamine//5-hydroxytryptamine receptor 1B//Serotonin receptor activity
Dihydroergotamine//Alpha-2A adrenergic receptor//Thioesterase binding
Dihydroergotamine//5-hydroxytryptamine receptor 2B//Serotonin receptor activity
Amitriptyline//Sodium-dependent noradrenaline transporter//Norepinephrine:sodium symporter activity
Amitriptyline//Sodium-dependent serotonin transporter//Serotonin:sodium symporter activity
Amitriptyline//5-hydroxytryptamine receptor 2A//Virus receptor activity
Amitriptyline//5-hydroxytryptamine receptor 1A//Serotonin receptor activity
Amitriptyline//Delta-type opioid receptor//Opioid receptor activity
Amitriptyline//Kappa-type opioid receptor//Opioid receptor activity
Amitriptyline//High affinity nerve growth factor receptor//Transmembrane receptor protein tyrosine kinase activity
Amitriptyline//BDNF/NT-3 growth factors receptor//Protein homodimerization activity
Amitriptyline//Alpha-1A adrenergic receptor//Protein heterodimerization activity
Amitriptyline//Alpha-1D adrenergic receptor//Alpha1-adrenergic receptor activity
Amitriptyline//Alpha-2A adrenergic receptor//Thioesterase binding
Amitriptyline//Histamine H1 receptor//Histamine receptor activity
Amitriptyline//Potassium voltage-gated channel subfamily KQT member 2//Voltage-gated potassium channel activity
Amitriptyline//Potassium voltage-gated channel subfamily A member 1//Voltage-gated potassium channel activity
Amitriptyline//Histamine H2 receptor//Histamine receptor activity
Amitriptyline//Histamine H4 receptor//Histamine receptor activity
Amitriptyline//Sigma non-opioid intracellular receptor 1//Opioid receptor activity
Amitriptyline//5-hydroxytryptamine receptor 2C//Serotonin receptor activity
Amitriptyline//Alpha-1B adrenergic receptor//Protein heterodimerization activity
Amitriptyline//5-hydroxytryptamine receptor 7//Serotonin receptor activity
Amitriptyline//5-hydroxytryptamine receptor 1D//Serotonin receptor activity
Amitriptyline//Mu-type opioid receptor//Voltage-gated calcium channel activity
Amitriptyline//5-hydroxytryptamine receptor 1B//Serotonin receptor activity
Amitriptyline//5-hydroxytryptamine receptor 6//Serotonin receptor activity
Amitriptyline//Potassium voltage-gated channel subfamily KQT member 3//Voltage-gated potassium channel activity
Amitriptyline//5-hydroxytryptamine receptor 2C//Serotonin receptor activity
Amitriptyline//Muscarinic acetylcholine receptor M1//Phosphatidylinositol phospholipase c activity
Amitriptyline//Muscarinic acetylcholine receptor M2//G-protein coupled acetylcholine receptor activity
Amitriptyline//Muscarinic acetylcholine receptor M3//Receptor activity
Amitriptyline//Muscarinic acetylcholine receptor M4//Guanyl-nucleotide exchange factor activity
Amitriptyline//Muscarinic acetylcholine receptor M5//Phosphatidylinositol phospholipase c activity
Amitriptyline//Potassium voltage-gated channel subfamily H member 2//Voltage-gated potassium channel activity involved in ventricular cardiac muscle cell action potential repolarization
Amitriptyline//Potassium voltage-gated channel subfamily H member 6//Voltage-gated potassium channel activity
Amitriptyline//Potassium voltage-gated channel subfamily H member 7//Voltage-gated potassium channel activity
Floxuridine//Thymidylate synthase//Thymidylate synthase activity
Fluorometholone//Glucocorticoid receptor//Zinc ion binding
Hydromorphone//Mu-type opioid receptor//Voltage-gated calcium channel activity
Hydromorphone//Delta-type opioid receptor//Opioid receptor activity
Hydromorphone//Kappa-type opioid receptor//Opioid receptor activity
Indomethacin//Prostaglandin G/H synthase 1//Prostaglandin-endoperoxide synthase activity
Indomethacin//Prostaglandin G/H synthase 2//Prostaglandin-endoperoxide synthase activity
Indomethacin//Phospholipase A2, membrane associated//Phospholipid binding
Indomethacin//Peroxisome proliferator-activated receptor gamma//Zinc ion binding
Indomethacin//Lactoylglutathione lyase//Zinc ion binding
Indomethacin//Peroxisome proliferator-activated receptor alpha//Zinc ion binding
Indomethacin//Aldo-keto reductase family 1 member C3//Trans-1,2-dihydrobenzene-1,2-diol dehydrogenase activity
Ipratropiumbromide//Muscarinic acetylcholine receptor M1//Phosphatidylinositol phospholipase c activity
Ipratropiumbromide//Muscarinic acetylcholine receptor M2//G-protein coupled acetylcholine receptor activity
Ipratropiumbromide//Muscarinic acetylcholine receptor M3//Receptor activity
Methadone//Mu-type opioid receptor//Voltage-gated calcium channel activity
Methadone//Glutamate receptor ionotropic, NMDA 1//Voltage-gated cation channel activity
Methadone//Glutamate receptor ionotropic, NMDA 2A//Zinc ion binding
Methadone//Glutamate receptor ionotropic, NMDA 2B//Zinc ion binding
Methadone//Glutamate receptor ionotropic, NMDA 2C//Nmda glutamate receptor activity
Methadone//Glutamate receptor ionotropic, NMDA 2D//Nmda glutamate receptor activity
Methadone//Glutamate receptor ionotropic, NMDA 3A//Protein phosphatase 2a binding
Methadone//Glutamate receptor ionotropic, NMDA 3B//Nmda glutamate receptor activity
Methadone//Delta-type opioid receptor//Opioid receptor activity
Methadone//5-hydroxytryptamine receptor 3A//Voltage-gated potassium channel activity
Methadone//Neuronal acetylcholine receptor subunit alpha-7//Toxic substance binding
Methadone//Neuronal acetylcholine receptor subunit alpha-3//Ligand-gated ion channel activity
Methadone//Neuronal acetylcholine receptor subunit alpha-4//Ligand-gated ion channel activity
Methadone//Neuronal acetylcholine receptor subunit beta-2//Ligand-gated ion channel activity
Diltiazem//Voltage-dependent calcium channel gamma-1 subunit//Voltage-gated calcium channel activity
Diltiazem//Voltage-dependent L-type calcium channel subunit alpha-1C//Voltage-gated calcium channel activity
Alfuzosin//Alpha-1A adrenergic receptor//Protein heterodimerization activity
Alfuzosin//Alpha-1B adrenergic receptor//Protein heterodimerization activity
Alfuzosin//Alpha-1D adrenergic receptor//Alpha1-adrenergic receptor activity
Alfuzosin//Potassium voltage-gated channel subfamily H member 2//Voltage-gated potassium channel activity involved in ventricular cardiac muscle cell action potential repolarization
Methylergometrine//D(1A) dopamine receptor//G-protein coupled amine receptor activity
Methylergometrine//5-hydroxytryptamine receptor 2B//Serotonin receptor activity
Chlorzoxazone//Calcium-activated potassium channel subunit alpha-1//Voltage-gated potassium channel activity
Aminoglutethimide//Aromatase//Oxygen binding
Aminoglutethimide//Cholesterol side-chain cleavage enzyme, mitochondrial//Oxidoreductase activity, acting on paired donors, with incorporation or reduction of molecular oxygen, nad(p)h as one donor, and incorporation of one atom of oxygen
Mefloquine//Adenosine receptor A2a//Identical protein binding
Clozapine//D(2) dopamine receptor//Potassium channel regulator activity
Clozapine//5-hydroxytryptamine receptor 2A//Virus receptor activity
Clozapine//D(1A) dopamine receptor//G-protein coupled amine receptor activity
Clozapine//D(3) dopamine receptor//G-protein coupled amine receptor activity
Clozapine//D(4) dopamine receptor//Sh3 domain binding
Clozapine//5-hydroxytryptamine receptor 1A//Serotonin receptor activity
Clozapine//5-hydroxytryptamine receptor 1B//Serotonin receptor activity
Clozapine//5-hydroxytryptamine receptor 1D//Serotonin receptor activity
Clozapine//5-hydroxytryptamine receptor 1E//Serotonin receptor activity
Clozapine//5-hydroxytryptamine receptor 3A//Voltage-gated potassium channel activity
Clozapine//5-hydroxytryptamine receptor 2C//Serotonin receptor activity
Clozapine//5-hydroxytryptamine receptor 7//Serotonin receptor activity
Clozapine//5-hydroxytryptamine receptor 6//Serotonin receptor activity
Clozapine//Histamine H1 receptor//Histamine receptor activity
Clozapine//Histamine H4 receptor//Histamine receptor activity
Clozapine//Alpha-1A adrenergic receptor//Protein heterodimerization activity
Clozapine//Alpha-1B adrenergic receptor//Protein heterodimerization activity
Clozapine//Alpha-2A adrenergic receptor//Thioesterase binding
Clozapine//Alpha-2B adrenergic receptor//Epinephrine binding
Clozapine//Alpha-2C adrenergic receptor//Protein homodimerization activity
Clozapine//Muscarinic acetylcholine receptor M1//Phosphatidylinositol phospholipase c activity
Clozapine//Muscarinic acetylcholine receptor M2//G-protein coupled acetylcholine receptor activity
Clozapine//Muscarinic acetylcholine receptor M3//Receptor activity
Clozapine//Muscarinic acetylcholine receptor M4//Guanyl-nucleotide exchange factor activity
Clozapine//Muscarinic acetylcholine receptor M5//Phosphatidylinositol phospholipase c activity
Clozapine//Glutathione S-transferase P//S-nitrosoglutathione binding
Doxylamine//Histamine H1 receptor//Histamine receptor activity
Doxylamine//Muscarinic acetylcholine receptor M1//Phosphatidylinositol phospholipase c activity
Doxylamine//Muscarinic acetylcholine receptor M2//G-protein coupled acetylcholine receptor activity
Doxylamine//Muscarinic acetylcholine receptor M3//Receptor activity
Doxylamine//Muscarinic acetylcholine receptor M4//Guanyl-nucleotide exchange factor activity
Doxylamine//Muscarinic acetylcholine receptor M5//Phosphatidylinositol phospholipase c activity
Doxylamine//Nuclear receptor subfamily 1 group I member 3//Zinc ion binding
Levonorgestrel//Progesterone receptor//Zinc ion binding
Levonorgestrel//3-oxo-5-alpha-steroid 4-dehydrogenase 1//Electron carrier activity
Levonorgestrel//Estrogen receptor//Zinc ion binding
Levonorgestrel//Androgen receptor//Zinc ion binding
Levonorgestrel//Sex hormone-binding globulin//Androgen binding
Levonorgestrel//Glucocorticoid receptor//Zinc ion binding
Mirtazapine//Alpha-2A adrenergic receptor//Thioesterase binding
Mirtazapine//Histamine H1 receptor//Histamine receptor activity
Mirtazapine//5-hydroxytryptamine receptor 2A//Virus receptor activity
Mirtazapine//5-hydroxytryptamine receptor 2C//Serotonin receptor activity
Mirtazapine//Kappa-type opioid receptor//Opioid receptor activity
Mirtazapine//Alpha-1A adrenergic receptor//Protein heterodimerization activity
Mirtazapine//Alpha-1B adrenergic receptor//Protein heterodimerization activity
Mirtazapine//Alpha-1D adrenergic receptor//Alpha1-adrenergic receptor activity
Meprobamate//Gamma-aminobutyric acid receptor subunit alpha-2//Inhibitory extracellular ligand-gated ion channel activity
Meprobamate//Gamma-aminobutyric acid receptor subunit alpha-5//Transporter activity
Meprobamate//Gamma-aminobutyric acid receptor subunit alpha-4//Inhibitory extracellular ligand-gated ion channel activity
Meprobamate//Gamma-aminobutyric acid receptor subunit alpha-3//Inhibitory extracellular ligand-gated ion channel activity
Meprobamate//Gamma-aminobutyric acid receptor subunit alpha-6//Inhibitory extracellular ligand-gated ion channel activity
Meprobamate//Gamma-aminobutyric acid receptor subunit alpha-1//Inhibitory extracellular ligand-gated ion channel activity
Meprobamate//Gamma-aminobutyric acid receptor subunit alpha-1//Inhibitory extracellular ligand-gated ion channel activity
Meprobamate//Gamma-aminobutyric acid receptor subunit alpha-2//Inhibitory extracellular ligand-gated ion channel activity
Meprobamate//Gamma-aminobutyric acid receptor subunit alpha-3//Inhibitory extracellular ligand-gated ion channel activity
Meprobamate//Gamma-aminobutyric acid receptor subunit alpha-4//Inhibitory extracellular ligand-gated ion channel activity
Meprobamate//Gamma-aminobutyric acid receptor subunit alpha-5//Transporter activity
Meprobamate//Gamma-aminobutyric acid receptor subunit alpha-6//Inhibitory extracellular ligand-gated ion channel activity
Meprobamate//Gamma-aminobutyric acid receptor subunit beta-1//Ligand-gated ion channel activity
Meprobamate//Gamma-aminobutyric acid receptor subunit beta-2//Inhibitory extracellular ligand-gated ion channel activity
Meprobamate//Gamma-aminobutyric acid receptor subunit beta-3//Gaba-gated chloride ion channel activity
Meprobamate//Gamma-aminobutyric acid receptor subunit delta//Gaba-a receptor activity
Meprobamate//Gamma-aminobutyric acid receptor subunit epsilon//Inhibitory extracellular ligand-gated ion channel activity
Meprobamate//Gamma-aminobutyric acid receptor subunit gamma-1//Inhibitory extracellular ligand-gated ion channel activity
Meprobamate//Gamma-aminobutyric acid receptor subunit gamma-2//Inhibitory extracellular ligand-gated ion channel activity
Meprobamate//Gamma-aminobutyric acid receptor subunit gamma-3//Inhibitory extracellular ligand-gated ion channel activity
Meprobamate//Gamma-aminobutyric acid receptor subunit pi//Gaba-a receptor activity
Meprobamate//Gamma-aminobutyric acid receptor subunit theta//Transmembrane signaling receptor activity
Mexiletine//Sodium channel protein type 5 subunit alpha//Voltage-gated sodium channel activity involved in sa node cell action potential
Mexiletine//Aryl hydrocarbon receptor//Transcription regulatory region dna binding
Amlodipine//Voltage-dependent L-type calcium channel subunit alpha-1C//Voltage-gated calcium channel activity
Amlodipine//Voltage-dependent L-type calcium channel subunit beta-1//Voltage-gated calcium channel activity
Amlodipine//Voltage-dependent N-type calcium channel subunit alpha-1B//Voltage-gated calcium channel activity
Amlodipine//Voltage-dependent calcium channel subunit alpha-2/delta-3//Voltage-gated ion channel activity
Amlodipine//Carbonic anhydrase 1//Zinc ion binding
Amlodipine//Sphingomyelin phosphodiesterase//Sphingomyelin phosphodiesterase activity
Amlodipine//Voltage-dependent T-type calcium channel subunit alpha-1I//Voltage-gated calcium channel activity
Amlodipine//Voltage-dependent N-type calcium channel subunit alpha-1B//Voltage-gated calcium channel activity
Carbimazole//Thyroid peroxidase//Peroxidase activity
Digoxin//Sodium/potassium-transporting ATPase subunit alpha-1//Steroid hormone binding
Ethopropazine//Muscarinic acetylcholine receptor M1//Phosphatidylinositol phospholipase c activity
Ethopropazine//Glutamate receptor ionotropic, NMDA 3A//Protein phosphatase 2a binding
Ethopropazine//Muscarinic acetylcholine receptor M2//G-protein coupled acetylcholine receptor activity
Beclomethasonedipropionate//Glucocorticoid receptor//Zinc ion binding
Carisoprodol//Gamma-aminobutyric acid receptor subunit alpha-1//Inhibitory extracellular ligand-gated ion channel activity
Carisoprodol//Gamma-aminobutyric acid receptor subunit beta-2//Inhibitory extracellular ligand-gated ion channel activity
Carisoprodol//Gamma-aminobutyric acid receptor subunit gamma-2//Inhibitory extracellular ligand-gated ion channel activity
Carisoprodol//Gamma-aminobutyric acid receptor subunit alpha-5//Transporter activity
Carisoprodol//Gamma-aminobutyric acid receptor subunit alpha-3//Inhibitory extracellular ligand-gated ion channel activity
Griseofulvin//Tubulin beta chain//Ubiquitin protein ligase binding
Griseofulvin//Keratin, type I cytoskeletal 12//Structural molecule activity
Eszopiclone//Gamma-aminobutyric acid receptor subunit alpha-1//Inhibitory extracellular ligand-gated ion channel activity
Eszopiclone//Gamma-aminobutyric acid receptor subunit alpha-2//Inhibitory extracellular ligand-gated ion channel activity
Eszopiclone//Gamma-aminobutyric acid receptor subunit alpha-5//Transporter activity
Eszopiclone//Gamma-aminobutyric acid receptor subunit alpha-3//Inhibitory extracellular ligand-gated ion channel activity
Eszopiclone//Gamma-aminobutyric acid receptor subunit alpha-1//Inhibitory extracellular ligand-gated ion channel activity
Eszopiclone//Gamma-aminobutyric acid receptor subunit alpha-2//Inhibitory extracellular ligand-gated ion channel activity
Eszopiclone//Gamma-aminobutyric acid receptor subunit alpha-3//Inhibitory extracellular ligand-gated ion channel activity
Eszopiclone//Gamma-aminobutyric acid receptor subunit alpha-4//Inhibitory extracellular ligand-gated ion channel activity
Eszopiclone//Gamma-aminobutyric acid receptor subunit alpha-5//Transporter activity
Eszopiclone//Gamma-aminobutyric acid receptor subunit alpha-6//Inhibitory extracellular ligand-gated ion channel activity
Eszopiclone//Gamma-aminobutyric acid receptor subunit beta-1//Ligand-gated ion channel activity
Eszopiclone//Gamma-aminobutyric acid receptor subunit beta-2//Inhibitory extracellular ligand-gated ion channel activity
Eszopiclone//Gamma-aminobutyric acid receptor subunit beta-3//Gaba-gated chloride ion channel activity
Eszopiclone//Gamma-aminobutyric acid receptor subunit delta//Gaba-a receptor activity
Eszopiclone//Gamma-aminobutyric acid receptor subunit epsilon//Inhibitory extracellular ligand-gated ion channel activity
Eszopiclone//Gamma-aminobutyric acid receptor subunit gamma-1//Inhibitory extracellular ligand-gated ion channel activity
Eszopiclone//Gamma-aminobutyric acid receptor subunit gamma-2//Inhibitory extracellular ligand-gated ion channel activity
Eszopiclone//Gamma-aminobutyric acid receptor subunit gamma-3//Inhibitory extracellular ligand-gated ion channel activity
Eszopiclone//Gamma-aminobutyric acid receptor subunit pi//Gaba-a receptor activity
Eszopiclone//Gamma-aminobutyric acid receptor subunit theta//Transmembrane signaling receptor activity
Carbachol//Muscarinic acetylcholine receptor M1//Phosphatidylinositol phospholipase c activity
Carbachol//Muscarinic acetylcholine receptor M2//G-protein coupled acetylcholine receptor activity
Carbachol//Neuronal acetylcholine receptor subunit alpha-2//Drug binding
Carbachol//Acetylcholinesterase//Serine hydrolase activity
Carbachol//Muscarinic acetylcholine receptor M3//Receptor activity
Carbachol//Muscarinic acetylcholine receptor M4//Guanyl-nucleotide exchange factor activity
Acetohexamide//ATP-sensitive inward rectifier potassium channel 1//Phosphatidylinositol-4,5-bisphosphate binding
Methylphenidate//Sodium-dependent noradrenaline transporter//Norepinephrine:sodium symporter activity
Methylphenidate//Sodium-dependent dopamine transporter//Monoamine transmembrane transporter activity
Methylphenidate//5-hydroxytryptamine receptor 1A//Serotonin receptor activity
Cyproheptadine//Histamine H1 receptor//Histamine receptor activity
Cyproheptadine//5-hydroxytryptamine receptor 2A//Virus receptor activity
Cyproheptadine//5-hydroxytryptamine receptor 2C//Serotonin receptor activity
Cyproheptadine//Muscarinic acetylcholine receptor M1//Phosphatidylinositol phospholipase c activity
Cyproheptadine//Muscarinic acetylcholine receptor M2//G-protein coupled acetylcholine receptor activity
Cyproheptadine//Muscarinic acetylcholine receptor M3//Receptor activity
Cyproheptadine//5-hydroxytryptamine receptor 7//Serotonin receptor activity
Bendroflumethiazide//Solute carrier family 12 member 3//Transporter activity
Bendroflumethiazide//Calcium-activated potassium channel subunit alpha-1//Voltage-gated potassium channel activity
Bendroflumethiazide//Carbonic anhydrase 1//Zinc ion binding
Bendroflumethiazide//Carbonic anhydrase 2//Zinc ion binding
Bendroflumethiazide//Carbonic anhydrase 4//Zinc ion binding
Allopurinol//Xanthine dehydrogenase/oxidase//Xanthine oxidase activity
Cerivastatin//3-hydroxy-3-methylglutaryl-coenzyme A reductase//Nadph binding
Gemcitabine//Ribonucleoside-diphosphate reductase large subunit//Ribonucleoside-diphosphate reductase activity, thioredoxin disulfide as acceptor
Gemcitabine//Thymidylate synthase//Thymidylate synthase activity
Betamethasone//Glucocorticoid receptor//Zinc ion binding
Epirubicin//DNA topoisomerase 2-alpha//Ubiquitin binding
Chloramphenicol//50S ribosomal protein L16//Trna binding
Chloramphenicol//Complement decay-accelerating factor//Virus receptor activity
Lansoprazole//Potassium-transporting ATPase alpha chain 1//Sodium:potassium-exchanging atpase activity
Lansoprazole//Microtubule-associated protein tau//Structural constituent of cytoskeleton
Levothyroxine//Thyroid hormone receptor beta//Zinc ion binding
Levothyroxine//Thyroid hormone receptor alpha//Zinc ion binding
Levothyroxine//Integrin alpha-V//Voltage-gated calcium channel activity
Levothyroxine//Integrin beta-3//Virus receptor activity
Loratadine//Histamine H1 receptor//Histamine receptor activity
Loratadine//Potassium voltage-gated channel subfamily H member 2//Voltage-gated potassium channel activity involved in ventricular cardiac muscle cell action potential repolarization
Imipramine//5-hydroxytryptamine receptor 2A//Virus receptor activity
Imipramine//Sodium-dependent noradrenaline transporter//Norepinephrine:sodium symporter activity
Imipramine//Sodium-dependent serotonin transporter//Serotonin:sodium symporter activity
Imipramine//Histamine H1 receptor//Histamine receptor activity
Imipramine//Alpha-1A adrenergic receptor//Protein heterodimerization activity
Imipramine//Alpha-1D adrenergic receptor//Alpha1-adrenergic receptor activity
Imipramine//Muscarinic acetylcholine receptor M3//Receptor activity
Imipramine//Muscarinic acetylcholine receptor M1//Phosphatidylinositol phospholipase c activity
Imipramine//Muscarinic acetylcholine receptor M4//Guanyl-nucleotide exchange factor activity
Imipramine//Muscarinic acetylcholine receptor M2//G-protein coupled acetylcholine receptor activity
Imipramine//Muscarinic acetylcholine receptor M5//Phosphatidylinositol phospholipase c activity
Imipramine//Potassium voltage-gated channel subfamily D member 2//Voltage-gated potassium channel activity
Imipramine//Potassium voltage-gated channel subfamily D member 3//Metal ion binding
Imipramine//5-hydroxytryptamine receptor 2C//Serotonin receptor activity
Imipramine//Alpha-1B adrenergic receptor//Protein heterodimerization activity
Imipramine//5-hydroxytryptamine receptor 7//Serotonin receptor activity
Imipramine//D(1A) dopamine receptor//G-protein coupled amine receptor activity
Imipramine//D(1B) dopamine receptor//G-protein coupled amine receptor activity
Imipramine//D(2) dopamine receptor//Potassium channel regulator activity
Imipramine//Potassium voltage-gated channel subfamily H member 2//Voltage-gated potassium channel activity involved in ventricular cardiac muscle cell action potential repolarization
Imipramine//Sodium-dependent dopamine transporter//Monoamine transmembrane transporter activity
Imipramine//5-hydroxytryptamine receptor 1A//Serotonin receptor activity
Imipramine//5-hydroxytryptamine receptor 6//Serotonin receptor activity
Imipramine//Potassium voltage-gated channel subfamily H member 1//Phosphorelay sensor kinase activity
Acitretin//Retinoic acid receptor RXR-alpha//Zinc ion binding
Acitretin//Retinoic acid receptor alpha//Zinc ion binding
Acitretin//Retinoic acid receptor beta//Zinc ion binding
Acitretin//Retinoic acid receptor gamma//Zinc ion binding
Acitretin//Retinoic acid receptor RXR-beta//Zinc ion binding
Acitretin//Retinoic acid receptor RXR-gamma//Zinc ion binding
Acitretin//Retinol-binding protein 1//Transporter activity
Nabumetone//Prostaglandin G/H synthase 2//Prostaglandin-endoperoxide synthase activity
Nabumetone//Prostaglandin G/H synthase 1//Prostaglandin-endoperoxide synthase activity
Enoxacin//DNA gyrase subunit A//Dna topoisomerase type ii (atp-hydrolyzing) activity
Enoxacin//DNA topoisomerase 4 subunit A//Dna topoisomerase type ii (atp-hydrolyzing) activity
Enoxacin//DNA topoisomerase 2-alpha//Ubiquitin binding
Dronabinol//Cannabinoid receptor 1//Drug binding
Dronabinol//Cannabinoid receptor 2//Cannabinoid receptor activity
Montelukast//Arachidonate 5-lipoxygenase//Iron ion binding
Fluoxetine//Sodium-dependent serotonin transporter//Serotonin:sodium symporter activity
Fluoxetine//5-hydroxytryptamine receptor 2C//Serotonin receptor activity
Fluoxetine//Neuronal acetylcholine receptor subunit alpha-2//Drug binding
Fluoxetine//Neuronal acetylcholine receptor subunit alpha-3//Ligand-gated ion channel activity
Fluoxetine//Neuronal acetylcholine receptor subunit beta-4//Ligand-gated ion channel activity
Fluoxetine//Cyclin-dependent kinases regulatory subunit 1//Cyclin-dependent protein serine/threonine kinase regulator activity
Fluoxetine//Potassium voltage-gated channel subfamily H member 2//Voltage-gated potassium channel activity involved in ventricular cardiac muscle cell action potential repolarization
Duloxetine//Sodium-dependent serotonin transporter//Serotonin:sodium symporter activity
Duloxetine//Sodium-dependent noradrenaline transporter//Norepinephrine:sodium symporter activity
Duloxetine//Sodium-dependent dopamine transporter//Monoamine transmembrane transporter activity
Chlorpromazine//D(2) dopamine receptor//Potassium channel regulator activity
Chlorpromazine//D(1A) dopamine receptor//G-protein coupled amine receptor activity
Chlorpromazine//5-hydroxytryptamine receptor 1A//Serotonin receptor activity
Chlorpromazine//5-hydroxytryptamine receptor 2A//Virus receptor activity
Chlorpromazine//Alpha-1A adrenergic receptor//Protein heterodimerization activity
Chlorpromazine//Alpha-1B adrenergic receptor//Protein heterodimerization activity
Chlorpromazine//Histamine H1 receptor//Histamine receptor activity
Chlorpromazine//Potassium voltage-gated channel subfamily H member 2//Voltage-gated potassium channel activity involved in ventricular cardiac muscle cell action potential repolarization
Chlorpromazine//D(1A) dopamine receptor//G-protein coupled amine receptor activity
Chlorpromazine//D(1B) dopamine receptor//G-protein coupled amine receptor activity
Chlorpromazine//D(3) dopamine receptor//G-protein coupled amine receptor activity
Chlorpromazine//D(4) dopamine receptor//Sh3 domain binding
Chlorpromazine//D(1B) dopamine receptor//G-protein coupled amine receptor activity
Chlorpromazine//5-hydroxytryptamine receptor 2C//Serotonin receptor activity
Chlorpromazine//5-hydroxytryptamine receptor 2A//Virus receptor activity
Chlorpromazine//5-hydroxytryptamine receptor 2B//Serotonin receptor activity
Chlorpromazine//5-hydroxytryptamine receptor 2C//Serotonin receptor activity
Chlorpromazine//Alpha-1A adrenergic receptor//Protein heterodimerization activity
Chlorpromazine//Alpha-1B adrenergic receptor//Protein heterodimerization activity
Chlorpromazine//Alpha-1D adrenergic receptor//Alpha1-adrenergic receptor activity
Chlorpromazine//Alpha-2A adrenergic receptor//Thioesterase binding
Chlorpromazine//Alpha-2B adrenergic receptor//Epinephrine binding
Chlorpromazine//Alpha-2C adrenergic receptor//Protein homodimerization activity
Chlorpromazine//Muscarinic acetylcholine receptor M1//Phosphatidylinositol phospholipase c activity
Chlorpromazine//Muscarinic acetylcholine receptor M3//Receptor activity
Chlorpromazine//Sphingomyelin phosphodiesterase//Sphingomyelin phosphodiesterase activity
Chlorpromazine//Calmodulin//Titin binding
Chlorpromazine//5-hydroxytryptamine receptor 6//Serotonin receptor activity
Chlorpromazine//5-hydroxytryptamine receptor 7//Serotonin receptor activity
Chlorpromazine//Histamine H4 receptor//Histamine receptor activity
Celecoxib//Prostaglandin G/H synthase 2//Prostaglandin-endoperoxide synthase activity
Celecoxib//3-phosphoinositide-dependent protein kinase 1//Protein serine/threonine kinase activity
Celecoxib//Carbonic anhydrase 2//Zinc ion binding
Celecoxib//Carbonic anhydrase 3//Zinc ion binding
Brimonidine//Alpha-2A adrenergic receptor//Thioesterase binding
Brimonidine//Alpha-2C adrenergic receptor//Protein homodimerization activity
Brimonidine//Alpha-2B adrenergic receptor//Epinephrine binding
Nabilone//Cannabinoid receptor 1//Drug binding
Nabilone//Cannabinoid receptor 2//Cannabinoid receptor activity
Buspirone//5-hydroxytryptamine receptor 1A//Serotonin receptor activity
Buspirone//D(2) dopamine receptor//Potassium channel regulator activity
Buspirone//D(3) dopamine receptor//G-protein coupled amine receptor activity
Buspirone//D(4) dopamine receptor//Sh3 domain binding
Buspirone//Alpha-1A adrenergic receptor//Protein heterodimerization activity
Buspirone//Alpha-1B adrenergic receptor//Protein heterodimerization activity
Buspirone//Alpha-1D adrenergic receptor//Alpha1-adrenergic receptor activity
Miglitol//Maltase-glucoamylase, intestinal//Maltose alpha-glucosidase activity
Miglitol//Lysosomal alpha-glucosidase//Maltose alpha-glucosidase activity
Miglitol//Neutral alpha-glucosidase AB//Poly(a) rna binding
Miglitol//Neutral alpha-glucosidase C//Maltose alpha-glucosidase activity
Entacapone//Catechol O-methyltransferase//O-methyltransferase activity
Darifenacin//Muscarinic acetylcholine receptor M3//Receptor activity
Darifenacin//Muscarinic acetylcholine receptor M1//Phosphatidylinositol phospholipase c activity
Darifenacin//Muscarinic acetylcholine receptor M2//G-protein coupled acetylcholine receptor activity
Darifenacin//Muscarinic acetylcholine receptor M4//Guanyl-nucleotide exchange factor activity
Darifenacin//Muscarinic acetylcholine receptor M5//Phosphatidylinositol phospholipase c activity
Flutamide//Androgen receptor//Zinc ion binding
Flutamide//Aryl hydrocarbon receptor//Transcription regulatory region dna binding
Flutamide//Nuclear receptor subfamily 1 group I member 2//Zinc ion binding
Cimetidine//Histamine H2 receptor//Histamine receptor activity
Haloperidol//D(1A) dopamine receptor//G-protein coupled amine receptor activity
Haloperidol//Glutamate receptor ionotropic, NMDA 2B//Zinc ion binding
Haloperidol//D(2) dopamine receptor//Potassium channel regulator activity
Haloperidol//5-hydroxytryptamine receptor 2A//Virus receptor activity
Haloperidol//D(3) dopamine receptor//G-protein coupled amine receptor activity
Haloperidol//Synaptic vesicular amine transporter//Monoamine transmembrane transporter activity
Haloperidol//5-hydroxytryptamine receptor 2C//Serotonin receptor activity
Haloperidol//Sigma non-opioid intracellular receptor 1//Opioid receptor activity
Haloperidol//Histamine H1 receptor//Histamine receptor activity
Haloperidol//Muscarinic acetylcholine receptor M3//Receptor activity
Haloperidol//Alpha-1A adrenergic receptor//Protein heterodimerization activity
Haloperidol//Alpha-2A adrenergic receptor//Thioesterase binding
Haloperidol//Alpha-2B adrenergic receptor//Epinephrine binding
Haloperidol//Alpha-2C adrenergic receptor//Protein homodimerization activity
Haloperidol//5-hydroxytryptamine receptor 1A//Serotonin receptor activity
Haloperidol//5-hydroxytryptamine receptor 6//Serotonin receptor activity
Haloperidol//5-hydroxytryptamine receptor 7//Serotonin receptor activity
Dextromethorphan//Sigma non-opioid intracellular receptor 1//Opioid receptor activity
Dextromethorphan//Glutamate receptor ionotropic, NMDA 3A//Protein phosphatase 2a binding
Dextromethorphan//Neuronal acetylcholine receptor subunit alpha-2//Drug binding
Dextromethorphan//Sodium-dependent serotonin transporter//Serotonin:sodium symporter activity
Dextromethorphan//Membrane-associated progesterone receptor component 1//Steroid binding
Dextromethorphan//Neuronal acetylcholine receptor subunit alpha-3//Ligand-gated ion channel activity
Dextromethorphan//Neuronal acetylcholine receptor subunit alpha-4//Ligand-gated ion channel activity
Dextromethorphan//Neuronal acetylcholine receptor subunit beta-4//Ligand-gated ion channel activity
Dextromethorphan//Neuronal acetylcholine receptor subunit beta-2//Ligand-gated ion channel activity
Dextromethorphan//Neuronal acetylcholine receptor subunit alpha-7//Toxic substance binding
Dextromethorphan//Mu-type opioid receptor//Voltage-gated calcium channel activity
Dextromethorphan//Delta-type opioid receptor//Opioid receptor activity
Dextromethorphan//Kappa-type opioid receptor//Opioid receptor activity
Dextromethorphan//Cytochrome b-245 heavy chain//Voltage-gated ion channel activity
Dextromethorphan//Ras-related C3 botulinum toxin substrate 1//Thioesterase binding
Dextromethorphan//Sodium-dependent noradrenaline transporter//Norepinephrine:sodium symporter activity
Albendazole//Tubulin alpha-1A chain//Tubulin is the major constituent of microtubules. It binds two moles of GTP, one at an exchangeable site on the beta chain and one at a non-exchangeable site on the alpha chain.
Albendazole//Tubulin beta-2 chain//Structural constituent of cytoskeleton
Albendazole//Tubulin beta-4B chain//Unfolded protein binding
Carteolol//Beta-1 adrenergic receptor//Receptor signaling protein activity
Carteolol//Beta-2 adrenergic receptor//Protein homodimerization activity
Alitretinoin//Retinoic acid receptor alpha//Zinc ion binding
Alitretinoin//Retinoic acid receptor RXR-alpha//Zinc ion binding
Alitretinoin//Retinoic acid receptor beta//Zinc ion binding
Alitretinoin//Retinoic acid receptor RXR-beta//Zinc ion binding
Alitretinoin//Retinoic acid receptor gamma//Zinc ion binding
Alitretinoin//Retinoic acid receptor RXR-gamma//Zinc ion binding
Cinchocaine//Sodium channel protein type 10 subunit alpha//Voltage-gated sodium channel activity
Cinchocaine//Sodium channel protein type 5 subunit alpha//Voltage-gated sodium channel activity involved in sa node cell action potential
Cinchocaine//Calmodulin//Titin binding
Lercanidipine//Voltage-dependent calcium channel gamma-1 subunit//Voltage-gated calcium channel activity
Erlotinib//Epidermal growth factor receptor//Ubiquitin protein ligase binding
Erlotinib//Nuclear receptor subfamily 1 group I member 2//Zinc ion binding
Cyclophosphamide//Nuclear receptor subfamily 1 group I member 2//Zinc ion binding
Ciprofloxacin//DNA topoisomerase 4 subunit A//Dna topoisomerase type ii (atp-hydrolyzing) activity
Ciprofloxacin//DNA gyrase subunit A//Dna topoisomerase type ii (atp-hydrolyzing) activity
Ciprofloxacin//DNA topoisomerase 2-alpha//Ubiquitin binding
Ciprofloxacin//Potassium voltage-gated channel subfamily H member 2//Voltage-gated potassium channel activity involved in ventricular cardiac muscle cell action potential repolarization
Ciprofloxacin//DNA gyrase subunit A//Dna topoisomerase type ii (atp-hydrolyzing) activity
Ciprofloxacin//DNA topoisomerase 4 subunit A//Dna topoisomerase type ii (atp-hydrolyzing) activity
Ciprofloxacin//DNA gyrase subunit A//Dna topoisomerase type ii (atp-hydrolyzing) activity
Ciprofloxacin//Multidrug resistance protein MdtK//Drug transmembrane transporter activity
Ciprofloxacin//Gyrase A//Dna topoisomerase type ii (atp-hydrolyzing) activity
Ciprofloxacin//DNA gyrase subunit A//Dna topoisomerase type ii (atp-hydrolyzing) activity
Benazepril//Angiotensin-converting enzyme//Zinc ion binding
Amoxapine//Sodium-dependent noradrenaline transporter//Norepinephrine:sodium symporter activity
Amoxapine//Sodium-dependent serotonin transporter//Serotonin:sodium symporter activity
Amoxapine//D(2) dopamine receptor//Potassium channel regulator activity
Amoxapine//D(1A) dopamine receptor//G-protein coupled amine receptor activity
Amoxapine//Alpha-2A adrenergic receptor//Thioesterase binding
Amoxapine//Alpha-1A adrenergic receptor//Protein heterodimerization activity
Amoxapine//Muscarinic acetylcholine receptor M1//Phosphatidylinositol phospholipase c activity
Amoxapine//Gamma-aminobutyric acid receptor subunit alpha-1//Inhibitory extracellular ligand-gated ion channel activity
Amoxapine//5-hydroxytryptamine receptor 2A//Virus receptor activity
Amoxapine//5-hydroxytryptamine receptor 2C//Serotonin receptor activity
Amoxapine//5-hydroxytryptamine receptor 6//Serotonin receptor activity
Amoxapine//5-hydroxytryptamine receptor 7//Serotonin receptor activity
Amoxapine//D(3) dopamine receptor//G-protein coupled amine receptor activity
Amoxapine//D(4) dopamine receptor//Sh3 domain binding
Amoxapine//Histamine H1 receptor//Histamine receptor activity
Amoxapine//Alpha-1A adrenergic receptor//Protein heterodimerization activity
Amoxapine//Alpha-1B adrenergic receptor//Protein heterodimerization activity
Amoxapine//Alpha-1D adrenergic receptor//Alpha1-adrenergic receptor activity
Amoxapine//Muscarinic acetylcholine receptor M1//Phosphatidylinositol phospholipase c activity
Amoxapine//Muscarinic acetylcholine receptor M2//G-protein coupled acetylcholine receptor activity
Amoxapine//Muscarinic acetylcholine receptor M3//Receptor activity
Amoxapine//Muscarinic acetylcholine receptor M4//Guanyl-nucleotide exchange factor activity
Amoxapine//Muscarinic acetylcholine receptor M5//Phosphatidylinositol phospholipase c activity
Amoxapine//5-hydroxytryptamine receptor 2B//Serotonin receptor activity
Amoxapine//5-hydroxytryptamine receptor 3A//Voltage-gated potassium channel activity
Amoxapine//5-hydroxytryptamine receptor 1A//Serotonin receptor activity
Amoxapine//5-hydroxytryptamine receptor 1B//Serotonin receptor activity
Amoxapine//Alpha-2A adrenergic receptor//Thioesterase binding
Amoxapine//Alpha-2B adrenergic receptor//Epinephrine binding
Amoxapine//Alpha-2C adrenergic receptor//Protein homodimerization activity
Amoxapine//Histamine H4 receptor//Histamine receptor activity
Amoxapine//Gamma-aminobutyric acid receptor subunit alpha-1//Inhibitory extracellular ligand-gated ion channel activity
Amoxapine//Gamma-aminobutyric acid receptor subunit alpha-2//Inhibitory extracellular ligand-gated ion channel activity
Amoxapine//Gamma-aminobutyric acid receptor subunit alpha-3//Inhibitory extracellular ligand-gated ion channel activity
Amoxapine//Gamma-aminobutyric acid receptor subunit alpha-4//Inhibitory extracellular ligand-gated ion channel activity
Amoxapine//Gamma-aminobutyric acid receptor subunit alpha-5//Transporter activity
Amoxapine//Gamma-aminobutyric acid receptor subunit alpha-6//Inhibitory extracellular ligand-gated ion channel activity
Amoxapine//Gamma-aminobutyric acid receptor subunit beta-1//Ligand-gated ion channel activity
Amoxapine//Gamma-aminobutyric acid receptor subunit beta-2//Inhibitory extracellular ligand-gated ion channel activity
Amoxapine//Gamma-aminobutyric acid receptor subunit beta-3//Gaba-gated chloride ion channel activity
Amoxapine//Gamma-aminobutyric acid receptor subunit delta//Gaba-a receptor activity
Amoxapine//Gamma-aminobutyric acid receptor subunit epsilon//Inhibitory extracellular ligand-gated ion channel activity
Amoxapine//Gamma-aminobutyric acid receptor subunit gamma-1//Inhibitory extracellular ligand-gated ion channel activity
Amoxapine//Gamma-aminobutyric acid receptor subunit gamma-2//Inhibitory extracellular ligand-gated ion channel activity
Amoxapine//Gamma-aminobutyric acid receptor subunit gamma-3//Inhibitory extracellular ligand-gated ion channel activity
Amoxapine//Gamma-aminobutyric acid receptor subunit pi//Gaba-a receptor activity
Amoxapine//Gamma-aminobutyric acid receptor subunit theta//Transmembrane signaling receptor activity
Amoxapine//Sodium-dependent dopamine transporter//Monoamine transmembrane transporter activity
Fluorouracil//Thymidylate synthase//Thymidylate synthase activity
Adinazolam//Gamma-aminobutyric acid receptor subunit alpha-1//Inhibitory extracellular ligand-gated ion channel activity
Adinazolam//Gamma-aminobutyric acid receptor subunit alpha-2//Inhibitory extracellular ligand-gated ion channel activity
Adinazolam//Gamma-aminobutyric acid receptor subunit alpha-3//Inhibitory extracellular ligand-gated ion channel activity
Adinazolam//Gamma-aminobutyric acid receptor subunit alpha-4//Inhibitory extracellular ligand-gated ion channel activity
Adinazolam//Gamma-aminobutyric acid receptor subunit alpha-5//Transporter activity
Adinazolam//Gamma-aminobutyric acid receptor subunit alpha-6//Inhibitory extracellular ligand-gated ion channel activity
Adinazolam//Gamma-aminobutyric acid receptor subunit beta-1//Ligand-gated ion channel activity
Adinazolam//Gamma-aminobutyric acid receptor subunit beta-2//Inhibitory extracellular ligand-gated ion channel activity
Adinazolam//Gamma-aminobutyric acid receptor subunit beta-3//Gaba-gated chloride ion channel activity
Adinazolam//Gamma-aminobutyric acid receptor subunit delta//Gaba-a receptor activity
Adinazolam//Gamma-aminobutyric acid receptor subunit epsilon//Inhibitory extracellular ligand-gated ion channel activity
Adinazolam//Gamma-aminobutyric acid receptor subunit gamma-1//Inhibitory extracellular ligand-gated ion channel activity
Adinazolam//Gamma-aminobutyric acid receptor subunit gamma-2//Inhibitory extracellular ligand-gated ion channel activity
Adinazolam//Gamma-aminobutyric acid receptor subunit gamma-3//Inhibitory extracellular ligand-gated ion channel activity
Adinazolam//Gamma-aminobutyric acid receptor subunit pi//Gaba-a receptor activity
Adinazolam//Gamma-aminobutyric acid receptor subunit theta//Transmembrane signaling receptor activity
Adinazolam//Gamma-aminobutyric acid receptor subunit alpha-1//Inhibitory extracellular ligand-gated ion channel activity
Adinazolam//Gamma-aminobutyric acid receptor subunit alpha-2//Inhibitory extracellular ligand-gated ion channel activity
Adinazolam//Gamma-aminobutyric acid receptor subunit alpha-3//Inhibitory extracellular ligand-gated ion channel activity
Adinazolam//Gamma-aminobutyric acid receptor subunit alpha-5//Transporter activity
Adinazolam//Gamma-aminobutyric acid receptor subunit gamma-1//Inhibitory extracellular ligand-gated ion channel activity
Adinazolam//Gamma-aminobutyric acid receptor subunit gamma-2//Inhibitory extracellular ligand-gated ion channel activity
Adinazolam//Gamma-aminobutyric acid receptor subunit gamma-3//Inhibitory extracellular ligand-gated ion channel activity
Lamotrigine//Voltage-dependent R-type calcium channel subunit alpha-1E//Voltage-sensitive calcium channels (VSCC) mediate the entry of calcium ions into excitable cells and are also involved in a variety of calcium-dependent processes, including muscle contraction, hormone or neurotransmitter release, gene expression, cell motility, cell division and cell death. The isoform alpha-1E gives rise to R-type calcium currents. R-type calcium channels belong to the 'high-voltage activated' (HVA) group and are blocked by nickel, and partially by omega-agatoxin-IIIA (omega-Aga-IIIA). They are however insensitive to dihydropyridines (DHP), omega-conotoxin-GVIA (omega-CTx-GVIA), and omega-agatoxin-IVA (omega-Aga-IVA). Calcium channels containing alpha-1E subunit could be involved in the modulation of firing patterns of neurons which is important for information processing.
Lamotrigine//Sodium channel protein type 1 subunit alpha//Voltage-gated sodium channel activity
Lamotrigine//Sodium channel protein type 10 subunit alpha//Voltage-gated sodium channel activity
Lamotrigine//Sodium channel protein type 11 subunit alpha//Voltage-gated sodium channel activity
Lamotrigine//Sodium channel protein type 2 subunit alpha//Voltage-gated sodium channel activity
Lamotrigine//Sodium channel protein type 3 subunit alpha//Voltage-gated sodium channel activity
Lamotrigine//Sodium channel protein type 4 subunit alpha//Voltage-gated sodium channel activity
Lamotrigine//Sodium channel protein type 5 subunit alpha//Voltage-gated sodium channel activity involved in sa node cell action potential
Lamotrigine//Sodium channel protein type 7 subunit alpha//Mediates the voltage-dependent sodium ion permeability of excitable membranes. Assuming opened or closed conformations in response to the voltage difference across the membrane, the protein forms a sodium-selective channel through which Na(+) ions may pass in accordance with their electrochemical gradient.
Lamotrigine//Sodium channel protein type 8 subunit alpha//Voltage-gated sodium channel activity
Lamotrigine//Sodium channel protein type 9 subunit alpha//Voltage-gated sodium channel activity
Lamotrigine//Adenosine receptor A1//Purine nucleoside binding
Lamotrigine//Adenosine receptor A2a//Identical protein binding
Lamotrigine//Alpha-1A adrenergic receptor//Protein heterodimerization activity
Lamotrigine//Alpha-2A adrenergic receptor//Thioesterase binding
Lamotrigine//Beta-1 adrenergic receptor//Receptor signaling protein activity
Lamotrigine//D(1A) dopamine receptor//G-protein coupled amine receptor activity
Lamotrigine//D(1B) dopamine receptor//G-protein coupled amine receptor activity
Lamotrigine//D(2) dopamine receptor//Potassium channel regulator activity
Lamotrigine//Gamma-aminobutyric acid receptor subunit alpha-1//Inhibitory extracellular ligand-gated ion channel activity
Lamotrigine//Gamma-aminobutyric acid receptor subunit alpha-2//Inhibitory extracellular ligand-gated ion channel activity
Lamotrigine//Gamma-aminobutyric acid receptor subunit alpha-3//Inhibitory extracellular ligand-gated ion channel activity
Lamotrigine//Gamma-aminobutyric acid receptor subunit alpha-4//Inhibitory extracellular ligand-gated ion channel activity
Lamotrigine//Gamma-aminobutyric acid receptor subunit alpha-5//Transporter activity
Lamotrigine//Gamma-aminobutyric acid receptor subunit alpha-6//Inhibitory extracellular ligand-gated ion channel activity
Lamotrigine//Gamma-aminobutyric acid receptor subunit beta-1//Ligand-gated ion channel activity
Lamotrigine//Gamma-aminobutyric acid receptor subunit beta-2//Inhibitory extracellular ligand-gated ion channel activity
Lamotrigine//Gamma-aminobutyric acid receptor subunit beta-3//Gaba-gated chloride ion channel activity
Lamotrigine//Gamma-aminobutyric acid receptor subunit delta//Gaba-a receptor activity
Lamotrigine//Gamma-aminobutyric acid receptor subunit epsilon//Inhibitory extracellular ligand-gated ion channel activity
Lamotrigine//Gamma-aminobutyric acid receptor subunit gamma-1//Inhibitory extracellular ligand-gated ion channel activity
Lamotrigine//Gamma-aminobutyric acid receptor subunit gamma-2//Inhibitory extracellular ligand-gated ion channel activity
Lamotrigine//Gamma-aminobutyric acid receptor subunit gamma-3//Inhibitory extracellular ligand-gated ion channel activity
Lamotrigine//Gamma-aminobutyric acid receptor subunit pi//Gaba-a receptor activity
Lamotrigine//Gamma-aminobutyric acid receptor subunit theta//Transmembrane signaling receptor activity
Lamotrigine//Gamma-aminobutyric acid receptor subunit alpha-1//Inhibitory extracellular ligand-gated ion channel activity
Lamotrigine//Gamma-aminobutyric acid receptor subunit alpha-2//Inhibitory extracellular ligand-gated ion channel activity
Lamotrigine//Gamma-aminobutyric acid receptor subunit alpha-3//Inhibitory extracellular ligand-gated ion channel activity
Lamotrigine//Gamma-aminobutyric acid receptor subunit alpha-5//Transporter activity
Lamotrigine//Gamma-aminobutyric acid receptor subunit gamma-1//Inhibitory extracellular ligand-gated ion channel activity
Lamotrigine//Gamma-aminobutyric acid receptor subunit gamma-2//Inhibitory extracellular ligand-gated ion channel activity
Lamotrigine//Gamma-aminobutyric acid receptor subunit gamma-3//Inhibitory extracellular ligand-gated ion channel activity
Lamotrigine//Histamine H1 receptor//Histamine receptor activity
Lamotrigine//Kappa-type opioid receptor//Opioid receptor activity
Lamotrigine//5-hydroxytryptamine receptor 2A//Virus receptor activity
Lamotrigine//5-hydroxytryptamine receptor 3A//Voltage-gated potassium channel activity
Lamotrigine//Glutamate receptor 1//Pdz domain binding
Hydroxyzine//Histamine H1 receptor//Histamine receptor activity
Hydroxyzine//Potassium voltage-gated channel subfamily H member 2//Voltage-gated potassium channel activity involved in ventricular cardiac muscle cell action potential repolarization
Bosentan//Endothelin B receptor//Peptide hormone binding
Bosentan//Endothelin-1 receptor//Phosphatidylinositol phospholipase c activity
Methotrexate//Dihydrofolate reductase//Nadph binding
Methotrexate//Thymidylate synthase//Thymidylate synthase activity
Methotrexate//Bifunctional purine biosynthesis protein PURH//Protein homodimerization activity
Carbamazepine//Sodium channel protein type 1 subunit alpha//Voltage-gated sodium channel activity
Carbamazepine//Sodium channel protein type 10 subunit alpha//Voltage-gated sodium channel activity
Carbamazepine//Sodium channel protein type 11 subunit alpha//Voltage-gated sodium channel activity
Carbamazepine//Sodium channel protein type 2 subunit alpha//Voltage-gated sodium channel activity
Carbamazepine//Sodium channel protein type 3 subunit alpha//Voltage-gated sodium channel activity
Carbamazepine//Sodium channel protein type 4 subunit alpha//Voltage-gated sodium channel activity
Carbamazepine//Sodium channel protein type 5 subunit alpha//Voltage-gated sodium channel activity involved in sa node cell action potential
Carbamazepine//Sodium channel protein type 7 subunit alpha//Mediates the voltage-dependent sodium ion permeability of excitable membranes. Assuming opened or closed conformations in response to the voltage difference across the membrane, the protein forms a sodium-selective channel through which Na(+) ions may pass in accordance with their electrochemical gradient.
Carbamazepine//Sodium channel protein type 8 subunit alpha//Voltage-gated sodium channel activity
Carbamazepine//Sodium channel protein type 9 subunit alpha//Voltage-gated sodium channel activity
Carbamazepine//Neuronal acetylcholine receptor subunit alpha-4//Ligand-gated ion channel activity
Carbamazepine//Nuclear receptor subfamily 1 group I member 2//Zinc ion binding
Cinnarizine//Histamine H1 receptor//Histamine receptor activity
Cinnarizine//Voltage-dependent L-type calcium channel subunit alpha-1C//Voltage-gated calcium channel activity
Cinnarizine//Voltage-dependent L-type calcium channel subunit alpha-1D//Voltage-gated calcium channel activity involved sa node cell action potential
Cinnarizine//Voltage-dependent L-type calcium channel subunit alpha-1F//Voltage-gated calcium channel activity
Cinnarizine//Voltage-dependent L-type calcium channel subunit alpha-1S//Voltage-gated calcium channel activity
Cinnarizine//Voltage-dependent T-type calcium channel subunit alpha-1G//Scaffold protein binding
Cinnarizine//Voltage-dependent T-type calcium channel subunit alpha-1I//Voltage-gated calcium channel activity
Cinnarizine//Voltage-dependent T-type calcium channel subunit alpha-1H//Scaffold protein binding
Cinnarizine//D(2) dopamine receptor//Potassium channel regulator activity
Cinnarizine//D(1A) dopamine receptor//G-protein coupled amine receptor activity
Cinnarizine//D(1B) dopamine receptor//G-protein coupled amine receptor activity
Cinnarizine//Muscarinic acetylcholine receptor M1//Phosphatidylinositol phospholipase c activity
Cinnarizine//Muscarinic acetylcholine receptor M2//G-protein coupled acetylcholine receptor activity
Cinnarizine//Muscarinic acetylcholine receptor M3//Receptor activity
Cinnarizine//Muscarinic acetylcholine receptor M4//Guanyl-nucleotide exchange factor activity
Cinnarizine//Muscarinic acetylcholine receptor M5//Phosphatidylinositol phospholipase c activity
Atropine//Muscarinic acetylcholine receptor M1//Phosphatidylinositol phospholipase c activity
Atropine//Muscarinic acetylcholine receptor M2//G-protein coupled acetylcholine receptor activity
Atropine//Muscarinic acetylcholine receptor M3//Receptor activity
Atropine//Muscarinic acetylcholine receptor M4//Guanyl-nucleotide exchange factor activity
Atropine//Muscarinic acetylcholine receptor M5//Phosphatidylinositol phospholipase c activity
Atropine//Glycine receptor subunit alpha-1//Transmitter-gated ion channel activity
Atropine//Neuronal acetylcholine receptor subunit alpha-4//Ligand-gated ion channel activity
Atropine//Neuronal acetylcholine receptor subunit beta-2//Ligand-gated ion channel activity
Fenfluramine//Sodium-dependent serotonin transporter//Serotonin:sodium symporter activity
Fenfluramine//5-hydroxytryptamine receptor 2B//Serotonin receptor activity
Fenfluramine//5-hydroxytryptamine receptor 2C//Serotonin receptor activity
Fenfluramine//5-hydroxytryptamine receptor 2A//Virus receptor activity
Clonidine//Alpha-2A adrenergic receptor//Thioesterase binding
Clonidine//Alpha-2B adrenergic receptor//Epinephrine binding
Clonidine//Alpha-2C adrenergic receptor//Protein homodimerization activity
Clonidine//Alpha-1A adrenergic receptor//Protein heterodimerization activity
Clonidine//Alpha-1B adrenergic receptor//Protein heterodimerization activity
Clonidine//Alpha-1D adrenergic receptor//Alpha1-adrenergic receptor activity
Enalapril//Angiotensin-converting enzyme//Zinc ion binding
Diclofenac//Prostaglandin G/H synthase 2//Prostaglandin-endoperoxide synthase activity
Diclofenac//Prostaglandin G/H synthase 1//Prostaglandin-endoperoxide synthase activity
Fluticasonepropionate//Glucocorticoid receptor//Zinc ion binding
Fluticasonepropionate//Progesterone receptor//Zinc ion binding
Fluticasonepropionate//Cytosolic phospholipase A2//Phospholipase a2 activity
Fluticasonepropionate//Mineralocorticoid receptor//Zinc ion binding
Lisuride//D(2) dopamine receptor//Potassium channel regulator activity
Lisuride//D(3) dopamine receptor//G-protein coupled amine receptor activity
Lisuride//D(4) dopamine receptor//Sh3 domain binding
Lisuride//D(1A) dopamine receptor//G-protein coupled amine receptor activity
Lisuride//D(1B) dopamine receptor//G-protein coupled amine receptor activity
Lisuride//5-hydroxytryptamine receptor 1A//Serotonin receptor activity
Lisuride//5-hydroxytryptamine receptor 1D//Serotonin receptor activity
Lisuride//5-hydroxytryptamine receptor 2B//Serotonin receptor activity
Lisuride//5-hydroxytryptamine receptor 2A//Virus receptor activity
Lisuride//5-hydroxytryptamine receptor 2C//Serotonin receptor activity
Lisuride//5-hydroxytryptamine receptor 1B//Serotonin receptor activity
Lisuride//Alpha-2A adrenergic receptor//Thioesterase binding
Lisuride//Alpha-2B adrenergic receptor//Epinephrine binding
Lisuride//Alpha-2C adrenergic receptor//Protein homodimerization activity
Lisuride//5-hydroxytryptamine receptor 7//Serotonin receptor activity
Doxazosin//Alpha-1A adrenergic receptor//Protein heterodimerization activity
Doxazosin//Alpha-1D adrenergic receptor//Alpha1-adrenergic receptor activity
Doxazosin//Potassium voltage-gated channel subfamily H member 2//Voltage-gated potassium channel activity involved in ventricular cardiac muscle cell action potential repolarization
Doxazosin//Potassium voltage-gated channel subfamily H member 6//Voltage-gated potassium channel activity
Doxazosin//Potassium voltage-gated channel subfamily H member 7//Voltage-gated potassium channel activity
Doxazosin//Alpha-1B adrenergic receptor//Protein heterodimerization activity
Fluocinoloneacetonide//Glucocorticoid receptor//Zinc ion binding
Fluocinoloneacetonide//Annexin A1//Structural molecule activity
Fluocinoloneacetonide//Annexin A2//S100 protein binding
Fluocinoloneacetonide//Annexin A5//Phospholipid binding
Ethosuximide//Voltage-dependent T-type calcium channel subunit alpha-1G//Scaffold protein binding
Amiloride//Amiloride-sensitive sodium channel subunit alpha//Ww domain binding
Amiloride//Amiloride-sensitive sodium channel subunit beta//Ww domain binding
Amiloride//Amiloride-sensitive sodium channel subunit gamma//Ww domain binding
Amiloride//Amiloride-sensitive sodium channel subunit delta//Ligand-gated sodium channel activity
Amiloride//Amiloride-sensitive amine oxidase [copper-containing]//Zinc ion binding
Amiloride//Acid-sensing ion channel 2//Ligand-gated sodium channel activity
Amiloride//Acid-sensing ion channel 1//Ligand-gated sodium channel activity
Amiloride//Urokinase-type plasminogen activator//Serine-type endopeptidase activity
Labetalol//Beta-1 adrenergic receptor//Receptor signaling protein activity
Labetalol//Beta-2 adrenergic receptor//Protein homodimerization activity
Labetalol//Alpha-1A adrenergic receptor//Protein heterodimerization activity
Labetalol//Alpha-1B adrenergic receptor//Protein heterodimerization activity
Labetalol//Alpha-1D adrenergic receptor//Alpha1-adrenergic receptor activity
Ivermectin//Glycine receptor subunit alpha-3//Transmitter-gated ion channel activity
Ivermectin//Gamma-aminobutyric acid receptor subunit beta-3//Gaba-gated chloride ion channel activity
Medroxyprogesteroneacetate//Progesterone receptor//Zinc ion binding
Medroxyprogesteroneacetate//Estrogen receptor//Zinc ion binding
Medroxyprogesteroneacetate//Multidrug resistance protein 1//Xenobiotic-transporting atpase activity
Medroxyprogesteroneacetate//Gamma-aminobutyric acid receptor subunit alpha-1//Inhibitory extracellular ligand-gated ion channel activity
Medroxyprogesteroneacetate//Gamma-aminobutyric acid receptor subunit alpha-2//Inhibitory extracellular ligand-gated ion channel activity
Medroxyprogesteroneacetate//Gamma-aminobutyric acid receptor subunit alpha-3//Inhibitory extracellular ligand-gated ion channel activity
Medroxyprogesteroneacetate//Gamma-aminobutyric acid receptor subunit alpha-4//Inhibitory extracellular ligand-gated ion channel activity
Medroxyprogesteroneacetate//Gamma-aminobutyric acid receptor subunit alpha-5//Transporter activity
Medroxyprogesteroneacetate//Gamma-aminobutyric acid receptor subunit alpha-6//Inhibitory extracellular ligand-gated ion channel activity
Medroxyprogesteroneacetate//Gamma-aminobutyric acid receptor subunit beta-1//Ligand-gated ion channel activity
Medroxyprogesteroneacetate//Gamma-aminobutyric acid receptor subunit beta-2//Inhibitory extracellular ligand-gated ion channel activity
Medroxyprogesteroneacetate//Gamma-aminobutyric acid receptor subunit beta-3//Gaba-gated chloride ion channel activity
Medroxyprogesteroneacetate//Gamma-aminobutyric acid receptor subunit delta//Gaba-a receptor activity
Medroxyprogesteroneacetate//Gamma-aminobutyric acid receptor subunit epsilon//Inhibitory extracellular ligand-gated ion channel activity
Medroxyprogesteroneacetate//Gamma-aminobutyric acid receptor subunit gamma-1//Inhibitory extracellular ligand-gated ion channel activity
Medroxyprogesteroneacetate//Gamma-aminobutyric acid receptor subunit gamma-2//Inhibitory extracellular ligand-gated ion channel activity
Medroxyprogesteroneacetate//Gamma-aminobutyric acid receptor subunit gamma-3//Inhibitory extracellular ligand-gated ion channel activity
Medroxyprogesteroneacetate//Gamma-aminobutyric acid receptor subunit pi//Gaba-a receptor activity
Medroxyprogesteroneacetate//Gamma-aminobutyric acid receptor subunit theta//Transmembrane signaling receptor activity
Cisapride//5-hydroxytryptamine receptor 4//Serotonin receptor activity
Cisapride//5-hydroxytryptamine receptor 3A//Voltage-gated potassium channel activity
Cisapride//5-hydroxytryptamine receptor 2A//Virus receptor activity
Cisapride//Potassium voltage-gated channel subfamily H member 2//Voltage-gated potassium channel activity involved in ventricular cardiac muscle cell action potential repolarization
Chloroquine//Tumor necrosis factor//Tumor necrosis factor receptor binding
Chloroquine//Glutathione S-transferase A2//Glutathione transferase activity
Chloroquine//Toll-like receptor 9//Transmembrane signaling receptor activity
Chloroquine//Glutathione S-transferase//Glutathione transferase activity
Chloroquine//High mobility group protein B1//Transcription factor binding
Chloroquine//Glutathione S-transferase Mu 1//Protein homodimerization activity
Chloroquine//Angiotensin-converting enzyme 2//Zinc ion binding
Bisoprolol//Beta-1 adrenergic receptor//Receptor signaling protein activity
Bisoprolol//Beta-2 adrenergic receptor//Protein homodimerization activity
Imatinib//Breakpoint cluster region protein//Rho guanyl-nucleotide exchange factor activity
Imatinib//Mast/stem cell growth factor receptor Kit//Transmembrane receptor protein tyrosine kinase activity
Imatinib//High affinity nerve growth factor receptor//Transmembrane receptor protein tyrosine kinase activity
Imatinib//Macrophage colony-stimulating factor 1 receptor//Protein homodimerization activity
Imatinib//Platelet-derived growth factor receptor alpha//Vascular endothelial growth factor-activated receptor activity
Imatinib//Epithelial discoidin domain-containing receptor 1//Transmembrane receptor protein tyrosine kinase activity
Imatinib//Tyrosine-protein kinase ABL1//Syntaxin binding
Imatinib//Platelet-derived growth factor receptor beta//Vascular endothelial growth factor binding
Nicardipine//Voltage-dependent L-type calcium channel subunit alpha-1C//Voltage-gated calcium channel activity
Nicardipine//Voltage-dependent L-type calcium channel subunit beta-2//Voltage-gated calcium channel activity
Nicardipine//Voltage-dependent calcium channel subunit alpha-2/delta-1//Voltage-gated calcium channel activity
Nicardipine//Voltage-dependent L-type calcium channel subunit alpha-1D//Voltage-gated calcium channel activity involved sa node cell action potential
Nicardipine//Calcium/calmodulin-dependent 3',5'-cyclic nucleotide phosphodiesterase 1A//Metal ion binding
Nicardipine//Calcium/calmodulin-dependent 3',5'-cyclic nucleotide phosphodiesterase 1B//Metal ion binding
Nicardipine//Alpha-1A adrenergic receptor//Protein heterodimerization activity
Nicardipine//Alpha-1B adrenergic receptor//Protein heterodimerization activity
Nicardipine//Alpha-1D adrenergic receptor//Alpha1-adrenergic receptor activity
Nicardipine//Muscarinic acetylcholine receptor M1//Phosphatidylinositol phospholipase c activity
Nicardipine//Muscarinic acetylcholine receptor M2//G-protein coupled acetylcholine receptor activity
Nicardipine//Muscarinic acetylcholine receptor M3//Receptor activity
Nicardipine//Muscarinic acetylcholine receptor M4//Guanyl-nucleotide exchange factor activity
Nicardipine//Muscarinic acetylcholine receptor M5//Phosphatidylinositol phospholipase c activity
Nicardipine//Calmodulin//Titin binding
Fluphenazine//D(2) dopamine receptor//Potassium channel regulator activity
Fluphenazine//D(1A) dopamine receptor//G-protein coupled amine receptor activity
Fluphenazine//Calmodulin//Titin binding
Fluphenazine//Androgen receptor//Zinc ion binding
Fluphenazine//5-hydroxytryptamine receptor 2A//Virus receptor activity
Fluphenazine//5-hydroxytryptamine receptor 2C//Serotonin receptor activity
Niacin//Hydroxycarboxylic acid receptor 3//G-protein coupled receptor activity
Niacin//Nicotinate-nucleotide pyrophosphorylase [carboxylating]//Protein homodimerization activity
Clorazepate//Gamma-aminobutyric acid receptor subunit alpha-1//Inhibitory extracellular ligand-gated ion channel activity
Clorazepate//Gamma-aminobutyric acid receptor subunit alpha-2//Inhibitory extracellular ligand-gated ion channel activity
Clorazepate//Gamma-aminobutyric acid receptor subunit alpha-3//Inhibitory extracellular ligand-gated ion channel activity
Clorazepate//Gamma-aminobutyric acid receptor subunit alpha-4//Inhibitory extracellular ligand-gated ion channel activity
Clorazepate//Gamma-aminobutyric acid receptor subunit alpha-5//Transporter activity
Clorazepate//Gamma-aminobutyric acid receptor subunit alpha-6//Inhibitory extracellular ligand-gated ion channel activity
Clorazepate//Gamma-aminobutyric acid receptor subunit beta-1//Ligand-gated ion channel activity
Clorazepate//Gamma-aminobutyric acid receptor subunit beta-2//Inhibitory extracellular ligand-gated ion channel activity
Clorazepate//Gamma-aminobutyric acid receptor subunit beta-3//Gaba-gated chloride ion channel activity
Clorazepate//Gamma-aminobutyric acid receptor subunit delta//Gaba-a receptor activity
Clorazepate//Gamma-aminobutyric acid receptor subunit epsilon//Inhibitory extracellular ligand-gated ion channel activity
Clorazepate//Gamma-aminobutyric acid receptor subunit gamma-1//Inhibitory extracellular ligand-gated ion channel activity
Clorazepate//Gamma-aminobutyric acid receptor subunit gamma-2//Inhibitory extracellular ligand-gated ion channel activity
Clorazepate//Gamma-aminobutyric acid receptor subunit gamma-3//Inhibitory extracellular ligand-gated ion channel activity
Clorazepate//Gamma-aminobutyric acid receptor subunit pi//Gaba-a receptor activity
Clorazepate//Gamma-aminobutyric acid receptor subunit theta//Transmembrane signaling receptor activity
Clorazepate//Gamma-aminobutyric acid receptor subunit alpha-1//Inhibitory extracellular ligand-gated ion channel activity
Clorazepate//Gamma-aminobutyric acid receptor subunit alpha-2//Inhibitory extracellular ligand-gated ion channel activity
Clorazepate//Gamma-aminobutyric acid receptor subunit alpha-3//Inhibitory extracellular ligand-gated ion channel activity
Clorazepate//Gamma-aminobutyric acid receptor subunit alpha-5//Transporter activity
Clorazepate//Gamma-aminobutyric acid receptor subunit gamma-1//Inhibitory extracellular ligand-gated ion channel activity
Clorazepate//Gamma-aminobutyric acid receptor subunit gamma-2//Inhibitory extracellular ligand-gated ion channel activity
Clorazepate//Gamma-aminobutyric acid receptor subunit gamma-3//Inhibitory extracellular ligand-gated ion channel activity
Guanabenz//Alpha-2A adrenergic receptor//Thioesterase binding
Guanabenz//Alpha-2B adrenergic receptor//Epinephrine binding
Clofarabine//Ribonucleoside-diphosphate reductase large subunit//Ribonucleoside-diphosphate reductase activity, thioredoxin disulfide as acceptor
Clofarabine//DNA polymerase alpha catalytic subunit//Protein kinase binding
Dexmedetomidine//Alpha-2A adrenergic receptor//Thioesterase binding
Clofibrate//Peroxisome proliferator-activated receptor alpha//Zinc ion binding
Astemizole//Histamine H1 receptor//Histamine receptor activity
Astemizole//Potassium voltage-gated channel subfamily H member 2//Voltage-gated potassium channel activity involved in ventricular cardiac muscle cell action potential repolarization
Astemizole//Potassium voltage-gated channel subfamily H member 1//Phosphorelay sensor kinase activity
Astemizole//Microtubule-associated protein tau//Structural constituent of cytoskeleton
Adenosine//Adenosine receptor A2a//Identical protein binding
Adenosine//Adenosine receptor A2b//G-protein coupled adenosine receptor activity
Adenosine//Adenosine receptor A3//G-protein coupled adenosine receptor activity
Adenosine//Adenosine receptor A1//Purine nucleoside binding
Mebendazole//Tubulin alpha-1A chain//Tubulin is the major constituent of microtubules. It binds two moles of GTP, one at an exchangeable site on the beta chain and one at a non-exchangeable site on the alpha chain.
Mebendazole//Tubulin beta-4B chain//Unfolded protein binding
Dextropropoxyphene//Delta-type opioid receptor//Opioid receptor activity
Dextropropoxyphene//Kappa-type opioid receptor//Opioid receptor activity
Dextropropoxyphene//Mu-type opioid receptor//Voltage-gated calcium channel activity
Dextropropoxyphene//Liver carboxylesterase 1//Triglyceride lipase activity
Mitotane//Adrenodoxin, mitochondrial//Iron ion binding
Mitotane//Cytochrome P450 11B1, mitochondrial//Steroid 11-beta-monooxygenase activity
Mitotane//Estrogen receptor//Zinc ion binding
Mitotane//Progesterone receptor//Zinc ion binding
Mitotane//Androgen receptor//Zinc ion binding
Estrone//Estrogen receptor//Zinc ion binding
Estrone//Estrogen receptor beta//Zinc ion binding
Estrone//Androgen receptor//Zinc ion binding
Estrone//Aromatase//Oxygen binding
Estrone//Sex hormone-binding globulin//Androgen binding
Epinephrine//Alpha-1A adrenergic receptor//Protein heterodimerization activity
Epinephrine//Alpha-1B adrenergic receptor//Protein heterodimerization activity
Epinephrine//Beta-1 adrenergic receptor//Receptor signaling protein activity
Epinephrine//Alpha-2A adrenergic receptor//Thioesterase binding
Epinephrine//Beta-2 adrenergic receptor//Protein homodimerization activity
Epinephrine//Alpha-2B adrenergic receptor//Epinephrine binding
Epinephrine//Alpha-1D adrenergic receptor//Alpha1-adrenergic receptor activity
Epinephrine//Tumor necrosis factor//Tumor necrosis factor receptor binding
Chlorpropamide//ATP-binding cassette sub-family C member 8//Sulfonylurea receptor activity
Aprepitant//Substance-P receptor//Tachykinin receptor activity
Galantamine//Acetylcholinesterase//Serine hydrolase activity
Galantamine//Neuronal acetylcholine receptor subunit alpha-7//Toxic substance binding
Galantamine//Cholinesterase//Identical protein binding
Isoflurophate//Acetylcholinesterase//Serine hydrolase activity
Isoflurophate//Cholinesterase//Identical protein binding
Losartan//Type-1 angiotensin II receptor//Protein heterodimerization activity
Midazolam//Gamma-aminobutyric acid receptor subunit alpha-1//Inhibitory extracellular ligand-gated ion channel activity
Midazolam//Gamma-aminobutyric acid receptor subunit alpha-2//Inhibitory extracellular ligand-gated ion channel activity
Midazolam//Gamma-aminobutyric acid receptor subunit alpha-3//Inhibitory extracellular ligand-gated ion channel activity
Midazolam//Gamma-aminobutyric acid receptor subunit alpha-4//Inhibitory extracellular ligand-gated ion channel activity
Midazolam//Gamma-aminobutyric acid receptor subunit alpha-5//Transporter activity
Midazolam//Gamma-aminobutyric acid receptor subunit alpha-6//Inhibitory extracellular ligand-gated ion channel activity
Midazolam//Gamma-aminobutyric acid receptor subunit beta-1//Ligand-gated ion channel activity
Midazolam//Gamma-aminobutyric acid receptor subunit beta-2//Inhibitory extracellular ligand-gated ion channel activity
Midazolam//Gamma-aminobutyric acid receptor subunit beta-3//Gaba-gated chloride ion channel activity
Midazolam//Gamma-aminobutyric acid receptor subunit delta//Gaba-a receptor activity
Midazolam//Gamma-aminobutyric acid receptor subunit epsilon//Inhibitory extracellular ligand-gated ion channel activity
Midazolam//Gamma-aminobutyric acid receptor subunit gamma-1//Inhibitory extracellular ligand-gated ion channel activity
Midazolam//Gamma-aminobutyric acid receptor subunit gamma-2//Inhibitory extracellular ligand-gated ion channel activity
Midazolam//Gamma-aminobutyric acid receptor subunit gamma-3//Inhibitory extracellular ligand-gated ion channel activity
Midazolam//Gamma-aminobutyric acid receptor subunit pi//Gaba-a receptor activity
Midazolam//Gamma-aminobutyric acid receptor subunit theta//Transmembrane signaling receptor activity
Midazolam//Gamma-aminobutyric acid receptor subunit alpha-1//Inhibitory extracellular ligand-gated ion channel activity
Midazolam//Gamma-aminobutyric acid receptor subunit alpha-2//Inhibitory extracellular ligand-gated ion channel activity
Midazolam//Gamma-aminobutyric acid receptor subunit alpha-3//Inhibitory extracellular ligand-gated ion channel activity
Midazolam//Gamma-aminobutyric acid receptor subunit alpha-5//Transporter activity
Midazolam//Gamma-aminobutyric acid receptor subunit gamma-1//Inhibitory extracellular ligand-gated ion channel activity
Midazolam//Gamma-aminobutyric acid receptor subunit gamma-2//Inhibitory extracellular ligand-gated ion channel activity
Midazolam//Gamma-aminobutyric acid receptor subunit gamma-3//Inhibitory extracellular ligand-gated ion channel activity
Mycophenolatemofetil//Inosine-5'-monophosphate dehydrogenase 1//Rna binding
Mycophenolatemofetil//Inosine-5'-monophosphate dehydrogenase 2//Rna binding
Mycophenolatemofetil//6-pyruvoyl tetrahydrobiopterin synthase//Metal ion binding
Flurazepam//Gamma-aminobutyric acid receptor subunit alpha-1//Inhibitory extracellular ligand-gated ion channel activity
Flurazepam//Gamma-aminobutyric acid receptor subunit alpha-2//Inhibitory extracellular ligand-gated ion channel activity
Flurazepam//Gamma-aminobutyric acid receptor subunit alpha-3//Inhibitory extracellular ligand-gated ion channel activity
Flurazepam//Gamma-aminobutyric acid receptor subunit alpha-4//Inhibitory extracellular ligand-gated ion channel activity
Flurazepam//Gamma-aminobutyric acid receptor subunit alpha-5//Transporter activity
Flurazepam//Gamma-aminobutyric acid receptor subunit alpha-6//Inhibitory extracellular ligand-gated ion channel activity
Flurazepam//Gamma-aminobutyric acid receptor subunit beta-1//Ligand-gated ion channel activity
Flurazepam//Gamma-aminobutyric acid receptor subunit beta-2//Inhibitory extracellular ligand-gated ion channel activity
Flurazepam//Gamma-aminobutyric acid receptor subunit beta-3//Gaba-gated chloride ion channel activity
Flurazepam//Gamma-aminobutyric acid receptor subunit delta//Gaba-a receptor activity
Flurazepam//Gamma-aminobutyric acid receptor subunit epsilon//Inhibitory extracellular ligand-gated ion channel activity
Flurazepam//Gamma-aminobutyric acid receptor subunit gamma-1//Inhibitory extracellular ligand-gated ion channel activity
Flurazepam//Gamma-aminobutyric acid receptor subunit gamma-2//Inhibitory extracellular ligand-gated ion channel activity
Flurazepam//Gamma-aminobutyric acid receptor subunit gamma-3//Inhibitory extracellular ligand-gated ion channel activity
Flurazepam//Gamma-aminobutyric acid receptor subunit pi//Gaba-a receptor activity
Flurazepam//Gamma-aminobutyric acid receptor subunit theta//Transmembrane signaling receptor activity
Flurazepam//Gamma-aminobutyric acid receptor subunit alpha-1//Inhibitory extracellular ligand-gated ion channel activity
Flurazepam//Gamma-aminobutyric acid receptor subunit alpha-2//Inhibitory extracellular ligand-gated ion channel activity
Flurazepam//Gamma-aminobutyric acid receptor subunit alpha-3//Inhibitory extracellular ligand-gated ion channel activity
Flurazepam//Gamma-aminobutyric acid receptor subunit alpha-5//Transporter activity
Flurazepam//Gamma-aminobutyric acid receptor subunit gamma-1//Inhibitory extracellular ligand-gated ion channel activity
Flurazepam//Gamma-aminobutyric acid receptor subunit gamma-2//Inhibitory extracellular ligand-gated ion channel activity
Flurazepam//Gamma-aminobutyric acid receptor subunit gamma-3//Inhibitory extracellular ligand-gated ion channel activity
Daunorubicin//DNA topoisomerase 2-alpha//Ubiquitin binding
Daunorubicin//DNA topoisomerase 2-beta//Protein kinase c binding
Furosemide//Solute carrier family 12 member 1//Sodium:potassium:chloride symporter activity
Furosemide//Carbonic anhydrase 2//Zinc ion binding
Furosemide//G-protein coupled receptor 35//G-protein coupled receptor activity
Ergotamine//5-hydroxytryptamine receptor 1D//Serotonin receptor activity
Ergotamine//5-hydroxytryptamine receptor 1B//Serotonin receptor activity
Ergotamine//5-hydroxytryptamine receptor 2A//Virus receptor activity
Ergotamine//D(2) dopamine receptor//Potassium channel regulator activity
Ergotamine//Alpha-1A adrenergic receptor//Protein heterodimerization activity
Ergotamine//Alpha-1B adrenergic receptor//Protein heterodimerization activity
Ergotamine//Alpha-1D adrenergic receptor//Alpha1-adrenergic receptor activity
Ergotamine//Alpha-2A adrenergic receptor//Thioesterase binding
Ergotamine//D(1A) dopamine receptor//G-protein coupled amine receptor activity
Ergotamine//D(1B) dopamine receptor//G-protein coupled amine receptor activity
Ergotamine//5-hydroxytryptamine receptor 1A//Serotonin receptor activity
Ergotamine//5-hydroxytryptamine receptor 1F//Serotonin receptor activity
Ergotamine//5-hydroxytryptamine receptor 2C//Serotonin receptor activity
Ergotamine//5-hydroxytryptamine receptor 2B//Serotonin receptor activity
Ergotamine//Alpha-2C adrenergic receptor//Protein homodimerization activity
Eplerenone//Mineralocorticoid receptor//Zinc ion binding
Methazolamide//Carbonic anhydrase 1//Zinc ion binding
Methazolamide//Carbonic anhydrase 2//Zinc ion binding
Methazolamide//Carbonic anhydrase 4//Zinc ion binding
Methazolamide//Carbonic anhydrase 3//Zinc ion binding
Methazolamide//Carbonic anhydrase 7//Zinc ion binding
Naltrexone//Delta-type opioid receptor//Opioid receptor activity
Naltrexone//Kappa-type opioid receptor//Opioid receptor activity
Naltrexone//Mu-type opioid receptor//Voltage-gated calcium channel activity
Diethylcarbamazine//Arachidonate 5-lipoxygenase//Iron ion binding
Diethylcarbamazine//Prostaglandin G/H synthase 1//Prostaglandin-endoperoxide synthase activity
Flurbiprofen//Prostaglandin G/H synthase 1//Prostaglandin-endoperoxide synthase activity
Flurbiprofen//Prostaglandin G/H synthase 2//Prostaglandin-endoperoxide synthase activity
Apomorphine//D(4) dopamine receptor//Sh3 domain binding
Apomorphine//D(2) dopamine receptor//Potassium channel regulator activity
Apomorphine//D(3) dopamine receptor//G-protein coupled amine receptor activity
Apomorphine//D(1B) dopamine receptor//G-protein coupled amine receptor activity
Apomorphine//D(1A) dopamine receptor//G-protein coupled amine receptor activity
Apomorphine//Alpha-2C adrenergic receptor//Protein homodimerization activity
Apomorphine//Alpha-2B adrenergic receptor//Epinephrine binding
Apomorphine//5-hydroxytryptamine receptor 1A//Serotonin receptor activity
Apomorphine//5-hydroxytryptamine receptor 2A//Virus receptor activity
Apomorphine//5-hydroxytryptamine receptor 2B//Serotonin receptor activity
Apomorphine//5-hydroxytryptamine receptor 2C//Serotonin receptor activity
Apomorphine//Alpha-2A adrenergic receptor//Thioesterase binding
Apomorphine//5-hydroxytryptamine receptor 1D//Serotonin receptor activity
Apomorphine//5-hydroxytryptamine receptor 1B//Serotonin receptor activity
Azatadine//Histamine H1 receptor//Histamine receptor activity
Clodronicacid//ADP/ATP translocase 2//Ubiquitin protein ligase binding
Imiquimod//Toll-like receptor 7//Transmembrane signaling receptor activity
Nateglinide//ATP-binding cassette sub-family C member 8//Sulfonylurea receptor activity
Nateglinide//Peroxisome proliferator-activated receptor gamma//Zinc ion binding
Esomeprazole//Potassium-transporting ATPase alpha chain 1//Sodium:potassium-exchanging atpase activity
Esomeprazole//N(G),N(G)-dimethylarginine dimethylaminohydrolase 1//Metal ion binding
Meclizine//Histamine H1 receptor//Histamine receptor activity
Meclizine//Nuclear receptor subfamily 1 group I member 3//Zinc ion binding
Hydrocortisone//Glucocorticoid receptor//Zinc ion binding
Hydrocortisone//Annexin A1//Structural molecule activity
Modafinil//Alpha-1B adrenergic receptor//Protein heterodimerization activity
Modafinil//Sodium-dependent dopamine transporter//Monoamine transmembrane transporter activity
Carbinoxamine//Histamine H1 receptor//Histamine receptor activity
Etodolac//Prostaglandin G/H synthase 2//Prostaglandin-endoperoxide synthase activity
Etodolac//Prostaglandin G/H synthase 1//Prostaglandin-endoperoxide synthase activity
Etodolac//Retinoic acid receptor RXR-alpha//Zinc ion binding
Epinastine//Histamine H1 receptor//Histamine receptor activity
Epinastine//Histamine H2 receptor//Histamine receptor activity
Epinastine//Alpha-1A adrenergic receptor//Protein heterodimerization activity
Epinastine//Alpha-2A adrenergic receptor//Thioesterase binding
Epinastine//5-hydroxytryptamine receptor 2A//Virus receptor activity
Epinastine//5-hydroxytryptamine receptor 7//Serotonin receptor activity
Isoflurane//Gamma-aminobutyric acid receptor subunit alpha-1//Inhibitory extracellular ligand-gated ion channel activity
Isoflurane//Calcium-transporting ATPase type 2C member 1//Signal transducer activity
Isoflurane//Glycine receptor subunit alpha-1//Transmitter-gated ion channel activity
Isoflurane//Glutamate receptor 1//Pdz domain binding
Isoflurane//Potassium voltage-gated channel subfamily A member 1//Voltage-gated potassium channel activity
Isoflurane//ATP synthase subunit delta, mitochondrial//Transporter activity
Isoflurane//Calmodulin//Titin binding
Isoflurane//Gamma-aminobutyric acid receptor subunit alpha-1//Inhibitory extracellular ligand-gated ion channel activity
Isoflurane//Gamma-aminobutyric acid receptor subunit alpha-2//Inhibitory extracellular ligand-gated ion channel activity
Isoflurane//Gamma-aminobutyric acid receptor subunit alpha-3//Inhibitory extracellular ligand-gated ion channel activity
Isoflurane//Gamma-aminobutyric acid receptor subunit alpha-4//Inhibitory extracellular ligand-gated ion channel activity
Isoflurane//Gamma-aminobutyric acid receptor subunit alpha-5//Transporter activity
Isoflurane//Gamma-aminobutyric acid receptor subunit alpha-6//Inhibitory extracellular ligand-gated ion channel activity
Isoflurane//Gamma-aminobutyric acid receptor subunit beta-1//Ligand-gated ion channel activity
Isoflurane//Gamma-aminobutyric acid receptor subunit beta-2//Inhibitory extracellular ligand-gated ion channel activity
Isoflurane//Gamma-aminobutyric acid receptor subunit beta-3//Gaba-gated chloride ion channel activity
Isoflurane//Gamma-aminobutyric acid receptor subunit delta//Gaba-a receptor activity
Isoflurane//Gamma-aminobutyric acid receptor subunit epsilon//Inhibitory extracellular ligand-gated ion channel activity
Isoflurane//Gamma-aminobutyric acid receptor subunit gamma-1//Inhibitory extracellular ligand-gated ion channel activity
Isoflurane//Gamma-aminobutyric acid receptor subunit gamma-2//Inhibitory extracellular ligand-gated ion channel activity
Isoflurane//Gamma-aminobutyric acid receptor subunit gamma-3//Inhibitory extracellular ligand-gated ion channel activity
Isoflurane//Gamma-aminobutyric acid receptor subunit pi//Gaba-a receptor activity
Isoflurane//Gamma-aminobutyric acid receptor subunit theta//Transmembrane signaling receptor activity
Isoflurane//Neuronal acetylcholine receptor subunit alpha-4//Ligand-gated ion channel activity
Isoflurane//Neuronal acetylcholine receptor subunit beta-2//Ligand-gated ion channel activity
Ethotoin//Sodium channel protein type 5 subunit alpha//Voltage-gated sodium channel activity involved in sa node cell action potential
Ethotoin//Nuclear receptor subfamily 1 group I member 2//Zinc ion binding
Dolasetron//5-hydroxytryptamine receptor 3A//Voltage-gated potassium channel activity
Clopidogrel//P2Y purinoceptor 12//Guanyl-nucleotide exchange factor activity
Irinotecan//DNA topoisomerase I, mitochondrial//Dna topoisomerase type ii (atp-hydrolyzing) activity
Methimazole//Thyroid peroxidase//Peroxidase activity
Mometasone//Glucocorticoid receptor//Zinc ion binding
Mometasone//Progesterone receptor//Zinc ion binding
Hydrocortamate//Glucocorticoid receptor//Zinc ion binding
Malathion//Cholinesterase//Identical protein binding
Etoposide//DNA topoisomerase 2-alpha//Ubiquitin binding
Etoposide//DNA topoisomerase 2-beta//Protein kinase c binding
Estradiol//Estrogen receptor//Zinc ion binding
Estradiol//Estrogen receptor beta//Zinc ion binding
Estradiol//Nuclear receptor subfamily 1 group I member 2//Zinc ion binding
Estradiol//Neuronal acetylcholine receptor subunit alpha-4//Ligand-gated ion channel activity
Estradiol//G-protein coupled estrogen receptor 1//Steroid hormone binding
Estradiol//ATP synthase subunit a//Mitochondrial membrane ATP synthase (F(1)F(0) ATP synthase or Complex V) produces ATP from ADP in the presence of a proton gradient across the membrane which is generated by electron transport complexes of the respiratory chain. F-type ATPases consist of two structural domains, F(1) - containing the extramembraneous catalytic core and F(0) - containing the membrane proton channel, linked together by a central stalk and a peripheral stalk. During catalysis, ATP synthesis in the catalytic domain of F(1) is coupled via a rotary mechanism of the central stalk subunits to proton translocation. Key component of the proton channel; it may play a direct role in the translocation of protons across the membrane.
Estradiol//Beclin-1//Plays a central role in autophagy (PubMed:23184933). Acts as core subunit of the PI3K complex that mediates formation of phosphatidylinositol 3-phosphate; different complex forms are believed to play a role in multiple membrane trafficking pathways: PI3KC3-C1 is involved in initiation of autophagosomes and PI3KC3-C2 in maturation of autophagosomes and endocytosis. Involved in regulation of degradative endocytic trafficking and required for the abcission step in cytokinesis, probably in the context of PI3KC3-C2 (PubMed:20643123, PubMed:20208530). Essential for the formation of PI3KC3-C2 but not PI3KC3-C1 PI3K complex forms. Involved in endocytosis (PubMed:25275521). Protects against infection by a neurovirulent strain of Sindbis virus (PubMed:9765397). May play a role in antiviral host defense.
Mefenamicacid//Prostaglandin G/H synthase 1//Prostaglandin-endoperoxide synthase activity
Mefenamicacid//Prostaglandin G/H synthase 2//Prostaglandin-endoperoxide synthase activity
Naproxen//Prostaglandin G/H synthase 1//Prostaglandin-endoperoxide synthase activity
Naproxen//Prostaglandin G/H synthase 2//Prostaglandin-endoperoxide synthase activity
Candesartancilexetil//Type-1 angiotensin II receptor//Protein heterodimerization activity
Alfentanil//Mu-type opioid receptor//Voltage-gated calcium channel activity
Dicyclomine//Muscarinic acetylcholine receptor M1//Phosphatidylinositol phospholipase c activity
Dicyclomine//Muscarinic acetylcholine receptor M2//G-protein coupled acetylcholine receptor activity
Minaprine//Amine oxidase [flavin-containing] A//Serotonin binding
Minaprine//5-hydroxytryptamine receptor 2B//Serotonin receptor activity
Minaprine//5-hydroxytryptamine receptor 2A//Virus receptor activity
Minaprine//5-hydroxytryptamine receptor 2C//Serotonin receptor activity
Minaprine//Acetylcholinesterase//Serine hydrolase activity
Minaprine//Sodium-dependent serotonin transporter//Serotonin:sodium symporter activity
Minaprine//D(1A) dopamine receptor//G-protein coupled amine receptor activity
Minaprine//D(2) dopamine receptor//Potassium channel regulator activity
Minaprine//Muscarinic acetylcholine receptor M1//Phosphatidylinositol phospholipase c activity
Indapamide//Solute carrier family 12 member 3//Transporter activity
Biperiden//Muscarinic acetylcholine receptor M1//Phosphatidylinositol phospholipase c activity
Fentanyl//Mu-type opioid receptor//Voltage-gated calcium channel activity
Fentanyl//Delta-type opioid receptor//Opioid receptor activity
Fentanyl//Kappa-type opioid receptor//Opioid receptor activity
Fentanyl//Multidrug resistance protein 1//Xenobiotic-transporting atpase activity
Meloxicam//Prostaglandin G/H synthase 2//Prostaglandin-endoperoxide synthase activity
Meloxicam//Prostaglandin G/H synthase 1//Prostaglandin-endoperoxide synthase activity
Acetazolamide//Carbonic anhydrase 1//Zinc ion binding
Acetazolamide//Carbonic anhydrase 2//Zinc ion binding
Acetazolamide//Carbonic anhydrase 4//Zinc ion binding
Acetazolamide//Carbonic anhydrase 12//Zinc ion binding
Acetazolamide//Carbonic anhydrase 14//Metal ion binding
Acetazolamide//Carbonic anhydrase 3//Zinc ion binding
Acetazolamide//Carbonic anhydrase 7//Zinc ion binding
Disulfiram//Aldehyde dehydrogenase, mitochondrial//Electron carrier activity
Disulfiram//Dopamine beta-hydroxylase//L-ascorbic acid binding
Diazepam//Gamma-aminobutyric acid receptor subunit alpha-1//Inhibitory extracellular ligand-gated ion channel activity
Diazepam//Gamma-aminobutyric acid receptor subunit alpha-2//Inhibitory extracellular ligand-gated ion channel activity
Diazepam//Gamma-aminobutyric acid receptor subunit alpha-3//Inhibitory extracellular ligand-gated ion channel activity
Diazepam//Gamma-aminobutyric acid receptor subunit alpha-4//Inhibitory extracellular ligand-gated ion channel activity
Diazepam//Gamma-aminobutyric acid receptor subunit alpha-5//Transporter activity
Diazepam//Gamma-aminobutyric acid receptor subunit alpha-6//Inhibitory extracellular ligand-gated ion channel activity
Diazepam//Gamma-aminobutyric acid receptor subunit beta-1//Ligand-gated ion channel activity
Diazepam//Gamma-aminobutyric acid receptor subunit beta-2//Inhibitory extracellular ligand-gated ion channel activity
Diazepam//Gamma-aminobutyric acid receptor subunit beta-3//Gaba-gated chloride ion channel activity
Diazepam//Gamma-aminobutyric acid receptor subunit delta//Gaba-a receptor activity
Diazepam//Gamma-aminobutyric acid receptor subunit epsilon//Inhibitory extracellular ligand-gated ion channel activity
Diazepam//Gamma-aminobutyric acid receptor subunit gamma-1//Inhibitory extracellular ligand-gated ion channel activity
Diazepam//Gamma-aminobutyric acid receptor subunit gamma-2//Inhibitory extracellular ligand-gated ion channel activity
Diazepam//Gamma-aminobutyric acid receptor subunit gamma-3//Inhibitory extracellular ligand-gated ion channel activity
Diazepam//Gamma-aminobutyric acid receptor subunit pi//Gaba-a receptor activity
Diazepam//Gamma-aminobutyric acid receptor subunit theta//Transmembrane signaling receptor activity
Diazepam//Gamma-aminobutyric acid receptor subunit alpha-1//Inhibitory extracellular ligand-gated ion channel activity
Diazepam//Gamma-aminobutyric acid receptor subunit alpha-2//Inhibitory extracellular ligand-gated ion channel activity
Diazepam//Gamma-aminobutyric acid receptor subunit alpha-3//Inhibitory extracellular ligand-gated ion channel activity
Diazepam//Gamma-aminobutyric acid receptor subunit alpha-5//Transporter activity
Diazepam//Gamma-aminobutyric acid receptor subunit gamma-1//Inhibitory extracellular ligand-gated ion channel activity
Diazepam//Gamma-aminobutyric acid receptor subunit gamma-2//Inhibitory extracellular ligand-gated ion channel activity
Diazepam//Gamma-aminobutyric acid receptor subunit gamma-3//Inhibitory extracellular ligand-gated ion channel activity
Mifepristone//Progesterone receptor//Zinc ion binding
Mifepristone//Glucocorticoid receptor//Zinc ion binding
Mifepristone//Nuclear receptor subfamily 1 group I member 2//Zinc ion binding
Brompheniramine//Histamine H1 receptor//Histamine receptor activity
Brompheniramine//Muscarinic acetylcholine receptor M1//Phosphatidylinositol phospholipase c activity
Brompheniramine//Muscarinic acetylcholine receptor M2//G-protein coupled acetylcholine receptor activity
Brompheniramine//Muscarinic acetylcholine receptor M3//Receptor activity
Brompheniramine//Muscarinic acetylcholine receptor M4//Guanyl-nucleotide exchange factor activity
Brompheniramine//Muscarinic acetylcholine receptor M5//Phosphatidylinositol phospholipase c activity
Loperamide//Mu-type opioid receptor//Voltage-gated calcium channel activity
Loperamide//Delta-type opioid receptor//Opioid receptor activity
Loperamide//Kappa-type opioid receptor//Opioid receptor activity
Loperamide//Voltage-dependent P/Q-type calcium channel subunit alpha-1A//Voltage-gated calcium channel activity
Loperamide//Calmodulin//Titin binding
Loperamide//Nuclear receptor subfamily 1 group I member 3//Zinc ion binding
Dobutamine//Beta-1 adrenergic receptor//Receptor signaling protein activity
Dobutamine//Beta-2 adrenergic receptor//Protein homodimerization activity
Dobutamine//Alpha-1A adrenergic receptor//Protein heterodimerization activity
Dobutamine//Alpha-1B adrenergic receptor//Protein heterodimerization activity
Dobutamine//Alpha-1D adrenergic receptor//Alpha1-adrenergic receptor activity
Dobutamine//Estrogen receptor//Zinc ion binding
Donepezil//Acetylcholinesterase//Serine hydrolase activity
Donepezil//5-hydroxytryptamine receptor 2A//Virus receptor activity
Donepezil//Cholinesterase//Identical protein binding
Donepezil//Nitric oxide synthase, brain//Tetrahydrobiopterin binding
Donepezil//Nuclear factor NF-kappa-B p100 subunit//Transcriptional activator activity, rna polymerase ii core promoter proximal region sequence-specific binding
Donepezil//Glutamate receptor ionotropic, NMDA 1//Voltage-gated cation channel activity
Donepezil//Glutamate receptor ionotropic, NMDA 2A//Zinc ion binding
Donepezil//Glutamate receptor ionotropic, NMDA 2B//Zinc ion binding
Donepezil//Glutamate receptor ionotropic, NMDA 2C//Nmda glutamate receptor activity
Donepezil//Glutamate receptor ionotropic, NMDA 2D//Nmda glutamate receptor activity
Donepezil//Glutamate receptor ionotropic, NMDA 3A//Protein phosphatase 2a binding
Donepezil//Glutamate receptor ionotropic, NMDA 3B//Nmda glutamate receptor activity
Clofazimine//Peroxisome proliferator-activated receptor gamma//Zinc ion binding
Clofazimine//Potassium voltage-gated channel subfamily A member 3//Voltage-gated ion channel activity
Cysteamine//Neuropeptide Y receptor type 2//Receptor activity
Methylphenobarbital//Gamma-aminobutyric acid receptor subunit alpha-1//Inhibitory extracellular ligand-gated ion channel activity
Methylphenobarbital//Gamma-aminobutyric acid receptor subunit alpha-2//Inhibitory extracellular ligand-gated ion channel activity
Methylphenobarbital//Gamma-aminobutyric acid receptor subunit alpha-3//Inhibitory extracellular ligand-gated ion channel activity
Methylphenobarbital//Gamma-aminobutyric acid receptor subunit alpha-4//Inhibitory extracellular ligand-gated ion channel activity
Methylphenobarbital//Gamma-aminobutyric acid receptor subunit alpha-5//Transporter activity
Methylphenobarbital//Gamma-aminobutyric acid receptor subunit alpha-6//Inhibitory extracellular ligand-gated ion channel activity
Methylphenobarbital//Neuronal acetylcholine receptor subunit alpha-4//Ligand-gated ion channel activity
Methylphenobarbital//Neuronal acetylcholine receptor subunit alpha-7//Toxic substance binding
Methylphenobarbital//Glutamate receptor 2//Ionotropic glutamate receptor activity
Methylphenobarbital//Glutamate receptor ionotropic, kainate 2//Kainate selective glutamate receptor activity
Methylphenobarbital//Nuclear receptor subfamily 1 group I member 2//Zinc ion binding
Dacarbazine//DNA polymerase alpha subunit B//Protein heterodimerization activity
Dacarbazine//6-phosphogluconate dehydrogenase, decarboxylating//Phosphogluconate dehydrogenase (decarboxylating) activity
Diflunisal//Prostaglandin G/H synthase 2//Prostaglandin-endoperoxide synthase activity
Diflunisal//Prostaglandin G/H synthase 1//Prostaglandin-endoperoxide synthase activity
Benzphetamine//Synaptic vesicular amine transporter//Monoamine transmembrane transporter activity
Benzphetamine//Alpha-2A adrenergic receptor//Thioesterase binding
Benzphetamine//Alpha-1A adrenergic receptor//Protein heterodimerization activity
Benzphetamine//Sodium-dependent dopamine transporter//Monoamine transmembrane transporter activity
Alprenolol//Beta-1 adrenergic receptor//Receptor signaling protein activity
Alprenolol//Beta-2 adrenergic receptor//Protein homodimerization activity
Alprenolol//5-hydroxytryptamine receptor 1A//Serotonin receptor activity
Alprenolol//Beta-3 adrenergic receptor//Protein homodimerization activity
Dorzolamide//Carbonic anhydrase 2//Zinc ion binding
Dorzolamide//Carbonic anhydrase 4//Zinc ion binding
Dorzolamide//Carbonic anhydrase 1//Zinc ion binding
Dorzolamide//Carbonic anhydrase 3//Zinc ion binding
Conivaptan//Vasopressin V1a receptor//Vasopressin receptor activity
Conivaptan//Vasopressin V2 receptor//Vasopressin receptor activity
Flupentixol//D(2) dopamine receptor//Potassium channel regulator activity
Flupentixol//5-hydroxytryptamine receptor 2A//Virus receptor activity
Flupentixol//D(1A) dopamine receptor//G-protein coupled amine receptor activity
Flupentixol//Alpha-1A adrenergic receptor//Protein heterodimerization activity
Flupentixol//Muscarinic acetylcholine receptor M1//Phosphatidylinositol phospholipase c activity
Eprosartan//Type-1 angiotensin II receptor//Protein heterodimerization activity
Clomifene//Estrogen receptor//Zinc ion binding
Clomifene//Sex hormone-binding globulin//Androgen binding
Isosorbidedinitrate//Atrial natriuretic peptide receptor 1//Protein kinase activity
Bumetanide//Solute carrier family 12 member 1//Sodium:potassium:chloride symporter activity
Bumetanide//Solute carrier family 12 member 2//Sodium:potassium:chloride symporter activity
Bumetanide//Solute carrier family 12 member 4//Protein kinase binding
Bumetanide//Solute carrier family 12 member 5//Protein kinase binding
Bumetanide//Cystic fibrosis transmembrane conductance regulator//Pdz domain binding
Granisetron//5-hydroxytryptamine receptor 3A//Voltage-gated potassium channel activity
Ethanol//Glycine receptor subunit alpha-1//Transmitter-gated ion channel activity
Ethanol//Glutamate receptor ionotropic, NMDA 3A//Protein phosphatase 2a binding
Ethanol//Glycine receptor subunit alpha-2//Transmitter-gated ion channel activity
Ethanol//Gamma-aminobutyric acid receptor subunit alpha-1//Inhibitory extracellular ligand-gated ion channel activity
Ethanol//Voltage-dependent L-type calcium channel subunit beta-1//Voltage-gated calcium channel activity
Ethanol//5-hydroxytryptamine receptor 3A//Voltage-gated potassium channel activity
Ethanol//Gamma-aminobutyric acid receptor subunit alpha-2//Inhibitory extracellular ligand-gated ion channel activity
Ethanol//Neuronal acetylcholine receptor subunit alpha-10//Receptor binding
Ethanol//Voltage-dependent L-type calcium channel subunit alpha-1C//Voltage-gated calcium channel activity
Ethanol//Gamma-aminobutyric acid receptor subunit alpha-5//Transporter activity
Ethanol//Gamma-aminobutyric acid receptor subunit alpha-4//Inhibitory extracellular ligand-gated ion channel activity
Ethanol//Gamma-aminobutyric acid receptor subunit alpha-3//Inhibitory extracellular ligand-gated ion channel activity
Ethanol//Glutamate receptor 1//Pdz domain binding
Ethanol//Voltage-dependent calcium channel gamma-1 subunit//Voltage-gated calcium channel activity
Ethanol//Neuronal acetylcholine receptor subunit alpha-2//Drug binding
Ethanol//Gamma-aminobutyric acid receptor subunit alpha-6//Inhibitory extracellular ligand-gated ion channel activity
Ethanol//Glutamate receptor 2//Ionotropic glutamate receptor activity
Ethanol//Glutamate receptor 4//Ionotropic glutamate receptor activity
Ethanol//Neuronal acetylcholine receptor subunit alpha-4//Ligand-gated ion channel activity
Ethanol//Neuronal acetylcholine receptor subunit beta-2//Ligand-gated ion channel activity
Ethanol//G protein-activated inward rectifier potassium channel 1//G-protein activated inward rectifier potassium channel activity
Ethanol//G protein-activated inward rectifier potassium channel 2//Inward rectifier potassium channel activity
Ethanol//Vascular cell adhesion protein 1//Primary amine oxidase activity
Ethanol//Equilibrative nucleoside transporter 1//Nucleoside transmembrane transporter activity
Ethanol//G protein-activated inward rectifier potassium channel 4//G-protein activated inward rectifier potassium channel activity
Ethanol//Neuronal acetylcholine receptor subunit alpha-7//Toxic substance binding
Ethanol//Neuronal acetylcholine receptor subunit alpha-9//Calcium channel activity
Ethanol//Gamma-aminobutyric acid receptor subunit beta-1//Ligand-gated ion channel activity
Ethanol//Gamma-aminobutyric acid receptor subunit beta-3//Gaba-gated chloride ion channel activity
Ethanol//Gamma-aminobutyric acid receptor subunit beta-2//Inhibitory extracellular ligand-gated ion channel activity
Ethanol//Voltage-dependent L-type calcium channel subunit alpha-1S//Voltage-gated calcium channel activity
Ethanol//Voltage-dependent L-type calcium channel subunit alpha-1D//Voltage-gated calcium channel activity involved sa node cell action potential
Ethanol//Neuronal acetylcholine receptor subunit beta-4//Ligand-gated ion channel activity
Ethanol//Neuronal acetylcholine receptor subunit alpha-3//Ligand-gated ion channel activity
Ethanol//Neuronal acetylcholine receptor subunit alpha-5//Ligand-gated ion channel activity
Ethanol//Neuronal acetylcholine receptor subunit beta-3//Drug binding
Ethanol//Gamma-aminobutyric acid receptor subunit gamma-1//Inhibitory extracellular ligand-gated ion channel activity
Ethanol//Gamma-aminobutyric acid receptor subunit gamma-3//Inhibitory extracellular ligand-gated ion channel activity
Ethanol//Gamma-aminobutyric acid receptor subunit epsilon//Inhibitory extracellular ligand-gated ion channel activity
Ethanol//Gamma-aminobutyric acid receptor subunit pi//Gaba-a receptor activity
Ethanol//Gamma-aminobutyric acid receptor subunit theta//Transmembrane signaling receptor activity
Ethanol//Gamma-aminobutyric acid receptor subunit delta//Gaba-a receptor activity
Ethanol//Equilibrative nucleoside transporter 2//Nucleoside transmembrane transporter activity
Ethanol//5-hydroxytryptamine receptor 3E//Serotonin-activated cation-selective channel activity
Ethanol//5-hydroxytryptamine receptor 3B//Serotonin-activated cation-selective channel activity
Ethanol//5-hydroxytryptamine receptor 3D//Serotonin-activated cation-selective channel activity
Ethanol//5-hydroxytryptamine receptor 3C//Serotonin-activated cation-selective channel activity
Ethanol//Voltage-dependent calcium channel gamma-2 subunit//Voltage-gated calcium channel activity
Ethanol//G protein-activated inward rectifier potassium channel 3//G-protein activated inward rectifier potassium channel activity
Etacrynicacid//Solute carrier family 12 member 1//Sodium:potassium:chloride symporter activity
Etacrynicacid//Sodium/potassium-transporting ATPase subunit alpha-1//Steroid hormone binding
Etacrynicacid//Glutathione S-transferase P//S-nitrosoglutathione binding
Cocaine//Sodium-dependent dopamine transporter//Monoamine transmembrane transporter activity
Cocaine//Sodium-dependent noradrenaline transporter//Norepinephrine:sodium symporter activity
Cocaine//Sodium-dependent serotonin transporter//Serotonin:sodium symporter activity
Cocaine//Sodium channel protein type 1 subunit alpha//Voltage-gated sodium channel activity
Cocaine//Sodium channel protein type 10 subunit alpha//Voltage-gated sodium channel activity
Cocaine//Sodium channel protein type 11 subunit alpha//Voltage-gated sodium channel activity
Cocaine//Sodium channel protein type 2 subunit alpha//Voltage-gated sodium channel activity
Cocaine//Sodium channel protein type 3 subunit alpha//Voltage-gated sodium channel activity
Cocaine//Sodium channel protein type 4 subunit alpha//Voltage-gated sodium channel activity
Cocaine//Sodium channel protein type 5 subunit alpha//Voltage-gated sodium channel activity involved in sa node cell action potential
Cocaine//Sodium channel protein type 7 subunit alpha//Mediates the voltage-dependent sodium ion permeability of excitable membranes. Assuming opened or closed conformations in response to the voltage difference across the membrane, the protein forms a sodium-selective channel through which Na(+) ions may pass in accordance with their electrochemical gradient.
Cocaine//Sodium channel protein type 8 subunit alpha//Voltage-gated sodium channel activity
Cocaine//Sodium channel protein type 9 subunit alpha//Voltage-gated sodium channel activity
Cocaine//Sodium channel subunit beta-2//Voltage-gated sodium channel activity involved in cardiac muscle cell action potential
Cocaine//Sodium channel subunit beta-3//Voltage-gated sodium channel activity involved in cardiac muscle cell action potential
Cocaine//Sodium channel subunit beta-4//Voltage-gated sodium channel activity involved in cardiac muscle cell action potential
Cocaine//Muscarinic acetylcholine receptor M1//Phosphatidylinositol phospholipase c activity
Cocaine//Muscarinic acetylcholine receptor M2//G-protein coupled acetylcholine receptor activity
Cocaine//Sigma non-opioid intracellular receptor 1//Opioid receptor activity
Cocaine//Liver carboxylesterase 1//Triglyceride lipase activity
Amantadine//Glutamate receptor ionotropic, NMDA 3A//Protein phosphatase 2a binding
Amantadine//D(2) dopamine receptor//Potassium channel regulator activity
Amantadine//Neuronal acetylcholine receptor subunit alpha-7//Toxic substance binding
Amantadine//Neuronal acetylcholine receptor subunit alpha-4//Ligand-gated ion channel activity
Amantadine//Neuronal acetylcholine receptor subunit alpha-3//Ligand-gated ion channel activity
Dinoprostone//Prostaglandin E2 receptor EP2 subtype//Prostaglandin e receptor activity
Dinoprostone//Prostaglandin E2 receptor EP1 subtype//Prostaglandin e receptor activity
Dinoprostone//Prostaglandin E2 receptor EP4 subtype//Prostaglandin e receptor activity
Almotriptan//5-hydroxytryptamine receptor 1D//Serotonin receptor activity
Almotriptan//5-hydroxytryptamine receptor 1B//Serotonin receptor activity
Buprenorphine//Kappa-type opioid receptor//Opioid receptor activity
Buprenorphine//Mu-type opioid receptor//Voltage-gated calcium channel activity
Buprenorphine//Delta-type opioid receptor//Opioid receptor activity
Cyclobenzaprine//5-hydroxytryptamine receptor 2A//Virus receptor activity
Cyclobenzaprine//5-hydroxytryptamine receptor 2B//Serotonin receptor activity
Cyclobenzaprine//5-hydroxytryptamine receptor 2C//Serotonin receptor activity
Cyclobenzaprine//5-hydroxytryptamine receptor 6//Serotonin receptor activity
Cyclobenzaprine//Sodium-dependent serotonin transporter//Serotonin:sodium symporter activity
Cyclobenzaprine//Sodium-dependent noradrenaline transporter//Norepinephrine:sodium symporter activity
Cyclobenzaprine//5-hydroxytryptamine receptor 7//Serotonin receptor activity
Cyclobenzaprine//Toll-like receptor 4//Transmembrane signaling receptor activity
Cyclobenzaprine//Aldehyde oxidase//Xanthine dehydrogenase activity
Famotidine//Histamine H2 receptor//Histamine receptor activity
Azacitidine//DNA (cytosine-5)-methyltransferase 1//Zinc ion binding
Mesoridazine//5-hydroxytryptamine receptor 2A//Virus receptor activity
Mesoridazine//D(2) dopamine receptor//Potassium channel regulator activity
Maprotiline//Sodium-dependent noradrenaline transporter//Norepinephrine:sodium symporter activity
Maprotiline//Muscarinic acetylcholine receptor M1//Phosphatidylinositol phospholipase c activity
Maprotiline//Histamine H1 receptor//Histamine receptor activity
Maprotiline//Muscarinic acetylcholine receptor M2//G-protein coupled acetylcholine receptor activity
Maprotiline//Muscarinic acetylcholine receptor M3//Receptor activity
Maprotiline//Muscarinic acetylcholine receptor M4//Guanyl-nucleotide exchange factor activity
Maprotiline//Muscarinic acetylcholine receptor M5//Phosphatidylinositol phospholipase c activity
Maprotiline//Alpha-1A adrenergic receptor//Protein heterodimerization activity
Maprotiline//Alpha-1B adrenergic receptor//Protein heterodimerization activity
Maprotiline//Alpha-1D adrenergic receptor//Alpha1-adrenergic receptor activity
Maprotiline//5-hydroxytryptamine receptor 2A//Virus receptor activity
Maprotiline//5-hydroxytryptamine receptor 2C//Serotonin receptor activity
Maprotiline//5-hydroxytryptamine receptor 7//Serotonin receptor activity
Maprotiline//D(2) dopamine receptor//Potassium channel regulator activity
Maprotiline//Alpha-2A adrenergic receptor//Thioesterase binding
Maprotiline//Alpha-2B adrenergic receptor//Epinephrine binding
Maprotiline//Alpha-2C adrenergic receptor//Protein homodimerization activity
Acetylsalicylicacid//Prostaglandin G/H synthase 1//Prostaglandin-endoperoxide synthase activity
Acetylsalicylicacid//Prostaglandin G/H synthase 2//Prostaglandin-endoperoxide synthase activity
Acetylsalicylicacid//Aldo-keto reductase family 1 member C1//Trans-1,2-dihydrobenzene-1,2-diol dehydrogenase activity
Acetylsalicylicacid//5'-AMP-activated protein kinase catalytic subunit alpha-1//Tau-protein kinase activity
Acetylsalicylicacid//5'-AMP-activated protein kinase catalytic subunit alpha-2//Protein serine/threonine/tyrosine kinase activity
Acetylsalicylicacid//5'-AMP-activated protein kinase subunit beta-1//Protein kinase activity
Acetylsalicylicacid//5'-AMP-activated protein kinase subunit beta-2//Identical protein binding
Acetylsalicylicacid//5'-AMP-activated protein kinase subunit gamma-1//Protein kinase binding
Acetylsalicylicacid//5'-AMP-activated protein kinase subunit gamma-2//Protein kinase binding
Acetylsalicylicacid//5'-AMP-activated protein kinase subunit gamma-3//Protein kinase binding
Acetylsalicylicacid//Endothelin-1 receptor//Phosphatidylinositol phospholipase c activity
Acetylsalicylicacid//78 kDa glucose-regulated protein//Unfolded protein binding
Acetylsalicylicacid//Ribosomal protein S6 kinase alpha-3//Ribosomal protein s6 kinase activity
Acetylsalicylicacid//NF-kappa-B inhibitor alpha//Ubiquitin protein ligase binding
Acetylsalicylicacid//Inhibitor of nuclear factor kappa-B kinase subunit beta//Scaffold protein binding
Acetylsalicylicacid//Mitogen-activated protein kinase 1//Rna polymerase ii carboxy-terminal domain kinase activity
Acetylsalicylicacid//G1/S-specific cyclin-D1//Transcription factor binding
Acetylsalicylicacid//Myc proto-oncogene protein//Transcriptional activator activity, rna polymerase ii core promoter proximal region sequence-specific binding
Fulvestrant//Estrogen receptor//Zinc ion binding
Felbamate//Glutamate receptor ionotropic, NMDA 2B//Zinc ion binding
Felbamate//Glutamate receptor ionotropic, NMDA 2A//Zinc ion binding
Fexofenadine//Histamine H1 receptor//Histamine receptor activity
Isoniazid//Cytochrome P450 2C8//Steroid hydroxylase activity
Isoniazid//Cytochrome P450 1A2//Oxidoreductase activity, acting on paired donors, with incorporation or reduction of molecular oxygen, reduced flavin or flavoprotein as one donor, and incorporation of one atom of oxygen
Isoniazid//Cytochrome P450 3A4//Vitamin d3 25-hydroxylase activity
Isoniazid//Cytochrome P450 2C19//Steroid hydroxylase activity
Isoniazid//Dihydrofolate reductase//Nadph binding
Naratriptan//5-hydroxytryptamine receptor 1F//Serotonin receptor activity
Naratriptan//5-hydroxytryptamine receptor 1D//Serotonin receptor activity
Naratriptan//5-hydroxytryptamine receptor 1B//Serotonin receptor activity
Naratriptan//5-hydroxytryptamine receptor 1A//Serotonin receptor activity
Hydrocodone//Delta-type opioid receptor//Opioid receptor activity
Hydrocodone//Mu-type opioid receptor//Voltage-gated calcium channel activity
Hydrocodone//Sigma non-opioid intracellular receptor 1//Opioid receptor activity
Methylprednisolone//Glucocorticoid receptor//Zinc ion binding
Methylprednisolone//Annexin A1//Structural molecule activity
Bromfenac//Prostaglandin G/H synthase 2//Prostaglandin-endoperoxide synthase activity
Bromfenac//Prostaglandin G/H synthase 1//Prostaglandin-endoperoxide synthase activity
Desloratadine//Histamine H1 receptor//Histamine receptor activity
Methyldopa//Alpha-2A adrenergic receptor//Thioesterase binding
Methyldopa//Aromatic-L-amino-acid decarboxylase//Pyridoxal phosphate binding
Alosetron//5-hydroxytryptamine receptor 3A//Voltage-gated potassium channel activity
Azelastine//Histamine H1 receptor//Histamine receptor activity
Azelastine//Histamine H2 receptor//Histamine receptor activity
Azelastine//Phospholipase A2//Receptor binding
Azelastine//Leukotriene C4 synthase//Lipid binding
Ezetimibe//Aminopeptidase N//Zinc ion binding
Ethinylestradiol//Estrogen receptor//Zinc ion binding
Ethinylestradiol//Nuclear receptor subfamily 1 group I member 2//Zinc ion binding
Lomefloxacin//DNA gyrase subunit A//Dna topoisomerase type ii (atp-hydrolyzing) activity
Lomefloxacin//DNA topoisomerase 4 subunit A//Dna topoisomerase type ii (atp-hydrolyzing) activity
Lomefloxacin//DNA topoisomerase 2-alpha//Ubiquitin binding
Cyclopentolate//Muscarinic acetylcholine receptor M1//Phosphatidylinositol phospholipase c activity
Formoterol//Beta-2 adrenergic receptor//Protein homodimerization activity
Formoterol//Beta-1 adrenergic receptor//Receptor signaling protein activity
Formoterol//Beta-3 adrenergic receptor//Protein homodimerization activity
Dopamine//D(2) dopamine receptor//Potassium channel regulator activity
Dopamine//D(1A) dopamine receptor//G-protein coupled amine receptor activity
Dopamine//D(1B) dopamine receptor//G-protein coupled amine receptor activity
Dopamine//D(3) dopamine receptor//G-protein coupled amine receptor activity
Dopamine//D(4) dopamine receptor//Sh3 domain binding
Dopamine//Sodium-dependent dopamine transporter//Monoamine transmembrane transporter activity
Dopamine//Dopamine beta-hydroxylase//L-ascorbic acid binding
Dopamine//5-hydroxytryptamine receptor 1A//Serotonin receptor activity
Dopamine//5-hydroxytryptamine receptor 7//Serotonin receptor activity
Dopamine//D(1A) dopamine receptor//G-protein coupled amine receptor activity
Dopamine//D(1B) dopamine receptor//G-protein coupled amine receptor activity
Dopamine//Sodium-dependent noradrenaline transporter//Norepinephrine:sodium symporter activity
Dopamine//Sodium-dependent serotonin transporter//Serotonin:sodium symporter activity
Dopamine//5-hydroxytryptamine receptor 3A//Voltage-gated potassium channel activity
Dopamine//5-hydroxytryptamine receptor 3B//Serotonin-activated cation-selective channel activity
Dopamine//Superoxide dismutase [Cu-Zn]//Zinc ion binding
Dopamine//Synaptic vesicular amine transporter//Monoamine transmembrane transporter activity
Exemestane//Aromatase//Oxygen binding
Azathioprine//Ras-related C3 botulinum toxin substrate 1//Thioesterase binding
Gabapentin//Voltage-dependent calcium channel subunit alpha-2/delta-1//Voltage-gated calcium channel activity
Gabapentin//Voltage-dependent calcium channel subunit alpha-2/delta-2//Voltage-gated calcium channel activity
Gabapentin//Voltage-dependent N-type calcium channel subunit alpha-1B//Voltage-gated calcium channel activity
Gabapentin//Adenosine receptor A1//Purine nucleoside binding
Gabapentin//Potassium voltage-gated channel subfamily KQT member 3//Voltage-gated potassium channel activity
Gabapentin//Potassium voltage-gated channel subfamily KQT member 5//Voltage-gated potassium channel activity
Doxorubicin//DNA topoisomerase 2-alpha//Ubiquitin binding
Doxorubicin//Nucleolar and coiled-body phosphoprotein 1//Poly(a) rna binding
Frovatriptan//5-hydroxytryptamine receptor 1D//Serotonin receptor activity
Frovatriptan//5-hydroxytryptamine receptor 1B//Serotonin receptor activity
Levobupivacaine//Sodium channel protein type 10 subunit alpha//Voltage-gated sodium channel activity
Hydroxyurea//Ribonucleoside-diphosphate reductase large subunit//Ribonucleoside-diphosphate reductase activity, thioredoxin disulfide as acceptor
Letrozole//Aromatase//Oxygen binding
Ketoprofen//Prostaglandin G/H synthase 1//Prostaglandin-endoperoxide synthase activity
Ketoprofen//Prostaglandin G/H synthase 2//Prostaglandin-endoperoxide synthase activity
Metyrapone//Cytochrome P450 11B1, mitochondrial//Steroid 11-beta-monooxygenase activity
Metyrapone//Camphor 5-monooxygenase//Iron ion binding
Cinacalcet//Extracellular calcium-sensing receptor//Phosphatidylinositol phospholipase c activity
Clobetasolpropionate//Glucocorticoid receptor//Zinc ion binding
Clobetasolpropionate//Annexin A1//Structural molecule activity
Clobetasolpropionate//Mineralocorticoid receptor//Zinc ion binding
Balsalazide//Peroxisome proliferator-activated receptor gamma//Zinc ion binding
Balsalazide//Prostaglandin G/H synthase 2//Prostaglandin-endoperoxide synthase activity
Balsalazide//Prostaglandin G/H synthase 1//Prostaglandin-endoperoxide synthase activity
Balsalazide//Arachidonate 5-lipoxygenase//Iron ion binding
Glyburide//ATP-binding cassette sub-family C member 8//Sulfonylurea receptor activity
Glyburide//ATP-sensitive inward rectifier potassium channel 11//Voltage-gated potassium channel activity
Glyburide//ATP-binding cassette sub-family C member 9//Transporter activity
Glyburide//Bile salt export pump//Transporter activity
Glyburide//ATP-binding cassette sub-family A member 1//Syntaxin binding
Glyburide//Cystic fibrosis transmembrane conductance regulator//Pdz domain binding
Glyburide//ATP-sensitive inward rectifier potassium channel 11//Voltage-gated potassium channel activity
Glyburide//ATP-sensitive inward rectifier potassium channel 8//Inward rectifier potassium channel activity
Guanfacine//Alpha-2A adrenergic receptor//Thioesterase binding
Guanfacine//Alpha-2B adrenergic receptor//Epinephrine binding
Isosorbidemononitrate//Guanylate cyclase soluble subunit alpha-2//Heme binding
Felodipine//Voltage-dependent L-type calcium channel subunit alpha-1C//Voltage-gated calcium channel activity
Felodipine//Voltage-dependent calcium channel subunit alpha-2/delta-1//Voltage-gated calcium channel activity
Felodipine//Voltage-dependent L-type calcium channel subunit beta-2//Voltage-gated calcium channel activity
Felodipine//Voltage-dependent L-type calcium channel subunit alpha-1D//Voltage-gated calcium channel activity involved sa node cell action potential
Felodipine//Voltage-dependent L-type calcium channel subunit alpha-1S//Voltage-gated calcium channel activity
Felodipine//Voltage-dependent T-type calcium channel subunit alpha-1H//Scaffold protein binding
Felodipine//Voltage-dependent calcium channel subunit alpha-2/delta-2//Voltage-gated calcium channel activity
Felodipine//Calmodulin//Titin binding
Felodipine//Calcium/calmodulin-dependent 3',5'-cyclic nucleotide phosphodiesterase 1B//Metal ion binding
Felodipine//Calcium/calmodulin-dependent 3',5'-cyclic nucleotide phosphodiesterase 1A//Metal ion binding
Felodipine//Mineralocorticoid receptor//Zinc ion binding
Felodipine//Troponin C, skeletal muscle//Calcium ion binding
Mycophenolicacid//Inosine-5'-monophosphate dehydrogenase 2//Rna binding
Mycophenolicacid//Inosine-5'-monophosphate dehydrogenase 1//Rna binding
Ketoconazole//Lanosterol 14-alpha demethylase//Sterol 14-demethylase activity
Ketoconazole//Androgen receptor//Zinc ion binding
Ketoconazole//Steroid 17-alpha-hydroxylase/17,20 lyase//Steroid 17-alpha-monooxygenase activity
Ketoconazole//Steroid 21-hydroxylase//Steroid hydroxylase activity
Ketoconazole//Potassium voltage-gated channel subfamily H member 2//Voltage-gated potassium channel activity involved in ventricular cardiac muscle cell action potential repolarization
Ketoconazole//Nuclear receptor subfamily 1 group I member 2//Zinc ion binding
Ketoconazole//Nuclear receptor subfamily 1 group I member 3//Zinc ion binding
Methoxyflurane//Gamma-aminobutyric acid receptor subunit alpha-1//Inhibitory extracellular ligand-gated ion channel activity
Methoxyflurane//Glutamate receptor 1//Pdz domain binding
Methoxyflurane//Glycine receptor subunit alpha-1//Transmitter-gated ion channel activity
Methoxyflurane//Calcium-transporting ATPase type 2C member 1//Signal transducer activity
Methoxyflurane//Potassium voltage-gated channel subfamily A member 1//Voltage-gated potassium channel activity
Methoxyflurane//NADH-ubiquinone oxidoreductase chain 1//Nadh dehydrogenase (ubiquinone) activity
Methoxyflurane//Gamma-aminobutyric acid receptor subunit alpha-1//Inhibitory extracellular ligand-gated ion channel activity
Methoxyflurane//Gamma-aminobutyric acid receptor subunit alpha-2//Inhibitory extracellular ligand-gated ion channel activity
Methoxyflurane//Gamma-aminobutyric acid receptor subunit alpha-3//Inhibitory extracellular ligand-gated ion channel activity
Methoxyflurane//Gamma-aminobutyric acid receptor subunit alpha-4//Inhibitory extracellular ligand-gated ion channel activity
Methoxyflurane//Gamma-aminobutyric acid receptor subunit alpha-5//Transporter activity
Methoxyflurane//Gamma-aminobutyric acid receptor subunit alpha-6//Inhibitory extracellular ligand-gated ion channel activity
Methoxyflurane//Gamma-aminobutyric acid receptor subunit beta-1//Ligand-gated ion channel activity
Methoxyflurane//Gamma-aminobutyric acid receptor subunit beta-2//Inhibitory extracellular ligand-gated ion channel activity
Methoxyflurane//Gamma-aminobutyric acid receptor subunit beta-3//Gaba-gated chloride ion channel activity
Methoxyflurane//Gamma-aminobutyric acid receptor subunit delta//Gaba-a receptor activity
Methoxyflurane//Gamma-aminobutyric acid receptor subunit epsilon//Inhibitory extracellular ligand-gated ion channel activity
Methoxyflurane//Gamma-aminobutyric acid receptor subunit gamma-1//Inhibitory extracellular ligand-gated ion channel activity
Methoxyflurane//Gamma-aminobutyric acid receptor subunit gamma-2//Inhibitory extracellular ligand-gated ion channel activity
Methoxyflurane//Gamma-aminobutyric acid receptor subunit gamma-3//Inhibitory extracellular ligand-gated ion channel activity
Methoxyflurane//Gamma-aminobutyric acid receptor subunit pi//Gaba-a receptor activity
Methoxyflurane//Gamma-aminobutyric acid receptor subunit theta//Transmembrane signaling receptor activity
Irbesartan//Type-1 angiotensin II receptor//Protein heterodimerization activity
Irbesartan//Transcription factor AP-1//Transcriptional activator activity, rna polymerase ii transcription factor binding
Mercaptopurine//Hypoxanthine-guanine phosphoribosyltransferase//Protein homodimerization activity
Mercaptopurine//Amidophosphoribosyltransferase//Metal ion binding
Mercaptopurine//Inosine-5'-monophosphate dehydrogenase 1//Rna binding
Mercaptopurine//Inosine-5'-monophosphate dehydrogenase 2//Rna binding
Fenofibrate//Peroxisome proliferator-activated receptor alpha//Zinc ion binding
Fenofibrate//Nuclear receptor subfamily 1 group I member 2//Zinc ion binding
Memantine//5-hydroxytryptamine receptor 3A//Voltage-gated potassium channel activity
Memantine//D(2) dopamine receptor//Potassium channel regulator activity
Memantine//Glutamate receptor ionotropic, NMDA 1//Voltage-gated cation channel activity
Memantine//Glutamate receptor ionotropic, NMDA 1//Voltage-gated cation channel activity
Memantine//Glutamate receptor ionotropic, NMDA 2A//Zinc ion binding
Memantine//Glutamate receptor ionotropic, NMDA 2B//Zinc ion binding
Memantine//Glutamate receptor ionotropic, NMDA 2C//Nmda glutamate receptor activity
Memantine//Glutamate receptor ionotropic, NMDA 2D//Nmda glutamate receptor activity
Memantine//Glutamate receptor ionotropic, NMDA 3A//Protein phosphatase 2a binding
Memantine//Glutamate receptor ionotropic, NMDA 3B//Nmda glutamate receptor activity
Memantine//Gamma-aminobutyric acid receptor subunit alpha-1//Inhibitory extracellular ligand-gated ion channel activity
Memantine//Gamma-aminobutyric acid receptor subunit alpha-2//Inhibitory extracellular ligand-gated ion channel activity
Memantine//Gamma-aminobutyric acid receptor subunit alpha-3//Inhibitory extracellular ligand-gated ion channel activity
Memantine//Gamma-aminobutyric acid receptor subunit alpha-4//Inhibitory extracellular ligand-gated ion channel activity
Memantine//Gamma-aminobutyric acid receptor subunit alpha-5//Transporter activity
Memantine//Gamma-aminobutyric acid receptor subunit alpha-6//Inhibitory extracellular ligand-gated ion channel activity
Memantine//Gamma-aminobutyric acid receptor subunit beta-1//Ligand-gated ion channel activity
Memantine//Gamma-aminobutyric acid receptor subunit beta-2//Inhibitory extracellular ligand-gated ion channel activity
Memantine//Gamma-aminobutyric acid receptor subunit beta-3//Gaba-gated chloride ion channel activity
Memantine//Gamma-aminobutyric acid receptor subunit delta//Gaba-a receptor activity
Memantine//Gamma-aminobutyric acid receptor subunit epsilon//Inhibitory extracellular ligand-gated ion channel activity
Memantine//Gamma-aminobutyric acid receptor subunit gamma-1//Inhibitory extracellular ligand-gated ion channel activity
Memantine//Gamma-aminobutyric acid receptor subunit gamma-2//Inhibitory extracellular ligand-gated ion channel activity
Memantine//Gamma-aminobutyric acid receptor subunit gamma-3//Inhibitory extracellular ligand-gated ion channel activity
Memantine//Gamma-aminobutyric acid receptor subunit pi//Gaba-a receptor activity
Memantine//Gamma-aminobutyric acid receptor subunit theta//Transmembrane signaling receptor activity
Memantine//Glycine receptor subunit alpha-1//Transmitter-gated ion channel activity
Memantine//Glycine receptor subunit alpha-2//Transmitter-gated ion channel activity
Memantine//Glycine receptor subunit alpha-3//Transmitter-gated ion channel activity
Memantine//Glycine receptor subunit beta//Glycine binding
Ibuprofen//Prostaglandin G/H synthase 2//Prostaglandin-endoperoxide synthase activity
Ibuprofen//Prostaglandin G/H synthase 1//Prostaglandin-endoperoxide synthase activity
Ibuprofen//Apoptosis regulator Bcl-2//Ubiquitin protein ligase binding
Ibuprofen//Thrombomodulin//Transmembrane signaling receptor activity
Ibuprofen//Fatty acid-binding protein, intestinal//Transporter activity
Ibuprofen//Peroxisome proliferator-activated receptor gamma//Zinc ion binding
Ibuprofen//Cystic fibrosis transmembrane conductance regulator//Pdz domain binding
Ibuprofen//Peroxisome proliferator-activated receptor alpha//Zinc ion binding
Ibuprofen//Protein S100-A7//Zinc ion binding
Isoprenaline//Beta-1 adrenergic receptor//Receptor signaling protein activity
Isoprenaline//Beta-2 adrenergic receptor//Protein homodimerization activity
Isoprenaline//Beta-3 adrenergic receptor//Protein homodimerization activity
Isoprenaline//Mitogen-activated protein kinase 1//Rna polymerase ii carboxy-terminal domain kinase activity
Isoprenaline//CAMP phosphodiesterase//Metal ion binding
Isoprenaline//Superoxide dismutase [Cu-Zn]//Zinc ion binding
Melatonin//Estrogen receptor//Zinc ion binding
Melatonin//Nuclear receptor ROR-beta//Zinc ion binding
Melatonin//Calmodulin//Titin binding
Melatonin//Myeloperoxidase//Peroxidase activity
Melatonin//Eosinophil peroxidase//Peroxidase activity
Melatonin//Calreticulin//Zinc ion binding
Melatonin//Acetylserotonin O-methyltransferase//Protein homodimerization activity
Melatonin//Ribosyldihydronicotinamide dehydrogenase [quinone]//Nadph dehydrogenase (quinone) activity
Glipizide//ATP-binding cassette sub-family C member 8//Sulfonylurea receptor activity
Glipizide//Peroxisome proliferator-activated receptor gamma//Zinc ion binding
Clonazepam//Gamma-aminobutyric acid receptor subunit alpha-1//Inhibitory extracellular ligand-gated ion channel activity
Clonazepam//Gamma-aminobutyric acid receptor subunit alpha-2//Inhibitory extracellular ligand-gated ion channel activity
Clonazepam//Gamma-aminobutyric acid receptor subunit alpha-3//Inhibitory extracellular ligand-gated ion channel activity
Clonazepam//Gamma-aminobutyric acid receptor subunit alpha-4//Inhibitory extracellular ligand-gated ion channel activity
Clonazepam//Gamma-aminobutyric acid receptor subunit alpha-5//Transporter activity
Clonazepam//Gamma-aminobutyric acid receptor subunit alpha-6//Inhibitory extracellular ligand-gated ion channel activity
Clonazepam//Gamma-aminobutyric acid receptor subunit beta-1//Ligand-gated ion channel activity
Clonazepam//Gamma-aminobutyric acid receptor subunit beta-2//Inhibitory extracellular ligand-gated ion channel activity
Clonazepam//Gamma-aminobutyric acid receptor subunit beta-3//Gaba-gated chloride ion channel activity
Clonazepam//Gamma-aminobutyric acid receptor subunit delta//Gaba-a receptor activity
Clonazepam//Gamma-aminobutyric acid receptor subunit epsilon//Inhibitory extracellular ligand-gated ion channel activity
Clonazepam//Gamma-aminobutyric acid receptor subunit gamma-1//Inhibitory extracellular ligand-gated ion channel activity
Clonazepam//Gamma-aminobutyric acid receptor subunit gamma-2//Inhibitory extracellular ligand-gated ion channel activity
Clonazepam//Gamma-aminobutyric acid receptor subunit gamma-3//Inhibitory extracellular ligand-gated ion channel activity
Clonazepam//Gamma-aminobutyric acid receptor subunit pi//Gaba-a receptor activity
Clonazepam//Gamma-aminobutyric acid receptor subunit theta//Transmembrane signaling receptor activity
Clonazepam//Gamma-aminobutyric acid receptor subunit alpha-1//Inhibitory extracellular ligand-gated ion channel activity
Clonazepam//Gamma-aminobutyric acid receptor subunit alpha-2//Inhibitory extracellular ligand-gated ion channel activity
Clonazepam//Gamma-aminobutyric acid receptor subunit alpha-3//Inhibitory extracellular ligand-gated ion channel activity
Clonazepam//Gamma-aminobutyric acid receptor subunit alpha-5//Transporter activity
Clonazepam//Gamma-aminobutyric acid receptor subunit gamma-1//Inhibitory extracellular ligand-gated ion channel activity
Clonazepam//Gamma-aminobutyric acid receptor subunit gamma-2//Inhibitory extracellular ligand-gated ion channel activity
Clonazepam//Gamma-aminobutyric acid receptor subunit gamma-3//Inhibitory extracellular ligand-gated ion channel activity
Clonazepam//Nuclear receptor subfamily 1 group I member 2//Zinc ion binding
Mequitazine//Histamine H1 receptor//Histamine receptor activity
Diphenhydramine//Histamine H1 receptor//Histamine receptor activity
Diphenhydramine//Muscarinic acetylcholine receptor M2//G-protein coupled acetylcholine receptor activity
Atorvastatin//3-hydroxy-3-methylglutaryl-coenzyme A reductase//Nadph binding
Atorvastatin//Dipeptidyl peptidase 4//Virus receptor activity
Atorvastatin//Aryl hydrocarbon receptor//Transcription regulatory region dna binding
Atorvastatin//Histone deacetylase 2//Transcription factor binding
Atorvastatin//Nuclear receptor subfamily 1 group I member 3//Zinc ion binding
Benzocaine//Sodium channel protein type 10 subunit alpha//Voltage-gated sodium channel activity
Hesperetin//Microsomal triglyceride transfer protein large subunit//Protein heterodimerization activity
Hesperetin//Sterol O-acyltransferase 2//Transferase activity, transferring acyl groups
Hesperetin//Sex hormone-binding globulin//Androgen binding
Fluvastatin//3-hydroxy-3-methylglutaryl-coenzyme A reductase//Nadph binding
Fluvastatin//Histone deacetylase 2//Transcription factor binding
Leflunomide//Dihydroorotate dehydrogenase (quinone), mitochondrial//Ubiquinone binding
Leflunomide//Aryl hydrocarbon receptor//Transcription regulatory region dna binding
Leflunomide//Protein-tyrosine kinase 2-beta//Signal transducer activity
Capecitabine//Thymidylate synthase//Thymidylate synthase activity
Methyprylon//Gamma-aminobutyric acid receptor subunit alpha-1//Inhibitory extracellular ligand-gated ion channel activity
Methyprylon//Gamma-aminobutyric acid receptor subunit alpha-1//Inhibitory extracellular ligand-gated ion channel activity
Methyprylon//Gamma-aminobutyric acid receptor subunit alpha-2//Inhibitory extracellular ligand-gated ion channel activity
Methyprylon//Gamma-aminobutyric acid receptor subunit alpha-3//Inhibitory extracellular ligand-gated ion channel activity
Methyprylon//Gamma-aminobutyric acid receptor subunit alpha-4//Inhibitory extracellular ligand-gated ion channel activity
Methyprylon//Gamma-aminobutyric acid receptor subunit alpha-5//Transporter activity
Methyprylon//Gamma-aminobutyric acid receptor subunit alpha-6//Inhibitory extracellular ligand-gated ion channel activity
Methyprylon//Gamma-aminobutyric acid receptor subunit beta-1//Ligand-gated ion channel activity
Methyprylon//Gamma-aminobutyric acid receptor subunit beta-2//Inhibitory extracellular ligand-gated ion channel activity
Methyprylon//Gamma-aminobutyric acid receptor subunit beta-3//Gaba-gated chloride ion channel activity
Methyprylon//Gamma-aminobutyric acid receptor subunit delta//Gaba-a receptor activity
Methyprylon//Gamma-aminobutyric acid receptor subunit epsilon//Inhibitory extracellular ligand-gated ion channel activity
Methyprylon//Gamma-aminobutyric acid receptor subunit gamma-1//Inhibitory extracellular ligand-gated ion channel activity
Methyprylon//Gamma-aminobutyric acid receptor subunit gamma-2//Inhibitory extracellular ligand-gated ion channel activity
Methyprylon//Gamma-aminobutyric acid receptor subunit gamma-3//Inhibitory extracellular ligand-gated ion channel activity
Methyprylon//Gamma-aminobutyric acid receptor subunit pi//Gaba-a receptor activity
Methyprylon//Gamma-aminobutyric acid receptor subunit theta//Transmembrane signaling receptor activity
Miconazole//Lanosterol 14-alpha demethylase//Sterol 14-demethylase activity
Miconazole//Nitric oxide synthase, endothelial//Tetrahydrobiopterin binding
Miconazole//Nitric oxide synthase, inducible//Tetrahydrobiopterin binding
Miconazole//Nuclear receptor subfamily 1 group I member 2//Zinc ion binding
Miconazole//Calcium-activated potassium channel subunit alpha-1//Voltage-gated potassium channel activity
Miconazole//Calcium-activated potassium channel subunit beta-1//Potassium channel regulator activity
Miconazole//Calcium-activated potassium channel subunit beta-2//Potassium channel regulator activity
Miconazole//Calcium-activated potassium channel subunit beta-3//Potassium channel regulator activity
Miconazole//Calcium-activated potassium channel subunit beta-4//Potassium channel regulator activity
Miconazole//Intermediate conductance calcium-activated potassium channel protein 4//Protein phosphatase binding
Miconazole//Small conductance calcium-activated potassium channel protein 1//Small conductance calcium-activated potassium channel activity
Miconazole//Small conductance calcium-activated potassium channel protein 2//Small conductance calcium-activated potassium channel activity
Miconazole//Small conductance calcium-activated potassium channel protein 3//Small conductance calcium-activated potassium channel activity
Miconazole//Potassium voltage-gated channel subfamily A member 1//Voltage-gated potassium channel activity
Miconazole//Potassium voltage-gated channel subfamily A member 10//Intracellular cyclic nucleotide activated cation channel activity
Miconazole//Potassium voltage-gated channel subfamily A member 2//Voltage-gated potassium channel activity
Miconazole//Potassium voltage-gated channel subfamily A member 3//Voltage-gated ion channel activity
Miconazole//Potassium voltage-gated channel subfamily A member 4//Voltage-gated potassium channel activity
Miconazole//Potassium voltage-gated channel subfamily A member 5//Voltage-gated potassium channel activity involved in sa node cell action potential repolarization
Miconazole//Potassium voltage-gated channel subfamily A member 6//Voltage-gated potassium channel activity
Miconazole//Potassium voltage-gated channel subfamily B member 1//Ubiquitin-like protein binding
Miconazole//Potassium voltage-gated channel subfamily B member 2//Protein heterodimerization activity
Miconazole//Potassium voltage-gated channel subfamily C member 1//Voltage-gated potassium channel activity
Miconazole//Potassium voltage-gated channel subfamily C member 2//Voltage-gated potassium channel activity
Miconazole//Potassium voltage-gated channel subfamily C member 3//Voltage-gated potassium channel activity
Miconazole//Potassium voltage-gated channel subfamily C member 4//Voltage-gated potassium channel activity
Miconazole//Potassium voltage-gated channel subfamily D member 1//Metal ion binding
Miconazole//Potassium voltage-gated channel subfamily D member 2//Voltage-gated potassium channel activity
Miconazole//Potassium voltage-gated channel subfamily D member 3//Metal ion binding
Miconazole//Potassium voltage-gated channel subfamily G member 1//Potassium channel subunit that does not form functional channels by itself. Can form functional heterotetrameric channels with KCNB1; modulates the delayed rectifier voltage-gated potassium channel activation and deactivation rates of KCNB1 (PubMed:19074135).
Miconazole//Potassium voltage-gated channel subfamily G member 2//Potassium channel subunit. Modulates channel activity by shifting the threshold and the half-maximal activation to more negative values.
Miconazole//Potassium voltage-gated channel subfamily G member 4//Potassium channel subunit that does not form functional channels by itself. Can form functional heterotetrameric channels with KCNB1; modulates the delayed rectifier voltage-gated potassium channel activation and deactivation rates of KCNB1 (PubMed:19074135).
Miconazole//Potassium voltage-gated channel subfamily H member 1//Phosphorelay sensor kinase activity
Miconazole//Potassium voltage-gated channel subfamily H member 2//Voltage-gated potassium channel activity involved in ventricular cardiac muscle cell action potential repolarization
Miconazole//Potassium voltage-gated channel subfamily H member 6//Voltage-gated potassium channel activity
Miconazole//Potassium voltage-gated channel subfamily H member 7//Voltage-gated potassium channel activity
Miconazole//Potassium voltage-gated channel subfamily KQT member 1//Voltage-gated potassium channel activity involved in ventricular cardiac muscle cell action potential repolarization
Miconazole//Potassium voltage-gated channel subfamily KQT member 2//Voltage-gated potassium channel activity
Miconazole//Potassium voltage-gated channel subfamily KQT member 3//Voltage-gated potassium channel activity
Miconazole//Potassium voltage-gated channel subfamily KQT member 4//Potassium channel activity
Miconazole//Potassium voltage-gated channel subfamily KQT member 5//Voltage-gated potassium channel activity
Miconazole//Potassium voltage-gated channel subfamily V member 2//Potassium channel subunit. Modulates channel activity by shifting the threshold and the half-maximal activation to more negative values.
Miconazole//ATP-sensitive inward rectifier potassium channel 12//Inward rectifier potassium channel activity
Miconazole//ATP-sensitive inward rectifier potassium channel 14//Inward rectifier potassium channels are characterized by a greater tendency to allow potassium to flow into the cell rather than out of it. Their voltage dependence is regulated by the concentration of extracellular potassium; as external potassium is raised, the voltage range of the channel opening shifts to more positive voltages. The inward rectification is mainly due to the blockage of outward current by internal magnesium. KCNJ14 gives rise to low-conductance channels with a low affinity to the channel blockers Barium and Cesium (By similarity).
Miconazole//Inward rectifier potassium channel 2//Probably participates in establishing action potential waveform and excitability of neuronal and muscle tissues. Inward rectifier potassium channels are characterized by a greater tendency to allow potassium to flow into the cell rather than out of it. Their voltage dependence is regulated by the concentration of extracellular potassium; as external potassium is raised, the voltage range of the channel opening shifts to more positive voltages. The inward rectification is mainly due to the blockage of outward current by internal magnesium. Can be blocked by extracellular barium or cesium.
Miconazole//Inward rectifier potassium channel 4//Pdz domain binding
Miconazole//Voltage-dependent L-type calcium channel subunit alpha-1C//Voltage-gated calcium channel activity
Miconazole//Voltage-dependent L-type calcium channel subunit alpha-1D//Voltage-gated calcium channel activity involved sa node cell action potential
Miconazole//Voltage-dependent L-type calcium channel subunit alpha-1F//Voltage-gated calcium channel activity
Miconazole//Voltage-dependent L-type calcium channel subunit alpha-1S//Voltage-gated calcium channel activity
Miconazole//Voltage-dependent L-type calcium channel subunit beta-1//Voltage-gated calcium channel activity
Miconazole//Voltage-dependent L-type calcium channel subunit beta-2//Voltage-gated calcium channel activity
Miconazole//Voltage-dependent L-type calcium channel subunit beta-3//Voltage-gated calcium channel activity
Miconazole//Voltage-dependent L-type calcium channel subunit beta-4//Voltage-gated calcium channel activity
Chlorphenamine//Histamine H1 receptor//Histamine receptor activity
Chlorphenamine//Sodium-dependent serotonin transporter//Serotonin:sodium symporter activity
Chlorphenamine//Sodium-dependent noradrenaline transporter//Norepinephrine:sodium symporter activity
Chlorphenamine//Sodium-dependent dopamine transporter//Monoamine transmembrane transporter activity
Atovaquone//Cytochrome b//Oxidoreductase activity
Atovaquone//Dihydroorotate dehydrogenase (quinone), mitochondrial//Ubiquinone binding
Atovaquone//Dihydroorotate dehydrogenase (quinone), mitochondrial//Ubiquinone binding
Amiodarone//Potassium voltage-gated channel subfamily H member 2//Voltage-gated potassium channel activity involved in ventricular cardiac muscle cell action potential repolarization
Amiodarone//Potassium voltage-gated channel subfamily H member 6//Voltage-gated potassium channel activity
Amiodarone//Potassium voltage-gated channel subfamily H member 7//Voltage-gated potassium channel activity
Amiodarone//Beta-1 adrenergic receptor//Receptor signaling protein activity
Amiodarone//Beta-2 adrenergic receptor//Protein homodimerization activity
Amiodarone//Beta-3 adrenergic receptor//Protein homodimerization activity
Amiodarone//Voltage-dependent T-type calcium channel subunit alpha-1I//Voltage-gated calcium channel activity
Amiodarone//Voltage-dependent L-type calcium channel subunit alpha-1C//Voltage-gated calcium channel activity
Amiodarone//Voltage-dependent L-type calcium channel subunit alpha-1D//Voltage-gated calcium channel activity involved sa node cell action potential
Amiodarone//Voltage-dependent L-type calcium channel subunit alpha-1F//Voltage-gated calcium channel activity
Amiodarone//Voltage-dependent L-type calcium channel subunit alpha-1S//Voltage-gated calcium channel activity
Amiodarone//Voltage-dependent L-type calcium channel subunit beta-1//Voltage-gated calcium channel activity
Amiodarone//Voltage-dependent L-type calcium channel subunit beta-2//Voltage-gated calcium channel activity
Amiodarone//Voltage-dependent L-type calcium channel subunit beta-3//Voltage-gated calcium channel activity
Amiodarone//Voltage-dependent L-type calcium channel subunit beta-4//Voltage-gated calcium channel activity
Amiodarone//Thyroid hormone receptor alpha//Zinc ion binding
Amiodarone//Thyroid hormone receptor beta//Zinc ion binding
Amiodarone//Peroxisome proliferator-activated receptor gamma//Zinc ion binding
Amiodarone//Peroxisome proliferator-activated receptor alpha//Zinc ion binding
Diazoxide//ATP-sensitive inward rectifier potassium channel 11//Voltage-gated potassium channel activity
Diazoxide//Carbonic anhydrase 1//Zinc ion binding
Diazoxide//Carbonic anhydrase 2//Zinc ion binding
Diazoxide//Sodium/potassium-transporting ATPase subunit alpha-1//Steroid hormone binding
Diazoxide//Calcium-activated potassium channel subunit alpha-1//Voltage-gated potassium channel activity
Gliclazide//ATP-binding cassette sub-family C member 8//Sulfonylurea receptor activity
Ambenonium//Acetylcholinesterase//Serine hydrolase activity
Dutasteride//3-oxo-5-alpha-steroid 4-dehydrogenase 1//Electron carrier activity
Dutasteride//3-oxo-5-alpha-steroid 4-dehydrogenase 2//Sterol 5-alpha reductase activity
Econazole//Lanosterol 14-alpha demethylase//Sterol 14-demethylase activity
Econazole//Nuclear receptor subfamily 1 group I member 2//Zinc ion binding
Bicalutamide//Androgen receptor//Zinc ion binding
Doxacuriumchloride//Neuronal acetylcholine receptor subunit alpha-2//Drug binding
Doxacuriumchloride//Muscarinic acetylcholine receptor M2//G-protein coupled acetylcholine receptor activity
Carvedilol//Beta-1 adrenergic receptor//Receptor signaling protein activity
Carvedilol//Alpha-1A adrenergic receptor//Protein heterodimerization activity
Carvedilol//NADH dehydrogenase [ubiquinone] 1 subunit C2//Nadh dehydrogenase (ubiquinone) activity
Carvedilol//Beta-2 adrenergic receptor//Protein homodimerization activity
Carvedilol//Natriuretic peptides B//Receptor binding
Carvedilol//Gap junction alpha-1 protein//Signal transducer activity
Carvedilol//Potassium voltage-gated channel subfamily H member 2//Voltage-gated potassium channel activity involved in ventricular cardiac muscle cell action potential repolarization
Carvedilol//Vascular cell adhesion protein 1//Primary amine oxidase activity
Carvedilol//Alpha-1D adrenergic receptor//Alpha1-adrenergic receptor activity
Carvedilol//Alpha-1B adrenergic receptor//Protein heterodimerization activity
Carvedilol//Alpha-2C adrenergic receptor//Protein homodimerization activity
Carvedilol//Alpha-2B adrenergic receptor//Epinephrine binding
Carvedilol//Alpha-2A adrenergic receptor//Thioesterase binding
Carvedilol//E-selectin//Transmembrane signaling receptor activity
Carvedilol//Hypoxia-inducible factor 1-alpha//Ubiquitin protein ligase binding
Carvedilol//Inward rectifier potassium channel 4//Pdz domain binding
Carvedilol//Inward rectifier potassium channel 2//Probably participates in establishing action potential waveform and excitability of neuronal and muscle tissues. Inward rectifier potassium channels are characterized by a greater tendency to allow potassium to flow into the cell rather than out of it. Their voltage dependence is regulated by the concentration of extracellular potassium; as external potassium is raised, the voltage range of the channel opening shifts to more positive voltages. The inward rectification is mainly due to the blockage of outward current by internal magnesium. Can be blocked by extracellular barium or cesium.
Carvedilol//Alpha-1A adrenergic receptor//Protein heterodimerization activity
Carvedilol//Alpha-1B adrenergic receptor//Protein heterodimerization activity
Carvedilol//Alpha-1D adrenergic receptor//Alpha1-adrenergic receptor activity
Levofloxacin//DNA gyrase subunit A//Dna topoisomerase type ii (atp-hydrolyzing) activity
Levofloxacin//DNA topoisomerase 4 subunit A//Dna topoisomerase type ii (atp-hydrolyzing) activity
Doxepin//Histamine H1 receptor//Histamine receptor activity
Doxepin//Histamine H2 receptor//Histamine receptor activity
Doxepin//Sodium-dependent noradrenaline transporter//Norepinephrine:sodium symporter activity
Doxepin//Sodium-dependent serotonin transporter//Serotonin:sodium symporter activity
Doxepin//5-hydroxytryptamine receptor 2A//Virus receptor activity
Doxepin//5-hydroxytryptamine receptor 2B//Serotonin receptor activity
Doxepin//5-hydroxytryptamine receptor 2C//Serotonin receptor activity
Doxepin//Muscarinic acetylcholine receptor M1//Phosphatidylinositol phospholipase c activity
Doxepin//Muscarinic acetylcholine receptor M2//G-protein coupled acetylcholine receptor activity
Doxepin//Muscarinic acetylcholine receptor M3//Receptor activity
Doxepin//Muscarinic acetylcholine receptor M4//Guanyl-nucleotide exchange factor activity
Doxepin//Muscarinic acetylcholine receptor M5//Phosphatidylinositol phospholipase c activity
Doxepin//Alpha-1A adrenergic receptor//Protein heterodimerization activity
Doxepin//Alpha-1B adrenergic receptor//Protein heterodimerization activity
Doxepin//Alpha-1D adrenergic receptor//Alpha1-adrenergic receptor activity
Doxepin//5-hydroxytryptamine receptor 1A//Serotonin receptor activity
Doxepin//5-hydroxytryptamine receptor 6//Serotonin receptor activity
Doxepin//Histamine H4 receptor//Histamine receptor activity
Doxepin//Potassium voltage-gated channel subfamily H member 2//Voltage-gated potassium channel activity involved in ventricular cardiac muscle cell action potential repolarization
Amifostine//Alkaline phosphatase, placental-like//Metal ion binding
Diclofenamide//Carbonic anhydrase 1//Zinc ion binding
Diclofenamide//Carbonic anhydrase 2//Zinc ion binding
Diclofenamide//Carbonic anhydrase 4//Zinc ion binding
Diclofenamide//Carbonic anhydrase 7//Zinc ion binding
Diclofenamide//Carbonic anhydrase 3//Zinc ion binding
Nefazodone//5-hydroxytryptamine receptor 2A//Virus receptor activity
Nefazodone//5-hydroxytryptamine receptor 2C//Serotonin receptor activity
Nefazodone//Sodium-dependent serotonin transporter//Serotonin:sodium symporter activity
Nefazodone//5-hydroxytryptamine receptor 1A//Serotonin receptor activity
Nefazodone//Sodium-dependent noradrenaline transporter//Norepinephrine:sodium symporter activity
Nefazodone//Sodium-dependent dopamine transporter//Monoamine transmembrane transporter activity
Nefazodone//Alpha-1B adrenergic receptor//Protein heterodimerization activity
Nefazodone//Alpha-2A adrenergic receptor//Thioesterase binding
Nefazodone//Alpha-1A adrenergic receptor//Protein heterodimerization activity
Nefazodone//Potassium voltage-gated channel subfamily H member 2//Voltage-gated potassium channel activity involved in ventricular cardiac muscle cell action potential repolarization
Desipramine//Sodium-dependent noradrenaline transporter//Norepinephrine:sodium symporter activity
Desipramine//5-hydroxytryptamine receptor 2A//Virus receptor activity
Desipramine//Beta-2 adrenergic receptor//Protein homodimerization activity
Desipramine//Sodium-dependent serotonin transporter//Serotonin:sodium symporter activity
Desipramine//Beta-1 adrenergic receptor//Receptor signaling protein activity
Desipramine//Histamine H1 receptor//Histamine receptor activity
Desipramine//Sphingomyelin phosphodiesterase//Sphingomyelin phosphodiesterase activity
Desipramine//Alpha-1A adrenergic receptor//Protein heterodimerization activity
Desipramine//Alpha-1B adrenergic receptor//Protein heterodimerization activity
Desipramine//Alpha-1D adrenergic receptor//Alpha1-adrenergic receptor activity
Desipramine//Muscarinic acetylcholine receptor M1//Phosphatidylinositol phospholipase c activity
Desipramine//Muscarinic acetylcholine receptor M2//G-protein coupled acetylcholine receptor activity
Desipramine//Muscarinic acetylcholine receptor M3//Receptor activity
Desipramine//Muscarinic acetylcholine receptor M4//Guanyl-nucleotide exchange factor activity
Desipramine//Muscarinic acetylcholine receptor M5//Phosphatidylinositol phospholipase c activity
Desipramine//5-hydroxytryptamine receptor 1A//Serotonin receptor activity
Desipramine//5-hydroxytryptamine receptor 2C//Serotonin receptor activity
Desipramine//D(2) dopamine receptor//Potassium channel regulator activity
Desipramine//Alpha-2A adrenergic receptor//Thioesterase binding
Desipramine//Alpha-2B adrenergic receptor//Epinephrine binding
Desipramine//Alpha-2C adrenergic receptor//Protein homodimerization activity
Bupropion//Sodium-dependent dopamine transporter//Monoamine transmembrane transporter activity
Bupropion//Sodium-dependent noradrenaline transporter//Norepinephrine:sodium symporter activity
Bupropion//Neuronal acetylcholine receptor subunit alpha-3//Ligand-gated ion channel activity
Bupropion//5-hydroxytryptamine receptor 3A//Voltage-gated potassium channel activity
Halothane//Potassium channel subfamily K member 3//S100 protein binding
Halothane//Potassium channel subfamily K member 9//Voltage-gated potassium channel activity
Halothane//Calcium-activated potassium channel subunit alpha-1//Voltage-gated potassium channel activity
Halothane//Glutamate receptor ionotropic, NMDA 3A//Protein phosphatase 2a binding
Halothane//Glutamate receptor ionotropic, NMDA 3B//Nmda glutamate receptor activity
Halothane//Glutamate receptor ionotropic, NMDA 2A//Zinc ion binding
Halothane//Glycine receptor subunit alpha-1//Transmitter-gated ion channel activity
Halothane//G protein-activated inward rectifier potassium channel 2//Inward rectifier potassium channel activity
Halothane//G protein-activated inward rectifier potassium channel 1//G-protein activated inward rectifier potassium channel activity
Halothane//NADH-ubiquinone oxidoreductase chain 1//Nadh dehydrogenase (ubiquinone) activity
Halothane//Intermediate conductance calcium-activated potassium channel protein 4//Protein phosphatase binding
Halothane//Gamma-aminobutyric acid receptor subunit alpha-1//Inhibitory extracellular ligand-gated ion channel activity
Halothane//Guanine nucleotide-binding protein G(I)/G(S)/G(O) subunit gamma-2//Signal transducer activity
Halothane//Neuropeptide S receptor//Vasopressin receptor activity
Halothane//Gamma-aminobutyric acid receptor subunit alpha-1//Inhibitory extracellular ligand-gated ion channel activity
Halothane//Gamma-aminobutyric acid receptor subunit alpha-2//Inhibitory extracellular ligand-gated ion channel activity
Halothane//Gamma-aminobutyric acid receptor subunit alpha-3//Inhibitory extracellular ligand-gated ion channel activity
Halothane//Gamma-aminobutyric acid receptor subunit alpha-4//Inhibitory extracellular ligand-gated ion channel activity
Halothane//Gamma-aminobutyric acid receptor subunit alpha-5//Transporter activity
Halothane//Gamma-aminobutyric acid receptor subunit alpha-6//Inhibitory extracellular ligand-gated ion channel activity
Halothane//Gamma-aminobutyric acid receptor subunit beta-1//Ligand-gated ion channel activity
Halothane//Gamma-aminobutyric acid receptor subunit beta-2//Inhibitory extracellular ligand-gated ion channel activity
Halothane//Gamma-aminobutyric acid receptor subunit beta-3//Gaba-gated chloride ion channel activity
Halothane//Gamma-aminobutyric acid receptor subunit delta//Gaba-a receptor activity
Halothane//Gamma-aminobutyric acid receptor subunit epsilon//Inhibitory extracellular ligand-gated ion channel activity
Halothane//Gamma-aminobutyric acid receptor subunit gamma-1//Inhibitory extracellular ligand-gated ion channel activity
Halothane//Gamma-aminobutyric acid receptor subunit gamma-2//Inhibitory extracellular ligand-gated ion channel activity
Halothane//Gamma-aminobutyric acid receptor subunit gamma-3//Inhibitory extracellular ligand-gated ion channel activity
Halothane//Gamma-aminobutyric acid receptor subunit pi//Gaba-a receptor activity
Halothane//Gamma-aminobutyric acid receptor subunit theta//Transmembrane signaling receptor activity
Chloroprocaine//Sodium channel protein type 10 subunit alpha//Voltage-gated sodium channel activity
Chloroprocaine//Sodium-dependent dopamine transporter//Monoamine transmembrane transporter activity
Cilostazol//cGMP-inhibited 3',5'-cyclic phosphodiesterase A//Metal ion binding
Itraconazole//Lanosterol 14-alpha demethylase//Sterol 14-demethylase activity
Itraconazole//Lanosterol 14-alpha demethylase//Sterol 14-demethylase activity
Arsenictrioxide//Inhibitor of nuclear factor kappa-B kinase subunit beta//Scaffold protein binding
Arsenictrioxide//Transcription factor AP-1//Transcriptional activator activity, rna polymerase ii transcription factor binding
Arsenictrioxide//G1/S-specific cyclin-D1//Transcription factor binding
Arsenictrioxide//Mitogen-activated protein kinase 1//Rna polymerase ii carboxy-terminal domain kinase activity
Arsenictrioxide//RAC-alpha serine/threonine-protein kinase//Protein serine/threonine/tyrosine kinase activity
Guanethidine//Sodium-dependent noradrenaline transporter//Norepinephrine:sodium symporter activity
Moclobemide//Amine oxidase [flavin-containing] A//Serotonin binding
Moclobemide//Amine oxidase [flavin-containing] A//Serotonin binding
Moclobemide//Amine oxidase [flavin-containing] B//Primary amine oxidase activity
Moclobemide//Amine oxidase [flavin-containing] B//Primary amine oxidase activity
Escitalopram//Sodium-dependent serotonin transporter//Serotonin:sodium symporter activity
Escitalopram//Muscarinic acetylcholine receptor M1//Phosphatidylinositol phospholipase c activity
Escitalopram//Histamine H1 receptor//Histamine receptor activity
Escitalopram//5-hydroxytryptamine receptor 1A//Serotonin receptor activity
Escitalopram//5-hydroxytryptamine receptor 2A//Virus receptor activity
Escitalopram//Alpha-1A adrenergic receptor//Protein heterodimerization activity
Escitalopram//Alpha-1B adrenergic receptor//Protein heterodimerization activity
Escitalopram//Alpha-1D adrenergic receptor//Alpha1-adrenergic receptor activity
Escitalopram//5-hydroxytryptamine receptor 2C//Serotonin receptor activity
Escitalopram//Alpha-2A adrenergic receptor//Thioesterase binding
Escitalopram//Alpha-2B adrenergic receptor//Epinephrine binding
Escitalopram//Alpha-2C adrenergic receptor//Protein homodimerization activity
Escitalopram//D(2) dopamine receptor//Potassium channel regulator activity
Escitalopram//Sodium-dependent noradrenaline transporter//Norepinephrine:sodium symporter activity
Escitalopram//Sodium-dependent dopamine transporter//Monoamine transmembrane transporter activity
Cyclizine//Histamine H1 receptor//Histamine receptor activity
Cyclizine//Estrogen sulfotransferase//Sulfotransferase activity
Idarubicin//DNA topoisomerase 2-alpha//Ubiquitin binding
Ifosfamide//Nuclear receptor subfamily 1 group I member 2//Zinc ion binding
Naloxone//Mu-type opioid receptor//Voltage-gated calcium channel activity
Naloxone//Delta-type opioid receptor//Opioid receptor activity
Naloxone//Kappa-type opioid receptor//Opioid receptor activity
Naloxone//Cyclic AMP-responsive element-binding protein 1//Transcriptional activator activity, rna polymerase ii transcription factor binding
Naloxone//Estrogen receptor//Zinc ion binding
Naloxone//Toll-like receptor 4//Transmembrane signaling receptor activity
Naloxone//Liver carboxylesterase 1//Triglyceride lipase activity
Domperidone//D(2) dopamine receptor//Potassium channel regulator activity
Domperidone//D(3) dopamine receptor//G-protein coupled amine receptor activity
Dexfenfluramine//Sodium-dependent serotonin transporter//Serotonin:sodium symporter activity
Dexfenfluramine//5-hydroxytryptamine receptor 2C//Serotonin receptor activity
Acebutolol//Beta-1 adrenergic receptor//Receptor signaling protein activity
Acebutolol//Beta-2 adrenergic receptor//Protein homodimerization activity
Brinzolamide//Carbonic anhydrase 2//Zinc ion binding
Brinzolamide//Carbonic anhydrase 1//Zinc ion binding
Brinzolamide//Carbonic anhydrase 4//Zinc ion binding
Brinzolamide//Carbonic anhydrase 5A, mitochondrial//Zinc ion binding
Brinzolamide//Carbonic anhydrase 3//Zinc ion binding
Flecainide//Sodium channel protein type 5 subunit alpha//Voltage-gated sodium channel activity involved in sa node cell action potential
Flecainide//Sodium channel protein type 4 subunit alpha//Voltage-gated sodium channel activity
Flecainide//Potassium voltage-gated channel subfamily H member 2//Voltage-gated potassium channel activity involved in ventricular cardiac muscle cell action potential repolarization
Estramustine//Estrogen receptor//Zinc ion binding
Estramustine//Estrogen receptor beta//Zinc ion binding
Estramustine//Microtubule-associated protein 2//Structural molecule activity
Estramustine//Microtubule-associated protein 1A//Structural molecule activity
Captopril//Angiotensin-converting enzyme//Zinc ion binding
Captopril//72 kDa type IV collagenase//Zinc ion binding
Captopril//Matrix metalloproteinase-9//Zinc ion binding
Captopril//Leukotriene A-4 hydrolase//Zinc ion binding
Bromocriptine//D(2) dopamine receptor//Potassium channel regulator activity
Bromocriptine//D(3) dopamine receptor//G-protein coupled amine receptor activity
Bromocriptine//5-hydroxytryptamine receptor 1D//Serotonin receptor activity
Bromocriptine//Alpha-2A adrenergic receptor//Thioesterase binding
Bromocriptine//5-hydroxytryptamine receptor 1A//Serotonin receptor activity
Bromocriptine//Alpha-2C adrenergic receptor//Protein homodimerization activity
Bromocriptine//Alpha-2B adrenergic receptor//Epinephrine binding
Bromocriptine//5-hydroxytryptamine receptor 2B//Serotonin receptor activity
Bromocriptine//D(4) dopamine receptor//Sh3 domain binding
Bromocriptine//5-hydroxytryptamine receptor 2A//Virus receptor activity
Bromocriptine//5-hydroxytryptamine receptor 1B//Serotonin receptor activity
Bromocriptine//5-hydroxytryptamine receptor 2C//Serotonin receptor activity
Bromocriptine//D(1B) dopamine receptor//G-protein coupled amine receptor activity
Bromocriptine//D(1A) dopamine receptor//G-protein coupled amine receptor activity
Bromocriptine//Alpha-1A adrenergic receptor//Protein heterodimerization activity
Bromocriptine//Alpha-1B adrenergic receptor//Protein heterodimerization activity
Bromocriptine//Alpha-1D adrenergic receptor//Alpha1-adrenergic receptor activity
Bromocriptine//5-hydroxytryptamine receptor 7//Serotonin receptor activity
Mitoxantrone//DNA topoisomerase 2-alpha//Ubiquitin binding
Clarithromycin//50S ribosomal protein L10//Structural constituent of ribosome
Clarithromycin//Potassium voltage-gated channel subfamily H member 2//Voltage-gated potassium channel activity involved in ventricular cardiac muscle cell action potential repolarization
Clarithromycin//Solute carrier organic anion transporter family member 1B1//Sodium-independent organic anion transmembrane transporter activity
Clarithromycin//Solute carrier organic anion transporter family member 1B3//Sodium-independent organic anion transmembrane transporter activity
Ceftriaxone//Solute carrier family 22 member 11//Sodium-independent organic anion transmembrane transporter activity
Ceftriaxone//Solute carrier family 22 member 6//Sodium-independent organic anion transmembrane transporter activity
Ceftriaxone//Solute carrier family 22 member 8//Sodium-independent organic anion transmembrane transporter activity
Ceftriaxone//Solute carrier family 15 member 1//Proton-dependent oligopeptide secondary active transmembrane transporter activity
Fomepizole//Alcohol dehydrogenase 1A//Zinc ion binding
Fomepizole//Alcohol dehydrogenase 1B//Zinc ion binding
Fomepizole//Alcohol dehydrogenase 1C//Zinc ion binding
Fomepizole//Catalase//Receptor binding
Estazolam//Gamma-aminobutyric acid receptor subunit alpha-1//Inhibitory extracellular ligand-gated ion channel activity
Estazolam//Gamma-aminobutyric acid receptor subunit alpha-2//Inhibitory extracellular ligand-gated ion channel activity
Estazolam//Gamma-aminobutyric acid receptor subunit alpha-3//Inhibitory extracellular ligand-gated ion channel activity
Estazolam//Gamma-aminobutyric acid receptor subunit alpha-4//Inhibitory extracellular ligand-gated ion channel activity
Estazolam//Gamma-aminobutyric acid receptor subunit alpha-5//Transporter activity
Estazolam//Gamma-aminobutyric acid receptor subunit alpha-6//Inhibitory extracellular ligand-gated ion channel activity
Estazolam//Gamma-aminobutyric acid receptor subunit beta-1//Ligand-gated ion channel activity
Estazolam//Gamma-aminobutyric acid receptor subunit beta-2//Inhibitory extracellular ligand-gated ion channel activity
Estazolam//Gamma-aminobutyric acid receptor subunit beta-3//Gaba-gated chloride ion channel activity
Estazolam//Gamma-aminobutyric acid receptor subunit delta//Gaba-a receptor activity
Estazolam//Gamma-aminobutyric acid receptor subunit epsilon//Inhibitory extracellular ligand-gated ion channel activity
Estazolam//Gamma-aminobutyric acid receptor subunit gamma-1//Inhibitory extracellular ligand-gated ion channel activity
Estazolam//Gamma-aminobutyric acid receptor subunit gamma-2//Inhibitory extracellular ligand-gated ion channel activity
Estazolam//Gamma-aminobutyric acid receptor subunit gamma-3//Inhibitory extracellular ligand-gated ion channel activity
Estazolam//Gamma-aminobutyric acid receptor subunit pi//Gaba-a receptor activity
Estazolam//Gamma-aminobutyric acid receptor subunit theta//Transmembrane signaling receptor activity
Estazolam//Gamma-aminobutyric acid receptor subunit alpha-1//Inhibitory extracellular ligand-gated ion channel activity
Estazolam//Gamma-aminobutyric acid receptor subunit alpha-2//Inhibitory extracellular ligand-gated ion channel activity
Estazolam//Gamma-aminobutyric acid receptor subunit alpha-3//Inhibitory extracellular ligand-gated ion channel activity
Estazolam//Gamma-aminobutyric acid receptor subunit alpha-5//Transporter activity
Estazolam//Gamma-aminobutyric acid receptor subunit gamma-1//Inhibitory extracellular ligand-gated ion channel activity
Estazolam//Gamma-aminobutyric acid receptor subunit gamma-2//Inhibitory extracellular ligand-gated ion channel activity
Estazolam//Gamma-aminobutyric acid receptor subunit gamma-3//Inhibitory extracellular ligand-gated ion channel activity
Finasteride//3-oxo-5-alpha-steroid 4-dehydrogenase 2//Sterol 5-alpha reductase activity
Finasteride//3-oxo-5-alpha-steroid 4-dehydrogenase 1//Electron carrier activity
Finasteride//3-oxo-5-beta-steroid 4-dehydrogenase//Steroid binding
Anastrozole//Aromatase//Oxygen binding
Halofantrine//Potassium voltage-gated channel subfamily H member 2//Voltage-gated potassium channel activity involved in ventricular cardiac muscle cell action potential repolarization
Dantrolene//Ryanodine receptor 1//Voltage-gated calcium channel activity
Ketamine//Glutamate receptor ionotropic, NMDA 3A//Protein phosphatase 2a binding
Ketamine//Substance-P receptor//Tachykinin receptor activity
Ketamine//D(2) dopamine receptor//Potassium channel regulator activity
Ketamine//Delta-type opioid receptor//Opioid receptor activity
Ketamine//Sodium-dependent noradrenaline transporter//Norepinephrine:sodium symporter activity
Ketamine//Kappa-type opioid receptor//Opioid receptor activity
Ketamine//Mu-type opioid receptor//Voltage-gated calcium channel activity
Ketamine//Muscarinic acetylcholine receptor M1//Phosphatidylinositol phospholipase c activity
Ketamine//Muscarinic acetylcholine receptor M2//G-protein coupled acetylcholine receptor activity
Ketamine//Muscarinic acetylcholine receptor M3//Receptor activity
Ketamine//Muscarinic acetylcholine receptor M4//Guanyl-nucleotide exchange factor activity
Ketamine//Muscarinic acetylcholine receptor M5//Phosphatidylinositol phospholipase c activity
Ketamine//5-hydroxytryptamine receptor 2A//Virus receptor activity
Ketamine//5-hydroxytryptamine receptor 2B//Serotonin receptor activity
Ketamine//5-hydroxytryptamine receptor 2C//Serotonin receptor activity
Ketamine//5-hydroxytryptamine receptor 1A//Serotonin receptor activity
Ketamine//5-hydroxytryptamine receptor 1B//Serotonin receptor activity
Ketamine//5-hydroxytryptamine receptor 1D//Serotonin receptor activity
Ketamine//5-hydroxytryptamine receptor 1E//Serotonin receptor activity
Ketamine//5-hydroxytryptamine receptor 1F//Serotonin receptor activity
Ketamine//5-hydroxytryptamine receptor 3A//Voltage-gated potassium channel activity
Ketamine//Cholinesterase//Identical protein binding
Ketamine//Nitric oxide synthase, brain//Tetrahydrobiopterin binding
Budesonide//Glucocorticoid receptor//Zinc ion binding
Budesonide//Annexin A1//Structural molecule activity
Aminophylline//cGMP-inhibited 3',5'-cyclic phosphodiesterase A//Metal ion binding
Aminophylline//Adenosine receptor A1//Purine nucleoside binding
Aminophylline//Adenosine receptor A3//G-protein coupled adenosine receptor activity
Aminophylline//Histone deacetylase 2//Transcription factor binding
Levomethadylacetate//Mu-type opioid receptor//Voltage-gated calcium channel activity
Levomethadylacetate//Neuronal acetylcholine receptor subunit beta-4//Ligand-gated ion channel activity
Levomethadylacetate//Neuronal acetylcholine receptor subunit alpha-3//Ligand-gated ion channel activity
Encainide//Sodium channel protein type 5 subunit alpha//Voltage-gated sodium channel activity involved in sa node cell action potential
Metoclopramide//Muscarinic acetylcholine receptor M1//Phosphatidylinositol phospholipase c activity
Metoclopramide//D(2) dopamine receptor//Potassium channel regulator activity
Metoclopramide//5-hydroxytryptamine receptor 4//Serotonin receptor activity
Metoclopramide//5-hydroxytryptamine receptor 3A//Voltage-gated potassium channel activity
Dexamethasone//Glucocorticoid receptor//Zinc ion binding
Dexamethasone//Nuclear receptor subfamily 0 group B member 1//Transcription factor binding
Dexamethasone//Annexin A1//Structural molecule activity
Dexamethasone//Nitric oxide synthase, inducible//Tetrahydrobiopterin binding
Dexamethasone//Nuclear receptor subfamily 1 group I member 2//Zinc ion binding
Levodopa//D(1A) dopamine receptor//G-protein coupled amine receptor activity
Levodopa//D(1B) dopamine receptor//G-protein coupled amine receptor activity
Levodopa//D(2) dopamine receptor//Potassium channel regulator activity
Levodopa//D(3) dopamine receptor//G-protein coupled amine receptor activity
Levodopa//D(4) dopamine receptor//Sh3 domain binding
Aripiprazole//5-hydroxytryptamine receptor 1A//Serotonin receptor activity
Aripiprazole//D(2) dopamine receptor//Potassium channel regulator activity
Aripiprazole//5-hydroxytryptamine receptor 2A//Virus receptor activity
Aripiprazole//Alpha-1A adrenergic receptor//Protein heterodimerization activity
Aripiprazole//Alpha-1B adrenergic receptor//Protein heterodimerization activity
Aripiprazole//D(3) dopamine receptor//G-protein coupled amine receptor activity
Aripiprazole//5-hydroxytryptamine receptor 1D//Serotonin receptor activity
Aripiprazole//5-hydroxytryptamine receptor 7//Serotonin receptor activity
Aripiprazole//Alpha-2A adrenergic receptor//Thioesterase binding
Aripiprazole//Alpha-2C adrenergic receptor//Protein homodimerization activity
Aripiprazole//Histamine H1 receptor//Histamine receptor activity
Aripiprazole//5-hydroxytryptamine receptor 1B//Serotonin receptor activity
Aripiprazole//5-hydroxytryptamine receptor 2C//Serotonin receptor activity
Aripiprazole//5-hydroxytryptamine receptor 3A//Voltage-gated potassium channel activity
Aripiprazole//5-hydroxytryptamine receptor 6//Serotonin receptor activity
Aripiprazole//D(1A) dopamine receptor//G-protein coupled amine receptor activity
Aripiprazole//D(4) dopamine receptor//Sh3 domain binding
Aripiprazole//Alpha-2B adrenergic receptor//Epinephrine binding
Aripiprazole//5-hydroxytryptamine receptor 1E//Serotonin receptor activity
Aripiprazole//D(1B) dopamine receptor//G-protein coupled amine receptor activity
Aripiprazole//5-hydroxytryptamine receptor 2B//Serotonin receptor activity
Aripiprazole//5-hydroxytryptamine receptor 5A//Serotonin receptor activity
Aripiprazole//Beta-1 adrenergic receptor//Receptor signaling protein activity
Aripiprazole//Beta-2 adrenergic receptor//Protein homodimerization activity
Aripiprazole//Histamine H2 receptor//Histamine receptor activity
Aripiprazole//Histamine H3 receptor//Histamine receptor activity
Aripiprazole//Histamine H4 receptor//Histamine receptor activity
Aripiprazole//Muscarinic acetylcholine receptor M1//Phosphatidylinositol phospholipase c activity
Aripiprazole//Muscarinic acetylcholine receptor M2//G-protein coupled acetylcholine receptor activity
Aripiprazole//Muscarinic acetylcholine receptor M3//Receptor activity
Aripiprazole//Muscarinic acetylcholine receptor M4//Guanyl-nucleotide exchange factor activity
Aripiprazole//Muscarinic acetylcholine receptor M5//Phosphatidylinositol phospholipase c activity
Aripiprazole//Kappa-type opioid receptor//Opioid receptor activity
Aripiprazole//Mu-type opioid receptor//Voltage-gated calcium channel activity
Aripiprazole//Delta-type opioid receptor//Opioid receptor activity
Aripiprazole//Glutamate receptor ionotropic, NMDA 1//Voltage-gated cation channel activity
Aripiprazole//Glutamate receptor ionotropic, NMDA 2A//Zinc ion binding
Aripiprazole//Glutamate receptor ionotropic, NMDA 2B//Zinc ion binding
Aripiprazole//Glutamate receptor ionotropic, NMDA 2C//Nmda glutamate receptor activity
Aripiprazole//Glutamate receptor ionotropic, NMDA 2D//Nmda glutamate receptor activity
Aripiprazole//Glutamate receptor ionotropic, NMDA 3A//Protein phosphatase 2a binding
Aripiprazole//Glutamate receptor ionotropic, NMDA 3B//Nmda glutamate receptor activity
Aripiprazole//Sodium-dependent dopamine transporter//Monoamine transmembrane transporter activity
Aripiprazole//Sodium-dependent serotonin transporter//Serotonin:sodium symporter activity
Epoprostenol//P2Y purinoceptor 12//Guanyl-nucleotide exchange factor activity
Epoprostenol//Prostacyclin receptor//Guanyl-nucleotide exchange factor activity
Gemfibrozil//Peroxisome proliferator-activated receptor alpha//Zinc ion binding
Gemfibrozil//Solute carrier organic anion transporter family member 1B1//Sodium-independent organic anion transmembrane transporter activity
Gemfibrozil//Solute carrier family 22 member 8//Sodium-independent organic anion transmembrane transporter activity
Gemfibrozil//Solute carrier organic anion transporter family member 2B1//Sodium-independent organic anion transmembrane transporter activity
Gemfibrozil//Solute carrier organic anion transporter family member 1B3//Sodium-independent organic anion transmembrane transporter activity
Clomipramine//Sodium-dependent serotonin transporter//Serotonin:sodium symporter activity
Clomipramine//5-hydroxytryptamine receptor 2A//Virus receptor activity
Clomipramine//5-hydroxytryptamine receptor 2B//Serotonin receptor activity
Clomipramine//5-hydroxytryptamine receptor 2C//Serotonin receptor activity
Clomipramine//Sodium-dependent noradrenaline transporter//Norepinephrine:sodium symporter activity
Clomipramine//Glutathione S-transferase P//S-nitrosoglutathione binding
Bepridil//Voltage-dependent P/Q-type calcium channel subunit alpha-1A//Voltage-gated calcium channel activity
Bepridil//Voltage-dependent T-type calcium channel subunit alpha-1H//Scaffold protein binding
Bepridil//Voltage-dependent calcium channel subunit alpha-2/delta-2//Voltage-gated calcium channel activity
Bepridil//Sodium/potassium-transporting ATPase subunit alpha-1//Steroid hormone binding
Bepridil//Potassium voltage-gated channel subfamily KQT member 1//Voltage-gated potassium channel activity involved in ventricular cardiac muscle cell action potential repolarization
Bepridil//Calmodulin//Titin binding
Bepridil//Calcium/calmodulin-dependent 3',5'-cyclic nucleotide phosphodiesterase 1B//Metal ion binding
Bepridil//Calcium/calmodulin-dependent 3',5'-cyclic nucleotide phosphodiesterase 1A//Metal ion binding
Bepridil//Potassium voltage-gated channel subfamily H member 2//Voltage-gated potassium channel activity involved in ventricular cardiac muscle cell action potential repolarization
Decamethonium//Acetylcholinesterase//Serine hydrolase activity
Decamethonium//Neuronal acetylcholine receptor subunit alpha-2//Drug binding
Decamethonium//Neuronal acetylcholine receptor subunit alpha-4//Ligand-gated ion channel activity
Decamethonium//Neuronal acetylcholine receptor subunit beta-2//Ligand-gated ion channel activity
Alimemazine//Histamine H1 receptor//Histamine receptor activity
Docetaxel//Tubulin beta-1 chain//Structural constituent of cytoskeleton
Docetaxel//Apoptosis regulator Bcl-2//Ubiquitin protein ligase binding
Docetaxel//Microtubule-associated protein 2//Structural molecule activity
Docetaxel//Microtubule-associated protein 4//Structural molecule activity
Docetaxel//Microtubule-associated protein tau//Structural constituent of cytoskeleton
Docetaxel//Nuclear receptor subfamily 1 group I member 2//Zinc ion binding
Mitiglinide//ATP-binding cassette sub-family C member 8//Sulfonylurea receptor activity
Mitiglinide//Peroxisome proliferator-activated receptor gamma//Zinc ion binding
Ergonovine//Alpha-1A adrenergic receptor//Protein heterodimerization activity
Dasatinib//Tyrosine-protein kinase ABL1//Syntaxin binding
Dasatinib//Proto-oncogene tyrosine-protein kinase Src//Sh3/sh2 adaptor activity
Dasatinib//Ephrin type-A receptor 2//Transmembrane receptor protein tyrosine kinase activity
Dasatinib//Tyrosine-protein kinase Lck//Sh2 domain binding
Dasatinib//Tyrosine-protein kinase Yes//Receptor binding
Dasatinib//Mast/stem cell growth factor receptor Kit//Transmembrane receptor protein tyrosine kinase activity
Dasatinib//Platelet-derived growth factor receptor beta//Vascular endothelial growth factor binding
Dasatinib//Abelson tyrosine-protein kinase 2//Receptor binding
Dasatinib//Tyrosine-protein kinase Fyn//Protein tyrosine kinase activity
Dasatinib//Tyrosine-protein kinase BTK//Protein tyrosine kinase activity
Dasatinib//Breakpoint cluster region protein//Rho guanyl-nucleotide exchange factor activity
Dasatinib//Tyrosine-protein kinase CSK//Receptor binding
Dasatinib//Ephrin type-A receptor 5//Transmembrane-ephrin receptor activity
Dasatinib//Ephrin type-B receptor 4//Transmembrane receptor protein tyrosine kinase activity
Dasatinib//Tyrosine-protein kinase Fgr//Protein tyrosine kinase activity
Dasatinib//Tyrosine-protein kinase FRK//Receptor binding
Dasatinib//Heat shock cognate 71 kDa protein//Unfolded protein binding
Dasatinib//Tyrosine-protein kinase Lyn//Receptor signaling protein tyrosine kinase activity
Dasatinib//Mitogen-activated protein kinase kinase kinase MLT//Protein serine/threonine kinase activity
Dasatinib//Mitogen-activated protein kinase 14//Protein serine/threonine kinase activity
Dasatinib//Amidophosphoribosyltransferase//Metal ion binding
Lapatinib//Receptor tyrosine-protein kinase erbB-2//Transmembrane signaling receptor activity
Lapatinib//Epidermal growth factor receptor//Ubiquitin protein ligase binding
Decitabine//DNA (cytosine-5)-methyltransferase 1//Zinc ion binding
Arformoterol//Beta-2 adrenergic receptor//Protein homodimerization activity
Hydralazine//Hypoxia-inducible factor 1-alpha//Ubiquitin protein ligase binding
Nelarabine//DNA polymerase alpha catalytic subunit//Protein kinase binding
Lumiracoxib//Prostaglandin G/H synthase 1//Prostaglandin-endoperoxide synthase activity
Lumiracoxib//Prostaglandin G/H synthase 2//Prostaglandin-endoperoxide synthase activity
Glucosamine//Matrix metalloproteinase-9//Zinc ion binding
Glucosamine//Tumor necrosis factor//Tumor necrosis factor receptor binding
Glucosamine//Nuclear factor NF-kappa-B p100 subunit//Transcriptional activator activity, rna polymerase ii core promoter proximal region sequence-specific binding
Fosphenytoin//Sodium channel protein type 5 subunit alpha//Voltage-gated sodium channel activity involved in sa node cell action potential
Cefazolin//Serum paraoxonase/arylesterase 1//Protein homodimerization activity
Amobarbital//Gamma-aminobutyric acid receptor subunit alpha-1//Inhibitory extracellular ligand-gated ion channel activity
Amobarbital//Gamma-aminobutyric acid receptor subunit alpha-2//Inhibitory extracellular ligand-gated ion channel activity
Amobarbital//Gamma-aminobutyric acid receptor subunit alpha-3//Inhibitory extracellular ligand-gated ion channel activity
Amobarbital//Gamma-aminobutyric acid receptor subunit alpha-4//Inhibitory extracellular ligand-gated ion channel activity
Amobarbital//Gamma-aminobutyric acid receptor subunit alpha-5//Transporter activity
Amobarbital//Gamma-aminobutyric acid receptor subunit alpha-6//Inhibitory extracellular ligand-gated ion channel activity
Amobarbital//Neuronal acetylcholine receptor subunit alpha-4//Ligand-gated ion channel activity
Amobarbital//Neuronal acetylcholine receptor subunit alpha-7//Toxic substance binding
Amobarbital//Glutamate receptor 2//Ionotropic glutamate receptor activity
Amobarbital//Glutamate receptor ionotropic, kainate 2//Kainate selective glutamate receptor activity
Hexobarbital//Gamma-aminobutyric acid receptor subunit alpha-1//Inhibitory extracellular ligand-gated ion channel activity
Hexobarbital//Gamma-aminobutyric acid receptor subunit alpha-2//Inhibitory extracellular ligand-gated ion channel activity
Hexobarbital//Gamma-aminobutyric acid receptor subunit alpha-3//Inhibitory extracellular ligand-gated ion channel activity
Hexobarbital//Gamma-aminobutyric acid receptor subunit alpha-4//Inhibitory extracellular ligand-gated ion channel activity
Hexobarbital//Gamma-aminobutyric acid receptor subunit alpha-5//Transporter activity
Hexobarbital//Gamma-aminobutyric acid receptor subunit alpha-6//Inhibitory extracellular ligand-gated ion channel activity
Hexobarbital//Neuronal acetylcholine receptor subunit alpha-4//Ligand-gated ion channel activity
Hexobarbital//Neuronal acetylcholine receptor subunit alpha-7//Toxic substance binding
Hexobarbital//Glutamate receptor 2//Ionotropic glutamate receptor activity
Hexobarbital//Glutamate receptor ionotropic, kainate 2//Kainate selective glutamate receptor activity
Mestranol//Estrogen receptor//Zinc ion binding
Ephedrine//Sodium-dependent noradrenaline transporter//Norepinephrine:sodium symporter activity
Ephedrine//Alpha-1A adrenergic receptor//Protein heterodimerization activity
Ephedrine//Beta-1 adrenergic receptor//Receptor signaling protein activity
Ephedrine//Beta-2 adrenergic receptor//Protein homodimerization activity
Cortisoneacetate//Glucocorticoid receptor//Zinc ion binding
Bezafibrate//Peroxisome proliferator-activated receptor alpha//Zinc ion binding
Bezafibrate//Peroxisome proliferator-activated receptor delta//Zinc ion binding
Bezafibrate//Peroxisome proliferator-activated receptor gamma//Zinc ion binding
Bezafibrate//Nuclear receptor subfamily 1 group I member 2//Zinc ion binding
Bezafibrate//Retinoic acid receptor RXR-alpha//Zinc ion binding
Bezafibrate//Retinoic acid receptor RXR-beta//Zinc ion binding
Bezafibrate//Retinoic acid receptor RXR-gamma//Zinc ion binding
Colchicine//Tubulin beta chain//Ubiquitin protein ligase binding
Drospirenone//Progesterone receptor//Zinc ion binding
Drospirenone//Mineralocorticoid receptor//Zinc ion binding
Drospirenone//Androgen receptor//Zinc ion binding
Drospirenone//Glucocorticoid receptor//Zinc ion binding
Digitoxin//Sodium/potassium-transporting ATPase subunit alpha-1//Steroid hormone binding
Neostigmine//Acetylcholinesterase//Serine hydrolase activity
Methotrimeprazine//D(2) dopamine receptor//Potassium channel regulator activity
Methotrimeprazine//D(1A) dopamine receptor//G-protein coupled amine receptor activity
Methotrimeprazine//D(1B) dopamine receptor//G-protein coupled amine receptor activity
Methotrimeprazine//D(3) dopamine receptor//G-protein coupled amine receptor activity
Methotrimeprazine//D(4) dopamine receptor//Sh3 domain binding
Methotrimeprazine//5-hydroxytryptamine receptor 2A//Virus receptor activity
Methotrimeprazine//5-hydroxytryptamine receptor 2C//Serotonin receptor activity
Methotrimeprazine//Histamine H1 receptor//Histamine receptor activity
Methotrimeprazine//Muscarinic acetylcholine receptor M1//Phosphatidylinositol phospholipase c activity
Methotrimeprazine//Muscarinic acetylcholine receptor M2//G-protein coupled acetylcholine receptor activity
Methotrimeprazine//Muscarinic acetylcholine receptor M3//Receptor activity
Methotrimeprazine//Muscarinic acetylcholine receptor M4//Guanyl-nucleotide exchange factor activity
Methotrimeprazine//Muscarinic acetylcholine receptor M5//Phosphatidylinositol phospholipase c activity
Methotrimeprazine//Alpha-1A adrenergic receptor//Protein heterodimerization activity
Methotrimeprazine//Alpha-1B adrenergic receptor//Protein heterodimerization activity
Methotrimeprazine//Alpha-1D adrenergic receptor//Alpha1-adrenergic receptor activity
Methotrimeprazine//Alpha-2A adrenergic receptor//Thioesterase binding
Methotrimeprazine//Alpha-2B adrenergic receptor//Epinephrine binding
Methotrimeprazine//Alpha-2C adrenergic receptor//Protein homodimerization activity
Danazol//Estrogen receptor//Zinc ion binding
Danazol//Androgen receptor//Zinc ion binding
Danazol//Progesterone receptor//Zinc ion binding
Clenbuterol//Beta-2 adrenergic receptor//Protein homodimerization activity
Clenbuterol//Beta-1 adrenergic receptor//Receptor signaling protein activity
Clenbuterol//Beta-3 adrenergic receptor//Protein homodimerization activity
Clenbuterol//Beta-nerve growth factor//Receptor signaling protein activity
Clenbuterol//Tumor necrosis factor//Tumor necrosis factor receptor binding
Bambuterol//Beta-2 adrenergic receptor//Protein homodimerization activity
Ciclesonide//Glucocorticoid receptor//Zinc ion binding
Acenocoumarol//Vitamin K epoxide reductase complex subunit 1//Vitamin-k-epoxide reductase (warfarin-sensitive) activity
Ajmaline//Sodium channel protein type 5 subunit alpha//Voltage-gated sodium channel activity involved in sa node cell action potential
Aprindine//Sodium channel protein type 5 subunit alpha//Voltage-gated sodium channel activity involved in sa node cell action potential
Aprindine//Calmodulin//Titin binding
Allylestrenol//Progesterone receptor//Zinc ion binding
Allylestrenol//Estrogen receptor//Zinc ion binding
Antipyrine//Prostaglandin G/H synthase 2//Prostaglandin-endoperoxide synthase activity
Antipyrine//Prostaglandin G/H synthase 1//Prostaglandin-endoperoxide synthase activity
Glutethimide//Gamma-aminobutyric acid receptor subunit alpha-1//Inhibitory extracellular ligand-gated ion channel activity
Glutethimide//Gamma-aminobutyric acid receptor subunit alpha-1//Inhibitory extracellular ligand-gated ion channel activity
Glutethimide//Gamma-aminobutyric acid receptor subunit alpha-2//Inhibitory extracellular ligand-gated ion channel activity
Glutethimide//Gamma-aminobutyric acid receptor subunit alpha-3//Inhibitory extracellular ligand-gated ion channel activity
Glutethimide//Gamma-aminobutyric acid receptor subunit alpha-4//Inhibitory extracellular ligand-gated ion channel activity
Glutethimide//Gamma-aminobutyric acid receptor subunit alpha-5//Transporter activity
Glutethimide//Gamma-aminobutyric acid receptor subunit alpha-6//Inhibitory extracellular ligand-gated ion channel activity
Glutethimide//Gamma-aminobutyric acid receptor subunit beta-1//Ligand-gated ion channel activity
Glutethimide//Gamma-aminobutyric acid receptor subunit beta-2//Inhibitory extracellular ligand-gated ion channel activity
Glutethimide//Gamma-aminobutyric acid receptor subunit beta-3//Gaba-gated chloride ion channel activity
Glutethimide//Gamma-aminobutyric acid receptor subunit delta//Gaba-a receptor activity
Glutethimide//Gamma-aminobutyric acid receptor subunit epsilon//Inhibitory extracellular ligand-gated ion channel activity
Glutethimide//Gamma-aminobutyric acid receptor subunit gamma-1//Inhibitory extracellular ligand-gated ion channel activity
Glutethimide//Gamma-aminobutyric acid receptor subunit gamma-2//Inhibitory extracellular ligand-gated ion channel activity
Glutethimide//Gamma-aminobutyric acid receptor subunit gamma-3//Inhibitory extracellular ligand-gated ion channel activity
Glutethimide//Gamma-aminobutyric acid receptor subunit pi//Gaba-a receptor activity
Glutethimide//Gamma-aminobutyric acid receptor subunit theta//Transmembrane signaling receptor activity
Ethylmorphine//Mu-type opioid receptor//Voltage-gated calcium channel activity
Flunitrazepam//Gamma-aminobutyric acid receptor subunit alpha-1//Inhibitory extracellular ligand-gated ion channel activity
Flunitrazepam//Gamma-aminobutyric acid receptor subunit alpha-2//Inhibitory extracellular ligand-gated ion channel activity
Flunitrazepam//Gamma-aminobutyric acid receptor subunit alpha-3//Inhibitory extracellular ligand-gated ion channel activity
Flunitrazepam//Gamma-aminobutyric acid receptor subunit alpha-4//Inhibitory extracellular ligand-gated ion channel activity
Flunitrazepam//Gamma-aminobutyric acid receptor subunit alpha-5//Transporter activity
Flunitrazepam//Gamma-aminobutyric acid receptor subunit alpha-6//Inhibitory extracellular ligand-gated ion channel activity
Flunitrazepam//Gamma-aminobutyric acid receptor subunit beta-1//Ligand-gated ion channel activity
Flunitrazepam//Gamma-aminobutyric acid receptor subunit beta-2//Inhibitory extracellular ligand-gated ion channel activity
Flunitrazepam//Gamma-aminobutyric acid receptor subunit beta-3//Gaba-gated chloride ion channel activity
Flunitrazepam//Gamma-aminobutyric acid receptor subunit delta//Gaba-a receptor activity
Flunitrazepam//Gamma-aminobutyric acid receptor subunit epsilon//Inhibitory extracellular ligand-gated ion channel activity
Flunitrazepam//Gamma-aminobutyric acid receptor subunit gamma-1//Inhibitory extracellular ligand-gated ion channel activity
Flunitrazepam//Gamma-aminobutyric acid receptor subunit gamma-2//Inhibitory extracellular ligand-gated ion channel activity
Flunitrazepam//Gamma-aminobutyric acid receptor subunit gamma-3//Inhibitory extracellular ligand-gated ion channel activity
Flunitrazepam//Gamma-aminobutyric acid receptor subunit pi//Gaba-a receptor activity
Flunitrazepam//Gamma-aminobutyric acid receptor subunit theta//Transmembrane signaling receptor activity
Flunitrazepam//Gamma-aminobutyric acid receptor subunit alpha-1//Inhibitory extracellular ligand-gated ion channel activity
Flunitrazepam//Gamma-aminobutyric acid receptor subunit alpha-2//Inhibitory extracellular ligand-gated ion channel activity
Flunitrazepam//Gamma-aminobutyric acid receptor subunit alpha-3//Inhibitory extracellular ligand-gated ion channel activity
Flunitrazepam//Gamma-aminobutyric acid receptor subunit alpha-5//Transporter activity
Flunitrazepam//Gamma-aminobutyric acid receptor subunit gamma-1//Inhibitory extracellular ligand-gated ion channel activity
Flunitrazepam//Gamma-aminobutyric acid receptor subunit gamma-2//Inhibitory extracellular ligand-gated ion channel activity
Flunitrazepam//Gamma-aminobutyric acid receptor subunit gamma-3//Inhibitory extracellular ligand-gated ion channel activity
Bromazepam//Gamma-aminobutyric acid receptor subunit alpha-1//Inhibitory extracellular ligand-gated ion channel activity
Bromazepam//Gamma-aminobutyric acid receptor subunit alpha-2//Inhibitory extracellular ligand-gated ion channel activity
Bromazepam//Gamma-aminobutyric acid receptor subunit alpha-3//Inhibitory extracellular ligand-gated ion channel activity
Bromazepam//Gamma-aminobutyric acid receptor subunit alpha-4//Inhibitory extracellular ligand-gated ion channel activity
Bromazepam//Gamma-aminobutyric acid receptor subunit alpha-5//Transporter activity
Bromazepam//Gamma-aminobutyric acid receptor subunit alpha-6//Inhibitory extracellular ligand-gated ion channel activity
Bromazepam//Gamma-aminobutyric acid receptor subunit beta-1//Ligand-gated ion channel activity
Bromazepam//Gamma-aminobutyric acid receptor subunit beta-2//Inhibitory extracellular ligand-gated ion channel activity
Bromazepam//Gamma-aminobutyric acid receptor subunit beta-3//Gaba-gated chloride ion channel activity
Bromazepam//Gamma-aminobutyric acid receptor subunit delta//Gaba-a receptor activity
Bromazepam//Gamma-aminobutyric acid receptor subunit epsilon//Inhibitory extracellular ligand-gated ion channel activity
Bromazepam//Gamma-aminobutyric acid receptor subunit gamma-1//Inhibitory extracellular ligand-gated ion channel activity
Bromazepam//Gamma-aminobutyric acid receptor subunit gamma-2//Inhibitory extracellular ligand-gated ion channel activity
Bromazepam//Gamma-aminobutyric acid receptor subunit gamma-3//Inhibitory extracellular ligand-gated ion channel activity
Bromazepam//Gamma-aminobutyric acid receptor subunit pi//Gaba-a receptor activity
Bromazepam//Gamma-aminobutyric acid receptor subunit theta//Transmembrane signaling receptor activity
Bromazepam//Gamma-aminobutyric acid receptor subunit alpha-1//Inhibitory extracellular ligand-gated ion channel activity
Bromazepam//Gamma-aminobutyric acid receptor subunit alpha-2//Inhibitory extracellular ligand-gated ion channel activity
Bromazepam//Gamma-aminobutyric acid receptor subunit alpha-3//Inhibitory extracellular ligand-gated ion channel activity
Bromazepam//Gamma-aminobutyric acid receptor subunit alpha-5//Transporter activity
Bromazepam//Gamma-aminobutyric acid receptor subunit gamma-1//Inhibitory extracellular ligand-gated ion channel activity
Bromazepam//Gamma-aminobutyric acid receptor subunit gamma-2//Inhibitory extracellular ligand-gated ion channel activity
Bromazepam//Gamma-aminobutyric acid receptor subunit gamma-3//Inhibitory extracellular ligand-gated ion channel activity
Clotiazepam//Gamma-aminobutyric acid receptor subunit alpha-1//Inhibitory extracellular ligand-gated ion channel activity
Clotiazepam//Gamma-aminobutyric acid receptor subunit alpha-2//Inhibitory extracellular ligand-gated ion channel activity
Clotiazepam//Gamma-aminobutyric acid receptor subunit alpha-3//Inhibitory extracellular ligand-gated ion channel activity
Clotiazepam//Gamma-aminobutyric acid receptor subunit alpha-4//Inhibitory extracellular ligand-gated ion channel activity
Clotiazepam//Gamma-aminobutyric acid receptor subunit alpha-5//Transporter activity
Clotiazepam//Gamma-aminobutyric acid receptor subunit alpha-6//Inhibitory extracellular ligand-gated ion channel activity
Clotiazepam//Gamma-aminobutyric acid receptor subunit beta-1//Ligand-gated ion channel activity
Clotiazepam//Gamma-aminobutyric acid receptor subunit beta-2//Inhibitory extracellular ligand-gated ion channel activity
Clotiazepam//Gamma-aminobutyric acid receptor subunit beta-3//Gaba-gated chloride ion channel activity
Clotiazepam//Gamma-aminobutyric acid receptor subunit delta//Gaba-a receptor activity
Clotiazepam//Gamma-aminobutyric acid receptor subunit epsilon//Inhibitory extracellular ligand-gated ion channel activity
Clotiazepam//Gamma-aminobutyric acid receptor subunit gamma-1//Inhibitory extracellular ligand-gated ion channel activity
Clotiazepam//Gamma-aminobutyric acid receptor subunit gamma-2//Inhibitory extracellular ligand-gated ion channel activity
Clotiazepam//Gamma-aminobutyric acid receptor subunit gamma-3//Inhibitory extracellular ligand-gated ion channel activity
Clotiazepam//Gamma-aminobutyric acid receptor subunit pi//Gaba-a receptor activity
Clotiazepam//Gamma-aminobutyric acid receptor subunit theta//Transmembrane signaling receptor activity
Clotiazepam//Gamma-aminobutyric acid receptor subunit alpha-1//Inhibitory extracellular ligand-gated ion channel activity
Clotiazepam//Gamma-aminobutyric acid receptor subunit alpha-2//Inhibitory extracellular ligand-gated ion channel activity
Clotiazepam//Gamma-aminobutyric acid receptor subunit alpha-3//Inhibitory extracellular ligand-gated ion channel activity
Clotiazepam//Gamma-aminobutyric acid receptor subunit alpha-5//Transporter activity
Clotiazepam//Gamma-aminobutyric acid receptor subunit gamma-1//Inhibitory extracellular ligand-gated ion channel activity
Clotiazepam//Gamma-aminobutyric acid receptor subunit gamma-2//Inhibitory extracellular ligand-gated ion channel activity
Clotiazepam//Gamma-aminobutyric acid receptor subunit gamma-3//Inhibitory extracellular ligand-gated ion channel activity
Dextroamphetamine//Synaptic vesicular amine transporter//Monoamine transmembrane transporter activity
Dextroamphetamine//Sodium-dependent noradrenaline transporter//Norepinephrine:sodium symporter activity
Dextroamphetamine//Sodium-dependent dopamine transporter//Monoamine transmembrane transporter activity
Dextroamphetamine//Trace amine-associated receptor 1//Trace-amine receptor activity
Dextroamphetamine//Alpha-1B adrenergic receptor//Protein heterodimerization activity
Dextroamphetamine//Alpha-1A adrenergic receptor//Protein heterodimerization activity
Dextroamphetamine//Alpha-1B adrenergic receptor//Protein heterodimerization activity
Dextroamphetamine//Alpha-1D adrenergic receptor//Alpha1-adrenergic receptor activity
Dextroamphetamine//Alpha-2A adrenergic receptor//Thioesterase binding
Dextroamphetamine//Alpha-2B adrenergic receptor//Epinephrine binding
Dextroamphetamine//Alpha-2C adrenergic receptor//Protein homodimerization activity
Methamphetamine//Sodium-dependent dopamine transporter//Monoamine transmembrane transporter activity
Methamphetamine//Sodium-dependent serotonin transporter//Serotonin:sodium symporter activity
Methamphetamine//Sodium-dependent noradrenaline transporter//Norepinephrine:sodium symporter activity
Methamphetamine//Synaptic vesicular amine transporter//Monoamine transmembrane transporter activity
Methamphetamine//Trace amine-associated receptor 1//Trace-amine receptor activity
Methamphetamine//Alpha-2A adrenergic receptor//Thioesterase binding
Methamphetamine//Alpha-2B adrenergic receptor//Epinephrine binding
Methamphetamine//Alpha-2C adrenergic receptor//Protein homodimerization activity
Methamphetamine//Amine oxidase [flavin-containing] A//Serotonin binding
Methamphetamine//Amine oxidase [flavin-containing] B//Primary amine oxidase activity
Liotrix//Thyroid hormone receptor alpha//Zinc ion binding
Liotrix//Thyroid hormone receptor beta//Zinc ion binding
Ketazolam//Gamma-aminobutyric acid receptor subunit alpha-1//Inhibitory extracellular ligand-gated ion channel activity
Ketazolam//Gamma-aminobutyric acid receptor subunit alpha-2//Inhibitory extracellular ligand-gated ion channel activity
Ketazolam//Gamma-aminobutyric acid receptor subunit alpha-3//Inhibitory extracellular ligand-gated ion channel activity
Ketazolam//Gamma-aminobutyric acid receptor subunit alpha-4//Inhibitory extracellular ligand-gated ion channel activity
Ketazolam//Gamma-aminobutyric acid receptor subunit alpha-5//Transporter activity
Ketazolam//Gamma-aminobutyric acid receptor subunit alpha-6//Inhibitory extracellular ligand-gated ion channel activity
Ketazolam//Gamma-aminobutyric acid receptor subunit beta-1//Ligand-gated ion channel activity
Ketazolam//Gamma-aminobutyric acid receptor subunit beta-2//Inhibitory extracellular ligand-gated ion channel activity
Ketazolam//Gamma-aminobutyric acid receptor subunit beta-3//Gaba-gated chloride ion channel activity
Ketazolam//Gamma-aminobutyric acid receptor subunit delta//Gaba-a receptor activity
Ketazolam//Gamma-aminobutyric acid receptor subunit epsilon//Inhibitory extracellular ligand-gated ion channel activity
Ketazolam//Gamma-aminobutyric acid receptor subunit gamma-1//Inhibitory extracellular ligand-gated ion channel activity
Ketazolam//Gamma-aminobutyric acid receptor subunit gamma-2//Inhibitory extracellular ligand-gated ion channel activity
Ketazolam//Gamma-aminobutyric acid receptor subunit gamma-3//Inhibitory extracellular ligand-gated ion channel activity
Ketazolam//Gamma-aminobutyric acid receptor subunit pi//Gaba-a receptor activity
Ketazolam//Gamma-aminobutyric acid receptor subunit theta//Transmembrane signaling receptor activity
Ketazolam//Gamma-aminobutyric acid receptor subunit alpha-1//Inhibitory extracellular ligand-gated ion channel activity
Ketazolam//Gamma-aminobutyric acid receptor subunit alpha-2//Inhibitory extracellular ligand-gated ion channel activity
Ketazolam//Gamma-aminobutyric acid receptor subunit alpha-3//Inhibitory extracellular ligand-gated ion channel activity
Ketazolam//Gamma-aminobutyric acid receptor subunit alpha-5//Transporter activity
Ketazolam//Gamma-aminobutyric acid receptor subunit gamma-1//Inhibitory extracellular ligand-gated ion channel activity
Ketazolam//Gamma-aminobutyric acid receptor subunit gamma-2//Inhibitory extracellular ligand-gated ion channel activity
Ketazolam//Gamma-aminobutyric acid receptor subunit gamma-3//Inhibitory extracellular ligand-gated ion channel activity
Hydroxychloroquine//Toll-like receptor 7//Transmembrane signaling receptor activity
Hydroxychloroquine//Toll-like receptor 9//Transmembrane signaling receptor activity
Hydroxychloroquine//Angiotensin-converting enzyme 2//Zinc ion binding
Amylnitrite//Atrial natriuretic peptide receptor 1//Protein kinase activity
Etoricoxib//Prostaglandin G/H synthase 2//Prostaglandin-endoperoxide synthase activity
Calcipotriol//Vitamin D3 receptor//Zinc ion binding
Acetylcholine//Acetylcholinesterase//Serine hydrolase activity
Acetylcholine//Muscarinic acetylcholine receptor M1//Phosphatidylinositol phospholipase c activity
Acetylcholine//Muscarinic acetylcholine receptor M2//G-protein coupled acetylcholine receptor activity
Acetylcholine//Muscarinic acetylcholine receptor M3//Receptor activity
Acetylcholine//Muscarinic acetylcholine receptor M4//Guanyl-nucleotide exchange factor activity
Acetylcholine//Neuronal acetylcholine receptor subunit alpha-7//Toxic substance binding
Doconexent//Peroxisome proliferator-activated receptor alpha//Zinc ion binding
Doconexent//Peroxisome proliferator-activated receptor gamma//Zinc ion binding
Doconexent//Retinoic acid receptor RXR-alpha//Zinc ion binding
Doconexent//Retinoic acid receptor RXR-beta//Zinc ion binding
Doconexent//Retinoic acid receptor RXR-gamma//Zinc ion binding
Doconexent//Sterol regulatory element-binding protein 1//Transcriptional activator activity, rna polymerase ii core promoter proximal region sequence-specific binding
Estronesulfate//Estrogen receptor//Zinc ion binding
Estronesulfate//Estrogen receptor beta//Zinc ion binding
Bifonazole//Lanosterol 14-alpha demethylase//Sterol 14-demethylase activity
Bifonazole//Cytochrome P450 2B6//Steroid hydroxylase activity
Metamizole//Prostaglandin G/H synthase 1//Prostaglandin-endoperoxide synthase activity
Maraviroc//C-C chemokine receptor type 5//Virus receptor activity
Cyproteroneacetate//Androgen receptor//Zinc ion binding
Debrisoquin//Sodium-dependent noradrenaline transporter//Norepinephrine:sodium symporter activity
Flunarizine//Voltage-dependent T-type calcium channel subunit alpha-1G//Scaffold protein binding
Flunarizine//Voltage-dependent T-type calcium channel subunit alpha-1H//Scaffold protein binding
Flunarizine//Voltage-dependent T-type calcium channel subunit alpha-1I//Voltage-gated calcium channel activity
Flunarizine//Histamine H1 receptor//Histamine receptor activity
Flunarizine//Calmodulin//Titin binding
Ixabepilone//Tubulin beta-3 chain//Structural constituent of cytoskeleton
Celiprolol//Beta-1 adrenergic receptor//Receptor signaling protein activity
Celiprolol//Beta-2 adrenergic receptor//Protein homodimerization activity
Celiprolol//Beta-3 adrenergic receptor//Protein homodimerization activity
Celiprolol//Alpha-2A adrenergic receptor//Thioesterase binding
Celiprolol//Alpha-2B adrenergic receptor//Epinephrine binding
Celiprolol//Alpha-2C adrenergic receptor//Protein homodimerization activity
Dronedarone//Alpha-1A adrenergic receptor//Protein heterodimerization activity
Dronedarone//Alpha-1B adrenergic receptor//Protein heterodimerization activity
Dronedarone//Alpha-1D adrenergic receptor//Alpha1-adrenergic receptor activity
Dronedarone//Alpha-2A adrenergic receptor//Thioesterase binding
Dronedarone//Alpha-2B adrenergic receptor//Epinephrine binding
Dronedarone//Alpha-2C adrenergic receptor//Protein homodimerization activity
Dronedarone//Beta-1 adrenergic receptor//Receptor signaling protein activity
Dronedarone//Potassium voltage-gated channel subfamily H member 2//Voltage-gated potassium channel activity involved in ventricular cardiac muscle cell action potential repolarization
Dronedarone//Voltage-dependent L-type calcium channel subunit alpha-1C//Voltage-gated calcium channel activity
Dronedarone//Voltage-dependent L-type calcium channel subunit alpha-1D//Voltage-gated calcium channel activity involved sa node cell action potential
Dronedarone//Voltage-dependent L-type calcium channel subunit alpha-1F//Voltage-gated calcium channel activity
Dronedarone//Voltage-dependent L-type calcium channel subunit alpha-1S//Voltage-gated calcium channel activity
Dronedarone//Voltage-dependent L-type calcium channel subunit beta-1//Voltage-gated calcium channel activity
Dronedarone//Voltage-dependent L-type calcium channel subunit beta-2//Voltage-gated calcium channel activity
Dronedarone//Voltage-dependent L-type calcium channel subunit beta-3//Voltage-gated calcium channel activity
Dronedarone//Voltage-dependent L-type calcium channel subunit beta-4//Voltage-gated calcium channel activity
Dronedarone//Sodium channel protein type 5 subunit alpha//Voltage-gated sodium channel activity involved in sa node cell action potential
Dronedarone//G protein-activated inward rectifier potassium channel 1//G-protein activated inward rectifier potassium channel activity
Dronedarone//Potassium voltage-gated channel subfamily KQT member 1//Voltage-gated potassium channel activity involved in ventricular cardiac muscle cell action potential repolarization
Dronedarone//ATP-sensitive inward rectifier potassium channel 12//Inward rectifier potassium channel activity
Dronedarone//ATP-sensitive inward rectifier potassium channel 14//Inward rectifier potassium channels are characterized by a greater tendency to allow potassium to flow into the cell rather than out of it. Their voltage dependence is regulated by the concentration of extracellular potassium; as external potassium is raised, the voltage range of the channel opening shifts to more positive voltages. The inward rectification is mainly due to the blockage of outward current by internal magnesium. KCNJ14 gives rise to low-conductance channels with a low affinity to the channel blockers Barium and Cesium (By similarity).
Dronedarone//Inward rectifier potassium channel 2//Probably participates in establishing action potential waveform and excitability of neuronal and muscle tissues. Inward rectifier potassium channels are characterized by a greater tendency to allow potassium to flow into the cell rather than out of it. Their voltage dependence is regulated by the concentration of extracellular potassium; as external potassium is raised, the voltage range of the channel opening shifts to more positive voltages. The inward rectification is mainly due to the blockage of outward current by internal magnesium. Can be blocked by extracellular barium or cesium.
Dronedarone//Inward rectifier potassium channel 4//Pdz domain binding
Dronedarone//Potassium voltage-gated channel subfamily D member 3//Metal ion binding
Dronedarone//Thyroid hormone receptor alpha//Zinc ion binding
Nebivolol//Beta-1 adrenergic receptor//Receptor signaling protein activity
Nebivolol//Beta-2 adrenergic receptor//Protein homodimerization activity
Nebivolol//Beta-3 adrenergic receptor//Protein homodimerization activity
Lorcaserin//5-hydroxytryptamine receptor 2C//Serotonin receptor activity
Flibanserin//5-hydroxytryptamine receptor 1A//Serotonin receptor activity
Flibanserin//D(4) dopamine receptor//Sh3 domain binding
Flibanserin//5-hydroxytryptamine receptor 2A//Virus receptor activity
Clevidipine//Voltage-dependent L-type calcium channel subunit alpha-1C//Voltage-gated calcium channel activity
Clevidipine//Voltage-dependent L-type calcium channel subunit alpha-1S//Voltage-gated calcium channel activity
Clevidipine//Voltage-dependent L-type calcium channel subunit alpha-1F//Voltage-gated calcium channel activity
Clevidipine//Voltage-dependent L-type calcium channel subunit alpha-1D//Voltage-gated calcium channel activity involved sa node cell action potential
Iloperidone//5-hydroxytryptamine receptor 2A//Virus receptor activity
Iloperidone//D(2) dopamine receptor//Potassium channel regulator activity
Iloperidone//D(1A) dopamine receptor//G-protein coupled amine receptor activity
Iloperidone//D(3) dopamine receptor//G-protein coupled amine receptor activity
Iloperidone//D(4) dopamine receptor//Sh3 domain binding
Iloperidone//5-hydroxytryptamine receptor 1A//Serotonin receptor activity
Iloperidone//5-hydroxytryptamine receptor 6//Serotonin receptor activity
Iloperidone//5-hydroxytryptamine receptor 7//Serotonin receptor activity
Iloperidone//Alpha-1A adrenergic receptor//Protein heterodimerization activity
Iloperidone//Histamine H1 receptor//Histamine receptor activity
Iloperidone//Alpha-2C adrenergic receptor//Protein homodimerization activity
Ezogabine//Potassium voltage-gated channel subfamily KQT member 2//Voltage-gated potassium channel activity
Ezogabine//Potassium voltage-gated channel subfamily KQT member 3//Voltage-gated potassium channel activity
Ezogabine//Potassium voltage-gated channel subfamily KQT member 4//Potassium channel activity
Ezogabine//Potassium voltage-gated channel subfamily KQT member 5//Voltage-gated potassium channel activity
Indacaterol//Beta-2 adrenergic receptor//Protein homodimerization activity
Crisaborole//cAMP-specific 3',5'-cyclic phosphodiesterase 4B//Metal ion binding
Crisaborole//cAMP-specific 3',5'-cyclic phosphodiesterase 4A//Metal ion binding
Crisaborole//cAMP-specific 3',5'-cyclic phosphodiesterase 4D//Ubiquitin protein ligase binding
Crisaborole//cAMP-specific 3',5'-cyclic phosphodiesterase 4C//Metal ion binding
Methsuximide//Voltage-dependent T-type calcium channel subunit alpha-1G//Scaffold protein binding
Dexlansoprazole//Potassium-transporting ATPase alpha chain 1//Sodium:potassium-exchanging atpase activity
Dexlansoprazole//N(G),N(G)-dimethylarginine dimethylaminohydrolase 1//Metal ion binding
Histamine//Histamine H1 receptor//Histamine receptor activity
Histamine//Histamine H2 receptor//Histamine receptor activity
Histamine//Histamine H3 receptor//Histamine receptor activity
Histamine//Histamine H4 receptor//Histamine receptor activity
Histamine//Synaptic vesicular amine transporter//Monoamine transmembrane transporter activity
Brivaracetam//Synaptic vesicle glycoprotein 2A//Transmembrane transporter activity
Brivaracetam//Sodium channel protein type 1 subunit alpha//Voltage-gated sodium channel activity
Brivaracetam//Sodium channel protein type 10 subunit alpha//Voltage-gated sodium channel activity
Brivaracetam//Sodium channel protein type 11 subunit alpha//Voltage-gated sodium channel activity
Brivaracetam//Sodium channel protein type 2 subunit alpha//Voltage-gated sodium channel activity
Brivaracetam//Sodium channel protein type 3 subunit alpha//Voltage-gated sodium channel activity
Brivaracetam//Sodium channel protein type 4 subunit alpha//Voltage-gated sodium channel activity
Brivaracetam//Sodium channel protein type 5 subunit alpha//Voltage-gated sodium channel activity involved in sa node cell action potential
Brivaracetam//Sodium channel protein type 7 subunit alpha//Mediates the voltage-dependent sodium ion permeability of excitable membranes. Assuming opened or closed conformations in response to the voltage difference across the membrane, the protein forms a sodium-selective channel through which Na(+) ions may pass in accordance with their electrochemical gradient.
Brivaracetam//Sodium channel protein type 8 subunit alpha//Voltage-gated sodium channel activity
Brivaracetam//Sodium channel protein type 9 subunit alpha//Voltage-gated sodium channel activity
Brivaracetam//Sodium channel subunit beta-2//Voltage-gated sodium channel activity involved in cardiac muscle cell action potential
Brivaracetam//Sodium channel subunit beta-3//Voltage-gated sodium channel activity involved in cardiac muscle cell action potential
Brivaracetam//Sodium channel subunit beta-4//Voltage-gated sodium channel activity involved in cardiac muscle cell action potential
Abiraterone//Steroid 17-alpha-hydroxylase/17,20 lyase//Steroid 17-alpha-monooxygenase activity
Cariprazine//D(3) dopamine receptor//G-protein coupled amine receptor activity
Cariprazine//D(2) dopamine receptor//Potassium channel regulator activity
Cariprazine//5-hydroxytryptamine receptor 1A//Serotonin receptor activity
Cariprazine//5-hydroxytryptamine receptor 2B//Serotonin receptor activity
Cariprazine//5-hydroxytryptamine receptor 2A//Virus receptor activity
Cariprazine//Histamine H1 receptor//Histamine receptor activity
Mianserin//Alpha-2A adrenergic receptor//Thioesterase binding
Mianserin//5-hydroxytryptamine receptor 2A//Virus receptor activity
Mianserin//5-hydroxytryptamine receptor 2C//Serotonin receptor activity
Mianserin//Histamine H1 receptor//Histamine receptor activity
Mianserin//Sodium-dependent noradrenaline transporter//Norepinephrine:sodium symporter activity
Mianserin//Sodium-dependent serotonin transporter//Serotonin:sodium symporter activity
Mianserin//Histamine H4 receptor//Histamine receptor activity
Mianserin//5-hydroxytryptamine receptor 1A//Serotonin receptor activity
Mianserin//Alpha-2C adrenergic receptor//Protein homodimerization activity
Mianserin//5-hydroxytryptamine receptor 2B//Serotonin receptor activity
Mianserin//5-hydroxytryptamine receptor 1F//Serotonin receptor activity
Mianserin//Alpha-2B adrenergic receptor//Epinephrine binding
Mianserin//D(3) dopamine receptor//G-protein coupled amine receptor activity
Mianserin//Kappa-type opioid receptor//Opioid receptor activity
Mianserin//Sodium-dependent dopamine transporter//Monoamine transmembrane transporter activity
Mianserin//5-hydroxytryptamine receptor 7//Serotonin receptor activity
Mianserin//D(2) dopamine receptor//Potassium channel regulator activity
Mianserin//5-hydroxytryptamine receptor 6//Serotonin receptor activity
Mianserin//Alpha-1A adrenergic receptor//Protein heterodimerization activity
Mianserin//Alpha-1B adrenergic receptor//Protein heterodimerization activity
Mianserin//Alpha-1D adrenergic receptor//Alpha1-adrenergic receptor activity
Mianserin//D(1A) dopamine receptor//G-protein coupled amine receptor activity
Mianserin//D(1B) dopamine receptor//G-protein coupled amine receptor activity
Alogliptin//Dipeptidyl peptidase 4//Virus receptor activity
Eltrombopag//Thrombopoietin receptor//Transmembrane signaling receptor activity
Asenapine//5-hydroxytryptamine receptor 1A//Serotonin receptor activity
Asenapine//5-hydroxytryptamine receptor 1B//Serotonin receptor activity
Asenapine//5-hydroxytryptamine receptor 2A//Virus receptor activity
Asenapine//5-hydroxytryptamine receptor 2B//Serotonin receptor activity
Asenapine//5-hydroxytryptamine receptor 2C//Serotonin receptor activity
Asenapine//5-hydroxytryptamine receptor 5A//Serotonin receptor activity
Asenapine//5-hydroxytryptamine receptor 6//Serotonin receptor activity
Asenapine//5-hydroxytryptamine receptor 7//Serotonin receptor activity
Asenapine//D(2) dopamine receptor//Potassium channel regulator activity
Asenapine//D(3) dopamine receptor//G-protein coupled amine receptor activity
Asenapine//D(4) dopamine receptor//Sh3 domain binding
Asenapine//D(1A) dopamine receptor//G-protein coupled amine receptor activity
Asenapine//Alpha-1A adrenergic receptor//Protein heterodimerization activity
Asenapine//Alpha-2A adrenergic receptor//Thioesterase binding
Asenapine//Alpha-2B adrenergic receptor//Epinephrine binding
Asenapine//Alpha-2C adrenergic receptor//Protein homodimerization activity
Asenapine//Histamine H1 receptor//Histamine receptor activity
Asenapine//Histamine H2 receptor//Histamine receptor activity
Asenapine//Beta-1 adrenergic receptor//Receptor signaling protein activity
Asenapine//Beta-2 adrenergic receptor//Protein homodimerization activity
Nalmefene//Mu-type opioid receptor//Voltage-gated calcium channel activity
Nalmefene//Kappa-type opioid receptor//Opioid receptor activity
Nalmefene//Delta-type opioid receptor//Opioid receptor activity
Avanafil//cGMP-specific 3',5'-cyclic phosphodiesterase//Metal ion binding
Droxidopa//Alpha-1A adrenergic receptor//Protein heterodimerization activity
Droxidopa//Alpha-1B adrenergic receptor//Protein heterodimerization activity
Droxidopa//Alpha-1D adrenergic receptor//Alpha1-adrenergic receptor activity
Droxidopa//Alpha-2A adrenergic receptor//Thioesterase binding
Droxidopa//Alpha-2B adrenergic receptor//Epinephrine binding
Droxidopa//Alpha-2C adrenergic receptor//Protein homodimerization activity
Droxidopa//Beta-1 adrenergic receptor//Receptor signaling protein activity
Droxidopa//Beta-2 adrenergic receptor//Protein homodimerization activity
Droxidopa//Beta-3 adrenergic receptor//Protein homodimerization activity
Amrubicin//DNA topoisomerase 2-alpha//Ubiquitin binding
Levocetirizine//Histamine H1 receptor//Histamine receptor activity
Dapagliflozin//Sodium/glucose cotransporter 2//Low-affinity glucose:sodium symporter activity
Ambrisentan//Endothelin-1 receptor//Phosphatidylinositol phospholipase c activity
Ambrisentan//Endothelin B receptor//Peptide hormone binding
Doxercalciferol//Vitamin D3 receptor//Zinc ion binding
Armodafinil//Sodium-dependent dopamine transporter//Monoamine transmembrane transporter activity
Agomelatine//5-hydroxytryptamine receptor 2C//Serotonin receptor activity
Midostaurin//Receptor-type tyrosine-protein kinase FLT3//Vascular endothelial growth factor-activated receptor activity
Midostaurin//Platelet-derived growth factor receptor beta//Vascular endothelial growth factor binding
Midostaurin//Vascular endothelial growth factor receptor 2//Vascular endothelial growth factor-activated receptor activity
Midostaurin//Mast/stem cell growth factor receptor Kit//Transmembrane receptor protein tyrosine kinase activity
Midostaurin//Platelet-derived growth factor receptor alpha//Vascular endothelial growth factor-activated receptor activity
Midostaurin//Protein kinase C alpha type//Zinc ion binding
Apixaban//Coagulation factor X//Serine-type endopeptidase activity
Bosutinib//Breakpoint cluster region protein//Rho guanyl-nucleotide exchange factor activity
Bosutinib//Tyrosine-protein kinase ABL1//Syntaxin binding
Bosutinib//Tyrosine-protein kinase Lyn//Receptor signaling protein tyrosine kinase activity
Bosutinib//Tyrosine-protein kinase HCK//Receptor binding
Bosutinib//Proto-oncogene tyrosine-protein kinase Src//Sh3/sh2 adaptor activity
Bosutinib//Cyclin-dependent kinase 2//Metal ion binding
Bosutinib//Dual specificity mitogen-activated protein kinase kinase 2//Scaffold protein binding
Bosutinib//Mitogen-activated protein kinase kinase kinase 2//Protein serine/threonine kinase activity
Bosutinib//Calcium/calmodulin-dependent protein kinase type II subunit gamma//Protein homodimerization activity
Axitinib//Vascular endothelial growth factor receptor 3//Vascular endothelial growth factor-activated receptor activity
Axitinib//Vascular endothelial growth factor receptor 1//Vegf-b-activated receptor activity
Axitinib//Vascular endothelial growth factor receptor 2//Vascular endothelial growth factor-activated receptor activity
Dalfampridine//Potassium voltage-gated channel subfamily A member 1//Voltage-gated potassium channel activity
Dalfampridine//Potassium voltage-gated channel subfamily A member 2//Voltage-gated potassium channel activity
Dalfampridine//Potassium voltage-gated channel subfamily A member 3//Voltage-gated ion channel activity
Dalfampridine//Potassium voltage-gated channel subfamily A member 4//Voltage-gated potassium channel activity
Dalfampridine//Potassium voltage-gated channel subfamily A member 5//Voltage-gated potassium channel activity involved in sa node cell action potential repolarization
Dalfampridine//Potassium voltage-gated channel subfamily A member 6//Voltage-gated potassium channel activity
Dalfampridine//Potassium voltage-gated channel subfamily A member 10//Intracellular cyclic nucleotide activated cation channel activity
Dalfampridine//Potassium voltage-gated channel subfamily B member 1//Ubiquitin-like protein binding
Dalfampridine//Potassium voltage-gated channel subfamily B member 2//Protein heterodimerization activity
Dalfampridine//Potassium voltage-gated channel subfamily C member 1//Voltage-gated potassium channel activity
Dalfampridine//Potassium voltage-gated channel subfamily C member 2//Voltage-gated potassium channel activity
Dalfampridine//Potassium voltage-gated channel subfamily C member 3//Voltage-gated potassium channel activity
Dalfampridine//Potassium voltage-gated channel subfamily D member 1//Metal ion binding
Dalfampridine//Potassium voltage-gated channel subfamily D member 2//Voltage-gated potassium channel activity
Dalfampridine//Potassium voltage-gated channel subfamily D member 3//Metal ion binding
Ethanolamineoleate//Coagulation factor XII//Serine-type endopeptidase activity
Mepyramine//Histamine H1 receptor//Histamine receptor activity
Dabigatranetexilate//Prothrombin//Thrombospondin receptor activity
Desvenlafaxine//Sodium-dependent noradrenaline transporter//Norepinephrine:sodium symporter activity
Desvenlafaxine//Sodium-dependent serotonin transporter//Serotonin:sodium symporter activity
Desvenlafaxine//Sodium-dependent dopamine transporter//Monoamine transmembrane transporter activity
Dexmethylphenidate//Sodium-dependent dopamine transporter//Monoamine transmembrane transporter activity
Dexmethylphenidate//Sodium-dependent noradrenaline transporter//Norepinephrine:sodium symporter activity
Dexmethylphenidate//Sodium-dependent serotonin transporter//Serotonin:sodium symporter activity
Fesoterodine//Muscarinic acetylcholine receptor M3//Receptor activity
Fesoterodine//Muscarinic acetylcholine receptor M4//Guanyl-nucleotide exchange factor activity
Fesoterodine//Muscarinic acetylcholine receptor M1//Phosphatidylinositol phospholipase c activity
Fesoterodine//Muscarinic acetylcholine receptor M2//G-protein coupled acetylcholine receptor activity
Fesoterodine//Muscarinic acetylcholine receptor M5//Phosphatidylinositol phospholipase c activity
Methyltestosterone//Androgen receptor//Zinc ion binding
Methyltestosterone//Estrogen receptor//Zinc ion binding
Fospropofol//Gamma-aminobutyric acid receptor subunit beta-2//Inhibitory extracellular ligand-gated ion channel activity
Fospropofol//Gamma-aminobutyric acid receptor subunit beta-3//Gaba-gated chloride ion channel activity
Lornoxicam//Prostaglandin G/H synthase 1//Prostaglandin-endoperoxide synthase activity
Lornoxicam//Prostaglandin G/H synthase 2//Prostaglandin-endoperoxide synthase activity
Gestodene//Progesterone receptor//Zinc ion binding
Aceclofenac//Prostaglandin G/H synthase 2//Prostaglandin-endoperoxide synthase activity
Aceclofenac//Prostaglandin G/H synthase 1//Prostaglandin-endoperoxide synthase activity
Ketobemidone//Mu-type opioid receptor//Voltage-gated calcium channel activity
Ketobemidone//Kappa-type opioid receptor//Opioid receptor activity
Ketobemidone//Delta-type opioid receptor//Opioid receptor activity
Ketobemidone//Glutamate receptor ionotropic, NMDA 1//Voltage-gated cation channel activity
Ketobemidone//Glutamate receptor ionotropic, NMDA 2A//Zinc ion binding
Ketobemidone//Glutamate receptor ionotropic, NMDA 2B//Zinc ion binding
Ketobemidone//Glutamate receptor ionotropic, NMDA 2C//Nmda glutamate receptor activity
Ketobemidone//Glutamate receptor ionotropic, NMDA 2D//Nmda glutamate receptor activity
Ketobemidone//Glutamate receptor ionotropic, NMDA 3A//Protein phosphatase 2a binding
Ketobemidone//Glutamate receptor ionotropic, NMDA 3B//Nmda glutamate receptor activity
Cabazitaxel//Tubulin alpha-4A chain//Structural constituent of cytoskeleton
Cabazitaxel//Tubulin beta-1 chain//Structural constituent of cytoskeleton
Capsaicin//Transient receptor potential cation channel subfamily V member 1//Transmembrane signaling receptor activity
Chenodeoxycholicacid//Bile acid receptor//Zinc ion binding
Chenodeoxycholicacid//Nuclear receptor subfamily 1 group I member 2//Zinc ion binding
Chenodeoxycholicacid//Aldo-keto reductase family 1 member C2//Trans-1,2-dihydrobenzene-1,2-diol dehydrogenase activity
Hydroxyprogesteronecaproate//Progesterone receptor//Zinc ion binding
Methylnaltrexone//Mu-type opioid receptor//Voltage-gated calcium channel activity
Methylnaltrexone//Kappa-type opioid receptor//Opioid receptor activity
Nandrolonedecanoate//Androgen receptor//Zinc ion binding
Lurasidone//D(2) dopamine receptor//Potassium channel regulator activity
Lurasidone//5-hydroxytryptamine receptor 2A//Virus receptor activity
Lurasidone//5-hydroxytryptamine receptor 7//Serotonin receptor activity
Lurasidone//5-hydroxytryptamine receptor 1A//Serotonin receptor activity
Lurasidone//Alpha-2C adrenergic receptor//Protein homodimerization activity
Lurasidone//Alpha-2A adrenergic receptor//Thioesterase binding
Ivacaftor//Cystic fibrosis transmembrane conductance regulator//Pdz domain binding
Lomitapide//Microsomal triglyceride transfer protein large subunit//Protein heterodimerization activity
Crizotinib//ALK tyrosine kinase receptor//Transmembrane receptor protein tyrosine kinase activity
Crizotinib//Hepatocyte growth factor receptor//Protein tyrosine kinase activity
Fingolimod//Sphingosine 1-phosphate receptor 5//Sphingosine-1-phosphate receptor activity
Fingolimod//Sphingosine 1-phosphate receptor 1//Sphingosine-1-phosphate receptor activity
Cabozantinib//Hepatocyte growth factor receptor//Protein tyrosine kinase activity
Cabozantinib//Vascular endothelial growth factor receptor 2//Vascular endothelial growth factor-activated receptor activity
Cabozantinib//Proto-oncogene tyrosine-protein kinase receptor Ret//Transmembrane receptor protein tyrosine kinase activity
Linagliptin//Dipeptidyl peptidase 4//Virus receptor activity
Mirabegron//Beta-3 adrenergic receptor//Protein homodimerization activity
Aclidinium//Muscarinic acetylcholine receptor M1//Phosphatidylinositol phospholipase c activity
Aclidinium//Muscarinic acetylcholine receptor M2//G-protein coupled acetylcholine receptor activity
Aclidinium//Muscarinic acetylcholine receptor M3//Receptor activity
Aclidinium//Muscarinic acetylcholine receptor M4//Guanyl-nucleotide exchange factor activity
Aclidinium//Muscarinic acetylcholine receptor M5//Phosphatidylinositol phospholipase c activity
Enzalutamide//Androgen receptor//Zinc ion binding
Fluticasonefuroate//Glucocorticoid receptor//Zinc ion binding
Fluticasonefuroate//Progesterone receptor//Zinc ion binding
Fluticasonefuroate//Mineralocorticoid receptor//Zinc ion binding
Canagliflozin//Sodium/glucose cotransporter 2//Low-affinity glucose:sodium symporter activity
Dabrafenib//Serine/threonine-protein kinase B-raf//Protein serine/threonine kinase activity
Dabrafenib//RAF proto-oncogene serine/threonine-protein kinase//Protein serine/threonine kinase activity
Dabrafenib//Serine/threonine-protein kinase SIK1//Protein serine/threonine kinase activity
Dabrafenib//Serine/threonine-protein kinase Nek11//Protein serine/threonine kinase activity
Dabrafenib//LIM domain kinase 1//Zinc ion binding
Levomilnacipran//Sodium-dependent serotonin transporter//Serotonin:sodium symporter activity
Levomilnacipran//Sodium-dependent noradrenaline transporter//Norepinephrine:sodium symporter activity
Macitentan//Endothelin-1 receptor//Phosphatidylinositol phospholipase c activity
Macitentan//Endothelin B receptor//Peptide hormone binding
Aliskiren//Renin//Receptor binding
Miltefosine//Multidrug resistance protein 1//Xenobiotic-transporting atpase activity
Netupitant//Substance-P receptor//Tachykinin receptor activity
Naloxegol//Mu-type opioid receptor//Voltage-gated calcium channel activity
Ibrutinib//Tyrosine-protein kinase BTK//Protein tyrosine kinase activity
Cannabidiol//Cannabinoid receptor 1//Drug binding
Cannabidiol//Cannabinoid receptor 2//Cannabinoid receptor activity
Cannabidiol//Glycine receptor subunit alpha-1//Transmitter-gated ion channel activity
Cannabidiol//Glycine receptor subunit alpha-1//Transmitter-gated ion channel activity
Cannabidiol//Glycine receptor subunit beta//Glycine binding
Cannabidiol//Glycine receptor subunit alpha-3//Transmitter-gated ion channel activity
Cannabidiol//N-arachidonyl glycine receptor//G-protein coupled receptor activity
Cannabidiol//G-protein coupled receptor 55//G-protein coupled receptor activity
Cannabidiol//5-hydroxytryptamine receptor 1A//Serotonin receptor activity
Cannabidiol//5-hydroxytryptamine receptor 2A//Virus receptor activity
Cannabidiol//Neuronal acetylcholine receptor subunit alpha-7//Toxic substance binding
Cannabidiol//Delta-type opioid receptor//Opioid receptor activity
Cannabidiol//Mu-type opioid receptor//Voltage-gated calcium channel activity
Cannabidiol//Peroxisome proliferator-activated receptor gamma//Zinc ion binding
Cannabidiol//Transient receptor potential cation channel subfamily V member 1//Transmembrane signaling receptor activity
Cannabidiol//Voltage-dependent T-type calcium channel subunit alpha-1G//Scaffold protein binding
Cannabidiol//Voltage-dependent T-type calcium channel subunit alpha-1H//Scaffold protein binding
Cannabidiol//Voltage-dependent T-type calcium channel subunit alpha-1I//Voltage-gated calcium channel activity
Cannabidiol//Transient receptor potential cation channel subfamily A member 1//Temperature-gated cation channel activity
Cannabidiol//Transient receptor potential cation channel subfamily M member 8//Calcium channel activity
Cannabidiol//Transient receptor potential cation channel subfamily V member 3//Calcium channel activity
Cannabidiol//Transient receptor potential cation channel subfamily V member 4//Non-selective calcium permeant cation channel involved in osmotic sensitivity and mechanosensitivity. Activation by exposure to hypotonicity within the physiological range exhibits an outward rectification (PubMed:18826956, PubMed:18695040). Also activated by heat, low pH, citrate and phorbol esters (PubMed:18826956, PubMed:18695040). Increase of intracellular Ca(2+) potentiates currents. Channel activity seems to be regulated by a calmodulin-dependent mechanism with a negative feedback mechanism (PubMed:12724311, PubMed:18826956). Promotes cell-cell junction formation in skin keratinocytes and plays an important role in the formation and/or maintenance of functional intercellular barriers (By similarity). Acts as a regulator of intracellular Ca(2+) in synoviocytes (PubMed:19759329). Plays an obligatory role as a molecular component in the nonselective cation channel activation induced by 4-alpha-phorbol 12,13-didecanoate and hypotonic stimulation in synoviocytes and also regulates production of IL-8 (PubMed:19759329). Together with PKD2, forms mechano- and thermosensitive channels in cilium (PubMed:18695040). Negatively regulates expression of PPARGC1A, UCP1, oxidative metabolism and respiration in adipocytes (By similarity). Regulates expression of chemokines and cytokines related to proinflammatory pathway in adipocytes (By similarity). Together with AQP5, controls regulatory volume decrease in salivary epithelial cells (By similarity). Required for normal development and maintenance of bone and cartilage (PubMed:26249260).
Cannabidiol//5-hydroxytryptamine receptor 3A//Voltage-gated potassium channel activity
Cannabidiol//Adenosine receptor A1//Purine nucleoside binding
Cannabidiol//Prostaglandin G/H synthase 1//Prostaglandin-endoperoxide synthase activity
Cannabidiol//Prostaglandin G/H synthase 2//Prostaglandin-endoperoxide synthase activity
Cannabidiol//Acetyl-CoA acetyltransferase, mitochondrial//Metal ion binding
Cannabidiol//Steroid 17-alpha-hydroxylase/17,20 lyase//Steroid 17-alpha-monooxygenase activity
Cannabidiol//3-hydroxy-3-methylglutaryl-coenzyme A reductase//Nadph binding
Cannabidiol//Glutathione reductase, mitochondrial//Nadp binding
Cannabidiol//Glutathione peroxidase 1//Sh3 domain binding
Cannabidiol//Indoleamine 2,3-dioxygenase 1//Tryptophan 2,3-dioxygenase activity
Cannabidiol//Cytochrome P450 1B1//Oxygen binding
Cannabidiol//NAD(P)H dehydrogenase [quinone] 1//Superoxide dismutase activity
Cannabidiol//Catalase//Receptor binding
Cannabidiol//Cytochrome P450 3A5//Oxygen binding
Cannabidiol//Cytochrome P450 2D6//Steroid hydroxylase activity
Cannabidiol//Superoxide dismutase [Cu-Zn]//Zinc ion binding
Cannabidiol//Cytochrome P450 1A2//Oxidoreductase activity, acting on paired donors, with incorporation or reduction of molecular oxygen, reduced flavin or flavoprotein as one donor, and incorporation of one atom of oxygen
Cannabidiol//Cytochrome P450 3A7//Oxygen binding
Ceritinib//ALK tyrosine kinase receptor//Transmembrane receptor protein tyrosine kinase activity
Lenvatinib//Vascular endothelial growth factor receptor 1//Vegf-b-activated receptor activity
Lenvatinib//Vascular endothelial growth factor receptor 2//Vascular endothelial growth factor-activated receptor activity
Lenvatinib//Vascular endothelial growth factor receptor 3//Vascular endothelial growth factor-activated receptor activity
Lenvatinib//Fibroblast growth factor receptor 1//Protein tyrosine kinase activity
Lenvatinib//Fibroblast growth factor receptor 2//Protein tyrosine kinase activity
Lenvatinib//Fibroblast growth factor receptor 3//Protein tyrosine kinase activity
Lenvatinib//Fibroblast growth factor receptor 4//Protein tyrosine kinase activity
Lenvatinib//Platelet-derived growth factor receptor alpha//Vascular endothelial growth factor-activated receptor activity
Lenvatinib//Proto-oncogene tyrosine-protein kinase receptor Ret//Transmembrane receptor protein tyrosine kinase activity
Lenvatinib//Mast/stem cell growth factor receptor Kit//Transmembrane receptor protein tyrosine kinase activity
Eslicarbazepineacetate//P2X purinoceptor 4//Zinc ion binding
Dienogest//Progesterone receptor//Zinc ion binding
Dienogest//Androgen receptor//Zinc ion binding
Brexpiprazole//5-hydroxytryptamine receptor 1A//Serotonin receptor activity
Brexpiprazole//D(2) dopamine receptor//Potassium channel regulator activity
Brexpiprazole//5-hydroxytryptamine receptor 2A//Virus receptor activity
Brexpiprazole//Alpha-2C adrenergic receptor//Protein homodimerization activity
Brexpiprazole//Alpha-1B adrenergic receptor//Protein heterodimerization activity
Etizolam//Gamma-aminobutyric acid receptor subunit alpha-1//Inhibitory extracellular ligand-gated ion channel activity
Etizolam//Gamma-aminobutyric acid receptor subunit alpha-2//Inhibitory extracellular ligand-gated ion channel activity
Etizolam//Gamma-aminobutyric acid receptor subunit alpha-3//Inhibitory extracellular ligand-gated ion channel activity
Etizolam//Gamma-aminobutyric acid receptor subunit alpha-4//Inhibitory extracellular ligand-gated ion channel activity
Etizolam//Gamma-aminobutyric acid receptor subunit alpha-5//Transporter activity
Etizolam//Gamma-aminobutyric acid receptor subunit alpha-6//Inhibitory extracellular ligand-gated ion channel activity
Etizolam//Gamma-aminobutyric acid receptor subunit beta-1//Ligand-gated ion channel activity
Etizolam//Gamma-aminobutyric acid receptor subunit beta-2//Inhibitory extracellular ligand-gated ion channel activity
Etizolam//Gamma-aminobutyric acid receptor subunit beta-3//Gaba-gated chloride ion channel activity
Etizolam//Gamma-aminobutyric acid receptor subunit delta//Gaba-a receptor activity
Etizolam//Gamma-aminobutyric acid receptor subunit epsilon//Inhibitory extracellular ligand-gated ion channel activity
Etizolam//Gamma-aminobutyric acid receptor subunit gamma-1//Inhibitory extracellular ligand-gated ion channel activity
Etizolam//Gamma-aminobutyric acid receptor subunit gamma-2//Inhibitory extracellular ligand-gated ion channel activity
Etizolam//Gamma-aminobutyric acid receptor subunit gamma-3//Inhibitory extracellular ligand-gated ion channel activity
Etizolam//Gamma-aminobutyric acid receptor subunit pi//Gaba-a receptor activity
Etizolam//Gamma-aminobutyric acid receptor subunit theta//Transmembrane signaling receptor activity
Etizolam//Gamma-aminobutyric acid receptor subunit alpha-1//Inhibitory extracellular ligand-gated ion channel activity
Etizolam//Gamma-aminobutyric acid receptor subunit alpha-2//Inhibitory extracellular ligand-gated ion channel activity
Etizolam//Gamma-aminobutyric acid receptor subunit alpha-3//Inhibitory extracellular ligand-gated ion channel activity
Etizolam//Gamma-aminobutyric acid receptor subunit alpha-5//Transporter activity
Etizolam//Gamma-aminobutyric acid receptor subunit gamma-1//Inhibitory extracellular ligand-gated ion channel activity
Etizolam//Gamma-aminobutyric acid receptor subunit gamma-2//Inhibitory extracellular ligand-gated ion channel activity
Etizolam//Gamma-aminobutyric acid receptor subunit gamma-3//Inhibitory extracellular ligand-gated ion channel activity
Dosulepin//5-hydroxytryptamine receptor 1A//Serotonin receptor activity
Dosulepin//5-hydroxytryptamine receptor 2A//Virus receptor activity
Dosulepin//Histamine H1 receptor//Histamine receptor activity
Dosulepin//Muscarinic acetylcholine receptor M1//Phosphatidylinositol phospholipase c activity
Dosulepin//Muscarinic acetylcholine receptor M2//G-protein coupled acetylcholine receptor activity
Dosulepin//Muscarinic acetylcholine receptor M3//Receptor activity
Dosulepin//Muscarinic acetylcholine receptor M4//Guanyl-nucleotide exchange factor activity
Dosulepin//Muscarinic acetylcholine receptor M5//Phosphatidylinositol phospholipase c activity
Dosulepin//Alpha-2A adrenergic receptor//Thioesterase binding
Dosulepin//Alpha-2B adrenergic receptor//Epinephrine binding
Dosulepin//Alpha-2C adrenergic receptor//Protein homodimerization activity
Dosulepin//Alpha-1A adrenergic receptor//Protein heterodimerization activity
Dosulepin//Alpha-1B adrenergic receptor//Protein heterodimerization activity
Dosulepin//Alpha-1D adrenergic receptor//Alpha1-adrenergic receptor activity
Dosulepin//Sodium-dependent noradrenaline transporter//Norepinephrine:sodium symporter activity
Dosulepin//Sodium-dependent serotonin transporter//Serotonin:sodium symporter activity
Lorpiprazole//5-hydroxytryptamine receptor 2A//Virus receptor activity
Lorpiprazole//5-hydroxytryptamine receptor 2C//Serotonin receptor activity
Lorpiprazole//Alpha-1A adrenergic receptor//Protein heterodimerization activity
Lorpiprazole//Alpha-1B adrenergic receptor//Protein heterodimerization activity
Lorpiprazole//Alpha-1D adrenergic receptor//Alpha1-adrenergic receptor activity
Lorpiprazole//Alpha-2A adrenergic receptor//Thioesterase binding
Lorpiprazole//Alpha-2B adrenergic receptor//Epinephrine binding
Lorpiprazole//Alpha-2C adrenergic receptor//Protein homodimerization activity
Lorpiprazole//Histamine H1 receptor//Histamine receptor activity
Lorpiprazole//Sodium-dependent serotonin transporter//Serotonin:sodium symporter activity
Lobeglitazone//Peroxisome proliferator-activated receptor gamma//Zinc ion binding
Loxoprofen//Prostaglandin G/H synthase 2//Prostaglandin-endoperoxide synthase activity
Loxoprofen//Prostaglandin G/H synthase 1//Prostaglandin-endoperoxide synthase activity
Dexketoprofen//Prostaglandin G/H synthase 1//Prostaglandin-endoperoxide synthase activity
Dexketoprofen//Prostaglandin G/H synthase 2//Prostaglandin-endoperoxide synthase activity
Blonanserin//D(2) dopamine receptor//Potassium channel regulator activity
Blonanserin//D(3) dopamine receptor//G-protein coupled amine receptor activity
Blonanserin//5-hydroxytryptamine receptor 2A//Virus receptor activity
Melperone//D(2) dopamine receptor//Potassium channel regulator activity
Aranidipine//Voltage-dependent L-type calcium channel subunit alpha-1C//Voltage-gated calcium channel activity
Aranidipine//Voltage-dependent L-type calcium channel subunit alpha-1D//Voltage-gated calcium channel activity involved sa node cell action potential
Aranidipine//Voltage-dependent L-type calcium channel subunit alpha-1F//Voltage-gated calcium channel activity
Aranidipine//Voltage-dependent L-type calcium channel subunit alpha-1S//Voltage-gated calcium channel activity
Aranidipine//Alpha-1A adrenergic receptor//Protein heterodimerization activity
Aranidipine//Alpha-1B adrenergic receptor//Protein heterodimerization activity
Aranidipine//Alpha-1D adrenergic receptor//Alpha1-adrenergic receptor activity
Aranidipine//Alpha-2A adrenergic receptor//Thioesterase binding
Aranidipine//Alpha-2B adrenergic receptor//Epinephrine binding
Aranidipine//Alpha-2C adrenergic receptor//Protein homodimerization activity
Azelnidipine//Voltage-dependent L-type calcium channel subunit beta-1//Voltage-gated calcium channel activity
Benidipine//Voltage-dependent L-type calcium channel subunit alpha-1C//Voltage-gated calcium channel activity
Benidipine//Voltage-dependent L-type calcium channel subunit alpha-1D//Voltage-gated calcium channel activity involved sa node cell action potential
Benidipine//Voltage-dependent L-type calcium channel subunit alpha-1F//Voltage-gated calcium channel activity
Benidipine//Voltage-dependent L-type calcium channel subunit alpha-1S//Voltage-gated calcium channel activity
Benidipine//Voltage-dependent L-type calcium channel subunit beta-1//Voltage-gated calcium channel activity
Benidipine//Voltage-dependent L-type calcium channel subunit beta-2//Voltage-gated calcium channel activity
Benidipine//Voltage-dependent L-type calcium channel subunit beta-3//Voltage-gated calcium channel activity
Benidipine//Voltage-dependent L-type calcium channel subunit beta-4//Voltage-gated calcium channel activity
Benidipine//Voltage-dependent P/Q-type calcium channel subunit alpha-1A//Voltage-gated calcium channel activity
Benidipine//Voltage-dependent N-type calcium channel subunit alpha-1B//Voltage-gated calcium channel activity
Benidipine//Voltage-dependent T-type calcium channel subunit alpha-1G//Scaffold protein binding
Benidipine//Voltage-dependent T-type calcium channel subunit alpha-1H//Scaffold protein binding
Benidipine//Voltage-dependent T-type calcium channel subunit alpha-1I//Voltage-gated calcium channel activity
Cilnidipine//Voltage-dependent N-type calcium channel subunit alpha-1B//Voltage-gated calcium channel activity
Cilnidipine//Voltage-dependent L-type calcium channel subunit alpha-1C//Voltage-gated calcium channel activity
Cilnidipine//Voltage-dependent L-type calcium channel subunit alpha-1D//Voltage-gated calcium channel activity involved sa node cell action potential
Cilnidipine//Voltage-dependent L-type calcium channel subunit alpha-1F//Voltage-gated calcium channel activity
Cilnidipine//Voltage-dependent L-type calcium channel subunit alpha-1S//Voltage-gated calcium channel activity
Cilnidipine//Voltage-dependent L-type calcium channel subunit beta-1//Voltage-gated calcium channel activity
Cilnidipine//Voltage-dependent L-type calcium channel subunit beta-2//Voltage-gated calcium channel activity
Cilnidipine//Voltage-dependent L-type calcium channel subunit beta-3//Voltage-gated calcium channel activity
Cilnidipine//Voltage-dependent L-type calcium channel subunit beta-4//Voltage-gated calcium channel activity
Cilnidipine//Voltage-dependent P/Q-type calcium channel subunit alpha-1A//Voltage-gated calcium channel activity
Efonidipine//Voltage-dependent T-type calcium channel subunit alpha-1I//Voltage-gated calcium channel activity
Efonidipine//Voltage-dependent L-type calcium channel subunit alpha-1C//Voltage-gated calcium channel activity
Imidafenacin//Muscarinic acetylcholine receptor M1//Phosphatidylinositol phospholipase c activity
Imidafenacin//Muscarinic acetylcholine receptor M2//G-protein coupled acetylcholine receptor activity
Imidafenacin//Muscarinic acetylcholine receptor M3//Receptor activity
Lumacaftor//Cystic fibrosis transmembrane conductance regulator//Pdz domain binding
Molsidomine//Guanylate cyclase soluble subunit alpha-2//Heme binding
Morniflumate//Arachidonate 5-lipoxygenase//Iron ion binding
Morniflumate//Prostaglandin G/H synthase 2//Prostaglandin-endoperoxide synthase activity
Mersalyl//Alkaline phosphatase, tissue-nonspecific isozyme//Pyrophosphatase activity
Mersalyl//Monocarboxylate transporter 1//Symporter activity
Glycerin//Peroxisome proliferator-activated receptor delta//Zinc ion binding
Glycerin//Group IIE secretory phospholipase A2//Phospholipase a2 activity
Glycerin//Alcohol dehydrogenase 1B//Zinc ion binding
Glycerin//Alpha-N-acetylgalactosaminidase//Protein homodimerization activity
Glycerin//ADP-ribosylation factor 1//Receptor signaling protein activity
Glycerin//Ribonucleoside-diphosphate reductase 1 subunit beta//Ribonucleoside-diphosphate reductase activity, thioredoxin disulfide as acceptor
Glycerin//Adenine DNA glycosylase//Metal ion binding
Glycerin//Maleylacetoacetate isomerase//Protein homodimerization activity
Dexchlorpheniraminemaleate//Histamine H1 receptor//Histamine receptor activity
Butamben//Voltage-dependent calcium channel gamma-1 subunit//Voltage-gated calcium channel activity
Butamben//Voltage-dependent calcium channel gamma-2 subunit//Voltage-gated calcium channel activity
Butamben//Voltage-dependent calcium channel gamma-3 subunit//Regulates the trafficking to the somatodendritic compartment and gating properties of AMPA-selective glutamate receptors (AMPARs). Promotes their targeting to the cell membrane and synapses and modulates their gating properties by slowing their rates of activation, deactivation and desensitization. Does not show subunit-specific AMPA receptor regulation and regulates all AMPAR subunits. Thought to stabilize the calcium channel in an inactivated (closed) state.
Butamben//Voltage-dependent calcium channel gamma-4 subunit//Regulates the trafficking and gating properties of AMPA-selective glutamate receptors (AMPARs). Promotes their targeting to the cell membrane and synapses and modulates their gating properties by slowing their rates of activation, deactivation and desensitization and by mediating their resensitization. Does not show subunit-specific AMPA receptor regulation and regulates all AMPAR subunits. Thought to stabilize the calcium channel in an inactivated (closed) state.
Butamben//Voltage-dependent calcium channel gamma-5 subunit//Regulates the gating properties of AMPA-selective glutamate receptors (AMPARs). Modulates their gating properties by accelerating their rates of activation, deactivation and desensitization. Displays subunit-specific AMPA receptor regulation. Shows specificity for GRIA1, GRIA4 and the long isoform of GRIA2. Thought to stabilize the calcium channel in an inactivated (closed) state (By similarity).
Butamben//Voltage-dependent calcium channel gamma-6 subunit//Thought to stabilize the calcium channel in an inactivated (closed) state.
Butamben//Voltage-dependent calcium channel gamma-7 subunit//Regulates the trafficking and gating properties of AMPA-selective glutamate receptors (AMPARs). Promotes their targeting to the cell membrane and synapses and modulates their gating properties by slowing their rates of activation, deactivation and desensitization and by mediating their resensitization. Displays subunit-specific AMPA receptor regulation. Shows specificity only for GRIA1 and GRIA2. Thought to stabilize the calcium channel in an inactivated (closed) state.
Butamben//Voltage-dependent calcium channel gamma-8 subunit//Regulates the trafficking and gating properties of AMPA-selective glutamate receptors (AMPARs). Promotes their targeting to the cell membrane and synapses and modulates their gating properties by slowing their rates of activation, deactivation and desensitization and by mediating their resensitization. Does not show subunit-specific AMPA receptor regulation and regulates all AMPAR subunits. Thought to stabilize the calcium channel in an inactivated (closed) state.
Butamben//Voltage-dependent calcium channel subunit alpha-2/delta-1//Voltage-gated calcium channel activity
Butamben//Voltage-dependent calcium channel subunit alpha-2/delta-2//Voltage-gated calcium channel activity
Butamben//Voltage-dependent calcium channel subunit alpha-2/delta-3//Voltage-gated ion channel activity
Butamben//Voltage-dependent calcium channel subunit alpha-2/delta-4//The alpha-2/delta subunit of voltage-dependent calcium channels regulates calcium current density and activation/inactivation kinetics of the calcium channel.
Butamben//Voltage-dependent L-type calcium channel subunit alpha-1C//Voltage-gated calcium channel activity
Butamben//Voltage-dependent L-type calcium channel subunit alpha-1D//Voltage-gated calcium channel activity involved sa node cell action potential
Butamben//Voltage-dependent L-type calcium channel subunit alpha-1F//Voltage-gated calcium channel activity
Butamben//Voltage-dependent L-type calcium channel subunit alpha-1S//Voltage-gated calcium channel activity
Butamben//Voltage-dependent L-type calcium channel subunit beta-1//Voltage-gated calcium channel activity
Butamben//Voltage-dependent L-type calcium channel subunit beta-2//Voltage-gated calcium channel activity
Butamben//Voltage-dependent L-type calcium channel subunit beta-3//Voltage-gated calcium channel activity
Butamben//Voltage-dependent L-type calcium channel subunit beta-4//Voltage-gated calcium channel activity
Butamben//Voltage-dependent N-type calcium channel subunit alpha-1B//Voltage-gated calcium channel activity
Butamben//Voltage-dependent P/Q-type calcium channel subunit alpha-1A//Voltage-gated calcium channel activity
Butamben//Voltage-dependent R-type calcium channel subunit alpha-1E//Voltage-sensitive calcium channels (VSCC) mediate the entry of calcium ions into excitable cells and are also involved in a variety of calcium-dependent processes, including muscle contraction, hormone or neurotransmitter release, gene expression, cell motility, cell division and cell death. The isoform alpha-1E gives rise to R-type calcium currents. R-type calcium channels belong to the 'high-voltage activated' (HVA) group and are blocked by nickel, and partially by omega-agatoxin-IIIA (omega-Aga-IIIA). They are however insensitive to dihydropyridines (DHP), omega-conotoxin-GVIA (omega-CTx-GVIA), and omega-agatoxin-IVA (omega-Aga-IVA). Calcium channels containing alpha-1E subunit could be involved in the modulation of firing patterns of neurons which is important for information processing.
Butamben//Voltage-dependent T-type calcium channel subunit alpha-1G//Scaffold protein binding
Butamben//Voltage-dependent T-type calcium channel subunit alpha-1H//Scaffold protein binding
Butamben//Voltage-dependent T-type calcium channel subunit alpha-1I//Voltage-gated calcium channel activity
Butamben//ATP-sensitive inward rectifier potassium channel 1//Phosphatidylinositol-4,5-bisphosphate binding
Butamben//ATP-sensitive inward rectifier potassium channel 11//Voltage-gated potassium channel activity
Butamben//ATP-sensitive inward rectifier potassium channel 12//Inward rectifier potassium channel activity
Butamben//ATP-sensitive inward rectifier potassium channel 14//Inward rectifier potassium channels are characterized by a greater tendency to allow potassium to flow into the cell rather than out of it. Their voltage dependence is regulated by the concentration of extracellular potassium; as external potassium is raised, the voltage range of the channel opening shifts to more positive voltages. The inward rectification is mainly due to the blockage of outward current by internal magnesium. KCNJ14 gives rise to low-conductance channels with a low affinity to the channel blockers Barium and Cesium (By similarity).
Butamben//ATP-sensitive inward rectifier potassium channel 8//Inward rectifier potassium channel activity
Butamben//Transient receptor potential cation channel subfamily A member 1//Temperature-gated cation channel activity
Butamben//Transient receptor potential cation channel subfamily V member 4//Non-selective calcium permeant cation channel involved in osmotic sensitivity and mechanosensitivity. Activation by exposure to hypotonicity within the physiological range exhibits an outward rectification (PubMed:18826956, PubMed:18695040). Also activated by heat, low pH, citrate and phorbol esters (PubMed:18826956, PubMed:18695040). Increase of intracellular Ca(2+) potentiates currents. Channel activity seems to be regulated by a calmodulin-dependent mechanism with a negative feedback mechanism (PubMed:12724311, PubMed:18826956). Promotes cell-cell junction formation in skin keratinocytes and plays an important role in the formation and/or maintenance of functional intercellular barriers (By similarity). Acts as a regulator of intracellular Ca(2+) in synoviocytes (PubMed:19759329). Plays an obligatory role as a molecular component in the nonselective cation channel activation induced by 4-alpha-phorbol 12,13-didecanoate and hypotonic stimulation in synoviocytes and also regulates production of IL-8 (PubMed:19759329). Together with PKD2, forms mechano- and thermosensitive channels in cilium (PubMed:18695040). Negatively regulates expression of PPARGC1A, UCP1, oxidative metabolism and respiration in adipocytes (By similarity). Regulates expression of chemokines and cytokines related to proinflammatory pathway in adipocytes (By similarity). Together with AQP5, controls regulatory volume decrease in salivary epithelial cells (By similarity). Required for normal development and maintenance of bone and cartilage (PubMed:26249260).
Homatropine//Muscarinic acetylcholine receptor M1//Phosphatidylinositol phospholipase c activity
Homatropine//Muscarinic acetylcholine receptor M2//G-protein coupled acetylcholine receptor activity
Homatropine//Muscarinic acetylcholine receptor M3//Receptor activity
Homatropine//Muscarinic acetylcholine receptor M4//Guanyl-nucleotide exchange factor activity
Homatropine//Muscarinic acetylcholine receptor M5//Phosphatidylinositol phospholipase c activity
Lesinurad//Solute carrier family 22 member 11//Sodium-independent organic anion transmembrane transporter activity
Isavuconazole//Lanosterol 14-alpha demethylase//Sterol 14-demethylase activity
Isavuconazole//Potassium voltage-gated channel subfamily H member 2//Voltage-gated potassium channel activity involved in ventricular cardiac muscle cell action potential repolarization
Isavuconazole//Voltage-dependent L-type calcium channel subunit alpha-1C//Voltage-gated calcium channel activity
Isavuconazole//G protein-activated inward rectifier potassium channel 2//Inward rectifier potassium channel activity
Isavuconazole//G protein-activated inward rectifier potassium channel 3//G-protein activated inward rectifier potassium channel activity
Isavuconazole//ATP-sensitive inward rectifier potassium channel 11//Voltage-gated potassium channel activity
Isavuconazole//Potassium voltage-gated channel subfamily A member 5//Voltage-gated potassium channel activity involved in sa node cell action potential repolarization
Isavuconazole//Potassium voltage-gated channel subfamily D member 3//Metal ion binding
Isavuconazole//Potassium voltage-gated channel subfamily KQT member 1//Voltage-gated potassium channel activity involved in ventricular cardiac muscle cell action potential repolarization
Isavuconazole//Sodium channel protein type 5 subunit alpha//Voltage-gated sodium channel activity involved in sa node cell action potential
Artenimol//Actin, cytoplasmic 2//Ubiquitin protein ligase binding
Artenimol//Annexin A2//S100 protein binding
Artenimol//ATP synthase subunit alpha, mitochondrial//Transmembrane transporter activity
Artenimol//Calpastatin//Poly(a) rna binding
Artenimol//T-complex protein 1 subunit gamma//Unfolded protein binding
Artenimol//Chloride intracellular channel protein 1//Voltage-gated ion channel activity
Artenimol//Elongation factor 1-alpha 1//Trna binding
Artenimol//Glucose-6-phosphate 1-dehydrogenase//Nadp binding
Artenimol//Glyceraldehyde-3-phosphate dehydrogenase, testis-specific//Nadp binding
Artenimol//Glucose-6-phosphate isomerase//Ubiquitin protein ligase binding
Artenimol//Heat shock protein beta-1//Ubiquitin binding
Artenimol//L-lactate dehydrogenase A chain//Nad binding
Artenimol//L-lactate dehydrogenase B chain//Nad binding
Artenimol//Galectin-1//Signal transducer activity
Artenimol//Microtubule-associated protein 4//Structural molecule activity
Artenimol//Malate dehydrogenase, cytoplasmic//Nad binding
Artenimol//Puromycin-sensitive aminopeptidase//Zinc ion binding
Artenimol//60S ribosomal protein L10//Component of the large ribosomal subunit.
Artenimol//60S ribosomal protein L14//Component of the large ribosomal subunit.
Artenimol//60S ribosomal protein L18//Component of the large ribosomal subunit.
Artenimol//60S ribosomal protein L23a//Structural constituent of ribosome
Artenimol//60S ribosomal protein L35//Component of the large ribosomal subunit.
Artenimol//Signal recognition particle 14 kDa protein//Rna binding
Artenimol//Triosephosphate isomerase//Ubiquitin protein ligase binding
Artenimol//Tubulin alpha-1A chain//Tubulin is the major constituent of microtubules. It binds two moles of GTP, one at an exchangeable site on the beta chain and one at a non-exchangeable site on the alpha chain.
Artenimol//Heat shock cognate 71 kDa protein//Unfolded protein binding
Artenimol//Tubulin beta-6 chain//Structural constituent of cytoskeleton
Artenimol//Tubulin beta-4A chain//Structural constituent of cytoskeleton
Artenimol//Tubulin beta chain//Ubiquitin protein ligase binding
Artenimol//Cytochrome c//Metal ion binding
Artenimol//Protein disulfide-isomerase//Protein heterodimerization activity
Artenimol//Serine hydroxymethyltransferase, mitochondrial//Pyridoxal phosphate binding
Artenimol//Protein disulfide-isomerase//Protein heterodimerization activity
Artenimol//Tubulin alpha chain//Tubulin is the major constituent of microtubules. It binds two moles of GTP, one at an exchangeable site on the beta chain and one at a non-exchangeable site on the alpha chain.
Artenimol//S-adenosylmethionine synthase//Methionine adenosyltransferase activity
Artenimol//60S ribosomal protein L3//Structural constituent of ribosome
Artenimol//Tubulin beta chain//Ubiquitin protein ligase binding
Artenimol//Purine nucleotide phosphorylase, putative//Uridine phosphorylase activity
Artenimol//Adenosylhomocysteinase//Nad binding
Artenimol//Adenosine deaminase//Zinc ion binding
Artenimol//Methionine--tRNA ligase//Zinc ion binding
Artenimol//60S ribosomal protein L23//Structural constituent of ribosome
Artenimol//GTP-binding nuclear protein Ran//Transcription coactivator activity
Artenimol//Serum albumin//Toxic substance binding
Naldemedine//Mu-type opioid receptor//Voltage-gated calcium channel activity
Naldemedine//Delta-type opioid receptor//Opioid receptor activity
Naldemedine//Kappa-type opioid receptor//Opioid receptor activity
Icotinib//Epidermal growth factor receptor//Ubiquitin protein ligase binding
Baricitinib//Tyrosine-protein kinase JAK1//Ubiquitin protein ligase binding
Baricitinib//Tyrosine-protein kinase JAK2//Sh2 domain binding
Baricitinib//Protein-tyrosine kinase 2-beta//Signal transducer activity
Baricitinib//Tyrosine-protein kinase JAK3//Protein tyrosine kinase activity
Ertugliflozin//Sodium/glucose cotransporter 2//Low-affinity glucose:sodium symporter activity
Neratinib//Epidermal growth factor receptor//Ubiquitin protein ligase binding
Apalutamide//Androgen receptor//Zinc ion binding
Apalutamide//Gamma-aminobutyric acid receptor subunit alpha-1//Inhibitory extracellular ligand-gated ion channel activity
Apalutamide//Gamma-aminobutyric acid receptor subunit alpha-2//Inhibitory extracellular ligand-gated ion channel activity
Apalutamide//Gamma-aminobutyric acid receptor subunit alpha-3//Inhibitory extracellular ligand-gated ion channel activity
Apalutamide//Gamma-aminobutyric acid receptor subunit alpha-4//Inhibitory extracellular ligand-gated ion channel activity
Apalutamide//Gamma-aminobutyric acid receptor subunit alpha-5//Transporter activity
Apalutamide//Gamma-aminobutyric acid receptor subunit alpha-6//Inhibitory extracellular ligand-gated ion channel activity
Apalutamide//Gamma-aminobutyric acid receptor subunit beta-1//Ligand-gated ion channel activity
Apalutamide//Gamma-aminobutyric acid receptor subunit beta-2//Inhibitory extracellular ligand-gated ion channel activity
Apalutamide//Gamma-aminobutyric acid receptor subunit beta-3//Gaba-gated chloride ion channel activity
Apalutamide//Gamma-aminobutyric acid receptor subunit delta//Gaba-a receptor activity
Apalutamide//Gamma-aminobutyric acid receptor subunit epsilon//Inhibitory extracellular ligand-gated ion channel activity
Apalutamide//Gamma-aminobutyric acid receptor subunit gamma-1//Inhibitory extracellular ligand-gated ion channel activity
Apalutamide//Gamma-aminobutyric acid receptor subunit gamma-2//Inhibitory extracellular ligand-gated ion channel activity
Apalutamide//Gamma-aminobutyric acid receptor subunit gamma-3//Inhibitory extracellular ligand-gated ion channel activity
Apalutamide//Gamma-aminobutyric acid receptor subunit pi//Gaba-a receptor activity
Apalutamide//Gamma-aminobutyric acid receptor subunit theta//Transmembrane signaling receptor activity
Abemaciclib//Cyclin-dependent kinase 4//Cyclin-dependent protein serine/threonine kinase regulator activity
Fostamatinib//Tyrosine-protein kinase SYK//Receptor signaling protein tyrosine kinase activity
Fostamatinib//Adenosine receptor A3//G-protein coupled adenosine receptor activity
Fostamatinib//Fatty-acid amide hydrolase 1//Fatty acid amide hydrolase activity
Fostamatinib//Equilibrative nucleoside transporter 1//Nucleoside transmembrane transporter activity
Fostamatinib//UDP-glucuronosyltransferase 1-1//Steroid binding
Fostamatinib//cGMP-specific 3',5'-cyclic phosphodiesterase//Metal ion binding
Fostamatinib//Arachidonate 5-lipoxygenase//Iron ion binding
Fostamatinib//Tyrosine-protein kinase ABL1//Syntaxin binding
Fostamatinib//Non-receptor tyrosine-protein kinase TYK2//Protein tyrosine kinase activity
Fostamatinib//Tyrosine-protein kinase JAK1//Ubiquitin protein ligase binding
Fostamatinib//Hepatocyte growth factor receptor//Protein tyrosine kinase activity
Fostamatinib//Serine/threonine-protein kinase 26//Protein serine/threonine kinase activity
Fostamatinib//cAMP-dependent protein kinase catalytic subunit alpha//Ubiquitin protein ligase binding
Fostamatinib//Serine/threonine-protein kinase TAO2//Protein serine/threonine kinase activity
Fostamatinib//Angiopoietin-1 receptor//Transmembrane receptor protein tyrosine kinase activity
Fostamatinib//Activated CDC42 kinase 1//Ww domain binding
Fostamatinib//Dual specificity protein kinase TTK//Protein tyrosine kinase activity
Fostamatinib//Wee1-like protein kinase//Protein tyrosine kinase activity
Fostamatinib//Tyrosine-protein kinase Yes//Receptor binding
Fostamatinib//Mitogen-activated protein kinase kinase kinase MLT//Protein serine/threonine kinase activity
Fostamatinib//Tyrosine-protein kinase ZAP-70//Receptor binding
Fostamatinib//Abelson tyrosine-protein kinase 2//Receptor binding
Fostamatinib//Activin receptor type-1B//Ubiquitin protein ligase binding
Fostamatinib//ALK tyrosine kinase receptor//Transmembrane receptor protein tyrosine kinase activity
Fostamatinib//Aurora kinase A//Protein serine/threonine/tyrosine kinase activity
Fostamatinib//Aurora kinase B//Protein serine/threonine/tyrosine kinase activity
Fostamatinib//Aurora kinase C//Protein serine/threonine/tyrosine kinase activity
Fostamatinib//Serine/threonine-protein kinase B-raf//Protein serine/threonine kinase activity
Fostamatinib//Tyrosine-protein kinase BTK//Protein tyrosine kinase activity
Fostamatinib//Calcium/calmodulin-dependent protein kinase type II subunit alpha//Protein serine/threonine kinase activity
Fostamatinib//Calcium/calmodulin-dependent protein kinase type II subunit beta//Protein homodimerization activity
Fostamatinib//Calcium/calmodulin-dependent protein kinase type II subunit delta//Titin binding
Fostamatinib//Calcium/calmodulin-dependent protein kinase type II subunit gamma//Protein homodimerization activity
Fostamatinib//Peripheral plasma membrane protein CASK//Protein serine/threonine kinase activity
Fostamatinib//Cyclin-dependent kinase 1//Rna polymerase ii carboxy-terminal domain kinase activity
Fostamatinib//Cyclin-dependent kinase 4//Cyclin-dependent protein serine/threonine kinase regulator activity
Fostamatinib//Serine/threonine-protein kinase Chk1//Protein serine/threonine kinase activity
Fostamatinib//Serine/threonine-protein kinase Chk2//Ubiquitin protein ligase binding
Fostamatinib//Dual specificity protein kinase CLK1//Protein serine/threonine/tyrosine kinase activity
Fostamatinib//Dual specificity protein kinase CLK3//Protein tyrosine kinase activity
Fostamatinib//Macrophage colony-stimulating factor 1 receptor//Protein homodimerization activity
Fostamatinib//Tyrosine-protein kinase CSK//Receptor binding
Fostamatinib//Casein kinase II subunit alpha//Protein serine/threonine kinase activity
Fostamatinib//Casein kinase II subunit alpha'//Protein serine/threonine kinase activity
Fostamatinib//Epithelial discoidin domain-containing receptor 1//Transmembrane receptor protein tyrosine kinase activity
Fostamatinib//Discoidin domain-containing receptor 2//Transmembrane receptor protein tyrosine kinase activity
Fostamatinib//Epidermal growth factor receptor//Ubiquitin protein ligase binding
Fostamatinib//Ephrin type-A receptor 2//Transmembrane receptor protein tyrosine kinase activity
Fostamatinib//Ephrin type-A receptor 5//Transmembrane-ephrin receptor activity
Fostamatinib//Ephrin type-A receptor 7//Protein tyrosine kinase activity
Fostamatinib//Ephrin type-B receptor 2//Transmembrane-ephrin receptor activity
Fostamatinib//Ephrin type-B receptor 4//Transmembrane receptor protein tyrosine kinase activity
Fostamatinib//Receptor tyrosine-protein kinase erbB-2//Transmembrane signaling receptor activity
Fostamatinib//Receptor tyrosine-protein kinase erbB-4//Transmembrane receptor protein tyrosine kinase activity
Fostamatinib//Serine/threonine-protein kinase/endoribonuclease IRE1//Protein serine/threonine kinase activity
Fostamatinib//Fibroblast growth factor receptor 1//Protein tyrosine kinase activity
Fostamatinib//Fibroblast growth factor receptor 2//Protein tyrosine kinase activity
Fostamatinib//Fibroblast growth factor receptor 3//Protein tyrosine kinase activity
Fostamatinib//Tyrosine-protein kinase Fgr//Protein tyrosine kinase activity
Fostamatinib//Vascular endothelial growth factor receptor 1//Vegf-b-activated receptor activity
Fostamatinib//Receptor-type tyrosine-protein kinase FLT3//Vascular endothelial growth factor-activated receptor activity
Fostamatinib//Vascular endothelial growth factor receptor 3//Vascular endothelial growth factor-activated receptor activity
Fostamatinib//Tyrosine-protein kinase FRK//Receptor binding
Fostamatinib//Tyrosine-protein kinase Fyn//Protein tyrosine kinase activity
Fostamatinib//Glycogen synthase kinase-3 beta//Ubiquitin protein ligase binding
Fostamatinib//Tyrosine-protein kinase HCK//Receptor binding
Fostamatinib//Inhibitor of nuclear factor kappa-B kinase subunit beta//Scaffold protein binding
Fostamatinib//Insulin receptor//Receptor signaling protein tyrosine kinase activity
Fostamatinib//Interleukin-1 receptor-associated kinase 4//Protein serine/threonine kinase activity
Fostamatinib//Tyrosine-protein kinase JAK2//Sh2 domain binding
Fostamatinib//Tyrosine-protein kinase JAK3//Protein tyrosine kinase activity
Fostamatinib//Vascular endothelial growth factor receptor 2//Vascular endothelial growth factor-activated receptor activity
Fostamatinib//Mast/stem cell growth factor receptor Kit//Transmembrane receptor protein tyrosine kinase activity
Fostamatinib//Tyrosine-protein kinase Lck//Sh2 domain binding
Fostamatinib//LIM domain kinase 1//Zinc ion binding
Fostamatinib//Tyrosine-protein kinase Lyn//Receptor signaling protein tyrosine kinase activity
Fostamatinib//Dual specificity mitogen-activated protein kinase kinase 2//Scaffold protein binding
Fostamatinib//Mitogen-activated protein kinase kinase kinase 1//Zinc ion binding
Fostamatinib//Mitogen-activated protein kinase kinase kinase 2//Protein serine/threonine kinase activity
Fostamatinib//Mitogen-activated protein kinase kinase kinase 9//Protein tyrosine kinase activity
Fostamatinib//Mitogen-activated protein kinase 13//Protein serine/threonine kinase activity
Fostamatinib//Mitogen-activated protein kinase 14//Protein serine/threonine kinase activity
Fostamatinib//Mitogen-activated protein kinase 9//Transcription factor binding
Fostamatinib//Tyrosine-protein kinase Mer//Transmembrane receptor protein tyrosine kinase activity
Fostamatinib//Serine/threonine-protein kinase Nek11//Protein serine/threonine kinase activity
Fostamatinib//Serine/threonine-protein kinase Nek2//Protein serine/threonine kinase activity
Fostamatinib//High affinity nerve growth factor receptor//Transmembrane receptor protein tyrosine kinase activity
Fostamatinib//BDNF/NT-3 growth factors receptor//Protein homodimerization activity
Fostamatinib//Cyclin-dependent kinase 16//Protein serine/threonine kinase activity
Fostamatinib//Platelet-derived growth factor receptor alpha//Vascular endothelial growth factor-activated receptor activity
Fostamatinib//Platelet-derived growth factor receptor beta//Vascular endothelial growth factor binding
Fostamatinib//3-phosphoinositide-dependent protein kinase 1//Protein serine/threonine kinase activity
Fostamatinib//Cyclin-dependent kinase 15//Protein serine/threonine kinase activity
Fostamatinib//Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform//Phosphatidylinositol-4,5-bisphosphate 3-kinase activity
Fostamatinib//Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform//Protein serine/threonine kinase activity
Fostamatinib//Serine/threonine-protein kinase pim-1//Transcription factor binding
Fostamatinib//Serine/threonine-protein kinase PLK1//Protein serine/threonine kinase activity
Fostamatinib//5'-AMP-activated protein kinase catalytic subunit alpha-1//Tau-protein kinase activity
Fostamatinib//5'-AMP-activated protein kinase catalytic subunit alpha-1//Tau-protein kinase activity
Fostamatinib//5'-AMP-activated protein kinase catalytic subunit alpha-2//Protein serine/threonine/tyrosine kinase activity
Fostamatinib//5'-AMP-activated protein kinase subunit beta-1//Protein kinase activity
Fostamatinib//5'-AMP-activated protein kinase subunit beta-2//Identical protein binding
Fostamatinib//5'-AMP-activated protein kinase subunit gamma-1//Protein kinase binding
Fostamatinib//5'-AMP-activated protein kinase subunit gamma-2//Protein kinase binding
Fostamatinib//5'-AMP-activated protein kinase subunit gamma-3//Protein kinase binding
Fostamatinib//cAMP-dependent protein kinase catalytic subunit beta//Ubiquitin protein ligase binding
Fostamatinib//Protein kinase C delta type//Protein serine/threonine kinase activity
Fostamatinib//Protein kinase C epsilon type//Signal transducer activity
Fostamatinib//Protein kinase C iota type//Protein serine/threonine kinase activity
Fostamatinib//Focal adhesion kinase 1//Signal transducer activity
Fostamatinib//Protein-tyrosine kinase 2-beta//Signal transducer activity
Fostamatinib//Protein-tyrosine kinase 6//Receptor binding
Fostamatinib//RAF proto-oncogene serine/threonine-protein kinase//Protein serine/threonine kinase activity
Fostamatinib//Proto-oncogene tyrosine-protein kinase receptor Ret//Transmembrane receptor protein tyrosine kinase activity
Fostamatinib//Rho-associated protein kinase 2//Structural molecule activity
Fostamatinib//Ribosomal protein S6 kinase alpha-1//Ribosomal protein s6 kinase activity
Fostamatinib//Ribosomal protein S6 kinase alpha-3//Ribosomal protein s6 kinase activity
Fostamatinib//Serine/threonine-protein kinase SIK1//Protein serine/threonine kinase activity
Fostamatinib//STE20-like serine/threonine-protein kinase//Protein serine/threonine kinase activity
Fostamatinib//Proto-oncogene tyrosine-protein kinase Src//Sh3/sh2 adaptor activity
Fostamatinib//Serine/threonine-protein kinase 17B//Protein serine/threonine kinase activity
Deutetrabenazine//Synaptic vesicular amine transporter//Monoamine transmembrane transporter activity
Brigatinib//ALK tyrosine kinase receptor//Transmembrane receptor protein tyrosine kinase activity
Brigatinib//Epidermal growth factor receptor//Ubiquitin protein ligase binding
Brigatinib//Tyrosine-protein kinase ABL1//Syntaxin binding
Brigatinib//Insulin-like growth factor 1 receptor//Protein tyrosine kinase activity
Brigatinib//Receptor-type tyrosine-protein kinase FLT3//Vascular endothelial growth factor-activated receptor activity
Brigatinib//Insulin receptor//Receptor signaling protein tyrosine kinase activity
Brigatinib//Hepatocyte growth factor receptor//Protein tyrosine kinase activity
Brigatinib//Receptor tyrosine-protein kinase erbB-4//Transmembrane receptor protein tyrosine kinase activity
Brigatinib//Receptor tyrosine-protein kinase erbB-2//Transmembrane signaling receptor activity
Betrixaban//Coagulation factor X//Serine-type endopeptidase activity
Copanlisib//Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform//Protein serine/threonine kinase activity
Copanlisib//Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform//Phosphatidylinositol-4,5-bisphosphate 3-kinase activity
Macimorelin//Growth hormone secretagogue receptor type 1//Peptide hormone binding
Levosalbutamol//Beta-2 adrenergic receptor//Protein homodimerization activity
Acemetacin//Prostaglandin G/H synthase 1//Prostaglandin-endoperoxide synthase activity
Acemetacin//Prostaglandin G/H synthase 2//Prostaglandin-endoperoxide synthase activity
Enasidenib//Isocitrate dehydrogenase [NADP], mitochondrial//Nad binding
Estradiolacetate//Estrogen receptor//Zinc ion binding
Estradiolacetate//Nuclear receptor subfamily 1 group I member 2//Zinc ion binding
Estradiolacetate//Estrogen receptor beta//Zinc ion binding
Estradiolacetate//Neuronal acetylcholine receptor subunit alpha-4//Ligand-gated ion channel activity
Estradiolacetate//Nuclear receptor coactivator 2//Transcription coactivator activity
Estradiolacetate//G-protein coupled estrogen receptor 1//Steroid hormone binding
Estradiolacetate//ATP synthase subunit a//Mitochondrial membrane ATP synthase (F(1)F(0) ATP synthase or Complex V) produces ATP from ADP in the presence of a proton gradient across the membrane which is generated by electron transport complexes of the respiratory chain. F-type ATPases consist of two structural domains, F(1) - containing the extramembraneous catalytic core and F(0) - containing the membrane proton channel, linked together by a central stalk and a peripheral stalk. During catalysis, ATP synthesis in the catalytic domain of F(1) is coupled via a rotary mechanism of the central stalk subunits to proton translocation. Key component of the proton channel; it may play a direct role in the translocation of protons across the membrane.
Estradiolacetate//Beclin-1//Plays a central role in autophagy (PubMed:23184933). Acts as core subunit of the PI3K complex that mediates formation of phosphatidylinositol 3-phosphate; different complex forms are believed to play a role in multiple membrane trafficking pathways: PI3KC3-C1 is involved in initiation of autophagosomes and PI3KC3-C2 in maturation of autophagosomes and endocytosis. Involved in regulation of degradative endocytic trafficking and required for the abcission step in cytokinesis, probably in the context of PI3KC3-C2 (PubMed:20643123, PubMed:20208530). Essential for the formation of PI3KC3-C2 but not PI3KC3-C1 PI3K complex forms. Involved in endocytosis (PubMed:25275521). Protects against infection by a neurovirulent strain of Sindbis virus (PubMed:9765397). May play a role in antiviral host defense.
Estradiolacetate//Estradiol 17-beta-dehydrogenase 2//Testosterone dehydrogenase (nad+) activity
Estradiolacetate//Estrogen-related receptor gamma//Zinc ion binding
Estradiolbenzoate//Estrogen receptor//Zinc ion binding
Estradiolbenzoate//Nuclear receptor subfamily 1 group I member 2//Zinc ion binding
Estradiolbenzoate//Estrogen receptor beta//Zinc ion binding
Estradiolbenzoate//Neuronal acetylcholine receptor subunit alpha-4//Ligand-gated ion channel activity
Estradiolbenzoate//Nuclear receptor coactivator 2//Transcription coactivator activity
Estradiolbenzoate//G-protein coupled estrogen receptor 1//Steroid hormone binding
Estradiolbenzoate//ATP synthase subunit a//Mitochondrial membrane ATP synthase (F(1)F(0) ATP synthase or Complex V) produces ATP from ADP in the presence of a proton gradient across the membrane which is generated by electron transport complexes of the respiratory chain. F-type ATPases consist of two structural domains, F(1) - containing the extramembraneous catalytic core and F(0) - containing the membrane proton channel, linked together by a central stalk and a peripheral stalk. During catalysis, ATP synthesis in the catalytic domain of F(1) is coupled via a rotary mechanism of the central stalk subunits to proton translocation. Key component of the proton channel; it may play a direct role in the translocation of protons across the membrane.
Estradiolbenzoate//Beclin-1//Plays a central role in autophagy (PubMed:23184933). Acts as core subunit of the PI3K complex that mediates formation of phosphatidylinositol 3-phosphate; different complex forms are believed to play a role in multiple membrane trafficking pathways: PI3KC3-C1 is involved in initiation of autophagosomes and PI3KC3-C2 in maturation of autophagosomes and endocytosis. Involved in regulation of degradative endocytic trafficking and required for the abcission step in cytokinesis, probably in the context of PI3KC3-C2 (PubMed:20643123, PubMed:20208530). Essential for the formation of PI3KC3-C2 but not PI3KC3-C1 PI3K complex forms. Involved in endocytosis (PubMed:25275521). Protects against infection by a neurovirulent strain of Sindbis virus (PubMed:9765397). May play a role in antiviral host defense.
Estradiolbenzoate//Estradiol 17-beta-dehydrogenase 2//Testosterone dehydrogenase (nad+) activity
Estradiolbenzoate//Estrogen-related receptor gamma//Zinc ion binding
Estradiolcypionate//Estrogen receptor//Zinc ion binding
Estradiolcypionate//Nuclear receptor subfamily 1 group I member 2//Zinc ion binding
Estradiolcypionate//Estrogen receptor beta//Zinc ion binding
Estradiolcypionate//Neuronal acetylcholine receptor subunit alpha-4//Ligand-gated ion channel activity
Estradiolcypionate//Nuclear receptor coactivator 2//Transcription coactivator activity
Estradiolcypionate//G-protein coupled estrogen receptor 1//Steroid hormone binding
Estradiolcypionate//ATP synthase subunit a//Mitochondrial membrane ATP synthase (F(1)F(0) ATP synthase or Complex V) produces ATP from ADP in the presence of a proton gradient across the membrane which is generated by electron transport complexes of the respiratory chain. F-type ATPases consist of two structural domains, F(1) - containing the extramembraneous catalytic core and F(0) - containing the membrane proton channel, linked together by a central stalk and a peripheral stalk. During catalysis, ATP synthesis in the catalytic domain of F(1) is coupled via a rotary mechanism of the central stalk subunits to proton translocation. Key component of the proton channel; it may play a direct role in the translocation of protons across the membrane.
Estradiolcypionate//Beclin-1//Plays a central role in autophagy (PubMed:23184933). Acts as core subunit of the PI3K complex that mediates formation of phosphatidylinositol 3-phosphate; different complex forms are believed to play a role in multiple membrane trafficking pathways: PI3KC3-C1 is involved in initiation of autophagosomes and PI3KC3-C2 in maturation of autophagosomes and endocytosis. Involved in regulation of degradative endocytic trafficking and required for the abcission step in cytokinesis, probably in the context of PI3KC3-C2 (PubMed:20643123, PubMed:20208530). Essential for the formation of PI3KC3-C2 but not PI3KC3-C1 PI3K complex forms. Involved in endocytosis (PubMed:25275521). Protects against infection by a neurovirulent strain of Sindbis virus (PubMed:9765397). May play a role in antiviral host defense.
Estradiolcypionate//Estradiol 17-beta-dehydrogenase 2//Testosterone dehydrogenase (nad+) activity
Estradiolcypionate//Estrogen-related receptor gamma//Zinc ion binding
Estradioldienanthate//Estrogen receptor//Zinc ion binding
Estradioldienanthate//Nuclear receptor subfamily 1 group I member 2//Zinc ion binding
Estradioldienanthate//Estrogen receptor beta//Zinc ion binding
Estradioldienanthate//Neuronal acetylcholine receptor subunit alpha-4//Ligand-gated ion channel activity
Estradioldienanthate//Nuclear receptor coactivator 2//Transcription coactivator activity
Estradioldienanthate//G-protein coupled estrogen receptor 1//Steroid hormone binding
Estradioldienanthate//ATP synthase subunit a//Mitochondrial membrane ATP synthase (F(1)F(0) ATP synthase or Complex V) produces ATP from ADP in the presence of a proton gradient across the membrane which is generated by electron transport complexes of the respiratory chain. F-type ATPases consist of two structural domains, F(1) - containing the extramembraneous catalytic core and F(0) - containing the membrane proton channel, linked together by a central stalk and a peripheral stalk. During catalysis, ATP synthesis in the catalytic domain of F(1) is coupled via a rotary mechanism of the central stalk subunits to proton translocation. Key component of the proton channel; it may play a direct role in the translocation of protons across the membrane.
Estradioldienanthate//Beclin-1//Plays a central role in autophagy (PubMed:23184933). Acts as core subunit of the PI3K complex that mediates formation of phosphatidylinositol 3-phosphate; different complex forms are believed to play a role in multiple membrane trafficking pathways: PI3KC3-C1 is involved in initiation of autophagosomes and PI3KC3-C2 in maturation of autophagosomes and endocytosis. Involved in regulation of degradative endocytic trafficking and required for the abcission step in cytokinesis, probably in the context of PI3KC3-C2 (PubMed:20643123, PubMed:20208530). Essential for the formation of PI3KC3-C2 but not PI3KC3-C1 PI3K complex forms. Involved in endocytosis (PubMed:25275521). Protects against infection by a neurovirulent strain of Sindbis virus (PubMed:9765397). May play a role in antiviral host defense.
Estradioldienanthate//Estradiol 17-beta-dehydrogenase 2//Testosterone dehydrogenase (nad+) activity
Estradioldienanthate//Estrogen-related receptor gamma//Zinc ion binding
Estradiolvalerate//Estrogen receptor//Zinc ion binding
Estradiolvalerate//Nuclear receptor subfamily 1 group I member 2//Zinc ion binding
Estradiolvalerate//Estrogen receptor beta//Zinc ion binding
Estradiolvalerate//Neuronal acetylcholine receptor subunit alpha-4//Ligand-gated ion channel activity
Estradiolvalerate//Nuclear receptor coactivator 2//Transcription coactivator activity
Estradiolvalerate//G-protein coupled estrogen receptor 1//Steroid hormone binding
Estradiolvalerate//ATP synthase subunit a//Mitochondrial membrane ATP synthase (F(1)F(0) ATP synthase or Complex V) produces ATP from ADP in the presence of a proton gradient across the membrane which is generated by electron transport complexes of the respiratory chain. F-type ATPases consist of two structural domains, F(1) - containing the extramembraneous catalytic core and F(0) - containing the membrane proton channel, linked together by a central stalk and a peripheral stalk. During catalysis, ATP synthesis in the catalytic domain of F(1) is coupled via a rotary mechanism of the central stalk subunits to proton translocation. Key component of the proton channel; it may play a direct role in the translocation of protons across the membrane.
Estradiolvalerate//Beclin-1//Plays a central role in autophagy (PubMed:23184933). Acts as core subunit of the PI3K complex that mediates formation of phosphatidylinositol 3-phosphate; different complex forms are believed to play a role in multiple membrane trafficking pathways: PI3KC3-C1 is involved in initiation of autophagosomes and PI3KC3-C2 in maturation of autophagosomes and endocytosis. Involved in regulation of degradative endocytic trafficking and required for the abcission step in cytokinesis, probably in the context of PI3KC3-C2 (PubMed:20643123, PubMed:20208530). Essential for the formation of PI3KC3-C2 but not PI3KC3-C1 PI3K complex forms. Involved in endocytosis (PubMed:25275521). Protects against infection by a neurovirulent strain of Sindbis virus (PubMed:9765397). May play a role in antiviral host defense.
Estradiolvalerate//Estradiol 17-beta-dehydrogenase 2//Testosterone dehydrogenase (nad+) activity
Estradiolvalerate//Estrogen-related receptor gamma//Zinc ion binding
Cholinesalicylate//Acetylcholinesterase//Serine hydrolase activity
Cholinesalicylate//Choline-phosphate cytidylyltransferase A//Lipid binding
Cholinesalicylate//Phospholipase D2//Phospholipase d activity
Cholinesalicylate//Cholinesterase//Identical protein binding
Cholinesalicylate//Phospholipase D1//Phospholipase d activity
Cholinesalicylate//Neuronal acetylcholine receptor subunit alpha-7//Toxic substance binding
Nabiximols//Cannabinoid receptor 1//Drug binding
Nabiximols//Cannabinoid receptor 2//Cannabinoid receptor activity
Nabiximols//Glycine receptor subunit alpha-1//Transmitter-gated ion channel activity
Nabiximols//Glycine receptor subunit alpha-1//Transmitter-gated ion channel activity
Nabiximols//Glycine receptor subunit beta//Glycine binding
Nabiximols//Glycine receptor subunit alpha-3//Transmitter-gated ion channel activity
Nabiximols//N-arachidonyl glycine receptor//G-protein coupled receptor activity
Nabiximols//G-protein coupled receptor 55//G-protein coupled receptor activity
Nabiximols//5-hydroxytryptamine receptor 1A//Serotonin receptor activity
Nabiximols//5-hydroxytryptamine receptor 2A//Virus receptor activity
Nabiximols//Neuronal acetylcholine receptor subunit alpha-7//Toxic substance binding
Nabiximols//Delta-type opioid receptor//Opioid receptor activity
Nabiximols//Mu-type opioid receptor//Voltage-gated calcium channel activity
Nabiximols//Peroxisome proliferator-activated receptor gamma//Zinc ion binding
Nabiximols//Transient receptor potential cation channel subfamily V member 1//Transmembrane signaling receptor activity
Nabiximols//Voltage-dependent T-type calcium channel subunit alpha-1G//Scaffold protein binding
Nabiximols//Voltage-dependent T-type calcium channel subunit alpha-1H//Scaffold protein binding
Nabiximols//Voltage-dependent T-type calcium channel subunit alpha-1I//Voltage-gated calcium channel activity
Nabiximols//Transient receptor potential cation channel subfamily A member 1//Temperature-gated cation channel activity
Nabiximols//Transient receptor potential cation channel subfamily M member 8//Calcium channel activity
Nabiximols//Transient receptor potential cation channel subfamily V member 3//Calcium channel activity
Nabiximols//Transient receptor potential cation channel subfamily V member 4//Non-selective calcium permeant cation channel involved in osmotic sensitivity and mechanosensitivity. Activation by exposure to hypotonicity within the physiological range exhibits an outward rectification (PubMed:18826956, PubMed:18695040). Also activated by heat, low pH, citrate and phorbol esters (PubMed:18826956, PubMed:18695040). Increase of intracellular Ca(2+) potentiates currents. Channel activity seems to be regulated by a calmodulin-dependent mechanism with a negative feedback mechanism (PubMed:12724311, PubMed:18826956). Promotes cell-cell junction formation in skin keratinocytes and plays an important role in the formation and/or maintenance of functional intercellular barriers (By similarity). Acts as a regulator of intracellular Ca(2+) in synoviocytes (PubMed:19759329). Plays an obligatory role as a molecular component in the nonselective cation channel activation induced by 4-alpha-phorbol 12,13-didecanoate and hypotonic stimulation in synoviocytes and also regulates production of IL-8 (PubMed:19759329). Together with PKD2, forms mechano- and thermosensitive channels in cilium (PubMed:18695040). Negatively regulates expression of PPARGC1A, UCP1, oxidative metabolism and respiration in adipocytes (By similarity). Regulates expression of chemokines and cytokines related to proinflammatory pathway in adipocytes (By similarity). Together with AQP5, controls regulatory volume decrease in salivary epithelial cells (By similarity). Required for normal development and maintenance of bone and cartilage (PubMed:26249260).
Nabiximols//Prostaglandin G/H synthase 1//Prostaglandin-endoperoxide synthase activity
Nabiximols//Prostaglandin G/H synthase 2//Prostaglandin-endoperoxide synthase activity
Nabiximols//Acetyl-CoA acetyltransferase, mitochondrial//Metal ion binding
Nabiximols//Steroid 17-alpha-hydroxylase/17,20 lyase//Steroid 17-alpha-monooxygenase activity
Nabiximols//3-hydroxy-3-methylglutaryl-coenzyme A reductase//Nadph binding
Nabiximols//Glutathione reductase, mitochondrial//Nadp binding
Nabiximols//Glutathione peroxidase 1//Sh3 domain binding
Nabiximols//Indoleamine 2,3-dioxygenase 1//Tryptophan 2,3-dioxygenase activity
Nabiximols//Cytochrome P450 1B1//Oxygen binding
Nabiximols//Cytochrome P450 3A5//Oxygen binding
Nabiximols//Cytochrome P450 2D6//Steroid hydroxylase activity
Nabiximols//Cytochrome P450 1A2//Oxidoreductase activity, acting on paired donors, with incorporation or reduction of molecular oxygen, reduced flavin or flavoprotein as one donor, and incorporation of one atom of oxygen
Nabiximols//Cytochrome P450 1A1//Vitamin d 24-hydroxylase activity
Nabiximols//Cytochrome P450 3A7//Oxygen binding
Nabiximols//Quinone oxidoreductase//Zinc ion binding
Nabiximols//Catalase//Receptor binding
Nabiximols//Fatty-acid amide hydrolase 1//Fatty acid amide hydrolase activity
Nabiximols//Superoxide dismutase [Cu-Zn]//Zinc ion binding
